Page last updated: 2024-08-24

1h-tetrazole and triazoles

1h-tetrazole has been researched along with triazoles in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19902 (18.18)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's8 (72.73)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Fotsch, C; St Jean, DJ1
Bron, S; Colau, D; Grosdidier, A; Majjigapu, SR; Michielin, O; Pilotte, L; Röhrig, UF; Stroobant, V; Van den Eynde, BJ; Vogel, P; Zoete, V1
Forsman, C; Lindskog, S; Simonsson, I; Tibell, L1
SICHENEDER, T1
Jia, Z; Nakatsu, K; Rahman, MN; Roman, G; Szarek, WA; Vukomanovic, D1
Avery, MA; Gut, J; Legac, J; Rosenthal, PJ; Shah, F; Sherman, W; Shivakumar, D1
Campidelli, S; Jégou, P; Jousselme, B; Morozan, A; Palacin, S; Pinault, M1
Boukraa, M; Doutheau, A; Efrit, ML; Fontaine, F; Grand, L; Queneau, Y; Sabbah, M; Soulère, L1
Adarsh, NN; Garcia, Y; Naik, AD1
Kappes, MM; Karmazin, L; Lebedkin, S; Ruben, M; Schäfer, B; Senthil Kumar, K1
Finiuk, N; Klyuchivska, O; Matiychuk, V; Obushak, M; Pokhodylo, N; Stoika, R1

Reviews

2 review(s) available for 1h-tetrazole and triazoles

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012
Crystal engineering of Fe(II) spin crossover coordination polymers derived from triazole or tetrazole ligands.
    Chimia, 2013, Volume: 67, Issue:6

    Topics: Crystallography, X-Ray; Ferrous Compounds; Magnetics; Models, Molecular; Molecular Structure; Organometallic Compounds; Polymers; Spin Labels; Tetrazoles; Triazoles

2013

Other Studies

9 other study(ies) available for 1h-tetrazole and triazoles

ArticleYear
Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition.
    Journal of medicinal chemistry, 2012, Jun-14, Volume: 55, Issue:11

    Topics: Animals; Catalytic Domain; Cell Line; Drug Design; Enzyme Assays; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Imidazoles; Indoleamine-Pyrrole 2,3,-Dioxygenase; Ligands; Mice; Models, Molecular; Protein Binding; Protein Conformation; Quantitative Structure-Activity Relationship; Quantum Theory; Static Electricity; Triazoles; Tryptophan Oxygenase

2012
The inhibition of human carbonic anhydrase II by some organic compounds.
    Biochimica et biophysica acta, 1985, Jun-10, Volume: 829, Issue:2

    Topics: Binding, Competitive; Carbonic Anhydrase Inhibitors; Chloral Hydrate; Humans; In Vitro Techniques; Kinetics; Nitrophenols; Tetrazoles; Triazoles

1985
[Insulin shock, electro-, tetrazole, triazole convulsions and the peripheral vascular system].
    Therapie der Gegenwart, 1957, Volume: 96, Issue:9

    Topics: Cardiovascular Diseases; Cardiovascular System; Convulsive Therapy; Insulin Coma; Seizures; Sympathomimetics; Tetrazoles; Triazoles

1957
Heme oxygenase inhibition by 2-oxy-substituted 1-azolyl-4-phenylbutanes: effect of variation of the azole moiety. X-ray crystal structure of human heme oxygenase-1 in complex with 4-phenyl-1-(1H-1,2,4-triazol-1-yl)-2-butanone.
    Chemical biology & drug design, 2010, Volume: 75, Issue:1

    Topics: Crystallography, X-Ray; Dioxolanes; Heme Oxygenase (Decyclizing); Heme Oxygenase-1; Humans; Hydrophobic and Hydrophilic Interactions; Imidazoles; Microsomes, Liver; Models, Molecular; Molecular Structure; Structure-Activity Relationship; Tetrazoles; Triazoles; X-Rays

2010
Computer-aided drug design of falcipain inhibitors: virtual screening, structure-activity relationships, hydration site thermodynamics, and reactivity analysis.
    Journal of chemical information and modeling, 2012, Mar-26, Volume: 52, Issue:3

    Topics: Binding Sites; Cysteine Endopeptidases; Drug Design; Drug Evaluation, Preclinical; Humans; Models, Molecular; Molecular Conformation; Protease Inhibitors; Protein Conformation; Quinazolines; Small Molecule Libraries; Structure-Activity Relationship; Tetrazoles; Thermodynamics; Triazoles; User-Computer Interface; Water

2012
Metal-free nitrogen-containing carbon nanotubes prepared from triazole and tetrazole derivatives show high electrocatalytic activity towards the oxygen reduction reaction in alkaline media.
    ChemSusChem, 2012, Volume: 5, Issue:4

    Topics: Catalysis; Electrochemistry; Hydrogen-Ion Concentration; Nanotubes, Carbon; Nitrogen; Oxidation-Reduction; Oxygen; Tetrazoles; Triazoles

2012
Synthesis and biological evaluation of new N-acyl-homoserine-lactone analogues, based on triazole and tetrazole scaffolds, acting as LuxR-dependent quorum sensing modulators.
    Bioorganic & medicinal chemistry, 2012, Aug-01, Volume: 20, Issue:15

    Topics: Homoserine; Lactones; Models, Molecular; Molecular Structure; Repressor Proteins; Structure-Activity Relationship; Tetrazoles; Trans-Activators; Triazoles

2012
Highly luminescent charge-neutral europium(iii) and terbium(iii) complexes with tridentate nitrogen ligands.
    Dalton transactions (Cambridge, England : 2003), 2015, Sep-21, Volume: 44, Issue:35

    Topics: Coordination Complexes; Crystallography, X-Ray; Europium; Lanthanoid Series Elements; Luminescence; Luminescent Agents; Models, Molecular; Nitrogen; Pyridines; Terbium; Tetrazoles; Triazoles

2015
Bioisosteric replacement of 1H-1,2,3-triazole with 1H-tetrazole ring enhances anti-leukemic activity of (5-benzylthiazol-2-yl)benzamides.
    European journal of medicinal chemistry, 2023, Mar-15, Volume: 250

    Topics: Amides; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Cell Proliferation; Structure-Activity Relationship; Triazoles

2023