2-amino-5-phosphonovalerate and diazepam

2-amino-5-phosphonovalerate has been researched along with diazepam in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-19906 (19.35)18.7374
1990's18 (58.06)18.2507
2000's3 (9.68)29.6817
2010's4 (12.90)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Sage, GP; Sethy, VH1
Bagetta, G; Bowery, NG; Britton, P; Nisticó, G; Whitton, P1
Baron, BM; Chi, EM; Harrison, BL; Kehne, JH; McCloskey, TC; Palfreyman, MG; Whitten, JP1
Luhmann, HJ; Prince, DA1
Czuczwar, SJ; Janusz, W; Kleinrok, Z; Wamil, A1
De Prins, E; Marrannes, R; Wauquier, A; Willems, R1
Grützner, M; Meldrum, BS; Schneider, C; Stephens, DN; Weidmann, R1
Amrick, CL; Bennett, DA1
Goddard, GV; Holmes, KH; Morimoto, K1
Balm, M; Coyle, JT; Markl, A; Zaczek, R1
Lowry, T; Simon, RP; Tanaka, K1
De Aguiar, JC; Graeff, FG; Guimarães, FS; Russo, AS1
Jessa, M; Nazar, M; Palejko, W; Plaznik, A1
Evans, RH; Long, SK; Siarey, RJ; Tulp, MT1
Daniels, AH; Fujikawa, DG; Kim, JS1
Block, F; Schwarz, M1
Faiman, CP; Skolnick, P; Trullas, R; Viu, E1
al-Zubaidy, ZA; Chapman, AG; Meldrum, BS; Smith, SE1
Brainard, MS; Feldman, DE; Knudsen, EI1
Bidzinski, A; Jessa, M; Nazar, M; Plaznik, A1
Graham, SH; Simon, RP; Tanaka, K1
Dunworth, SJ; Stephens, DN1
Bienkowski, P; Kostowski, W1
Balster, RL; Compton, AD; Holcomb, JD; McCallum, SE; Porter, JH; Varvel, SA; Wiley, JL1
Chojnacka-Wójcik, E; Przegaliński, E; Tatarczyńska, E1
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R1
Kang-Park, MH; Moore, SD; Wilson, WA1
Cao, J; Hu, XD; Li, S; Liu, YN; Shi, L; Suo, ZW; Yang, HB; Yang, X; Zheng, CR1
Liu, L; Mikler, J; Stewart, C; Wang, Y; Weiss, T1
Bähner, F; Both, M; Draguhn, A; Kostic, M; Viereckel, T1
Jang, HJ; Joo, K; Kim, MJ; Lee, C; Rhie, DJ1

Other Studies

31 other study(ies) available for 2-amino-5-phosphonovalerate and diazepam

ArticleYear
Modulation of release of acetylcholine from the striatum by a proposed excitatory amino acid antagonist U-54494A: comparison with known antagonists, diazepam and phenytoin.
    Neuropharmacology, 1992, Volume: 31, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Anticonvulsants; Corpus Striatum; Diazepam; Dizocilpine Maleate; In Vitro Techniques; N-Methylaspartate; Phencyclidine; Phenytoin; Potassium; Pyrrolidines; Rats

1992
Intrahippocampal tetanus toxin produces generalized convulsions and neurodegeneration in rats: antagonism by NMDA receptor blockers.
    Epilepsy research. Supplement, 1992, Volume: 9

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Carbamazepine; Diazepam; Dizocilpine Maleate; Epilepsy, Generalized; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hippocampus; Male; Nerve Degeneration; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Tetanus Toxin

1992
NMDA receptor complex antagonists have potential anxiolytic effects as measured with separation-induced ultrasonic vocalizations.
    European journal of pharmacology, 1991, Feb-14, Volume: 193, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anxiety, Separation; Behavior, Animal; Buspirone; Diazepam; Dioxins; Dizocilpine Maleate; Dose-Response Relationship, Drug; Indoles; Kynurenic Acid; Maternal Deprivation; Mephenesin; Piperidines; Quinolizines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin Antagonists; Spiro Compounds; Valine; Vocalization, Animal

1991
Control of NMDA receptor-mediated activity by GABAergic mechanisms in mature and developing rat neocortex.
    Brain research. Developmental brain research, 1990, Jul-01, Volume: 54, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Bicuculline; Diazepam; Electric Stimulation; Evoked Potentials; gamma-Aminobutyric Acid; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Somatosensory Cortex

1990
Inhibition of aminophylline-induced convulsions in mice by antiepileptic drugs and other agents.
    European journal of pharmacology, 1987, Dec-15, Volume: 144, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Aminophylline; Animals; Anticonvulsants; Aspartic Acid; Diazepam; Female; Mice; N-Methylaspartate; Phenobarbital; Seizures; Synaptic Transmission; Valproic Acid

