Page last updated: 2024-08-26

2-(2-aminoethyl)thiazole and dimaprit

2-(2-aminoethyl)thiazole has been researched along with dimaprit in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19908 (38.10)18.7374
1990's12 (57.14)18.2507
2000's1 (4.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH1
Nowak, JZ; Sek, B2
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P1
Madrid, JA; Pariente, JA; Salido, GM2
Raybould, HE; Yoneda, M1
Knigge, U; Matzen, S; Warberg, J2
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Guldvog, I; Linnestad, P; Schrumpf, E1
Badger, AM; Poste, G; Young, J1
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G1
Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Iinuma, K; Onodera, K; Watanabe, T; Yokoyama, H1
Malinowska, B; Schlicker, E1
Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J1
Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG; Leurs, R; Timmerman, H1
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G1

Other Studies

21 other study(ies) available for 2-(2-aminoethyl)thiazole and dimaprit

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins

1992
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil

1991
Role of histamine receptors in rabbit pancreatic exocrine secretion stimulated by cholecystokinin and secretin.
    Experimental physiology, 1990, Volume: 75, Issue:5

    Topics: Animals; Chlorpheniramine; Cholecystokinin; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Secretin; Thiazoles; Thiourea

1990
Capsaicin-sensitive vagal afferent fibers do not contribute to histamine H2 receptor agonist-induced gastric acid secretion in anesthetized rats.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Anesthesia; Animals; Capsaicin; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Injections, Subcutaneous; Male; Neurons, Afferent; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vagus Nerve

1990
Histamine receptors in unstimulated pancreatic exocrine secretion of the rabbit.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Kinetics; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1989
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Histaminergic regulation of prolactin secretion: involvement of tuberoinfundibular dopaminergic neurons.
    Neuroendocrinology, 1988, Volume: 48, Issue:2

    Topics: Animals; Cerebral Ventricles; Dimaprit; Dopamine; Histamine; Infusions, Intra-Arterial; Injections, Intraventricular; Male; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Reference Values; Thiazoles; Thiourea

1988
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
    Scandinavian journal of gastroenterology, 1983, Volume: 18, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea

1983
Inhibition of phytohaemagglutinin-induced proliferation of human peripheral blood lymphocytes by histamine and histamine H1 and H2 agonists.
    Clinical and experimental immunology, 1983, Volume: 51, Issue:1

    Topics: Cell Division; Cells, Cultured; Dimaprit; Dose-Response Relationship, Drug; Histamine; Humans; Imidazoles; Impromidine; Lymphocytes; Methylhistamines; Phytohemagglutinins; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
A possible physiological role of histamine H2-receptors in rat mesenteric circulation.
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Animals; Cimetidine; Dimaprit; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Splanchnic Circulation; Thiazoles; Thiourea; Vasodilation

1983
Effects of histamine receptor stimulation on regional myocardial blood flow.
    The American journal of physiology, 1983, Volume: 245, Issue:3

    Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium

1994
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
2-Thiazolylethylamine, a selective histamine H1 agonist, decreases seizure susceptibility in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Anticonvulsants; Dimaprit; Dose-Response Relationship, Drug; Electroshock; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Receptors, Histamine H1; Seizures; Thiazoles

1994
Identification of endothelial H1, vascular H2 and cardiac presynaptic H3 receptors in the pithed rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:1

    Topics: Animals; Blood Pressure; Blood Vessels; Cardiovascular System; Dimaprit; Electric Stimulation; Endothelium, Vascular; Heart Rate; Histamine Agonists; Male; Methylhistamines; Myocardium; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles

1993
The source and action of histamine in the isolated guinea-pig gallbladder.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1995, Volume: 44, Issue:10

    Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles

1995
Histamine H3 receptor inhibition of K(+)-evoked release of acetylcholine from rat cortex in vivo.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45 Suppl 1

    Topics: Acetylcholine; Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Microdialysis; Neurons; Parietal Lobe; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Histamine H3; Thiazoles

1996
Effects of histamine and related compounds on regional cerebral blood flow in rats.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors

1999