Page last updated: 2024-09-03

2-chloro-n(6)cyclopentyladenosine and colforsin

2-chloro-n(6)cyclopentyladenosine has been researched along with colforsin in 7 studies

Compound Research Comparison

Studies
(2-chloro-n(6)cyclopentyladenosine)
Trials
(2-chloro-n(6)cyclopentyladenosine)
Recent Studies (post-2010)
(2-chloro-n(6)cyclopentyladenosine)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
25204313,460461,298

Protein Interaction Comparison

ProteinTaxonomy2-chloro-n(6)cyclopentyladenosine (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (71.43)18.2507
2000's1 (14.29)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Banerjee, A; Bensard, DD; Brew, EC; Fullerton, DA; Hahn, AR; McIntyre, RC1
Schiele, JO; Schwabe, U1
Christofi, FL; Wood, JD1
Bottrill, FE; Hiley, CR; Richardson, PJ; Warnock, J1
Bagley, EE; Christie, MJ; Vaughan, CW1
Doering, A; Middlekauff, HR; Weiss, JN1
Dobson, JG; Fenton, RA; Ikebe, M; Komatsu, S; Shea, LG1

Other Studies

7 other study(ies) available for 2-chloro-n(6)cyclopentyladenosine and colforsin

ArticleYear
Adenosine A1-receptor mechanisms antagonize beta-adrenergic pulmonary vasodilation in hypoxia.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Adenosine; Animals; Colforsin; Isoproterenol; Oxygen; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Vasodilation

1994
Characterization of the adenosine receptor in microvascular coronary endothelial cells.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclase Inhibitors; Animals; Antihypertensive Agents; Cells, Cultured; Colforsin; Coronary Vessels; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; Guinea Pigs; Isoproterenol; Myocardium; Phenethylamines; Phenylisopropyladenosine; Receptors, Purinergic P1; Thioinosine; Vasodilator Agents

1994
Effects of PACAP on morphologically identified myenteric neurons in guinea pig small bowel.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 1

    Topics: Action Potentials; Adenosine; Animals; Colforsin; Guinea Pigs; Intestine, Small; Male; Myenteric Plexus; Neuroglia; Neurons; Neuropeptides; Neurotransmitter Agents; Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Cell Surface; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Pituitary Hormone

1993
Effects of pH on responses to adenosine, CGS 21680, carbachol and nitroprusside in the isolated perfused superior mesenteric arterial bed of the rat.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Carbachol; Colforsin; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Nitroprusside; Perfusion; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Vascular Resistance; Vasoconstrictor Agents; Vasodilator Agents; Xanthines

1995
Inhibition by adenosine receptor agonists of synaptic transmission in rat periaqueductal grey neurons.
    The Journal of physiology, 1999, Apr-01, Volume: 516 ( Pt 1)

    Topics: Action Potentials; Adenosine; Animals; Colforsin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Synaptic Transmission

1999
Adenosine enhances neuroexcitability by inhibiting a slow postspike afterhyperpolarization in rabbit vagal afferent neurons.
    Circulation, 2001, Mar-06, Volume: 103, Issue:9

    Topics: Action Potentials; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cadmium; Colforsin; Neurons, Afferent; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rabbits; Receptors, Purinergic P1; Time Factors; Vagus Nerve; Xanthines

2001
Crosstalk between adenosine A1 and β1-adrenergic receptors regulates translocation of PKCε in isolated rat cardiomyocytes.
    Journal of cellular physiology, 2012, Volume: 227, Issue:9

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adrenergic beta-1 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Intracellular Signaling Peptides and Proteins; Isoproterenol; Isoquinolines; Membrane Proteins; Myocardium; Myocytes, Cardiac; Organ Culture Techniques; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Protein Transport; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adrenergic, beta-1; Signal Transduction; Sulfonamides; Xanthines

2012