1987
Evidence for a role of the N-methyl-D-aspartate (NMDA) receptor in cortical spreading depression in the rat.
    Brain research, 1988, Aug-09, Volume: 457, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Aspartic Acid; Cortical Spreading Depression; Diazepam; Dibenzocycloheptenes; Dizocilpine Maleate; Ketamine; Male; N-Methylaspartate; Phencyclidine; Phenytoin; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1988
Does the excitatory amino acid receptor antagonist 2-APH exhibit anxiolytic activity?
    Psychopharmacology, 1986, Volume: 90, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Carbolines; Diazepam; Discrimination, Psychological; Drug Interactions; Male; Mice; Pentylenetetrazole; Rats; Rats, Inbred Strains

1986
2-Amino-7-phosphonoheptanoic acid (AP7) produces discriminative stimuli and anticonflict effects similar to diazepam.
    Life sciences, 1986, Dec-22, Volume: 39, Issue:25

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Anticonvulsants; Baclofen; Diazepam; Male; Methocarbamol; Muscle Relaxants, Central; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1986
Kindling-induced changes in EEG recorded during stimulation from the site of stimulation. III. Direct pharmacological manipulations of the kindled amygdala.
    Experimental neurology, 1987, Volume: 97, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amygdala; Animals; Atropine; Baclofen; Diazepam; Electroencephalography; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Muscimol; Neural Inhibition; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Valine

1987
A simple method for quantitative electroencephalographic assessment of drugs with convulsant and anticonvulsant properties.
    Journal of neuroscience methods, 1986, Volume: 18, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Aspartic Acid; Convulsants; Diazepam; Electroencephalography; Hippocampus; Injections; Kainic Acid; Male; N-Methylaspartate; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures

1986
Bilateral intranigral NMDA blockade increases status duration and neuronal injury from systemic kainic acid.
    Brain research, 1994, Oct-17, Volume: 660, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Blood Pressure; Carbon Dioxide; Diazepam; Drug Synergism; Electroencephalography; Functional Laterality; Heat-Shock Proteins; HSP72 Heat-Shock Proteins; Immunohistochemistry; Injections, Intravenous; Kainic Acid; Male; Microinjections; N-Methylaspartate; Neurons; Oxygen; Partial Pressure; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Substantia Nigra; Time Factors

1994
Role of benzodiazepine receptors located in the dorsal periaqueductal grey of rats in anxiety.
    Psychopharmacology, 1993, Volume: 110, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Anxiety; Appetite Depressants; Carbolines; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Male; Microinjections; Midazolam; Periaqueductal Gray; Rats; Rats, Wistar; Receptors, GABA-A

1993
Effects of antagonists at the NMDA receptor complex in two models of anxiety.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1994, Volume: 4, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anxiety; Behavior, Animal; Conflict, Psychological; Diazepam; Dizocilpine Maleate; Drinking; Electroshock; Exploratory Behavior; Injections, Intraventricular; Kynurenic Acid; Male; Motor Activity; Rats; Rats, Wistar; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1994
The effects of central myorelaxants on synaptically-evoked primary afferent depolarization in the immature rat spinal cord in vitro.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Adrenergic alpha-Agonists; Animals; Baclofen; Clonidine; Diazepam; Electric Stimulation; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Muscle Relaxants, Central; Nerve Fibers; Neurons, Afferent; Rats; Receptors, Adrenergic, alpha-2; Spinal Cord; Synapses

1994
The competitive NMDA receptor antagonist CGP 40116 protects against status epilepticus-induced neuronal damage.
    Epilepsy research, 1994, Volume: 17, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Behavior, Animal; Brain; Diazepam; Electroencephalography; Lithium; Male; Neurons; Phenobarbital; Pilocarpine; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Status Epilepticus

1994
The depressant effect of GYKI 52466 on spinal reflex transmission in rats is mediated via non-NMDA and benzodiazepine receptors.
    European journal of pharmacology, 1994, Apr-21, Volume: 256, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; H-Reflex; Injections, Spinal; Male; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex; Synaptic Transmission

1994
Differential effects of compounds that act at strychnine-insensitive glycine receptors in a punishment procedure.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Behavior, Animal; Diazepam; Learning; Male; Memory; Mice; N-Methylaspartate; Punishment; Reaction Time; Receptors, Glycine; Strychnine

1994
Excitatory amino acid antagonists, lamotrigine and BW 1003C87 as anticonvulsants in the genetically epilepsy-prone rat.
    Epilepsy research, 1993, Volume: 15, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acoustic Stimulation; Amino Acids; Amino Acids, Cyclic; Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Epilepsy; Female; Lamotrigine; Male; Motor Activity; Phenytoin; Pyrimidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Time Factors; Triazines

1993
Newly learned auditory responses mediated by NMDA receptors in the owl inferior colliculus.
    Science (New York, N.Y.), 1996, Jan-26, Volume: 271, Issue:5248

