1,3-dipropyl-8-cyclopentylxanthine and n(6)-cyclopentyladenosine

1,3-dipropyl-8-cyclopentylxanthine has been researched along with n(6)-cyclopentyladenosine in 152 studies

Research

Studies (152)

TimeframeStudies, this research(%)All Research%
pre-19901 (0.66)18.7374
1990's68 (44.74)18.2507
2000's68 (44.74)29.6817
2010's15 (9.87)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ijzerman, AP; Soudijn, W; van der Wenden, EM1
Ishii, A; Nonaka, H; Shimada, J; Suzuki, F1
Jacobson, KA; van Galen, PJ; Williams, M1
Jacobson, MA; Johnson, RG; Linden, J; Salvatore, CA; Taylor, HE1
Fredholm, BB; Hegler, J; Hessling, J; Klotz, KN; Kull, B; Lohse, MJ; Owman, C1
Barbhaiya, H; IJzerman, AP; Rivkees, SA1
Hess, S; Hölzl, J; Khudeir, N; Müller, CE; Scholle, S; Schumacher, B1
de Ligt, RA; IJzerman, AP; Leurs, R; Lorenzen, A; Rivkees, SA1
Beukers, MW; Brussee, J; Chang, LC; Ijzerman, AP; Mulder-Krieger, T; Roerink, SF; Spanjersberg, RF; van den Hout, G; von Frijtag Drabbe Künzel, JK1
Brussee, J; Chang, LC; Ijzerman, AP; Mulder-Krieger, T; Spangenberg, T; von Frijtag Drabbe Künzel, JK; Westerhout, J1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Beukers, MW; Brussee, J; Chang, LC; IJzerman, AP; Mulder-Krieger, T; Struensee-Link, R; van Veldhoven, JP; von Frijtag Drabbe Künzel, JK1
Beukers, MW; