2,5-dimethoxy-4-bromoamphetamine has been researched along with ketanserin in 22 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 7 (31.82) | 18.7374 |
| 1990's | 11 (50.00) | 18.2507 |
| 2000's | 2 (9.09) | 29.6817 |
| 2010's | 2 (9.09) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Glennon, RA; Lyon, RA; Roth, BL; Seggel, MR; Suba, EA; Titeler, M; Yousif, MY | 1 |
| Glennon, RA | 2 |
| Frescas, S; Gudelsky, GA; Huang, X; Marona-Lewicka, D; Nash, JF; Nichols, DE; Roth, BL | 1 |
| Egan, CT; Herrick-Davis, K; Teitler, M | 1 |
| Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
| Glennon, RA; Mosier, PD; Roth, BL; Runyon, SP; Westkaemper, RB | 1 |
| Barker, EL; Burris, KD; Sanders-Bush, E | 1 |
| Appel, NM; De Souza, EB; Glennon, RA; Leonhardt, S; Teitler, M | 1 |
| Ashby, CR; Jiang, LH; Kasser, RJ; Wang, RY | 1 |
| Adham, N; Branchek, T; Hartig, PR; Kao, HT; Macchi, M | 1 |
| Peroutka, SJ; Pierce, PA | 2 |
| Adrien, J; Gorea, E | 1 |
| Glennon, RA; Lyon, RA; Seggel, MR; Titeler, M | 1 |
| Buckholtz, NS; Freedman, DX; Zhou, DF | 1 |
| Davis, KH; Glennon, RA; Lyon, RA; Titeler, M | 1 |
| Grotewiel, MS; Sanders-Bush, E | 1 |
| Pritchett, DB; Szele, FG | 1 |
| Mutel, V; Sleight, AJ; Stam, NJ; Vanderheyden, PM | 1 |
| Chen, Z; Morimoto, Y; Nakata, Y; Nishio, H; Yoshikawa, S | 1 |
| Buchborn, T; Dieterich, DC; Grecksch, G; Höllt, V; Schröder, H | 1 |
1 review(s) available for 2,5-dimethoxy-4-bromoamphetamine and ketanserin
| Article | Year |
|---|---|
Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
21 other study(ies) available for 2,5-dimethoxy-4-bromoamphetamine and ketanserin
| Article | Year |
|---|---|
A structure-affinity study of the binding of 4-substituted analogues of 1-(2,5-dimethoxyphenyl)-2-aminopropane at 5-HT2 serotonin receptors.
Topics: Amphetamines; Animals; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Solubility; Structure-Activity Relationship | 1990 |
1-(2,5-Dimethoxy-4-(trifluoromethyl)phenyl)-2-aminopropane: a potent serotonin 5-HT2A/2C agonist.
Topics: 3T3 Cells; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Cell Line; Discrimination, Psychological; Frontal Lobe; Hippocampus; Iodine Radioisotopes; Ketanserin; Male; Mice; Phenethylamines; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Tritium | 1994 |
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; COS Cells; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship | 1998 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Potential modes of interaction of 9-aminomethyl-9,10-dihydroanthracene (AMDA) derivatives with the 5-HT2A receptor: a ligand structure-affinity relationship, receptor mutagenesis and receptor modeling investigation.
Topics: Animals; Anthracenes; Cattle; Humans; Ligands; Models, Molecular; Molecular Sequence Data; Molecular Structure; Mutagenesis; Protein Binding; Receptor, Serotonin, 5-HT2A; Sequence Alignment; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Structure-Activity Relationship | 2008 |
The 2014 Philip S. Portoghese Medicinal Chemistry Lectureship: The "Phenylalkylaminome" with a Focus on Selected Drugs of Abuse.
Topics: Animals; Central Nervous System Stimulants; Chemistry, Pharmaceutical; Dopamine; Drug Discovery; Hallucinogens; Humans; Illicit Drugs; Norepinephrine; Phenethylamines; Psychotropic Drugs; Receptors, Serotonin; Serotonin | 2017 |
Phosphoinositide hydrolysis linked 5-HT2 receptors in fibroblasts from choroid plexus.
Topics: Animals; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fibroblasts; Haloperidol; Hydrolysis; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Serotonin; Serotonin; Spiperone | 1991 |
Receptor pharmacology of MDMA and related hallucinogens.
