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2-aminothiazoline and thiazoles

2-aminothiazoline has been researched along with thiazoles in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199010 (40.00)18.7374
1990's1 (4.00)18.2507
2000's9 (36.00)29.6817
2010's4 (16.00)24.3611
2020's1 (4.00)2.80

Authors

AuthorsStudies
Kazarov, AR; Sobolev, AS; Tertov, VV1
Goncharenko, EN; Graevskaia, EE; Zolotareva, LT1
Ando, K; Nagatomi, H1
Ambrus, JL; Bock, FG; Mirand, EA; Pine, MJ1
Huertas, A; Smeyers, YG1
Díaz Gil, JJ; Trilla, C1
Brugarolas, A; Gosálvez, M1
Huang, ZX; May, PM; Williams, DR1
Benkö, G; Perjés, I; Rónai, E; Szabó, DL1
Fowler, M; Furfine, ES; Garvey, EP; Harmon, MF; Marshall, S; Oplinger, JA; Paith, JE; Sherman, PA; Tanoury, GJ1
Král, V; Li, H; Martásek, P; Masters, BS; Poulos, TL; Raman, CS1
Andriantsitohaina, R; Martínez, MC; Randriamboavonjy, V; Stoclet, J1
Simkeviciene, V; Straukas, J; Uleckiene, S1
TISLER, M1
Lynch, DE1
Li, Z; Qian, X; Yang, Q1
Bolos, CA; Chaviara, AT; Christidis, PC; Chrysogelou, E; Hadjipavlou-Litina, DJ; Papageorgiou, A1
Bolos, CA; Chaviara, AT; Hadjipavlou-Litina, D; Pontiki, E1
Caille, S; Cui, S; Faul, MM; Hwang, TL; Wang, X1
Bolos, CA; Cox, PJ; Psomas, G1
Bernacki, AL; Hennings, DD; Zhu, L1
Effertz, T; Schlittgen, R1
Atreya, HS; Chandrashekaran, IR; Debono, CO; Devine, SM; Jaipuria, G; Krishnarjuna, B; Lam, R; Lim, SS; MacRaild, CA; Norton, RS; Scammells, PJ; Scanlon, MJ; Yagi, H1
Bachurin, SO; Boltneva, NP; Lushchekina, SV; Makhaeva, GF; Proshin, AN; Richardson, RJ; Serebryakova, OG; Serkov, IV; Stupina, TS; Terentiev, AA1
Ahmed, N; Ali, S; Farooq, S; Hussain, M; Khan, MA; Khan, S; Shamim, S1

Trials

1 trial(s) available for 2-aminothiazoline and thiazoles

ArticleYear
Preliminary clinical results with norgamem (thioproline) and revercan (2-amino-2-thiazoline): the first inducers of reverse transformation.
    Recent results in cancer research. Fortschritte der Krebsforschung. Progres dans les recherches sur le cancer, 1982, Volume: 80

    Topics: Adult; Aged; Antineoplastic Agents; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Clinical Trials as Topic; Drug Evaluation; Female; Head and Neck Neoplasms; Humans; Male; Middle Aged; Neoplasms; Thiazoles; Thiazolidines; Urinary Bladder Neoplasms

1982

Other Studies

24 other study(ies) available for 2-aminothiazoline and thiazoles

ArticleYear
Effects of radioprotectors on the cAMP and cGMP systems.
    Radiation and environmental biophysics, 1984, Volume: 23, Issue:2

    Topics: Adenylyl Cyclases; Animals; beta-Aminoethyl Isothiourea; Biogenic Amines; Cyclic AMP; Cyclic GMP; Enzyme Activation; Guanylate Cyclase; Male; Mercaptoethylamines; Mice; Phosphoric Diester Hydrolases; Protein Kinases; Radiation-Protective Agents; Rats; Rats, Inbred Strains; Thiazoles; Thiourea

1984
[Effect of 2-amino-2-thiazoline on the sulfhydryl group content of yeasts of various degrees of radiosensitivity].
    Nauchnye doklady vysshei shkoly. Biologicheskie nauki, 1984, Issue:5

    Topics: Diploidy; Haploidy; Pichia; Radiation Tolerance; Radiation-Protective Agents; Saccharomyces cerevisiae; Sulfhydryl Compounds; Thiazoles; Yeasts

1984
Studies on the anti-inflammatory activity and ulcerogenic adverse effect of thiazole derivatives, especially 2-amino-thiazoleacetic acid derivatives.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:5

    Topics: Acetates; Animals; Anti-Inflammatory Agents; Edema; Erythrocytes; Hemolysis; Male; Protease Inhibitors; Protein Denaturation; Rats; Rats, Inbred Strains; Stomach Ulcer; Structure-Activity Relationship; Thiazoles

