1h-3-benzazepin-7-ol, 8-bromo-2,3,4,5-tetrahydro-3-methyl-5-phenyl- has been researched along with sk&f-38393 in 86 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (15.12) | 18.7374 |
1990's | 37 (43.02) | 18.2507 |
2000's | 23 (26.74) | 29.6817 |
2010's | 10 (11.63) | 24.3611 |
2020's | 3 (3.49) | 2.80 |
Authors | Studies |
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George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH | 1 |
Chang, JP; Peter, RE; Wong, AO | 2 |
Borrelli, L; Capasso, A; Carginale, V; Madonna, L; Parisi, E | 1 |
Rajashekhar, KP; Wilkens, JL | 1 |
Bell, C; Sunn, N; Woodman, OL | 1 |
O'Boyle, KM; Waddington, JL | 2 |
Cottrell, GA; Meyer, ME; Van Hartesveldt, C | 1 |
Cazin, L; Louiset, E; Valentijn, JA; Vaudry, H | 1 |
Dulka, JG; Peter, RE; Sloley, BD; Trudeau, VL | 1 |
Capasso, A; Carginale, V; De Petrocellis, B; Madonna, L; Mancaniello, D; Paolo De Prisco, P; Parisi, E; Scudiero, R | 1 |
Fukuda, H; Ito, H; Ono, H | 1 |
Kennedy, DA; Travis, ML; Weldon, DA | 1 |
Aronin, N; Baindur, N; Bakthavachalam, V; Canfield, DR; Difiglia, M; Madras, BK; Neumeyer, JL; Pfaelzer, C; Vittimberga, FJ | 1 |
Chang, JP; Peter, RE; Wong, AO; Yu, KL | 1 |
Claro, E; Wallace, MA | 1 |
Ball, SG; Balmforth, AJ; Vaughan, PF; Yasunari, K | 1 |
Feletou, M; Vanhoutte, PM | 1 |
Kopia, GA; Valocik, RE | 1 |
Crooke, ST; Flaim, KE; Gessner, GW; Heys, JR; Weinstock, J | 1 |
Barone, FC; Fine, CF; Fowler, PJ; Grous, M; Lombardi, DM; Ormsbee, HS; Phyall, WB; Rush, JA | 1 |
Mashurano, M; Molloy, AG; O'Boyle, KM; Waddington, JL | 1 |
Altar, CA; Boyar, WC; Gerhardt, SC; Liebman, JM; Wasley, A; Wood, PL | 1 |
Kebabian, JW; Yamamoto, T | 1 |
Molloy, AG; O'Boyle, KM; Pugh, MT; Waddington, JL | 1 |
Boyson, SJ; McGonigle, P; Molinoff, PB | 1 |
Berkowitz, BA; Ohlstein, EH | 1 |
Molloy, AG; Waddington, JL | 1 |
Emaduddin, M; Liu, GJ; Takeuchi, H | 1 |
Heistracher, M; Philippu, A; Prast, H | 1 |
Chuang, YC; Huang, WT; Lin, MT; Liu, HS; Won, SJ | 1 |
Katz, JL; Newman, AH; Nowak, G; Witkin, JM | 1 |
Farrell, CB; O'Boyle, KM | 1 |
Mittleman, G; Rosner, AL; Schaub, CL | 1 |
Cottrell, GA; Meyer, ME; Potter, TJ; Van Hartesveldt, C | 1 |
Gean, PW; Hsu, KS; Huang, CC; Yang, CH | 1 |
Harrison, MB; Login, IS | 1 |
Emaduddin, M; Takeuchi, H | 1 |
Braghiroli, L; De Feo, G; Giacomelli, S; Koppenaal, DW; Ponzianelli, A | 1 |
Gwag, BJ; Noh, JS | 1 |
Fritts, ME; Morris, L; Mueller, K | 2 |
Fischer, H; Philippu, A; Prast, H; Tran, MH | 1 |
Cheng, CY; Giacomelli, S; Palmery, M; Romanelli, L; Silvestrini, B | 1 |
Berndt, TJ; Knox, FG; LeClaire, MM | 1 |
Gáborján, A; Lendvai, B; Vizi, ES | 1 |
Philippu, A; Prast, H; Tran, MH | 1 |
Chen, SF; Cheng, FC; Chung, LJ; Hsueh, CM; Huang, HJ; Kuo, JS; Lin, RJ | 1 |
Lucas-Teixeira, VA; Pestana, M; Serrão, P; Soares-da-Silva, P; Vieira-Coelho, MA | 1 |
Cory-Slechta, DA; Zuch, CL | 1 |
Gomes, P; Soares-Da-Silva, P; Vieira-Coelho, MA | 1 |
Miller, JW; Roth, KA; Torack, RM | 1 |
Aberman, JE; Arizzi, MN; Cervone, KM; Salamone, JD; Sandoval, MD | 1 |
Gomes, P; Soares-Da-Silva, P | 1 |
Khorevin, VI; Rozumna, NM; Storozhuk, VM; Tetko, IV; Villa, AE | 1 |
Liang, PJ; Liu, Y; Luo, FJ | 1 |
Alonso, G; Duvoid, A; Hussy, N; Moos, F; Runquist, M | 1 |
Fraga, S; Jose, PA; Soares-da-Silva, P | 1 |
Kiehn, L; Mukai, ST; Saleuddin, AS | 1 |
Gomes, P; Hopfer, U; Jose, PA; Pedrosa, R; Soares-da-Silva, P; Zeng, C | 1 |
Xiang, G; Zhang, L; Zhou, R | 1 |
Canlon, B; Niu, X | 1 |
Asgari, K; Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Szabadi, E | 1 |
Domenger, D; Schwarting, RK | 1 |
Ariano, MA; Cepeda, C; Hernández-Echeagaray, E; Levine, MS; Lobo, MK; Sibley, DR | 1 |
Asgari, K; Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Glennon, JC; Szabadi, E | 1 |
Fraga, S; Jose, P; Luo, Y; Mount, DB; Soares-da-Silva, P; Zandi-Nejad, K | 1 |
Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Hampson, CL; Szabadi, E | 1 |
Chen, H; Ho, WZ; Liang, H; Song, L; Wang, SH; Wang, X; Wang, YJ; Ye, L; Zhou, L | 1 |
Griffin, WC; Krnjević, K; Li, KY; Olive, MF; Shao, XM; Xiao, C; Ye, JH; Zhou, C | 1 |
Coppa-Hopman, R; Galle, J; Pimkine, D | 1 |
Ali, S; Carr, KD; Patel, JC; Reith, ME; Rice, ME; Sarti, F; Stouffer, MA | 1 |
Diefenbach, TJ; Goldberg, JI; Kuang, S; Liu, MB; Muruganathan, SP; Pon, JR; Rich, DR; Tam, R | 1 |
Currie, PJ; Jacoby, SM | 1 |
Kawabe, K; Moriyama, M; Nakamura, Y; Takano, K; Tanaka, N | 1 |
Adelekun, AE; Hannaway, KE; Horiguchi, M; Huang, M; Jayathilake, K; Meltzer, HY | 1 |
Chen, L; Wang, L; Ye, JH; Zuo, W | 1 |
Bradshaw, CM; Cassaday, HJ; Olarte-Sánchez, CM; Szabadi, E; Valencia-Torres, L | 1 |
