2-amino-4-phosphonobutyric acid has been researched along with quisqualic acid in 48 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 18 (37.50) | 18.7374 |
1990's | 25 (52.08) | 18.2507 |
2000's | 5 (10.42) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Johnson, RL; Koerner, JF; Schulte, MK; Whittemore, ER | 1 |
Johnson, RL; Koerner, JF; Roon, RJ; Schulte, M; Subasinghe, N | 1 |
Garcia-Ladona, FJ; Girard, C; Gombos, G; Palacios, JM | 1 |
Cotman, CW; Whittemore, ER | 1 |
Harrison, PS; Kilpatrick, IC | 1 |
Adamson, P; Brammer, MJ; Campbell, IC; Hajimohammadreza, I; Meldrum, BS | 1 |
Boos, R; Müller, F; Wässle, H | 1 |
Koerner, JF; Whittemore, ER | 2 |
Pranzatelli, MR | 1 |
Clements, JD; Forsythe, ID | 1 |
Marchenko, SM | 1 |
Berry, BW; Boland, LM; Dingledine, R; Hoch, DB | 1 |
Cotman, CW; Monaghan, DT; Palmer, E | 1 |
Akoev, GN; Andrianov, IuN; Bromm, B; Sabo, T; Sherman, NO | 1 |
Johnson, BG; Schoepp, DD | 1 |
Hablitz, JJ | 1 |
Baudry, M; Cummins, JT; Kessler, M; Lynch, G; Way, S | 1 |
Costa, E; Iadarola, MJ; Nicoletti, F; Wroblewski, JT | 1 |
Gullak, MF; Mena, EE; Pagnozzi, MJ | 1 |
Koerner, JF; Marks, RL; Robinson, MB; Whittemore, ER | 1 |
Quinn, MR; Spraguer, PA | 1 |
Arqueros, L; Bustos, G; Fiedler, JL | 1 |
Cotman, CW; Harris, EW; Stevens, DR | 1 |
Alho, H; Costa, E; Eva, C; Fadda, E; Nicoletti, F; Wroblewski, JT | 1 |
Cowburn, RF; Hardy, JA; Roberts, PJ | 1 |
Sheardown, MJ | 1 |
Akaike, N; Carpenter, DO; Hori, N | 1 |
Cotman, CW; Fagg, GE; Foster, AC; Mena, EE | 1 |
Cavanni, P; Eistetter, H; Ferraguti, F; Ratti, E; Salvagno, C; Trist, DG | 1 |
Schultz, K; Weiler, R | 1 |
Turner, JP | 1 |
Haldeman, B; Hampson, DR; Mulvihill, ER; Pickering, DS; Suzdak, PD; Thomsen, C | 1 |
Barnes, S; Mahmud, F; Merchant, V | 1 |
Bigl, V; Grantyn, R; Rothe, T | 1 |
Koerner, JF; Roon, RJ; Schulte, MK | 1 |
Ebert, B; Hansen, JJ; Krogsgaard-Larsen, P; Madsen, U | 1 |
Neuman, RS; Rahman, S | 1 |
Nakamura, Y; Ogata, T; Schubert, P | 1 |
Sheardown, MJ; Thomsen, C | 1 |
Keirstead, SA; Miller, RF | 1 |
Ebert, B; Madsen, U; Vestergaard, HT; Vogensen, SB | 1 |
Allgeier, H; Knöpfel, T; Kuhn, R | 1 |
Johnson, RL; Koerner, JF; Roon, RJ; Schulte, MK; Venkatraman, S | 1 |
Bräuner-Osborne, H; Egebjerg, J; Krogsgaard-Larsen, P; Madsen, U; Nielsen, EO | 1 |
Acher, FC; Bertrand, HO; Bessis, AS; Pin, JP | 1 |
Acher, F; Bertrand, HO; Brabet, I; Pin, JP; Triballeau, N | 1 |
2 review(s) available for 2-amino-4-phosphonobutyric acid and quisqualic acid
Article | Year |
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Metabotropic glutamate receptors: novel targets for drug development.
Topics: Animals; Cloning, Molecular; Drug Design; Humans; Receptors, Metabotropic Glutamate | 1995 |
Ligands for glutamate receptors: design and therapeutic prospects.
Topics: Animals; Drug Design; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Humans; Ligands; N-Methylaspartate; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Synapses | 2000 |
46 other study(ies) available for 2-amino-4-phosphonobutyric acid and quisqualic acid
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Structure-function relationships for analogues of L-2-amino-4-phosphonobutanoic acid on the quisqualic acid-sensitive AP4 receptor of the rat hippocampus.
