2',4'-dichlorobenzamil amiloride has been researched along with amiloride in 16 studies
Studies (2',4'-dichlorobenzamil amiloride) | Trials (2',4'-dichlorobenzamil amiloride) | Recent Studies (post-2010) (2',4'-dichlorobenzamil amiloride) | Studies (amiloride) | Trials (amiloride) | Recent Studies (post-2010) (amiloride) |
---|---|---|---|---|---|
18 | 0 | 2 | 7,584 | 339 | 788 |
Protein | Taxonomy | 2',4'-dichlorobenzamil amiloride (IC50) | amiloride (IC50) |
---|---|---|---|
Urokinase-type plasminogen activator | Homo sapiens (human) | 4.7 | |
Urokinase-type plasminogen activator | Mus musculus (house mouse) | 2.3 | |
Amine oxidase [flavin-containing] A | Homo sapiens (human) | 3.909 | |
Sodium/hydrogen exchanger 1 | Rattus norvegicus (Norway rat) | 1 | |
Amiloride-sensitive sodium channel subunit alpha | Homo sapiens (human) | 0.776 | |
Sodium/hydrogen exchanger 2 | Oryctolagus cuniculus (rabbit) | 1 | |
Acid-sensing ion channel 3 | Homo sapiens (human) | 4.4 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (31.25) | 18.2507 |
2000's | 10 (62.50) | 29.6817 |
2010's | 1 (6.25) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Northover, BJ | 1 |
Feuvray, D; Lagadic-Gossmann, D | 1 |
Conner, JA; Hernández-Cruz, A; Santi, CM | 1 |
Hartung, K; Kappl, M | 1 |
Friis, UG; Johansen, T; Praetorius, HA; Praetorius, J | 1 |
Mayer, A; Pecht, I; Pilatus, U; Rumpel, E | 1 |
Eriksson, KS; Haas, HL; Stevens, DR | 1 |
Gupta, S; Patni, A; Reddy, PR; Sharma, A; Tiwary, AK | 1 |
Kato, M; Kitazono, T; Nakamura, U; Uchizono, Y; Wakisaka, M; Yoshinari, M; Yoshioka, M | 1 |
Garg, SK; Gupta, S; Patni, AK; Sharma, A; Tiwary, AK | 1 |
Hogg, DS; Kozlowski, RZ | 1 |
Au, AL; Chau, WH; Kwan, YW; Lau, WH; Lee, WH; Raymond, K | 1 |
Gupta, A; Gupta, S; Tiwary, AK | 1 |
Gupta, A; Gupta, S; Moudgil, P; Sharma, A; Tiwary, AK | 1 |
Choi, S; Kim, JA; Liang, GH; Park, S; Suh, SH | 1 |
Calafat, AM; Chiu, YH; Dadd, R; Hauser, R; Mínguez-Alarcón, L; Nassan, FL; Ospina, M; Segal, TR; Williams, PL | 1 |
16 other study(ies) available for 2',4'-dichlorobenzamil amiloride and amiloride
Article | Year |
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Effects of 8-(N,N-diethylamino)octyl 3,4,5-trimethoxybenzoate (TMB8) on rat atrial muscle.
Topics: Amiloride; Animals; Carrier Proteins; Fluorescent Dyes; Gallic Acid; Heart; Heart Atria; Indoles; Myocardium; Rats; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase | 1992 |
Decreased sensitivity of contraction to changes of intracellular pH in papillary muscle from diabetic rat hearts.
Topics: Amiloride; Ammonium Chloride; Animals; Caffeine; Diabetes Mellitus, Experimental; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Muscle Contraction; Papillary Muscles; Rats; Rats, Inbred Strains; Ryanodine | 1990 |
A significant fraction of calcium transients in intact guinea pig ventricular myocytes is mediated by Na(+)-Ca2+ exchange.
Topics: Amiloride; Animals; Biological Transport; Calcium; Calcium Channel Blockers; Calcium Channels; Carrier Proteins; Cells, Cultured; Guinea Pigs; Heart; Heart Ventricles; Membrane Potentials; Microscopy, Confocal; Microscopy, Fluorescence; Monensin; Muscle Proteins; Myocardium; Nickel; Ouabain; Potassium; Ryanodine; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Signal Transduction; Sodium-Calcium Exchanger; Verapamil | 1995 |
Rapid charge translocation by the cardiac Na(+)-Ca2+ exchanger after a Ca2+ concentration jump.
Topics: Amiloride; Animals; Calcium; Carrier Proteins; Cell-Free System; Cytoplasm; Electric Conductivity; Guinea Pigs; Heart; Kinetics; Myocardium; Nickel; Patch-Clamp Techniques; Rats; Sodium; Sodium-Calcium Exchanger; Temperature | 1996 |
Evidence for a Na+/Ca2+ exchange mechanism in rat peritoneal mast cells.