Bogard, AS; Brand, CS; Conley, JM; Dessauer, CW; Hockerman, GH; Ostrom, RS; Pratt, EP; Watts, VJ; Xu, R | 1 |
Bashir, ZI; Savalli, G; Warburton, EC | 1 |
Chien, ME; Hsu, KS; Wu, YJ; Yu, TH | 1 |
Alghorabi, AA; Alkhalifa, T; Almalki, AD; Almalki, AH; Almutairi, FM; Alsaab, HO; Alsanie, WF; Alshehri, FS; Althobaiti, YS; Altowairqi, E; Gaber, A; Hakami, AY; Hardy, AMG; Marghalani, AM; Shah, ZA | 1 |
Huang, H; Li, C; Wang, J; Zhang, B; Zheng, S; Zhu, X | 1 |
Baindur, N; Bakthavachalam, V; Madras, BK; Neumeyer, JL | 1 |
Alberts, I; Giri, R; Harding, WW; Namballa, HK; Sarker, A | 1 |
86 other study(ies) available for 1h-3-benzazepin-7-ol, 8-bromo-2,3,4,5-tetrahydro-3-methyl-5-phenyl- and sk&f-38393
Article | Year |
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Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection | 1991 |
Dopamine stimulates growth hormone release from the pituitary of goldfish, Carassius auratus, through the dopamine D1 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Bromocriptine; Domperidone; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Goldfish; Gonadotropin-Releasing Hormone; Growth Hormone; Pituitary Gland; Quinpirole; Radioimmunoassay; Receptors, Dopamine | 1992 |
Adenylate cyclase from sea urchin eggs is positively and negatively regulated by D-1 and D-2 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Dopamine; Dopamine Agents; Metergoline; Ovum; Phenethylamines; Receptors, Dopamine D1; Receptors, Dopamine D2; Sea Urchins | 1992 |
Dopamine and nicotine, but not serotonin, modulate the crustacean ventilatory pattern generator.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Brachyura; Domperidone; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Ganglia; Motor Neurons; Neural Pathways; Nicotine; Receptors, Dopamine D1; Respiration; Serotonin; Thorax | 1992 |
Involvement of dopamine in control of renal blood flow.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Blood Pressure; Coronary Circulation; Coronary Vessels; Dogs; Dopamine; Female; Glomerular Filtration Rate; Kidney; Kidney Function Tests; Male; Receptors, Dopamine D1; Renal Circulation | 1992 |
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1992 |
Dopamine D1 antagonists potentiate the durations of bar and cling catalepsy and the dorsal immobility response in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Catalepsy; Dopamine Antagonists; Male; Motor Activity; Rats; Receptors, Dopamine; Receptors, Dopamine D1 | 1992 |
Dopamine-induced inhibition of action potentials in cultured frog pituitary melanotrophs is mediated through activation of potassium channels and inhibition of calcium and sodium channels.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Calcium Channel Blockers; Calcium Chloride; Dopamine; In Vitro Techniques; Male; Melanins; Membrane Potentials; Pituitary Gland; Potassium Channels; Rana ridibunda; Sodium Channels; Sulpiride; Tetrodotoxin | 1991 |
Selective depletion of dopamine in the goldfish pituitary caused by domperidone.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Benzazepines; Body Weight; Brain Chemistry; Carbidopa; DOM 2,5-Dimethoxy-4-Methylamphetamine; Domperidone; Dopamine; Dose-Response Relationship, Drug; Female; Goldfish; Gonadotropins; Hypothalamus; Male; Methyltyrosines; Mice; Norepinephrine; Pituitary Gland; Receptors, Dopamine; Serotonin; Telencephalon; Tyrosine 3-Monooxygenase | 1991 |
A dopamine- and octopamine-sensitive adenylate cyclase in the nervous system of Octopus vulgaris.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Binding, Competitive; Cattle; Dopamine; Epinephrine; Female; Insecta; Male; Nervous System; Norepinephrine; Octopamine; Octopodiformes | 1991 |
2-phenylethylamine and methamphetamine enhance the spinal monosynaptic reflex by releasing noradrenaline from the terminals of descending fibers.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Blood Pressure; Hydroxydopamines; Male; Methamphetamine; Monoamine Oxidase Inhibitors; Nerve Endings; Neurons; Norepinephrine; Oxidopamine; Phenethylamines; Prazosin; Psychotropic Drugs; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reflex, Monosynaptic; Reserpine; Spinal Cord | 1991 |
Posttraining D1 receptor blockade impairs odor conditioning in neonatal rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Association Learning; Conditioning, Classical; Dopamine Antagonists; Female; Male; Odorants; Olfactory Bulb; Physical Stimulation; Rats; Receptors, Dopamine; Reinforcement, Psychology; Smell; Sodium Chloride | 1991 |
