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1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) and enkephalin, ala(2)-mephe(4)-gly(5)-

1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 3 studies

Compound Research Comparison

Studies
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Trials
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Recent Studies (post-2010)
(1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8))
Studies
(enkephalin, ala(2)-mephe(4)-gly(5)-)
Trials
(enkephalin, ala(2)-mephe(4)-gly(5)-)
Recent Studies (post-2010) (enkephalin, ala(2)-mephe(4)-gly(5)-)
3520151071
35202,7271374

Protein Interaction Comparison

ProteinTaxonomy1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) (IC50)enkephalin, ala(2)-mephe(4)-gly(5)- (IC50)
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.003
Delta-type opioid receptorMus musculus (house mouse)1.2415
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0132
Mu-type opioid receptorHomo sapiens (human)0.004
Delta-type opioid receptorHomo sapiens (human)0.0014
Mu-type opioid receptorMus musculus (house mouse)0.0048
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0283

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akil, H; Goldstein, A; Mansour, A; Meng, F; Thompson, RC; Watson, SJ; Xie, GX1
Herz, A; Shippenberg, TS; Spanagel, R1
Ableitner, A; Bals-Kubik, R; Herz, A; Shippenberg, TS1

Other Studies

3 other study(ies) available for 1-n-me-tyr(1)-7-n-me-arg-8-n-et-leunh2-dynorphin (1-8) and enkephalin, ala(2)-mephe(4)-gly(5)-

ArticleYear
Cloning and pharmacological characterization of a rat kappa opioid receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Nov-01, Volume: 90, Issue:21

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Analgesics; Animals; Benzeneacetamides; Cell Line; Cell Membrane; Cloning, Molecular; Corpus Striatum; Cyclic AMP; DNA Primers; DNA, Complementary; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Gene Library; In Situ Hybridization; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Molecular Sequence Data; Pyrrolidines; Rats; Receptors, Opioid, kappa; Restriction Mapping; RNA, Messenger; Transfection

1993
The effects of opioid peptides on dopamine release in the nucleus accumbens: an in vivo microdialysis study.
    Journal of neurochemistry, 1990, Volume: 55, Issue:5

    Topics: Analgesics; Animals; Dialysis; Dopamine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Magnesium; Male; Nucleus Accumbens; Peptide Fragments; Potassium; Rats; Rats, Inbred Strains; Tetrodotoxin

1990
Neuroanatomical sites mediating the motivational effects of opioids as mapped by the conditioned place preference paradigm in rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:1

    Topics: Amino Acid Sequence; Animals; Association Learning; Autoradiography; Brain Mapping; Conditioning, Operant; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hypothalamus, Middle; Injections, Intraventricular; Limbic System; Male; Microinjections; Molecular Sequence Data; Motivation; Narcotics; Nucleus Accumbens; Peptide Fragments; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substantia Nigra

1993