Page last updated: 2024-08-16

1-NA-PP1 and 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine

1-NA-PP1 has been researched along with 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cravatt, BF; Saghatelian, A1
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Bhandari, JG; Castellanos-Gonzalez, A; Keyloun, KR; Kim, JE; Larson, ET; Maly, DJ; Merritt, EA; Muller, NR; Murphy, RC; Ojo, KK; Perera, BG; Van Voorhis, WC; Verlinde, CL; White, AC1
Barks, J; Lopez, MS; Lourido, S; Shokat, KM; Sibley, LD; Tang, K; Wang, Q; Wildman, SA; Zhang, C1
Capretta, A; Egorova, O; Evdokimova, E; Savchenko, A; Shakya, T; Spanogiannopoulos, P; Stogios, PJ; Todorovic, N; Wright, GD1

Reviews

1 review(s) available for 1-NA-PP1 and 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine

ArticleYear
Assignment of protein function in the postgenomic era.
    Nature chemical biology, 2005, Volume: 1, Issue:3

    Topics: Amino Acid Sequence; Bacteria; Models, Biological; Molecular Structure; Protein Processing, Post-Translational; Proteins; Proteomics; Sequence Alignment

2005

Other Studies

4 other study(ies) available for 1-NA-PP1 and 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Discovery of Potent and Selective Inhibitors of Calcium-Dependent Protein Kinase 1 (CDPK1) from C. parvum and T. gondii.
    ACS medicinal chemistry letters, 2010, Oct-14, Volume: 1, Issue:7

    Topics:

2010
Optimizing small molecule inhibitors of calcium-dependent protein kinase 1 to prevent infection by Toxoplasma gondii.
    Journal of medicinal chemistry, 2013, Apr-11, Volume: 56, Issue:7

    Topics: Animals; Base Sequence; Disease Models, Animal; DNA Primers; Enzyme-Linked Immunosorbent Assay; Mice; Protein Kinase Inhibitors; Protein Kinases; Small Molecule Libraries; Toxoplasma; Toxoplasmosis

2013
Structure-guided optimization of protein kinase inhibitors reverses aminoglycoside antibiotic resistance.
    The Biochemical journal, 2013, Sep-01, Volume: 454, Issue:2

    Topics: Acinetobacter baumannii; Aminoglycosides; Anthracenes; Anti-Bacterial Agents; Bacterial Proteins; Binding Sites; Drug Design; Drug Resistance, Bacterial; Escherichia coli; Isoenzymes; Kanamycin; Kanamycin Kinase; Microbial Sensitivity Tests; Molecular Conformation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Quinazolines; Recombinant Proteins; Structure-Activity Relationship

2013