1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 3 studies
Studies (1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8)) | Trials (1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8)) | Recent Studies (post-2010) (1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8)) | Studies (enkephalin, ala(2)-mephe(4)-gly(5)-) | Trials (enkephalin, ala(2)-mephe(4)-gly(5)-) | Recent Studies (post-2010) (enkephalin, ala(2)-mephe(4)-gly(5)-) |
---|---|---|---|---|---|
35 | 2 | 0 | 151 | 0 | 71 |
35 | 2 | 0 | 2,727 | 1 | 374 |
Protein | Taxonomy | 1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) (IC50) | enkephalin, ala(2)-mephe(4)-gly(5)- (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 0.003 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 0.003 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 0.003 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 0.003 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 0.003 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 1.2415 | |
Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0132 | |
Mu-type opioid receptor | Homo sapiens (human) | 0.004 | |
Delta-type opioid receptor | Homo sapiens (human) | 0.0014 | |
Mu-type opioid receptor | Mus musculus (house mouse) | 0.0048 | |
Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0283 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Akil, H; Goldstein, A; Mansour, A; Meng, F; Thompson, RC; Watson, SJ; Xie, GX | 1 |
Herz, A; Shippenberg, TS; Spanagel, R | 1 |
Ableitner, A; Bals-Kubik, R; Herz, A; Shippenberg, TS | 1 |
3 other study(ies) available for 1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) and enkephalin, ala(2)-mephe(4)-gly(5)-
Article | Year |
---|---|
Cloning and pharmacological characterization of a rat kappa opioid receptor.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Analgesics; Animals; Benzeneacetamides; Cell Line; Cell Membrane; Cloning, Molecular; Corpus Striatum; Cyclic AMP; DNA Primers; DNA, Complementary; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Gene Library; In Situ Hybridization; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Molecular Sequence Data; Pyrrolidines; Rats; Receptors, Opioid, kappa; Restriction Mapping; RNA, Messenger; Transfection | 1993 |
The effects of opioid peptides on dopamine release in the nucleus accumbens: an in vivo microdialysis study.
Topics: Analgesics; Animals; Dialysis; Dopamine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Magnesium; Male; Nucleus Accumbens; Peptide Fragments; Potassium; Rats; Rats, Inbred Strains; Tetrodotoxin | 1990 |
Neuroanatomical sites mediating the motivational effects of opioids as mapped by the conditioned place preference paradigm in rats.
Topics: Amino Acid Sequence; Animals; Association Learning; Autoradiography; Brain Mapping; Conditioning, Operant; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hypothalamus, Middle; Injections, Intraventricular; Limbic System; Male; Microinjections; Molecular Sequence Data; Motivation; Narcotics; Nucleus Accumbens; Peptide Fragments; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substantia Nigra | 1993 |