Page last updated: 2024-08-18

1,3-ditolylguanidine and eliprodil

1,3-ditolylguanidine has been researched along with eliprodil in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's6 (75.00)24.3611
2020's2 (25.00)2.80

Authors

AuthorsStudies
Frehland, B; Schepmann, D; Schmidtke, KU; Tewes, B; Winckler, T; Wünsch, B1
Bonifazi, A; Gawaskar, S; Schepmann, D; Wünsch, B1
Bonifazi, A; Gawaskar, S; Robaa, D; Schepmann, D; Sippl, W; Wünsch, B1
Lütnant, I; Schepmann, D; Wünsch, B1
Dey, S; Frehland, B; Lehmkuhl, K; Schepmann, D; Schreiber, JA; Seebohm, G; Strutz-Seebohm, N; Temme, L; Wünsch, B1
Kitamura, M; Schepmann, D; Shuto, Y; Temme, L; Thum, S; Wünsch, B1
Baumeister, S; Schepmann, D; Wünsch, B1
Bechthold, E; Daniliuc, C; Ritter, N; Schepmann, D; Schreiber, JA; Seebohm, G; Wünsch, B1

Other Studies

8 other study(ies) available for 1,3-ditolylguanidine and eliprodil

ArticleYear
Conformationally constrained NR2B selective NMDA receptor antagonists derived from ifenprodil: Synthesis and biological evaluation of tetrahydro-3-benzazepine-1,7-diols.
    Bioorganic & medicinal chemistry, 2010, Nov-15, Volume: 18, Issue:22

    Topics: Analgesics; Animals; Benzazepines; Humans; Mice; Microsomes, Liver; Neuralgia; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2010
Synthesis, GluN2B affinity and selectivity of benzo[7]annulen-7-amines.
    Bioorganic & medicinal chemistry, 2014, Dec-01, Volume: 22, Issue:23

    Topics: Benzocycloheptenes; Dose-Response Relationship, Drug; Humans; Molecular Structure; Piperazines; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2014
Benzo[7]annulene-based GluN2B selective NMDA receptor antagonists: Surprising effect of a nitro group in 2-position.
    Bioorganic & medicinal chemistry letters, 2015, Dec-15, Volume: 25, Issue:24

    Topics: Amines; Binding Sites; Molecular Docking Simulation; Phenols; Piperidines; Protein Binding; Protein Structure, Tertiary; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2015
Benzimidazolone bioisosteres of potent GluN2B selective NMDA receptor antagonists.
    European journal of medicinal chemistry, 2016, Jun-30, Volume: 116

    Topics: Benzimidazoles; Drug Design; Humans; Receptors, N-Methyl-D-Aspartate

2016
Deconstruction - reconstruction approach to analyze the essential structural elements of tetrahydro-3-benzazepine-based antagonists of GluN2B subunit containing NMDA receptors.
    European journal of medicinal chemistry, 2017, Sep-29, Volume: 138

    Topics: Benzazepines; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Structure; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2017
Do GluN2B subunit containing NMDA receptors tolerate a fluorine atom in the phenylalkyl side chain?
    MedChemComm, 2017, May-01, Volume: 8, Issue:5

    Topics:

2017
Thiophene bioisosteres of GluN2B selective NMDA receptor antagonists: Synthesis and pharmacological evaluation of [7]annuleno[b]thiophen-6-amines.
    Bioorganic & medicinal chemistry, 2020, 01-15, Volume: 28, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Molecular Structure; Rats; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Thiophenes

2020
Synthesis and biological evaluation of conformationally restricted GluN2B ligands derived from eliprodil.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Ligands; Piperidines; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Tropanes

2022