Fluorescent and biotin probes for dopamine receptors: D1 and D2 receptor affinity and selectivity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Biotin; Brain; Female; Fluoresceins; Fluorescent Dyes; Macaca fascicularis; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin | 1990 |
Differential actions of dopamine receptor subtypes on gonadotropin and growth hormone release in vitro in goldfish.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Cells, Cultured; Cyprinidae; Domperidone; Dopamine Antagonists; Ergolines; Female; Goldfish; Gonadotropins, Pituitary; Growth Hormone; Male; Perfusion; Pituitary Gland; Pituitary Hormone-Releasing Hormones; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1990 |
A novel role for dopamine: inhibition of muscarinic cholinergic-stimulated phosphoinositide hydrolysis in rat brain cortical membranes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Carbachol; Cerebral Cortex; Dopamine; In Vitro Techniques; Male; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Muscarinic; Type C Phospholipases | 1990 |
Characterization of dopamine and beta-adrenergic receptors linked to cyclic AMP formation in intact cells of the clone D384 derived from a human astrocytoma.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic beta-Antagonists; Astrocytoma; Benzazepines; Cyclic AMP; Domperidone; Dopamine; Dopamine Antagonists; Humans; Isoproterenol; Practolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D1; Tetrahydronaphthalenes; Tumor Cells, Cultured | 1988 |
Tetrodotoxin-insensitive relaxation of coronary arterial smooth muscle to electrical stimulation: possible involvement of a dopaminergic mechanism.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Calcium; Cattle; Coronary Vessels; Dogs; Dopamine; Electric Stimulation; Female; Hydroxydopamines; In Vitro Techniques; Male; Oxidopamine; Receptors, Dopamine; Scorpion Venoms; Swine; Tetraethylammonium Compounds; Tetrodotoxin; Vasodilation | 1989 |
Demonstration of specific dopamine-1 receptor-mediated coronary vasodilation in the anesthetized dog.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Anesthesia; Angina Pectoris; Animals; Benzazepines; Coronary Circulation; Dogs; Domperidone; Dopamine; Female; Fenoldopam; Male; Receptors, Dopamine; Receptors, Dopamine D1; Vasodilation | 1989 |
Regulation of agonist and antagonist binding to striatal D-1 dopamine receptors: studies using the selective D-1 antagonist [3H]SK&F R-83566.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine Triphosphate; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Fenoldopam; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Lithium; Male; Membranes; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium | 1986 |
DA1 receptor mediates dopamine-induced relaxation of opossum lower esophageal sphincter in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Aporphines; Benzazepines; Deoxyepinephrine; Domperidone; Dopamine; Dose-Response Relationship, Drug; Esophagogastric Junction; Female; In Vitro Techniques; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Opossums; Receptors, Dopamine | 1986 |
Structural analogs of SCH 23390 as discriminators of dopamine receptor subtypes: behavioral interactions between D-1 and D-2 agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Brain; Humans; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Structure-Activity Relationship | 1986 |
Dopamine neurochemical profile of atypical antipsychotics resembles that of D-1 antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Behavior, Animal; Benzazepines; Brain Chemistry; Dopamine; Dopamine Antagonists; Male; Mice; Motor Activity; Pargyline; Stereotyped Behavior | 1988 |
Occurrence of the D-1 dopamine receptor in the substantia nigra of several mammalian species: identification in binding studies using [125I]SCH 23982.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Cats; Caudate Nucleus; Guinea Pigs; Ligands; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, GABA-A; Substantia Nigra | 1987 |
Locomotor behaviors in response to new selective D-1 and D-2 dopamine receptor agonists, and the influence of selective antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Flupenthixol; Isoquinolines; Male; Metoclopramide; Motor Activity; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stimulation, Chemical | 1986 |
Quantitative autoradiographic localization of the D1 and D2 subtypes of dopamine receptors in rat brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Brain Chemistry; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
