Page last updated: 2024-09-03

1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) and spiradoline

1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) has been researched along with spiradoline in 2 studies

Compound Research Comparison

Studies
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Trials
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Recent Studies (post-2010)
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Studies
(spiradoline)
Trials
(spiradoline)
Recent Studies (post-2010) (spiradoline)
3520132624

Protein Interaction Comparison

ProteinTaxonomy1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) (IC50)spiradoline (IC50)
Mu-type opioid receptorHomo sapiens (human)0.234
Kappa-type opioid receptorHomo sapiens (human)0.0083

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ohno, M; Ueki, S; Yamamoto, T1
Butelman, ER; Harris, TJ; Kreek, MJ1

Other Studies

2 other study(ies) available for 1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) and spiradoline

ArticleYear
Analgesic and discriminative stimulus properties of U-62,066E, the selective kappa-opioid receptor agonist, in the rat.
    Psychopharmacology, 1992, Volume: 106, Issue:1

    Topics: Analgesics; Animals; Benzomorphans; Cues; Discrimination, Psychological; Dopamine; Dopamine Antagonists; Dynorphins; Male; Morphine; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1992
Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys.
    Psychopharmacology, 1999, Volume: 147, Issue:1

    Topics: Animals; Azocines; Dose-Response Relationship, Drug; Dynorphins; Female; Hypnotics and Sedatives; Injections, Subcutaneous; Macaca mulatta; Male; Motor Activity; Muscle Relaxation; Naltrexone; Narcotic Antagonists; Peptide Fragments; Prolactin; Pyrrolidines; Receptors, Opioid, kappa; Time Factors

1999