Topics: Amiloride; Animals; Calcium; Electric Conductivity; Histamine Release; Lanthanum; Male; Mast Cells; Membrane Potentials; Ouabain; Patch-Clamp Techniques; Peritoneal Cavity; Rats; Rats, Sprague-Dawley; Sodium; Sodium-Calcium Exchanger | 1998 |
Na(+)-dependent Ca(2+) transport modulates the secretory response to the Fcepsilon receptor stimulus of mast cells.
Topics: Amiloride; Animals; beta-N-Acetylhexosaminidases; Biological Transport; Calcium; Cell Line; Cell Membrane; Fluorescent Dyes; Indoles; Kinetics; Magnetic Resonance Spectroscopy; Mast Cells; Models, Chemical; Rats; Receptors, IgE; Sodium; Strontium | 2000 |
Serotonin excites tuberomammillary neurons by activation of Na(+)/Ca(2+)-exchange.
Topics: Amiloride; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hypothalamic Area, Lateral; In Vitro Techniques; Ion Transport; Lithium; Male; Meglumine; Membrane Potentials; Neurons; Nickel; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Sodium; Sodium-Calcium Exchanger; Temperature; Tetrodotoxin | 2001 |
Effect of 2',4'-dichlorobenzamil hydrochloride, a Na(+)-Ca(2+) exchange inhibitor, on human spermatozoa.
Topics: Amiloride; Calcium; Cell Survival; Dose-Response Relationship, Drug; Glucose; Humans; Male; Sodium-Calcium Exchanger; Sperm Count; Sperm Motility; Spermatocidal Agents; Spermatozoa; Time Factors | 2001 |
Sodium-coupled glucose transporter as a functional glucose sensor of retinal microvascular circulation.
Topics: Amiloride; Angiotensin II; Animals; Calcium; Calcium Channel Blockers; Cattle; Cell Size; Deoxyglucose; Dose-Response Relationship, Drug; Extracellular Space; Glucose; Methylglucosides; Microcirculation; Monosaccharide Transport Proteins; Pericytes; Phlorhizin; Retinal Vessels; Sodium; Sodium-Calcium Exchanger; Vasoconstrictor Agents | 2001 |
Role of intracellular calcium in the spermicidal action of 2',4'-dichlorobenzamil, a novel contact spermicide.
Topics: Adrenergic beta-Antagonists; Adult; Amiloride; Calcium; Humans; In Vitro Techniques; Male; Propranolol; Semen; Sperm Motility; Spermatocidal Agents; Spermatozoa | 2001 |
Hypoxia activates a background conductance in freshly isolated pulmonary arterial endothelial cells of the rat.
Topics: Amiloride; Animals; Cell Hypoxia; Cells, Cultured; Electrophysiology; Endothelium, Vascular; Gadolinium; Lanthanum; Male; Oxygen; Potassium Channels; Pulmonary Artery; Rats; Rats, Wistar; Sodium-Calcium Exchanger | 2002 |
Role of Na+/H+ exchanger in acetylcholine-mediated pulmonary artery contraction of spontaneously hypertensive rats.
Topics: Acetylcholine; Amiloride; Animals; Calcium; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Hypertension; Imidazoles; In Vitro Techniques; Indoles; Male; Maleimides; Muscarinic Agonists; Muscarinic Antagonists; Neostigmine; Protein Kinase C; Pulmonary Artery; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Sodium; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Sodium-Potassium-Exchanging ATPase; Species Specificity; Thiourea; Vasoconstriction; Vasodilator Agents | 2003 |
Spermicidal efficacy of H2-receptor antagonists and potentiation with 2', 4'-dichlorobenzamil hydrochloride: role of intrasperm Ca2+.
Topics: Adult; Amiloride; Calcium; Cimetidine; Famotidine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Ranitidine; Receptors, Cytoplasmic and Nuclear; Sodium-Calcium Exchanger; Sperm Motility; Spermatocidal Agents; Spermatozoa; Time Factors | 2003 |
Potentiation of spermicidal activity of 2',4'-dichlorobenzamil by lidocaine.
Topics: Amiloride; Animals; Humans; Lidocaine; Male; Rabbits; Spermatocidal Agents; Spermatozoa | 2002 |
Stimulation of large-conductance Ca2+-activated K+ channels by the Na+/Ca2+ exchanger inhibitor dichlorobenzamil in cultured human umbilical vein endothelial cells and mouse aortic smooth muscle cells.
Topics: Amiloride; Animals; Aorta; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Mice; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Sodium-Calcium Exchanger; Umbilical Veins | 2009 |
Urinary concentrations of 3-(diethylcarbamoyl)benzoic acid (DCBA), a major metabolite of N,N-diethyl-m-toluamide (DEET) and semen parameters among men attending a fertility center.
Topics: Adult; Amiloride; Body Mass Index; DEET; Fertility; Humans; Infertility, Male; Insect Repellents; Male; Massachusetts; Middle Aged; Prospective Studies; Semen; Semen Analysis; Sperm Count; Sperm Motility; Young Adult | 2017 |