1984
Antitumor studies of 2-amino-2-thiazoline and other tumor-modifying agents.
    Journal of medicine, 1983, Volume: 14, Issue:5-6

    Topics: Animals; Antineoplastic Agents; Antioxidants; Cell Line; Dimethylhydrazines; Female; Methylcholanthrene; Mice; Neoplasm Transplantation; Neoplasms, Experimental; Thiazoles; Thiazolidines

1983
[Distribution of electric charges in 2 substances inducing tumor cell regression].
    Revista espanola de oncologia, 1983, Volume: 30, Issue:4

    Topics: Antineoplastic Agents; Electrochemistry; Thiazoles; Thiazolidines

1983
[Diminution of the rate of growth of HeLa cells caused by thioproline (Tp) and 2-aminothiazoline HCl (2-AT). Effect of L-proline].
    Revista espanola de oncologia, 1982, Volume: 29, Issue:4

    Topics: Growth Inhibitors; HeLa Cells; Humans; Proline; Thiazoles; Thiazolidines

1982
Reverse transformation agent and their ability to complex metal ions.
    European journal of cancer & clinical oncology, 1981, Volume: 17, Issue:10

    Topics: Ligands; Metals; Thiazoles; Thiazolidines

1981
[Quantitative determination of the ratio of 2-aminothiazoline contamination in IXECUR enteric-coated dragees].
    Acta pharmaceutica Hungarica, 1981, Volume: 51, Issue:4

    Topics: beta-Aminoethyl Isothiourea; Drug Contamination; Radiation-Protective Agents; Spectrophotometry; Thiazoles

1981
Potent and selective inhibition of human nitric oxide synthases. Inhibition by non-amino acid isothioureas.
    The Journal of biological chemistry, 1994, Oct-28, Volume: 269, Issue:43

    Topics: Amino Acid Oxidoreductases; Animals; Arginine; Endothelium, Vascular; Enzyme Induction; Humans; Isoenzymes; Isothiuronium; Kinetics; Mice; Models, Chemical; Neurons; Nitric Oxide Synthase; Species Specificity; Structure-Activity Relationship; Thiazoles; Thiourea

1994
Mapping the active site polarity in structures of endothelial nitric oxide synthase heme domain complexed with isothioureas.
    Journal of inorganic biochemistry, 2000, Aug-31, Volume: 81, Issue:3

    Topics: Binding Sites; Crystallography, X-Ray; Endothelium; Heme; Humans; Isothiuronium; Kinetics; Models, Molecular; Nitric Oxide Synthase; Protein Binding; Protein Conformation; Protein Structure, Secondary; Protein Structure, Tertiary; Thiazoles; Thiourea

2000
Potentiation by aminoethylisothiourea of the extra-cellular Ca(2+) component of norepinephrine-induced contraction in rat femoral arteries.
    Biochemical pharmacology, 2001, Jan-01, Volume: 61, Issue:1

    Topics: Animals; Calcium; Drug Synergism; Endothelium, Vascular; Enzyme Inhibitors; Femoral Artery; Guanidines; In Vitro Techniques; Male; Nitric Oxide Synthase; Norepinephrine; Prostaglandin-Endoperoxide Synthases; Protein Kinase C; Radiation-Protective Agents; Rats; Rats, Wistar; Thiazoles; Thiourea; Vasoconstriction

2001
N-acetil-l-cysteine and 2-amino-2-thiiazoline N-acetyl-l-cysteinate as a possible cancer chemopreventive agents in murine models.
    Acta biologica Hungarica, 2002, Volume: 53, Issue:3

    Topics: Acetylcysteine; Adenoma; Animals; Anticarcinogenic Agents; Dose-Response Relationship, Drug; Female; Lung Neoplasms; Mice; Mice, Inbred BALB C; Models, Animal; Thiazoles

2002
[Chemistry of substituted thiosemicarbazides and thioureas. V. Contribution on the synthesis and conversion of 1-substituted thiocarbamylethylene-imines in N-substituted derivatives of 2-amino-2-thiazoline].
    Archiv der Pharmazie und Berichte der Deutschen Pharmazeutischen Gesellschaft, 1958, Volume: 291/63, Issue:9

    Topics: Ethylamines; Imines; Semicarbazides; Thiazoles; Thiocarbamates; Thiourea

1958
2-Amino-2-thiazoline and its 1:1 organic salt with 2-naphthoxyacetic acid.
    Acta crystallographica. Section C, Crystal structure communications, 2004, Volume: 60, Issue:Pt 9

    Topics: Antineoplastic Agents; Crystallography, X-Ray; Glycolates; Hydrogen Bonding; Molecular Structure; Thiazoles