Topics: Aminobutyrates; Animals; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Molecular Structure; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Receptors, Neurotransmitter; Structure-Activity Relationship | 1992 |
Quisqualic acid analogues: synthesis of beta-heterocyclic 2-aminopropanoic acid derivatives and their activity at a novel quisqualate-sensitized site.
Topics: Aminobutyrates; Animals; Cyclization; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Evoked Potentials; Hippocampus; Imidazoles; Male; Maleimides; Molecular Structure; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Succinimides | 1992 |
Autoradiographic characterization of [3H]L-glutamate binding sites in developing mouse cerebellar cortex.
Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminobutyrates; Animals; Binding, Competitive; Calcium; Cerebellar Cortex; Chlorides; Glutamates; Glutamic Acid; Ibotenic Acid; Kainic Acid; Mice; N-Methylaspartate; Protein Binding; Quisqualic Acid; Receptors, Glutamate; Receptors, Neurotransmitter; Synapses | 1991 |
Agonists selective for phosphoinositide-coupled receptors sensitize neurons to depolarization by L-2-amino-4-phosphonobutanoic acid (L-AP4).
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aminobutyrates; Animals; Carbachol; Cerebral Cortex; Cycloleucine; Hippocampus; Ibotenic Acid; In Vitro Techniques; Male; Neuromuscular Depolarizing Agents; Neurons; Norepinephrine; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear | 1991 |
Hippocampal slices do not appear to accumulate low micromolar concentrations of quisqualate by an active uptake mechanism.
Topics: Amino Acids; Aminobutyrates; Animals; Hippocampus; Male; Quisqualic Acid; Rats; Rats, Inbred Strains | 1991 |
Presynaptic glutamate/quisqualate receptors: effects on synaptosomal free calcium concentrations.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aminobutyrates; Animals; Calcium; Excitatory Amino Acid Antagonists; Glutamates; Glutamic Acid; Ibotenic Acid; Male; Phosphoserine; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Glutamate; Receptors, Neurotransmitter; Synapses; Synaptosomes | 1990 |
Actions of excitatory amino acids on brisk ganglion cells in the cat retina.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Aminobutyrates; Anesthesia; Animals; Aspartic Acid; Cats; Electrodes; Glutamates; Glutamic Acid; Ibotenic Acid; Iontophoresis; Kainic Acid; N-Methylaspartate; Photic Stimulation; Quisqualic Acid; Retinal Ganglion Cells | 1990 |
Pre-exposure to L-homocysteinesulfinic acid blocks quisqualate-induced sensitization to L-2-amino-4-phosphonobutanoic acid.
Topics: Action Potentials; Aminobutyrates; Animals; Hippocampus; Homocysteine; In Vitro Techniques; Male; Quisqualic Acid; Rats; Rats, Inbred Strains; Time Factors | 1991 |
Antimyoclonic effect of MK-801: a possible role for NMDA receptors in developmental myoclonus of the neonatal rat.
Topics: Aminobutyrates; Analysis of Variance; Animals; Animals, Newborn; Anticonvulsants; Clonazepam; Diazepam; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Isoxazoles; Kynurenic Acid; Male; Myoclonus; N-Methylaspartate; Quisqualic Acid; Rats; Receptors, N-Methyl-D-Aspartate; Strychnine | 1990 |
Presynaptic glutamate receptors depress excitatory monosynaptic transmission between mouse hippocampal neurones.
Topics: Action Potentials; Aminobutyrates; Animals; Baclofen; Cells, Cultured; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Kainic Acid; Mice; Quisqualic Acid; Receptors, Glutamate; Receptors, Neurotransmitter; Synaptic Transmission | 1990 |
[The distribution of kainate and quisqualate receptors in the rat cerebellum].
Topics: Aminobutyrates; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Kainic Acid; Membrane Potentials; N-Methylaspartate; Purkinje Cells; Quisqualic Acid; Rats; Receptors, Drug | 1990 |
L-glutamate binding site on N18-RE-105 neuroblastoma hybrid cells is not coupled to an ion channel.
Topics: Aminobutyrates; Animals; Binding, Competitive; Calcium; Chlorides; Cystine; Electric Conductivity; Fluorescent Antibody Technique; Glutamates; Glutamic Acid; Hybrid Cells; Intermediate Filament Proteins; Ion Channels; Mice; Neuroblastoma; Neurofilament Proteins; Neurons; Oxadiazoles; Potassium; Quisqualic Acid; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Sodium; Tumor Cells, Cultured | 1988 |
Novel recognition site for L-quisqualate sensitizes neurons to depolarization by L-2-amino-4-phosphonobutanoate (L-AP4).