Topics: 3,4-Methylenedioxyamphetamine; Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Designer Drugs; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; Ketanserin; Kinetics; N-Methyl-3,4-methylenedioxyamphetamine; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1990 |
Electrophysiological characterization of 5-hydroxytryptamine2 receptors in the rat medial prefrontal cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Frontal Lobe; Ketanserin; Magnesium; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sodium Glutamate; Tetrahydronaphthalenes | 1990 |
[3H]-DOB(4-bromo-2,5-dimethoxyphenylisopropylamine) and [3H] ketanserin label two affinity states of the cloned human 5-hydroxytryptamine2 receptor.
Topics: Affinity Labels; Animals; Binding Sites; Binding, Competitive; Cell Line; Chlorocebus aethiops; Cloning, Molecular; DOM 2,5-Dimethoxy-4-Methylamphetamine; Genetic Vectors; Guanylyl Imidodiphosphate; Ketanserin; Mice; Receptors, Serotonin; Transfection; Tritium | 1990 |
Evidence for distinct 5-hydroxytryptamine2 binding site subtypes in cortical membrane preparations.
Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Cerebral Cortex; DOM 2,5-Dimethoxy-4-Methylamphetamine; Humans; Ketanserin; Rats; Receptors, Serotonin; Serotonin; Species Specificity | 1989 |
Antagonism of 5-hydroxytryptamine2 receptor-mediated phosphatidylinositol turnover by d-lysergic acid diethylamide.
Topics: Amphetamines; Animals; Cerebral Cortex; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Guanosine Triphosphate; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1988 |
Serotonergic regulation of noradrenergic coerulean neurons: electrophysiological evidence for the involvement of 5-HT2 receptors.
Topics: Action Potentials; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electrophysiology; Ketanserin; Locus Coeruleus; Male; Neurons; Norepinephrine; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Synapses | 1988 |
Indolealkylamine analogs share 5-HT2 binding characteristics with phenylalkylamine hallucinogens.
Topics: Amines; Animals; Cerebral Cortex; Computer Simulation; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; In Vitro Techniques; Indoles; Ketanserin; Methylation; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship | 1988 |
Serotonin2 agonist administration down-regulates rat brain serotonin2 receptors.
Topics: Amphetamines; Animals; Brain; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1988 |
Selectivity of serotonergic drugs for multiple brain serotonin receptors. Role of [3H]-4-bromo-2,5-dimethoxyphenylisopropylamine ([3H]DOB), a 5-HT2 agonist radioligand.
Topics: Amphetamines; Animals; Brain; DOM 2,5-Dimethoxy-4-Methylamphetamine; In Vitro Techniques; Ketanserin; Ligands; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tritium | 1987 |
Regulation of serotonin2A receptors in heterologous expression systems.
Topics: 3T3 Cells; Animals; Antiparkinson Agents; Binding, Competitive; Cell Line; Dogs; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Gene Expression Regulation; Ketanserin; Kidney; Kinetics; Mice; Pituitary Neoplasms; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Transfection; Tumor Cells, Cultured | 1994 |
High affinity agonist binding to cloned 5-hydroxytryptamine2 receptors is not sensitive to GTP analogs.
Topics: 3T3 Cells; Animals; Binding Sites; Cell Line; Cloning, Molecular; DOM 2,5-Dimethoxy-4-Methylamphetamine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Ketanserin; Kidney; Mice; Phosphatidylinositols; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists | 1993 |
Radiolabelling of the human 5-HT2A receptor with an agonist, a partial agonist and an antagonist: effects on apparent agonist affinities.
Topics: 3T3 Cells; Animals; Binding, Competitive; Cell Membrane; DOM 2,5-Dimethoxy-4-Methylamphetamine; Humans; Ketanserin; Mice; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1996 |
Binding affinity of sarpogrelate to 5-HT(2A) receptor ligand recognition sites in rat renal cortical and mesangial cells in culture.
Topics: Animals; Binding Sites; Binding, Competitive; Cells, Cultured; Cerebral Cortex; DOM 2,5-Dimethoxy-4-Methylamphetamine; Glomerular Mesangium; Ketanserin; Kidney Cortex; Male; Membranes; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Subcellular Fractions; Succinates; Tritium | 1999 |
Tolerance to LSD and DOB induced shaking behaviour: differential adaptations of frontocortical 5-HT(2A) and glutamate receptor binding sites.
Topics: Animals; Binding Sites; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Tolerance; Frontal Lobe; Glutamic Acid; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Motor Activity; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Glutamate; Serotonin Antagonists | 2015 |