Page last updated: 2024-09-03

1-naphthylacetylspermine and morphine

1-naphthylacetylspermine has been researched along with morphine in 1 studies

Compound Research Comparison

Studies
(1-naphthylacetylspermine)
Trials
(1-naphthylacetylspermine)
Recent Studies (post-2010)
(1-naphthylacetylspermine)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
5102244,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomy1-naphthylacetylspermine (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carusillo, B; Fakira, AK; Melyan, Z; MorĂ³n, JA; Portugal, GS1

Other Studies

1 other study(ies) available for 1-naphthylacetylspermine and morphine

ArticleYear
Increased small conductance calcium-activated potassium type 2 channel-mediated negative feedback on N-methyl-D-aspartate receptors impairs synaptic plasticity following context-dependent sensitization to morphine.
    Biological psychiatry, 2014, Jan-15, Volume: 75, Issue:2

    Topics: Animals; Apamin; Central Nervous System Sensitization; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Feedback, Physiological; Hippocampus; Long-Term Potentiation; Male; Mice; Morphine; Motor Activity; Neuronal Plasticity; Okadaic Acid; Protein Phosphatase 2; Protein Subunits; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Small-Conductance Calcium-Activated Potassium Channels; Spermine; Synaptic Potentials

2014