Page last updated: 2024-08-24

2,5-dimethoxy-4-bromoamphetamine and 2,4,5-trimethoxyphenylisopropylamine

2,5-dimethoxy-4-bromoamphetamine has been researched along with 2,4,5-trimethoxyphenylisopropylamine in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19906 (42.86)18.7374
1990's3 (21.43)18.2507
2000's4 (28.57)29.6817
2010's1 (7.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA; Liebowitz, SM; Mack, EC1
Hall, LH; Kier, LB1
Bartyzel, P; Glennon, RA; Leonhardt, S; Raghupathi, R; Teitler, M1
Glennon, RA; Lyon, RA; Roth, BL; Seggel, MR; Suba, EA; Titeler, M; Yousif, MY1
Glennon, RA2
Benington, F; Glennon, RA; Morin, RD; Young, R1
Anderson, GM; Castagnoli, N; Domelsmith, LN; Eaton, TA; Glennon, RA; Houk, KN; Kollman, PA; Shulgin, AT1
Anderson, GM; Glennon, RA; Liebowitz, SM1
Clare, BW1
Glennon, RA; Peddi, S; Roth, BL; Westkaemper, RB1
Glennon, RA; Mosier, PD; Roth, BL; Runyon, SP; Westkaemper, RB1
Berg, KA; Cassels, BK; Clarke, WP; Gutiérrez-Hernandez, MA; Moya, PR; Reyes-Parada, M; Sáez-Briones, P1
Ewald, AH; Maurer, HH1

Reviews

1 review(s) available for 2,5-dimethoxy-4-bromoamphetamine and 2,4,5-trimethoxyphenylisopropylamine

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Other Studies

13 other study(ies) available for 2,5-dimethoxy-4-bromoamphetamine and 2,4,5-trimethoxyphenylisopropylamine

ArticleYear
Serotonin receptor binding affinities of several hallucinogenic phenylalkylamine and N,N-dimethyltryptamine analogues.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:8

    Topics: Amines; Animals; Female; Hallucinogens; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; N,N-Dimethyltryptamine; Rats; Receptors, Serotonin; Stomach; Tryptamines

1978
Structure-activity studies on hallucinogenic amphetamines using molecular connectivity.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:12

    Topics: Amphetamines; Chemical Phenomena; Chemistry, Physical; Hallucinogens; Models, Chemical; Structure-Activity Relationship

1977
Binding of phenylalkylamine derivatives at 5-HT1C and 5-HT2 serotonin receptors: evidence for a lack of selectivity.
    Journal of medicinal chemistry, 1992, Feb-21, Volume: 35, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Ergolines; Ketanserin; Male; Molecular Structure; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Structure-Activity Relationship; Tritium

1992
A structure-affinity study of the binding of 4-substituted analogues of 1-(2,5-dimethoxyphenyl)-2-aminopropane at 5-HT2 serotonin receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:3

    Topics: Amphetamines; Animals; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Solubility; Structure-Activity Relationship

1990
Behavioral and serotonin receptor properties of 4-substituted derivatives of the hallucinogen 1-(2,5-dimethoxyphenyl)-2-aminopropane.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:10

    Topics: Amphetamines; Animals; Behavior, Animal; Discrimination Learning; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; In Vitro Techniques; Isomerism; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin

1982
Photoelectron spectra of psychotropic drugs. 6. Relationships between the physical properties and pharmacological actions of amphetamine analogues.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:12

    Topics: Amphetamines; Animals; Chemical Phenomena; Chemistry, Physical; Humans; Psychotropic Drugs; Rabbits; Spectrophotometry, Ultraviolet; Structure-Activity Relationship

1981
Serotonin receptor affinities of psychoactive phenalkylamine analogues.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:3

    Topics: Amines; Animals; Female; Hallucinogens; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rats; Receptors, Serotonin; Stomach; Structure-Activity Relationship

1980
The frontier orbital phase angles: novel QSAR descriptors for benzene derivatives, applied to phenylalkylamine hallucinogens.
    Journal of medicinal chemistry, 1998, Sep-24, Volume: 41, Issue:20

    Topics: Hallucinogens; Humans; Models, Molecular; Molecular Conformation; Phenethylamines; Quantum Theory

1998
Ring substituted analogues of 5-aminomethyl-10,11-dihydro-dibenzo[a,d]cycloheptene (AMDH): potential modes of binding to the 5-HT(2A) receptor.
    Bioorganic & medicinal chemistry letters, 2003, Aug-04, Volume: 13, Issue:15

    Topics: Cyclopentanes; Indicators and Reagents; Kinetics; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Serotonin Agents; Structure-Activity Relationship

2003
Potential modes of interaction of 9-aminomethyl-9,10-dihydroanthracene (AMDA) derivatives with the 5-HT2A receptor: a ligand structure-affinity relationship, receptor mutagenesis and receptor modeling investigation.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Animals; Anthracenes; Cattle; Humans; Ligands; Models, Molecular; Molecular Sequence Data; Molecular Structure; Mutagenesis; Protein Binding; Receptor, Serotonin, 5-HT2A; Sequence Alignment; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Structure-Activity Relationship

2008
The 2014 Philip S. Portoghese Medicinal Chemistry Lectureship: The "Phenylalkylaminome" with a Focus on Selected Drugs of Abuse.
    Journal of medicinal chemistry, 2017, 04-13, Volume: 60, Issue:7

    Topics: Animals; Central Nervous System Stimulants; Chemistry, Pharmaceutical; Dopamine; Drug Discovery; Hallucinogens; Humans; Illicit Drugs; Norepinephrine; Phenethylamines; Psychotropic Drugs; Receptors, Serotonin; Serotonin

2017
Functional selectivity of hallucinogenic phenethylamine and phenylisopropylamine derivatives at human 5-hydroxytryptamine (5-HT)2A and 5-HT2C receptors.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Amphetamines; Animals; Arachidonic Acid; Behavior, Animal; CHO Cells; Cricetinae; Cricetulus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; Humans; Inositol Phosphates; Male; Mescaline; Motor Activity; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Signal Transduction; Transfection

2007
2,5-Dimethoxyamphetamine-derived designer drugs: studies on the identification of cytochrome P450 (CYP) isoenzymes involved in formation of their main metabolites and on their capability to inhibit CYP2D6.
    Toxicology letters, 2008, Dec-15, Volume: 183, Issue:1-3

    Topics: Algorithms; Amphetamines; Animals; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP2D6 Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Designer Drugs; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fluoxetine; Gas Chromatography-Mass Spectrometry; Humans; Hydroxylation; Insecta; Kinetics; Microsomes, Liver; Molecular Structure; Quinidine; Spectrometry, Mass, Electrospray Ionization

2008