SCH 23390 and SK&F 83566 are antagonists at vascular dopamine and serotonin receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aorta, Thoracic; Benzazepines; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Rabbits; Receptors, Dopamine; Receptors, Serotonin; Serotonin | 1985 |
The enantiomers of SK&F 83566, a new selective D-1 dopamine antagonist, stereospecifically block stereotyped behaviour induced by apomorphine and by the selective D-2 agonist RU 24213.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Male; Motor Activity; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Stereotyped Behavior | 1985 |
Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Thioxanthenes | 1984 |
Effects of dopamine on snail neurones.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Membrane Potentials; Neurons; Snails; Sulpiride; Time Factors | 1995 |
Modulation by dopamine receptors of the histamine release in the rat hypothalamus.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine Agents; Dopamine Antagonists; Histamine Release; Hypothalamus; Male; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride | 1993 |
Suppression of natural killer cell activity in mouse spleen lymphocytes by several dopamine receptor antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cytotoxicity, Immunologic; Dopamine Antagonists; Flupenthixol; Fluphenazine; Killer Cells, Natural; Mice; Mice, Inbred C3H; Pimozide; Spiperone; Spleen; Thiothixene; Trifluoperazine | 1995 |
Role of dopamine D1 receptors in the lethal effects of cocaine and a quaternary methiodide analog.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cocaine; Dopamine D2 Receptor Antagonists; Fenoldopam; Lidocaine; Male; Mice; Motor Activity; Rats; Rats, Inbred F344; Receptors, Dopamine D1; Receptors, Dopamine D2; Seizures; Structure-Activity Relationship | 1993 |
The kinetics of [3H]SCH 23390 dissociation from rat striatal dopamine D1 receptors: effect of dopamine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Allosteric Site; Animals; Benzazepines; Binding, Competitive; Brain; Cell Membrane; Dopamine; Dopamine Antagonists; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1 | 1994 |
Polydipsia and dopamine: behavioral effects of dopamine D1 and D2 receptor agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Diazepam; Dopamine Agonists; Dopamine Antagonists; Drinking; Eating; Ergolines; Haloperidol; Male; Motor Activity; Quinpirole; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Thirst | 1994 |
Characterization of D1 receptors mediating dopamine-stimulated growth hormone release from pituitary cells of the goldfish, Carassius auratus.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Binding, Competitive; Domperidone; Dopamine; Ergolines; Goldfish; Growth Hormone; Kinetics; Pituitary Gland; Quinpirole; Receptors, Dopamine D1; Serotonin; Somatostatin | 1993 |
Effects of dopamine D1 antagonists SCH23390 and SK&F83566 on locomotor activities in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Benzazepines; Dose-Response Relationship, Drug; Male; Motor Activity; Rats; Receptors, Dopamine D1; Stereotyped Behavior; Time Factors | 1993 |
Presynaptic D2 dopaminergic receptors mediate inhibition of excitatory synaptic transmission in rat neostriatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Dopamine; Dopamine Antagonists; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Neostriatum; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Presynaptic; Sulpiride; Synaptic Transmission | 1995 |
A D1 dopamine agonist stimulates acetylcholine release from dissociated striatal cholinergic neurons.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Calcium; Choline; Corpus Striatum; Dopamine Antagonists; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Neurons; Rats; Receptors, Dopamine D1; Stereoisomerism; Tritium | 1996 |
Lineweaver-Burk analysis for the blocking effects of mammalian dopamine receptor antagonists on dopamine-induced currents in Achatina giant neurones.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ganglia, Invertebrate; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Receptors, Dopamine; Receptors, Dopamine D1; Snails; Sulpiride | 1996 |
A sensitive assay for studying dopaminergic activity in cultures of rat pituitary cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cell Count; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation, Preclinical; Female; Haloperidol; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Spiperone | 1997 |
Attenuation of oxidative neuronal necrosis by a dopamine D1 agonist in mouse cortical cell cultures.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antioxidants; Apoptosis; Cells, Cultured; Cerebral Cortex; Chromans; Culture Media, Serum-Free; Dopamine Agonists; Dopamine Antagonists; Mice; Necrosis; Neurons; Neuroprotective Agents; Oxidation-Reduction; Receptors, Dopamine D1; Vitamin E | 1997 |
