2',6'-dimethyltyrosine has been researched along with endomorphin 1 in 3 studies
| Studies (2',6'-dimethyltyrosine) | Trials (2',6'-dimethyltyrosine) | Recent Studies (post-2010) (2',6'-dimethyltyrosine) | Studies (endomorphin 1) | Trials (endomorphin 1) | Recent Studies (post-2010) (endomorphin 1) |
|---|---|---|---|---|---|
| 27 | 0 | 6 | 448 | 2 | 109 |
| Protein | Taxonomy | 2',6'-dimethyltyrosine (IC50) | endomorphin 1 (IC50) |
|---|---|---|---|
| Delta-type opioid receptor | Mus musculus (house mouse) | 0.026 | |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0005 | |
| Mu-type opioid receptor | Homo sapiens (human) | 0.0275 | |
| Mu-type opioid receptor | Mus musculus (house mouse) | 0.0363 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (66.67) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 1 (33.33) | 2.80 |
| Authors | Studies |
|---|---|
| Imam, MZ; Kong, D; Kuo, A; Smith, MT; Williams, CM | 1 |
| Blanchfield, JT; Koda, Y; Okada, Y; Shiotani, K; Toth, I; Tsuda, Y | 1 |
| Bryant, SD; Jinsmaa, Y; Lazarus, LH; Li, T; Marczak, ED; Okada, Y; Tsuda, Y | 1 |
3 other study(ies) available for 2',6'-dimethyltyrosine and endomorphin 1
| Article | Year |
|---|---|
Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources.
Topics: Analgesics, Opioid; Animals; Biological Products; Cell Line, Tumor; Chemistry, Pharmaceutical; Drug Discovery; Humans; Ligands; Pain; Peptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 2022 |
Comparison of the in vitro apparent permeability and stability of opioid mimetic compounds with that of the native peptide.
Topics: Analgesics, Opioid; Blood-Brain Barrier; Caco-2 Cells; Chemistry, Pharmaceutical; Drug Design; Humans; Inhibitory Concentration 50; Injections, Intraventricular; Kinetics; Molecular Conformation; Oligopeptides; Peptides; Permeability; Receptors, Opioid; Tyrosine | 2007 |
[N-allyl-Dmt1]-endomorphins are micro-opioid receptor antagonists lacking inverse agonist properties.
Topics: Analgesics, Opioid; Animals; Brain; Cell Line; Cell Membrane; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Male; Mice; Oligopeptides; Protein Binding; Radioligand Assay; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Tyrosine | 2007 |