Page last updated: 2024-09-02

1-hexadecyl-2-acetyl-glycero-3-phosphocholine and bisindolylmaleimide i

1-hexadecyl-2-acetyl-glycero-3-phosphocholine has been researched along with bisindolylmaleimide i in 5 studies

Compound Research Comparison

Studies
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Trials
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Recent Studies (post-2010)
(1-hexadecyl-2-acetyl-glycero-3-phosphocholine)
Studies
(bisindolylmaleimide i)
Trials
(bisindolylmaleimide i)
Recent Studies (post-2010) (bisindolylmaleimide i)
9,1561875521,1981174

Protein Interaction Comparison

ProteinTaxonomy1-hexadecyl-2-acetyl-glycero-3-phosphocholine (IC50)bisindolylmaleimide i (IC50)
Chain A, Protein kinase C, iotaHomo sapiens (human)5.8
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)9
G2/mitotic-specific cyclin-B2Homo sapiens (human)2.3
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.5
Protein kinase C gamma typeHomo sapiens (human)0.03
Protein kinase C beta typeHomo sapiens (human)0.0054
Cyclin-dependent kinase 1Homo sapiens (human)2.3
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.068
Cyclin-dependent kinase 4Homo sapiens (human)0.99
G2/mitotic-specific cyclin-B1Homo sapiens (human)2.3
Lethal factorBacillus anthracis1.5
Protein kinase C alpha typeHomo sapiens (human)0.0055
Glycogen synthase kinase-3 betaRattus norvegicus (Norway rat)0.36
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoformOryctolagus cuniculus (rabbit)0.7
G1/S-specific cyclin-D1Homo sapiens (human)0.99
Protein kinase C eta typeHomo sapiens (human)0.0066
G1/S-specific cyclin-E1Homo sapiens (human)0.99
Cyclin-dependent kinase 2Homo sapiens (human)0.99
cAMP-dependent protein kinase catalytic subunit alpha Rattus norvegicus (Norway rat)2
Protein kinase C iota typeHomo sapiens (human)3.463
Glycogen synthase kinase-3 betaHomo sapiens (human)0.19
Protein kinase C epsilon typeHomo sapiens (human)0.0067
Protein kinase C theta typeHomo sapiens (human)0.0061
Protein kinase C zeta typeHomo sapiens (human)5.8
Protein kinase C delta typeHomo sapiens (human)0.0096
Peroxisome proliferator-activated receptor alphaHomo sapiens (human)0.006
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)7.3
G2/mitotic-specific cyclin-B3Homo sapiens (human)2.3
Serine/threonine-protein kinase LMTK3Homo sapiens (human)0.0001

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Izumi, T; Kato, M; Kimura, H; Morikawa, A; Obinata, H; Suzuki, M; Tachibana, A; Takizawa, T; Tokuyama, K1
Bazan, NG; Bernatchez, PN; GĂ©linas, DS; Rollin, S; Sirois, MG1
Biffl, WL; Carnaggio, R; Gonzalez, RJ; Moore, EE; Offner, PJ; Silliman, CC; West, KE1
Chen, LW; Hsu, CM; Lin, MW1
Ajiro, Y; Giles, WR; Saegusa, N; Spitzer, KW; Stafforini, DM1

Other Studies

5 other study(ies) available for 1-hexadecyl-2-acetyl-glycero-3-phosphocholine and bisindolylmaleimide i

ArticleYear
Inhibition of protein kinases A and C demonstrates dual modes of response in human eosinophils stimulated with platelet-activating factor.
    The Journal of allergy and clinical immunology, 2002, Volume: 110, Issue:2

    Topics: Benzoquinones; Cell Adhesion; Cell Degranulation; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Eosinophils; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Indoles; Isoquinolines; Lactams, Macrocyclic; Macrophage-1 Antigen; Maleimides; Platelet Activating Factor; Protein Kinase C; Protein-Tyrosine Kinases; Quinones; Rifabutin; Signal Transduction; Sulfonamides; Superoxides; Up-Regulation; Virulence Factors, Bordetella

2002
Immediate and delayed VEGF-mediated NO synthesis in endothelial cells: role of PI3K, PKC and PLC pathways.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: 1-Methyl-3-isobutylxanthine; Androstadienes; Animals; Calcimycin; Calcium; Cattle; Cells, Cultured; Chelating Agents; Chromones; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Egtazic Acid; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Ginkgolides; Indoles; Intercellular Signaling Peptides and Proteins; Ionophores; Lactones; Lymphokines; Maleimides; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroprusside; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Serine; Signal Transduction; Time Factors; Type C Phospholipases; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin

2002
Neutrophil apoptosis is delayed by trauma patients' plasma via a mechanism involving proinflammatory phospholipids and protein kinase C.
    Surgical infections, 2001,Winter, Volume: 2, Issue:4

    Topics: Adolescent; Adult; Aged; Apoptosis; Azepines; Enzyme Inhibitors; Humans; In Vitro Techniques; Indoles; Injury Severity Score; Maleimides; Middle Aged; Neutrophils; Phospholipids; Plasma; Platelet Activating Factor; Platelet Aggregation Inhibitors; Protein Kinase C; Signal Transduction; Time Factors; Triazoles; Wounds and Injuries

2001
Different pathways leading to activation of extracellular signal-regulated kinase and p38 MAP kinase by formyl-methionyl-leucyl-phenylalanine or platelet activating factor in human neutrophils.
    Journal of biomedical science, 2005, Volume: 12, Issue:2

    Topics: Androstadienes; Aristolochic Acids; Calcium; Calcium Channel Blockers; Calcium Channels; Chromones; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Extracellular Signal-Regulated MAP Kinases; Humans; Imidazoles; Indoles; Maleimides; Models, Biological; Morpholines; N-Formylmethionine Leucyl-Phenylalanine; Naphthalenes; Neutrophils; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Phosphorylation; Platelet Activating Factor; Protein Isoforms; Protein Kinase C; Pyrrolidinones; Type C Phospholipases; Wortmannin

2005
Platelet-activating factor stimulates sodium-hydrogen exchange in ventricular myocytes.
    American journal of physiology. Heart and circulatory physiology, 2011, Volume: 301, Issue:6

    Topics: Acidosis; Alkalosis; Animals; Azepines; Benzophenanthridines; Dose-Response Relationship, Drug; Flavonoids; Guanidines; Guinea Pigs; Heart Ventricles; Hydrogen-Ion Concentration; Indoles; Ion Transport; Maleimides; Mitogen-Activated Protein Kinase Kinases; Myocytes, Cardiac; Phospholipid Ethers; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Kinase Inhibitors; Receptors, G-Protein-Coupled; Signal Transduction; Sodium; Sodium-Hydrogen Exchangers; Spectrometry, Fluorescence; Sulfones; Time Factors; Triazoles

2011