2004
Novel 2-aminothiazonaphthalimides as visible light activatable photonucleases: effects of intercalation, heterocyclic-fused area and side chains.
    Bioorganic & medicinal chemistry letters, 2005, Apr-01, Volume: 15, Issue:7

    Topics: Deoxyribonucleases; DNA Damage; Heterocyclic Compounds, 4 or More Rings; Intercalating Agents; Light; Nucleic Acid Conformation; Photolysis; Phthalimides; Structure-Activity Relationship; Superoxides; Thiazoles

2005
In vivo anticancer, anti-inflammatory, and toxicity studies of mixed-ligand Cu(II) complexes of dien and its Schiff dibases with heterocyclic aldehydes and 2-amino-2-thiazoline. Crystal structure of [Cu(dien)(Br)(2a-2tzn)](Br)(H(2)O).
    Journal of inorganic biochemistry, 2005, Volume: 99, Issue:11

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Copper; Crystallography, X-Ray; Female; Heterocyclic Compounds; Inflammation; Leukemia, Lymphoid; Ligands; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Polyamines; Rats; Schiff Bases; Spectrophotometry, Infrared; Thiazoles

2005
Evaluation of anti-inflammatory and antioxidant activities of mixed-ligand Cu(II) complexes of dien and its Schiff dibases with heterocyclic aldehydes and 2-amino-2-thiazoline.
    Bioorganic & medicinal chemistry letters, 2006, Apr-15, Volume: 16, Issue:8

    Topics: Aldehydes; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Carrageenan; Cations, Divalent; Copper; Edema; Free Radical Scavengers; Organometallic Compounds; Rats; Schiff Bases; Structure-Activity Relationship; Thiazoles

2006
Two asymmetric syntheses of AMG 221, an inhibitor of 11beta-hydroxysteroid dehydrogenase type 1.
    The Journal of organic chemistry, 2009, May-15, Volume: 74, Issue:10

    Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 1; Alcohols; Chlorides; Cyclization; Enzyme Inhibitors; Solvents; Stereoisomerism; Substrate Specificity; Thiazoles

2009
Characterization and DNA-interaction studies of 1,1-dicyano-2,2-ethylene dithiolate Ni(II) mixed-ligand complexes with 2-amino-5-methyl thiazole, 2-amino-2-thiazoline and imidazole. Crystal structure of [Ni(i-MNT)(2a-5mt)(2)].
    Bioorganic & medicinal chemistry, 2009, Aug-15, Volume: 17, Issue:16

    Topics: Animals; Cattle; Crystallography, X-Ray; DNA; Imidazoles; Ligands; Molecular Conformation; Nickel; Organometallic Compounds; Spectrophotometry, Ultraviolet; Thiazoles

2009
A selective and convenient method for the synthesis of 2-phenylaminothiazolines.
    Organic letters, 2010, Dec-03, Volume: 12, Issue:23

    Topics: Cyclization; Molecular Structure; Thiazoles

2010
[Cigarette prices, tobacco taxes and the proportion of contraband cigarettes in Germany].
    Gesundheitswesen (Bundesverband der Arzte des Offentlichen Gesundheitsdienstes (Germany)), 2013, Volume: 75, Issue:6

    Topics: Crime; Germany; Health Policy; Humans; Income; Prevalence; Smoking; Taxes; Thiazoles; Tobacco Industry; Tobacco Products

2013
Solution NMR characterization of apical membrane antigen 1 and small molecule interactions as a basis for designing new antimalarials.
    Journal of molecular recognition : JMR, 2016, Volume: 29, Issue:6

    Topics: Amino Acid Sequence; Antigens, Protozoan; Antimalarials; Benzimidazoles; Binding Sites; Drug Design; Humans; Membrane Proteins; Models, Molecular; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Protein Binding; Protein Conformation; Protozoan Proteins; Pyrazoles; Small Molecule Libraries; Thiazoles

2016
Synthesis, molecular docking and biological evaluation of N,N-disubstituted 2-aminothiazolines as a new class of butyrylcholinesterase and carboxylesterase inhibitors.
    Bioorganic & medicinal chemistry, 2016, Mar-01, Volume: 24, Issue:5

    Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carboxylesterase; Cholinesterase Inhibitors; Enzyme Inhibitors; Horses; Humans; Molecular Docking Simulation; Swine; Thiazoles

2016
Antimicrobial and synergistic activity of thiazoline derivatives in combination with conventional antibiotics against multidrug resistant Staphylococcus aureus isolated from abscess drainage samples.
    Pakistan journal of pharmaceutical sciences, 2020, Volume: 33, Issue:5(Suppleme

    Topics: Abscess; Anti-Bacterial Agents; Disk Diffusion Antimicrobial Tests; Drainage; Drug Resistance, Multiple, Bacterial; Drug Synergism; Drug Therapy, Combination; Humans; Ribotyping; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Thiazolidines

2020