Amphetamine-induced locomotor stereotypy in rats is reduced by a D1 but not a D2 antagonist.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Stereotyped Behavior; Sulpiride | 1997 |
Nitric oxide-induced release of acetylcholine in the nucleus accumbens: role of cyclic GMP, glutamate, and GABA.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Chromatography, High Pressure Liquid; Cyclic GMP; Diethylamines; Dopamine Antagonists; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Guanylate Cyclase; Male; Neurons; Nitric Oxide; Nitrogen Oxides; Nucleus Accumbens; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Receptors, Dopamine; Receptors, GABA; Receptors, Glutamate | 1998 |
Locomotor stereotypy produced by dexbenzetimide and scopolamine is reduced by SKF 83566, not sulpiride.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dexetimide; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Locomotion; Male; Muscarinic Antagonists; Rats; Rats, Wistar; Receptors, Dopamine D1; Scopolamine; Stereotyped Behavior; Sulpiride | 1998 |
Lysergic acid diethylamide (LSD) is a partial agonist of D2 dopaminergic receptors and it potentiates dopamine-mediated prolactin secretion in lactotrophs in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Lysergic Acid Diethylamide; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2 | 1998 |
Effect of renal interstitial infusion of L-dopa on sodium and phosphate excretions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Infusions, Parenteral; Kidney Tubules, Proximal; Levodopa; Male; Natriuresis; Phosphates; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium; Sulpiride | 1998 |
Neurochemical evidence of dopamine release by lateral olivocochlear efferents and its presynaptic modulation in guinea-pig cochlea.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Axons; Bromocriptine; Cadmium Chloride; Calcium Signaling; Cochlea; Cochlear Nucleus; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Efferent Pathways; Feedback; Guinea Pigs; Male; Models, Neurological; Neuroprotective Agents; Nomifensine; Olivary Nucleus; Piribedil; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Presynaptic; Sulpiride; Tetrodotoxin | 1999 |
Histaminergic H2 receptor ligands modulate acetylcholine release in the ventral striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Corpus Striatum; Dimaprit; Dopamine; Dopamine Agonists; Dopamine Antagonists; Famotidine; gamma-Aminobutyric Acid; Histamine; Histamine H2 Antagonists; Male; Neurons; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2 | 1999 |
Involvement of catecholamines in recall of the conditioned NK cell response.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amygdala; Animals; Atenolol; Brain Chemistry; Catecholamines; Cerebellum; Cerebral Cortex; Chromatography, High Pressure Liquid; Conditioning, Classical; Corpus Striatum; Dopamine; Dopamine Antagonists; Epinephrine; Female; Immunologic Memory; Killer Cells, Natural; Lymphocyte Activation; Mental Recall; Mice; Mice, Inbred BALB C; Norepinephrine; Oxathiins; Propanolamines; Salicylamides; Spleen; Yohimbine | 1999 |
Salt intake and sensitivity of intestinal and renal Na+-K+ atpase to inhibition by dopamine in spontaneous hypertensive and Wistar-Kyoto rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Diet, Sodium-Restricted; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Inhibitors; Hypertension; In Vitro Techniques; Jejunum; Kidney Tubules, Proximal; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Dopamine D1; Sodium-Potassium-Exchanging ATPase; Sodium, Dietary; Sulpiride | 2000 |
Stimulus properties of 7-OH-DPAT versus auto- and postsynaptic receptor-specific doses of quinpirole.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clozapine; Dopamine Antagonists; Female; Haloperidol; Maternal Behavior; Motivation; Motor Activity; Pimozide; Rats | 2001 |
Ouabain-insensitive acidification by dopamine in renal OK cells: primary control of the Na(+)/H(+) exchanger.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acids; Animals; Bicarbonates; Biological Transport; Cardiotonic Agents; Cell Line; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Inhibitors; Female; Hydrogen-Ion Concentration; Kidney Tubules, Proximal; Opossums; Ouabain; Radioligand Assay; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium-Hydrogen Exchangers; Sodium-Potassium-Exchanging ATPase; Tritium | 2001 |
