Page last updated: 2024-09-02

1-hexadecyl-2-acetyl-glycero-3-phosphocholine and sdz 64-412

1-hexadecyl-2-acetyl-glycero-3-phosphocholine has been researched along with sdz 64-412 in 6 studies

Compound Research Comparison

Studies
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Trials
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Recent Studies (post-2010)
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Studies
(sdz 64-412)
Trials
(sdz 64-412)
Recent Studies (post-2010) (sdz 64-412)
9,156187552600

Protein Interaction Comparison

ProteinTaxonomy1-hexadecyl-2-acetyl-glycero-3-phosphocholine (IC50)sdz 64-412 (IC50)
Platelet-activating factor receptorHomo sapiens (human)0.06

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19901 (16.67)18.7374
1990's5 (83.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Handley, DA; Havill, AM; Van Valen, RG1
Beattie, LL; Ishida, K; Schellenberg, RR; Thomson, RJ; Wiggs, B1
Handley, DA; Houlihan, WJ; Melden, MK; Saunders, RN; Van Valen, RG1
Athill, LV; Charnick, SB; Karara, AH; Lau, DT; Tse, FL; Yu, Z1
Cheon, SH; Handley, DA; Houlihan, WJ; Larson, DA; Parrino, VA1
Fleming, TP; Stoddart, NR; Wild, AE1

Other Studies

6 other study(ies) available for 1-hexadecyl-2-acetyl-glycero-3-phosphocholine and sdz 64-412

ArticleYear
Prevention of non-specific airway hyperreactivity after allergen challenge in guinea-pigs by the PAF receptor antagonist SDZ 64-412.
    British journal of pharmacology, 1990, Volume: 99, Issue:2

    Topics: Allergens; Animals; Azepines; Bronchi; Bronchoalveolar Lavage Fluid; Eosinophils; Guinea Pigs; Histamine; Hypersensitivity; In Vitro Techniques; Isoquinolines; Male; Methylprednisolone; Platelet Activating Factor; Triazines; Triazoles; Vagotomy; Vagus Nerve

1990
Inhibition of antigen-induced airway hyperresponsiveness, but not acute hypoxia nor airway eosinophilia, by an antagonist of platelet-activating factor.
    Journal of immunology (Baltimore, Md. : 1950), 1990, May-15, Volume: 144, Issue:10

    Topics: Acetylcholine; Airway Resistance; Animals; Bronchial Provocation Tests; Bronchial Spasm; Connective Tissue Cells; Eosinophils; Epithelial Cells; Guinea Pigs; Hypersensitivity; Isoquinolines; Ovalbumin; Platelet Activating Factor; Platelet Aggregation; Respiratory System

1990
Biological effects of the orally active platelet activating factor receptor antagonist SDZ 64-412.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2

    Topics: Adenosine Diphosphate; Animals; Blood Pressure; Bronchi; Cebus; Collagen; Dogs; Dose-Response Relationship, Drug; Epinephrine; Guinea Pigs; Isoquinolines; Mice; Platelet Activating Factor; Platelet Aggregation; Rats

1988
Pharmacokinetics of SDZ 64-412, a novel antiasthmatic agent, following intravenous, oral, and inhalation dosing in the rat.
    Biopharmaceutics & drug disposition, 1994, Volume: 15, Issue:4

    Topics: Administration, Inhalation; Administration, Oral; Animals; Atmosphere Exposure Chambers; Biological Availability; Dose-Response Relationship, Drug; Half-Life; Injections, Intravenous; Intestinal Absorption; Isoquinolines; Metabolic Clearance Rate; Platelet Activating Factor; Rats; Rats, Sprague-Dawley; Tissue Distribution

1994
Structural modification of 5-aryl-2,3-dihydroimidazo[2,1-a]isoquinoline platelet activating factor receptor antagonists.
    Journal of medicinal chemistry, 1993, Oct-15, Volume: 36, Issue:21

    Topics: Animals; Binding, Competitive; Bronchoconstriction; Guinea Pigs; Humans; Isoquinolines; Platelet Activating Factor; Platelet Membrane Glycoproteins; Pyridines; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Structure-Activity Relationship; Thienopyridines; Thiophenes

1993
Stimulation of development in vitro by platelet-activating factor receptor ligands released by mouse preimplantation embryos.
    Journal of reproduction and fertility, 1996, Volume: 108, Issue:1

    Topics: Animals; Blastocyst; Cell Culture Techniques; Embryonic and Fetal Development; Isoquinolines; Mice; Mice, Inbred Strains; Phospholipid Ethers; Platelet Activating Factor; Stimulation, Chemical

1996