Topics: Action Potentials; Aminobutyrates; Animals; Cyclic AMP; Hippocampus; In Vitro Techniques; Male; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface; Second Messenger Systems; Time Factors | 1989 |
Trans-ACPD, a selective agonist of the phosphoinositide-coupled excitatory amino acid receptor.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Aminobutyrates; Animals; Aspartic Acid; Cycloleucine; Hippocampus; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Neuromuscular Depolarizing Agents; Oxadiazoles; Phosphatidylinositols; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface | 1989 |
[Analysis of the effect of quisqualate, N-methyl-D- aspartate and several blockers of amino acid receptors on synaptic transmission in the ampullae of Lorenzini].
Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Aminobutyrates; Animals; Aspartic Acid; Electric Fish; Evoked Potentials; Magnesium; Membrane Potentials; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Sensory Receptor Cells; Skates, Fish; Synapses; Synaptic Transmission; Valine | 1989 |
Excitatory amino acid agonist-antagonist interactions at 2-amino-4-phosphonobutyric acid-sensitive quisqualate receptors coupled to phosphoinositide hydrolysis in slices of rat hippocampus.
Topics: Amino Acids; Aminobutyrates; Animals; Carbachol; Drug Interactions; Hippocampus; Hydrolysis; Ibotenic Acid; Male; Norepinephrine; Oxadiazoles; Phosphatidylinositols; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Drug | 1988 |
Action of excitatory amino acids and their antagonists on hippocampal neurons.
Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Aminobutyrates; Animals; Aspartic Acid; Excitatory Amino Acid Antagonists; Glutamic Acid; Guinea Pigs; Hippocampus; Iontophoresis; Manganese; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Tetrodotoxin; Valine | 1985 |
Induction of glutamate binding sites in hippocampal membranes by transient exposure to high concentrations of glutamate or glutamate analogs.
Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Aminobutyrates; Animals; Aspartic Acid; Binding Sites; Chlorides; Chromatography, High Pressure Liquid; Glutamates; Glutamic Acid; Hippocampus; Homocysteine; Kainic Acid; Kinetics; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Saponins; Sodium; Valine | 1986 |
Excitatory amino acid recognition sites coupled with inositol phospholipid metabolism: developmental changes and interaction with alpha 1-adrenoceptors.
Topics: Age Factors; Aminobutyrates; Animals; Aspartic Acid; Drug Interactions; Glutamates; Glutamic Acid; Hippocampus; Hydrolysis; Ibotenic Acid; Norepinephrine; Oxadiazoles; Oxazoles; Phosphatidylinositols; Phosphoserine; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Amino Acid; Receptors, Cell Surface | 1986 |
Characterization of L-glutamate binding sites in rat spinal cord synaptic membranes: evidence for multiple chloride ion-dependent sites.
Topics: Aminobutyrates; Animals; Anions; Brain; Calcium; Cations; Chlorides; Diencephalon; Glutamates; Glutamic Acid; Kinetics; Oxadiazoles; Quisqualic Acid; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Sodium; Spinal Cord; Synaptic Membranes; Telencephalon | 1986 |
Exposure of hippocampal slices to quisqualate sensitizes synaptic responses to phosphonate-containing analogues of glutamate.
Topics: 2-Amino-5-phosphonovalerate; Aminobutyrates; Animals; Evoked Potentials; Glutamates; Hippocampus; In Vitro Techniques; Male; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Stereoisomerism; Synapses; Valine | 1986 |
Chloride-dependent binding sites for L-[3H]glutamate on dendrodendritic synaptosomal membranes of rat olfactory bulb.
Topics: Aminobutyrates; Animals; Chlorides; Dendrites; Glutamates; Glutamic Acid; Male; Olfactory Bulb; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Glutamate; Receptors, Neurotransmitter; Synaptic Membranes | 1986 |
Specific binding of L-[3H]-glutamic acid to rat substantia nigra synaptic membranes.
Topics: 2-Aminoadipic Acid; Aminobutyrates; Animals; Glutamates; Glutamic Acid; Humans; In Vitro Techniques; Kinetics; Male; Oxadiazoles; Quisqualic Acid; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Glutamate; Receptors, Neurotransmitter; Substantia Nigra; Synaptic Membranes | 1986 |
Hippocampal cells primed with quisqualate are depolarized by AP4 and AP6, ligands for a putative glutamate uptake site.
Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminobutyrates; Aminocaproates; Animals; Aspartic Acid; Electric Stimulation; Glutamates; Glutamic Acid; Hippocampus; Ibotenic Acid; In Vitro Techniques; Male; Membrane Potentials; N-Methylaspartate; Norleucine; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Glutamate; Receptors, Neurotransmitter | 1987 |
Lesions of putative glutamatergic pathways potentiate the increase of inositol phospholipid hydrolysis elicited by excitatory amino acids.
Topics: Amino Acids; Aminobutyrates; Animals; Aspartic Acid; Colchicine; Corpus Striatum; Glutamates; Glutamic Acid; Hippocampus; Hydrolysis; Ibotenic Acid; Kainic Acid; Male; N-Methylaspartate; Oxadiazoles; Phosphatidylinositols; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface | 1987 |
Characterisation of Na+-independent L-[3H]glutamate binding sites in human temporal cortex.
Topics: 2-Amino-5-phosphonovalerate; Aged; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Aminobutyrates; Cell Membrane; Chlorides; Glutamates; Glutamic Acid; Humans; Ibotenic Acid; Kainic Acid; Male; Middle Aged; Oxadiazoles; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Sodium; Temporal Lobe | 1988 |
A new and specific non-NMDA receptor antagonist, FG 9065, blocks L-AP4-evoked depolarization in rat cerebral cortex.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aminobutyrates; Animals; Aspartic Acid; Cerebral Cortex; Evoked Potentials; In Vitro Techniques; N-Methylaspartate; Oxadiazoles; Quinoxalines; Quisqualic Acid; Rats; Receptors, Glutamate; Receptors, Neurotransmitter | 1988 |
Piriform cortex brain slices: techniques for isolation of synaptic inputs.
Topics: Aminobutyrates; Animals; Aspartic Acid; Cerebral Cortex; Dendrites; Electrophysiology; Evoked Potentials; In Vitro Techniques; Kainic Acid; Male; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Rats; Synapses | 1988 |
Chloride and calcium ions separate L-glutamate receptor populations in synaptic membranes.
Topics: Amino Acids, Dicarboxylic; Aminobutyrates; Animals; Calcium; Chlorides; Glutamates; Glutamic Acid; In Vitro Techniques; Oxadiazoles; Quisqualic Acid; Rats; Receptors, Cell Surface; Receptors, Glutamate; Synaptic Membranes | 1983 |
Competitive antagonism by phenylglycine derivatives at type I metabotropic glutamate receptors.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminobutyrates; Animals; Benzoates; Binding, Competitive; Calcium; Cells, Cultured; CHO Cells; Cricetinae; Cycloleucine; Cytidine Diphosphate Diglycerides; Excitatory Amino Acid Antagonists; Glutamates; Glutamic Acid; Glycine; Ibotenic Acid; Kainic Acid; Neurons; Neurotoxins; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Phosphoric Diester Hydrolases; Quisqualic Acid; Receptors, Metabotropic Glutamate; Recombinant Fusion Proteins; Signal Transduction | 1994 |
Ionotropic non-N-methyl-D-aspartate agonists induce retraction of dendritic spinules from retinal horizontal cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminobutyrates; Animals; Carps; Cell Movement; Cyclopentanes; Dendrites; Ibotenic Acid; N-Methylaspartate; Quisqualic Acid; Receptors, Neurotransmitter; Retina | 1993 |
Anion transport blockers inhibit DL-2-amino-4-phosphonobutyrate responses induced by quisqualate in the rat cerebral cortex.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Aminobutyrates; Animals; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Male; Neuromuscular Depolarizing Agents; Quisqualic Acid; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Glutamate | 1993 |
A pharmacological characterization of the mGluR1 alpha subtype of the metabotropic glutamate receptor expressed in a cloned baby hamster kidney cell line.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids, Diamino; Aminobutyrates; Animals; Binding, Competitive; Cell Line; Cell Membrane; Clone Cells; Cricetinae; Cyanobacteria Toxins; Dizocilpine Maleate; Glutamates; Glutamic Acid; Ibotenic Acid; Inositol Phosphates; Kidney; Kinetics; Neurotoxins; Pertussis Toxin; Quinoxalines; Quisqualic Acid; Receptors, Glutamate; Recombinant Proteins; Transfection; Virulence Factors, Bordetella | 1993 |
Modulation of transmission gain by protons at the photoreceptor output synapse.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Ambystoma; Aminobutyrates; Animals; Calcium Channels; Hydrogen-Ion Concentration; In Vitro Techniques; Kainic Acid; Light; Membrane Potentials; Photoreceptor Cells; Protons; Quisqualic Acid; Receptors, Glutamate; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells; Synapses; Synaptic Transmission | 1993 |
Potentiating and depressant effects of metabotropic glutamate receptor agonists on high-voltage-activated calcium currents in cultured retinal ganglion neurons from postnatal mice.