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Auditory Perception; Birds; Diazepam; Excitatory Amino Acid Antagonists; Inferior Colliculi; Ketamine; Kynurenic Acid; Learning; Neuronal Plasticity; Receptors, N-Methyl-D-Aspartate; Sound Localization; Synaptic Transmission; Visual Perception

1996
The effects of repeated administration of diazepam, MK-801 and CGP 37849 on rat behavior in two models of anxiety.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1996, Volume: 6, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anxiety; Behavior, Animal; Diazepam; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Rats; Rats, Wistar; Time Factors

1996
The role of excitatory neurotransmitters in seizure-induced neuronal injury in rats.
    Brain research, 1996, Oct-21, Volume: 737, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Blood Pressure; Cerebral Cortex; Diazepam; Electroencephalography; Excitatory Amino Acid Agonists; Glutamic Acid; Kainic Acid; Male; Microdialysis; Neurons; Neurotransmitter Agents; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Seizures; Status Epilepticus

1996
Sensitisation to repeated withdrawal, in mice treated chronically with diazepam, is blocked by an NMDA receptor antagonist.
    Psychopharmacology, 1998, Volume: 136, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Convulsants; Diazepam; Excitatory Amino Acid Antagonists; Glutamic Acid; Male; Mice; Mice, Inbred C57BL; Pentylenetetrazole; Receptors, N-Methyl-D-Aspartate; Seizures; Substance Withdrawal Syndrome; Synaptic Transmission

1998
Discrimination of ethanol in rats: effects of nicotine, diazepam, CGP 40116, and 1-(m-chlorophenyl)-biguanide.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Biguanides; Diazepam; Discrimination Learning; Drug Interactions; Ethanol; GABA Modulators; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Reinforcement Schedule; Serotonin Receptor Agonists

1998
Effects of modulation of NMDA neurotransmission on response rate and duration in a conflict procedure in rats.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 2-Amino-5-phosphonovalerate; Acetamides; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reward; Synaptic Transmission

1998
The influence of the benzodiazepine receptor antagonist flumazenil on the anxiolytic-like effects of CGP 37849 and ACPC in rats.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Amino Acids, Cyclic; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking Behavior; Electroshock; Excitatory Amino Acid Antagonists; Flumazenil; GABA-A Receptor Antagonists; Male; Maze Learning; Rats; Rats, Wistar; Seizures

2000
Neuronal mechanisms of the anoxia-induced network oscillations in the rat hippocampus in vitro.
    The Journal of physiology, 2001, Oct-15, Volume: 536, Issue:Pt 2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; Anesthetics, Local; Animals; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periodicity; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Xanthines

2001
Differential actions of diazepam and zolpidem in basolateral and central amygdala nuclei.
    Neuropharmacology, 2004, Volume: 46, Issue:1

    Topics: Amygdala; Animals; Animals, Newborn; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; GABA Modulators; In Vitro Techniques; Male; Neural Inhibition; Patch-Clamp Techniques; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Valine; Zolpidem

2004
GABAergic disinhibition induced pain hypersensitivity by upregulating NMDA receptor functions in spinal dorsal horn.
    Neuropharmacology, 2011, Volume: 60, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Bicuculline; Diazepam; Drug Interactions; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; Hyperalgesia; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Phosphorylation; Posterior Horn Cells; Protein Kinase Inhibitors; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Sulfonamides

2011
Effect of acute soman exposure on GABA(A) receptors in rat hippocampal slices and cultured hippocampal neurons.
    Neurotoxicity research, 2011, Volume: 20, Issue:4

    Topics: Animals; Animals, Newborn; Anticonvulsants; Atropine; Cells, Cultured; Cholinesterase Inhibitors; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Embryo, Mammalian; Endocytosis; Enzyme-Linked Immunosorbent Assay; Excitatory Amino Acid Antagonists; Female; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Membrane Potentials; Microscopy, Confocal; Muscarinic Antagonists; Neurons; Patch-Clamp Techniques; Pregnancy; Protein Transport; Rats; Receptors, GABA-A; Soman; Valine

2011
Effects of the GABA-uptake blocker NNC-711 on spontaneous sharp wave-ripple complexes in mouse hippocampal slices.
    Hippocampus, 2013, Volume: 23, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Diazepam; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; Fourier Analysis; GABA Antagonists; GABA Modulators; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Nerve Net; Neural Conduction; Nipecotic Acids; Oximes; Time Factors

2013
GluN2B-containing N-methyl-D-aspartate receptors compensate for the inhibitory control of synaptic plasticity during the early critical period in the rat visual cortex.
    Journal of neuroscience research, 2015, Volume: 93, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Modulators; GABA-A Receptor Antagonists; Gene Expression Regulation, Developmental; Long-Term Potentiation; Male; Neural Inhibition; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Visual Cortex

2015