Deafferentation-induced abnormal neurofilament phosphorylation in red nucleus neurones.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Afferent Pathways; Animals; Benzazepines; Dementia; Denervation; Dopamine Antagonists; Hippocampus; Immunohistochemistry; Neurofibrillary Tangles; Neurofilament Proteins; Parvalbumins; Phosphorylation; Rats; Receptors, Dopamine D2; Red Nucleus; Silver Staining; Ventral Tegmental Area | 2001 |
Dopamine antagonists alter response allocation but do not suppress appetite for food in rats: contrast between the effects of SKF 83566, raclopride, and fenfluramine on a concurrent choice task.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetite Depressants; Choice Behavior; Dopamine Antagonists; Eating; Fenfluramine; Food Preferences; Male; Raclopride; Rats; Rats, Sprague-Dawley; Reaction Time; Reinforcement, Psychology; Selective Serotonin Reuptake Inhibitors | 2002 |
D2-like receptor-mediated inhibition of Na+-K+-ATPase activity is dependent on the opening of K+ channels.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphotericin B; Animals; Antifungal Agents; Cardiotonic Agents; Cell Line; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Glyburide; GTP-Binding Protein alpha Subunits, Gi-Go; Hypoglycemic Agents; Ion Channel Gating; Kidney; Opossums; Pertussis Toxin; Pinacidil; Potassium Channels; Quinolines; Receptors, Dopamine D2; Sodium; Sodium-Potassium-Exchanging ATPase; Sulpiride; Vasodilator Agents; Virulence Factors, Bordetella | 2002 |
Dopamine modulation of activity of cat sensorimotor cortex neurons during conditioned reflexes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acoustic Stimulation; Action Potentials; Animals; Cats; Conditioning, Classical; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Electromyography; Male; Motor Cortex; Neurons; Pyramidal Cells; Quinpirole; Reaction Time; Sulpiride | 2002 |
Dopamine effect on the stimulus pattern related changes in response characteristics of R/G horizontal cells in carp retina.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic Agents; Animals; Carps; Dopamine; Dopamine Antagonists; Drug Interactions; In Vitro Techniques; Light; Membrane Potentials; Neurons; Oxidopamine; Receptors, Dopamine D2; Retina; Salicylamides; Time Factors | 2003 |
Age-related modifications of the morphological organization of pituicytes are associated with alteration of the GABAergic and dopaminergic innervation afferent to the neurohypophysial lobe.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Afferent Pathways; Aging; Animals; Astrocytes; Axons; Cell Count; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Isotonic Solutions; Male; Microscopy, Electron; Microscopy, Immunoelectron; Muscimol; Pyridazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Sulpiride; Tyrosine 3-Monooxygenase | 2003 |
Involvement of G protein-coupled receptor kinase 4 and 6 in rapid desensitization of dopamine D1 receptor in rat IEC-6 intestinal epithelial cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antibodies, Blocking; Blotting, Western; Cell Line; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Enzyme Inhibitors; Epithelial Cells; G-Protein-Coupled Receptor Kinase 4; G-Protein-Coupled Receptor Kinases; Heparin; Intestines; Isoenzymes; Protein Serine-Threonine Kinases; Rats; Receptors, Dopamine D1; Sodium-Hydrogen Exchangers | 2004 |
Dopamine stimulates snail albumen gland glycoprotein secretion through the activation of a D1-like receptor.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Exocrine Glands; Fresh Water; Glycoproteins; Phenanthridines; Receptors, Dopamine D1; Reproduction; Signal Transduction; Snails; Tetrahydronaphthalenes | 2004 |
Dopamine D3 receptor-mediated inhibition of Na+/H+ exchanger activity in normotensive and spontaneously hypertensive rat proximal tubular epithelial cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Blood Pressure; Cell Line, Transformed; Cells, Cultured; Dopamine; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Epithelial Cells; Hypertension; Kidney Tubules, Proximal; Male; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Dopamine D2; Receptors, Dopamine D3; Sodium-Hydrogen Exchangers | 2004 |
Stepholidine protects against H2O2 neurotoxicity in rat cortical neurons by activation of Akt.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Berberine; Blotting, Western; Cell Count; Cell Death; Cells, Cultured; Chromones; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Gene Expression Regulation; Haloperidol; Hydrogen Peroxide; Morpholines; Neurons; Neuroprotective Agents; Prefrontal Cortex; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Time Factors | 2005 |