Topics: Alanine; Aminobutyrates; Animals; Calcium; Calcium Channels; Cells, Cultured; Cycloleucine; Glutamates; Glutamic Acid; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Intracellular Fluid; Mice; omega-Conotoxin GVIA; Organophosphorus Compounds; Peptides; Quisqualic Acid; Receptors, Metabotropic Glutamate; Retinal Ganglion Cells | 1994 |
Quisqualic acid induced sensitization and the active uptake of L-quisqualic acid by hippocampal slices.
Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Aminobutyrates; Animals; Chromatography, High Pressure Liquid; Electrophysiology; Hippocampus; In Vitro Techniques; Male; Models, Biological; o-Phthalaldehyde; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Synapses | 1993 |
The non-depolarizing D-form of bromohomoibotenic acid enhances depolarizations evoked by the L-form or quisqualate.
Topics: Aminobutyrates; Animals; Brain; Electrophysiology; Ibotenic Acid; In Vitro Techniques; Quisqualic Acid; Rats; Stereoisomerism | 1993 |
Characterization of metabotropic glutamate receptor-mediated facilitation of N-methyl-D-aspartate depolarization of neocortical neurones.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Alanine; Alkaloids; Aminobutyrates; Animals; Cerebral Cortex; Cyclic GMP; Cycloleucine; Male; Neurons; Phorbol Esters; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Staurosporine | 1996 |
Potentiated cAMP rise in metabotropically stimulated rat cultured astrocytes by a Ca2+-related A1/A2 adenosine receptor cooperation.
Topics: Amino Acids, Dicarboxylic; Aminobutyrates; Animals; Astrocytes; Calcium; Cells, Cultured; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Agonists; Purinergic P1 Receptor Agonists; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Stimulation, Chemical | 1996 |
Phenylglycines can evoke quisqualate-primed depolarizations in rat cingulate cortex: an effect associated with [3H]DL-AP4 uptake.
Topics: Aminobutyrates; Animals; Cerebral Cortex; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; Glycine; Gyrus Cinguli; Osmolar Concentration; Piperazines; Quinoxalines; Quisqualic Acid; Rats; Tritium | 1996 |
Metabotropic glutamate receptor agonists evoke calcium waves in isolated Müller cells.
Topics: Adenosine Triphosphate; Ambystoma; Aminobutyrates; Animals; Calcium Channels; Cycloleucine; Excitatory Amino Acid Agonists; Fluorescent Dyes; Histocytochemistry; In Vitro Techniques; Neuroglia; Neuroprotective Agents; Quisqualic Acid; Receptors, Metabotropic Glutamate; Retina | 1997 |
Analogues of homoibotenic acid show potent and selective activity following sensitisation by quisqualic acid.
Topics: Aminobutyrates; Animals; Calcium Chloride; Cerebral Cortex; Electrophysiology; Excitatory Amino Acid Agonists; Glutamic Acid; Glycine; Ibotenic Acid; In Vitro Techniques; Male; Neurons; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Synaptosomes | 2004 |
Synthesis of oxadiazolidinedione derivatives as quisqualic acid analogues and their evaluation at a quisqualate-sensitized site in the rat hippocampus.
Topics: Animals; Hippocampus; In Vitro Techniques; Male; Oxadiazoles; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship | 1994 |
Common and selective molecular determinants involved in metabotopic glutamate receptor agonist activity.
Topics: Binding Sites; Crystallography, X-Ray; Excitatory Amino Acid Agonists; Glutamic Acid; Ligands; Models, Molecular; Receptors, Metabotropic Glutamate; Sequence Homology, Amino Acid; Structure-Activity Relationship | 2002 |
Virtual screening workflow development guided by the "receiver operating characteristic" curve approach. Application to high-throughput docking on metabotropic glutamate receptor subtype 4.
Topics: Binding Sites; Databases, Factual; Drug Design; Models, Molecular; Quantitative Structure-Activity Relationship; Receptors, Metabotropic Glutamate; ROC Curve | 2005 |