Compounds > 2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole
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2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole and fentanyl isothiocyanate

2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole has been researched along with fentanyl isothiocyanate in 7 studies

Compound Research Comparison

Studies
(2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole)		Trials
(2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole)		Recent Studies (post-2010)
(2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole)		Studies
(fentanyl isothiocyanate)		Trials
(fentanyl isothiocyanate)		Recent Studies (post-2010) (fentanyl isothiocyanate)
14022202

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19906 (85.71)18.7374
1990's1 (14.29)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bajwa, BS; Burke, TR; Jacobson, AE; Klee, WA; Rice, KC; Streaty, RA1
Chuang, DM; Coscia, CJ; McLean, S; Rice, KC; Roth, BL; Rothman, RB; Spain, JW1
Aceto, MD; Bajwa, BS; Harris, LS; Jacobson, AE; Klee, WA; Lessor, RA; May, EL; Rice, KC; Smith, CB; Streaty, RA1
Bowen, WD; Burke, TR; Bykov, V; Jacobson, AE; Pert, CB; Rice, KC; Rothman, RB; Schumacher, UK1
Burke, TR; Danks, JA; Jacobson, AE; Pert, CB; Rice, KC; Rothman, RB2
Mash, DC; Partilla, J; Rice, KC; Rothman, RB; Staley, JK1

Other Studies

7 other study(ies) available for 2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazole and fentanyl isothiocyanate

ArticleYear
Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for mu or delta opiate receptors.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Benzimidazoles; Cell Line; Cell Membrane; Chemical Phenomena; Chemistry; Drug Evaluation, Preclinical; Fentanyl; Glioma; Hybrid Cells; Indicators and Reagents; Ligands; Magnetic Resonance Spectroscopy; Mass Spectrometry; Mice; Narcotic Antagonists; Neuroblastoma; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Thebaine

1984
Cross-linking of [125I]beta-endorphin to mu-opioid receptors during development.
    Brain research. Developmental brain research, 1989, Feb-01, Volume: 45, Issue:2

    Topics: Alkylation; Animals; Autoradiography; beta-Endorphin; Cross-Linking Reagents; Electrophoresis, Polyacrylamide Gel; Female; Fentanyl; Isothiocyanates; Male; Microsomes; Rats; Receptors, Opioid; Receptors, Opioid, mu; Succinimides; Synaptic Membranes; Thiocyanates

1989
Probes for narcotic receptor mediated phenomena. 13. Potential irreversible narcotic antagonist-based ligands derived from 6,14-endo-ethenotetrahydronororipavine with 7-(methoxyfumaroyl)amino, (bromoacetyl)amino, or isothiocyanate electrophiles: chemistry
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:11

    Topics: Animals; Brain; Enkephalin, Leucine; Fentanyl; In Vitro Techniques; Isothiocyanates; Ligands; Male; Mice; Mice, Inbred ICR; Narcotic Antagonists; Oligopeptides; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Thebaine; Thiocyanates

1986
Preparation of rat brain membranes greatly enriched with either type-I-delta or type-II-delta opiate binding sites using site directed alkylating agents: evidence for a two-site allosteric model.
    Neuropeptides, 1984, Volume: 4, Issue:3

    Topics: Alkylating Agents; Allosteric Regulation; Animals; Brain; Cell Membrane; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Fentanyl; Isothiocyanates; Kinetics; Male; Oxymorphone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Thiocyanates

1984
Ionic conditions differentially affect 3H-DADL binding to type-I and type-II opiate delta receptors in vitro.
    Neuropeptides, 1984, Volume: 4, Issue:3

    Topics: Animals; Brain; Calcium; Cell Membrane; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Fentanyl; Isothiocyanates; Kinetics; Manganese; Osmolar Concentration; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Sodium; Thiocyanates

1984
Tritiated-6-beta-fluoro-6-desoxy-oxymorphone: a highly selective ligand for the opiate mu receptor whose binding is characterized by low nonspecific binding.
    Neuropeptides, 1984, Volume: 4, Issue:4

    Topics: Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Fentanyl; Hydromorphone; Isothiocyanates; Kinetics; Oxymorphone; Rats; Receptors, Opioid; Receptors, Opioid, mu; Thiocyanates; Tomography, Emission-Computed

1984
Kappa2 opioid receptors in limbic areas of the human brain are upregulated by cocaine in fatal overdose victims.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adult; Amygdala; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Brain Chemistry; Caudate Nucleus; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Drug Overdose; Female; Fentanyl; Gyrus Cinguli; Humans; Isothiocyanates; Kinetics; Male; Morphinans; Protein Binding; Pyrrolidines; Receptors, Opioid, kappa; Tissue Distribution; Up-Regulation

1997