The signal transduction pathway for the dopamine D1 receptor in the guinea-pig cochlea.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Blotting, Western; Cochlea; Cochlear Nerve; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Dopamine and cAMP-Regulated Phosphoprotein 32; Female; Guinea Pigs; Immunohistochemistry; Isoquinolines; Male; Oxidopamine; Perfusion; Receptors, AMPA; Receptors, Dopamine D1; Signal Transduction; Sulfonamides; Sympathectomy, Chemical; Sympatholytics | 2006 |
Evidence for a role of D1 dopamine receptors in d-amphetamine's effect on timing behaviour in the free-operant psychophysical procedure.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Conditioning, Operant; Dextroamphetamine; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Motor Activity; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Time Perception | 2006 |
The serial reaction time task in the rat: effects of D1 and D2 dopamine-receptor antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Conditioning, Operant; Dopamine Antagonists; Male; Practice, Psychological; Psychomotor Performance; Raclopride; Random Allocation; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Receptors, Dopamine D2; Serial Learning; Statistics, Nonparametric | 2006 |
Dopamine reduction of GABA currents in striatal medium-sized spiny neurons is mediated principally by the D(1) receptor subtype.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Mice; Mice, Knockout; Patch-Clamp Techniques; Receptors, Dopamine D1; Receptors, Dopamine D5; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; Sulpiride | 2007 |
Effects of d-amphetamine and DOI (2,5-dimethoxy-4-iodoamphetamine) on timing behavior: interaction between D1 and 5-HT2A receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Amphetamines; Animals; Conditioning, Operant; Drug Interactions; Female; Fluorobenzenes; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists; Time Perception | 2006 |
Dopamine D1-like receptor-mediated inhibition of Cl/HCO3- exchanger activity in rat intestinal epithelial IEC-6 cells is regulated by G protein-coupled receptor kinase 6 (GRK 6).
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cells, Cultured; Chloride-Bicarbonate Antiporters; Dopamine Agonists; Dopamine Antagonists; G-Protein-Coupled Receptor Kinase 4; G-Protein-Coupled Receptor Kinases; Gene Expression; Heparin; Heparin Antagonists; Immunohistochemistry; Intestinal Mucosa; Intestines; Protein Serine-Threonine Kinases; Rats; Receptors, Dopamine D1; RNA, Messenger | 2006 |
Evidence for the sensitivity of operant timing behaviour to stimulation of D1 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Psychometrics; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Time Perception | 2007 |
Methamphetamine enhances HIV infection of macrophages.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Cells, Cultured; Central Nervous System Stimulants; Down-Regulation; HIV-1; Humans; Interferon-alpha; Macrophages; Methamphetamine; Receptors, CCR5; Receptors, Dopamine D1; STAT1 Transcription Factor; Virus Replication | 2008 |
Ethanol facilitates glutamatergic transmission to dopamine neurons in the ventral tegmental area.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Ethanol; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Neurons; Piperazines; Quinoxalines; Raclopride; Rats; Receptors, AMPA; Receptors, Dopamine D1; Reserpine; Synaptic Transmission; Ventral Tegmental Area | 2009 |
D1 receptor antagonist-induced long-term depression in the medial prefrontal cortex of rat, in vivo: an animal model of psychiatric hypofrontality.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Chromans; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Male; Neuronal Plasticity; Prefrontal Cortex; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate | 2009 |
SKF-83566, a D1-dopamine receptor antagonist, inhibits the dopamine transporter.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; In Vitro Techniques; Male; Nomifensine; Prosencephalon; Protein Binding; Rats; Rats, Sprague-Dawley; Tritium; Tropanes | 2011 |
Identification and evolutionary implications of neurotransmitter-ciliary interactions underlying the behavioral response to hypoxia in Lymnaea stagnalis embryos.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Anaerobiosis; Animals; Behavior, Animal; Biological Evolution; Cilia; Dopamine; Embryo, Nonmammalian; Fluorescent Antibody Technique; Lymnaea; Mianserin; Neurotransmitter Agents; Rotation; Serotonin; Time Factors | 2011 |
