Page last updated: 2024-08-18

1,3-ditolylguanidine and e-52862

1,3-ditolylguanidine has been researched along with e-52862 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Chen, Y; Lan, Y; Liu, BF; Liu, S; Liu, X; Qiu, Y; Xu, X; Zhang, G1
Gao, ZB; Gunosewoyo, H; Liu, T; Pang, T; Shi, JJ; Shi, M; Sun, H; Tang, J; Xu, YZ; Yang, F; Yu, LF; Zhang, W; Zheng, YM1
Iyamu, ID; Lv, W; Malik, N; Mishra, RK; Schiltz, GE1
Almansa, C; Álvarez, I; Caamaño, AM; Cendán, CM; de la Puente, B; Díaz, JL; Enjo, J; García, M; Lorente, A; Maldonado, R; Martín, M; Montero, A; Port, A; Sicre, C; Torrens, A; Vela, JM; Vidal-Torres, A; Yeste, S1

Other Studies

4 other study(ies) available for 1,3-ditolylguanidine and e-52862

ArticleYear
Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesic.
    European journal of medicinal chemistry, 2014, May-22, Volume: 79

    Topics: Analgesics; Animals; Brain; Dose-Response Relationship, Drug; Formaldehyde; Guinea Pigs; Hydroquinones; Mice; Mice, Inbred Strains; Molecular Structure; Nociceptive Pain; Pain Measurement; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship

2014
Development of Novel Alkoxyisoxazoles as Sigma-1 Receptor Antagonists with Antinociceptive Efficacy.
    Journal of medicinal chemistry, 2016, 07-14, Volume: 59, Issue:13

    Topics: Analgesics; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Formaldehyde; Injections, Intraperitoneal; Isoxazoles; Ligands; Mice; Mice, Inbred Strains; Molecular Structure; Pain; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship

2016
Discovery of a novel class of potent and selective tetrahydroindazole-based sigma-1 receptor ligands.
    Bioorganic & medicinal chemistry, 2019, 05-01, Volume: 27, Issue:9

    Topics: Animals; Binding Sites; Indazoles; Ligands; Mice; Microsomes, Liver; Molecular Docking Simulation; Protein Structure, Tertiary; Receptors, sigma; Sigma-1 Receptor; Solubility; Structure-Activity Relationship

2019
EST64454: a Highly Soluble σ
    Journal of medicinal chemistry, 2020, 12-10, Volume: 63, Issue:23

    Topics: Analgesics; Animals; Caco-2 Cells; Humans; Mice; Molecular Structure; Pain; Piperazines; Pyrazoles; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship

2020