2-chloro-n(6)cyclopentyladenosine has been researched along with isoproterenol in 11 studies
Studies (2-chloro-n(6)cyclopentyladenosine) | Trials (2-chloro-n(6)cyclopentyladenosine) | Recent Studies (post-2010) (2-chloro-n(6)cyclopentyladenosine) | Studies (isoproterenol) | Trials (isoproterenol) | Recent Studies (post-2010) (isoproterenol) |
---|---|---|---|---|---|
252 | 0 | 43 | 30,780 | 803 | 2,640 |
Protein | Taxonomy | 2-chloro-n(6)cyclopentyladenosine (IC50) | isoproterenol (IC50) |
---|---|---|---|
Beta-2 adrenergic receptor | Homo sapiens (human) | 0.246 | |
Beta-1 adrenergic receptor | Homo sapiens (human) | 0.333 | |
Beta-2 adrenergic receptor | Rattus norvegicus (Norway rat) | 0.2125 | |
Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | 1.77 | |
Beta-1 adrenergic receptor | Rattus norvegicus (Norway rat) | 0.2125 | |
Beta-3 adrenergic receptor | Rattus norvegicus (Norway rat) | 0.2125 | |
Beta-2 adrenergic receptor | Canis lupus familiaris (dog) | 0.6667 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (54.55) | 18.2507 |
2000's | 4 (36.36) | 29.6817 |
2010's | 1 (9.09) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Klotz, KN; Schwabe, U; Tawfik-Schlieper, H; Wilken, A | 1 |
Banerjee, A; Bensard, DD; Brew, EC; Fullerton, DA; Hahn, AR; McIntyre, RC | 1 |
Schiele, JO; Schwabe, U | 1 |
Armstrong, S; Downey, JM; Ganote, CE | 1 |
Adkins, WK; Allison, RC; Barnard, JW; Moore, TM; Prasad, VR; Taylor, AE | 1 |
Dobson, JG; Fenton, RA; Sawmiller, DR | 1 |
Lasley, RD; Mentzer, RM; Narayan, P | 1 |
Chung, ES; Dobson, JG; Fenton, RA; Lorbar, M; Meyer, TE; Norton, GR; Perlini, S; Woodiwiss, AJ | 1 |
Dobson, JG; Fenton, RA; Shea, LG | 1 |
Dobson, JG; Fenton, RA; Tikh, EI | 1 |
Dobson, JG; Fenton, RA; Ikebe, M; Komatsu, S; Shea, LG | 1 |
11 other study(ies) available for 2-chloro-n(6)cyclopentyladenosine and isoproterenol
Article | Year |
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Pharmacological characterization of the adenylate cyclase-coupled adenosine receptor in isolated guinea pig atrial myocytes.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Carrier Proteins; Cyclic AMP; Cyclic AMP Receptor Protein; Female; Guinea Pigs; Heart Atria; Isoproterenol; Male; Myocardium; Pertussis Toxin; Virulence Factors, Bordetella | 1990 |
Adenosine A1-receptor mechanisms antagonize beta-adrenergic pulmonary vasodilation in hypoxia.
Topics: Adenosine; Animals; Colforsin; Isoproterenol; Oxygen; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Vasodilation | 1994 |
Characterization of the adenosine receptor in microvascular coronary endothelial cells.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclase Inhibitors; Animals; Antihypertensive Agents; Cells, Cultured; Colforsin; Coronary Vessels; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; Guinea Pigs; Isoproterenol; Myocardium; Phenethylamines; Phenylisopropyladenosine; Receptors, Purinergic P1; Thioinosine; Vasodilator Agents | 1994 |
Adenosine and A1 selective agonists offer minimal protection against ischaemic injury to isolated rat cardiomyocytes.
Topics: Adenosine; Animals; Carbachol; Cell Death; Cells, Cultured; Iodoacetates; Iodoacetic Acid; Isoproterenol; Male; Myocardial Ischemia; Myocardium; Rats; Rats, Sprague-Dawley; Theophylline | 1993 |
Adenosine prevents PMA-induced lung injury via an A2 receptor mechanism.
Topics: Adenosine; Animals; Blood Pressure; Capillary Permeability; Cyclic AMP; Dogs; Endothelium; Female; In Vitro Techniques; Isoproterenol; Lung Diseases; Male; Neutrophils; Pulmonary Circulation; Purinergic Antagonists; Receptors, Purinergic; Tetradecanoylphorbol Acetate; Vascular Resistance; Xanthines | 1993 |
Myocardial adenosine A1-receptor sensitivity during juvenile and adult stages of maturation.
Topics: Adenosine; Adenylyl Cyclases; Adrenergic beta-Agonists; Aging; Animals; Heart; Heart Rate; Isoproterenol; Male; Myocardial Contraction; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Vasodilator Agents; Xanthines | 1998 |
Phosphatase inhibitor cantharidin blocks adenosine A(1) receptor anti-adrenergic effect in rat cardiac myocytes.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adrenergic beta-Agonists; Animals; Calcium; Cantharidin; Cyclic AMP; Enzyme Inhibitors; Intracellular Membranes; Isoproterenol; Male; Myocardial Contraction; Myocardium; Phosphoric Monoester Hydrolases; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1 | 2000 |
Antiadrenergic effects of adenosine in pressure overload hypertrophy.
Topics: Adenosine; Adrenergic Antagonists; Adrenergic beta-Agonists; Animals; Blood Pressure; Body Weight; Caffeine; Calcium; Cardiomegaly; Cells, Cultured; Coronary Circulation; Disease Models, Animal; Echocardiography; In Vitro Techniques; Inosine; Isoproterenol; Male; Myocardial Contraction; Myocardium; Organ Size; Perfusion; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley | 2001 |
Beta-adrenergic and antiadrenergic modulation of cardiac adenylyl cyclase is influenced by phosphorylation.
Topics: Adenosine; Adenylyl Cyclases; Adrenergic beta-Agonists; Alkaline Phosphatase; Animals; Cyclic AMP-Dependent Protein Kinases; Heart Ventricles; Isoproterenol; Membrane Proteins; Myocardium; Phosphorylation; Precipitin Tests; Purinergic P1 Receptor Agonists; Rats; Receptors, Adrenergic, beta-1; Receptors, Purinergic P1 | 2003 |
Contractile effects of adenosine A1 and A2A receptors in isolated murine hearts.
Topics: Adenosine; Animals; Heart; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Myocardial Contraction; Myocardial Ischemia; Phenethylamines; Receptor, Adenosine A1; Receptor, Adenosine A2A; Xanthines | 2006 |
Crosstalk between adenosine A1 and β1-adrenergic receptors regulates translocation of PKCε in isolated rat cardiomyocytes.
Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adrenergic beta-1 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Intracellular Signaling Peptides and Proteins; Isoproterenol; Isoquinolines; Membrane Proteins; Myocardium; Myocytes, Cardiac; Organ Culture Techniques; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Protein Transport; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adrenergic, beta-1; Signal Transduction; Sulfonamides; Xanthines | 2012 |