SKF 83566 attenuates the effects of ghrelin on performance in the object location memory task.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetite; Dopamine; Dopamine Antagonists; Eating; Exploratory Behavior; Ghrelin; Injections, Intraventricular; Long-Term Potentiation; Male; Memory Disorders; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spatial Behavior | 2011 |
Extracellular superoxide dismutase induced by dopamine in cultured astrocytes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Astrocytes; Blotting, Western; Cell Survival; Cells, Cultured; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Extracellular Space; Nerve Tissue Proteins; NF-kappa B; Piperazines; Rats; Reactive Oxygen Species; Real-Time Polymerase Chain Reaction; RNA, Messenger; Stimulation, Chemical; Superoxide Dismutase | 2013 |
D(1) receptor agonists reverse the subchronic phencyclidine (PCP)-induced novel object recognition (NOR) deficit in female rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Female; Isoindoles; Phencyclidine; Piperazines; Pyrimidines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D1; Recognition, Psychology; Serotonin 5-HT1 Receptor Agonists | 2013 |
Cocaine facilitates glutamatergic transmission and activates lateral habenular neurons.
Topics: 2-Amino-5-phosphonovalerate; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Calcium Channels; Cocaine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABAergic Neurons; Glutamic Acid; Habenula; Male; Miniature Postsynaptic Potentials; Piperazines; Quinoxalines; Quinpirole; Raclopride; Rats; Receptors, Dopamine; Receptors, Glutamate; Sodium Channels; Synaptic Transmission | 2013 |
Effects of SKF-83566 and haloperidol on performance on progressive ratio schedules maintained by sucrose and corn oil reinforcement: quantitative analysis using a new model derived from the Mathematical Principles of Reinforcement (MPR).
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Conditioning, Operant; Corn Oil; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Injections, Intraperitoneal; Models, Theoretical; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Reinforcement Schedule; Sucrose | 2013 |
Development of a high-throughput screening paradigm for the discovery of small-molecule modulators of adenylyl cyclase: identification of an adenylyl cyclase 2 inhibitor.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Membrane; Cyclic AMP; Enzyme Inhibitors; HEK293 Cells; High-Throughput Screening Assays; Humans; Mice; Myocytes, Smooth Muscle; Sf9 Cells; Small Molecule Libraries; Spodoptera; Transfection | 2013 |
Regionally selective requirement for D1/D5 dopaminergic neurotransmission in the medial prefrontal cortex in object-in-place associative recognition memory.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Association Learning; Benzazepines; Dopamine Antagonists; Male; Prefrontal Cortex; Rats; Receptors, Dopamine D1; Receptors, Dopamine D5; Recognition, Psychology; Spatial Memory; Synaptic Transmission | 2015 |
Transcranial direct current stimulation induces hippocampal metaplasticity mediated by brain-derived neurotrophic factor.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic beta-Antagonists; Animals; Avoidance Learning; Azepines; Benzamides; Brain-Derived Neurotrophic Factor; CA1 Region, Hippocampal; Long-Term Potentiation; Male; Memory; Propranolol; Random Allocation; Rats, Sprague-Dawley; Receptor, trkB; Receptors, Dopamine D1; Synapses; Tissue Culture Techniques; Transcranial Direct Current Stimulation | 2019 |
Involvement of the dopaminergic system in the reward-related behavior of pregabalin.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Behavior, Animal; Dopaminergic Neurons; Male; Mice, Inbred BALB C; Pregabalin; Random Allocation; Receptors, Dopamine D1; Reward | 2021 |
The effects of aging and dopaminergic inhibition on large scale maze learning in rhesus monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Intravenous; Aging; Animals; Dopamine Antagonists; Haloperidol; Macaca mulatta; Male; Maze Learning; Psychomotor Performance; Spatial Navigation | 2021 |
Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine Antagonists; Fluorescent Dyes; Ligands; Macaca fascicularis; Oxadiazoles; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship | 1991 |
Synthesis and dopamine receptor pharmacological evaluations on ring C ortho halogenated 1-phenylbenzazepines.
Topics: Benzazepines; Dopamine Antagonists; Dose-Response Relationship, Drug; Halogenation; Molecular Structure; Receptors, Dopamine D1; Structure-Activity Relationship | 2020 |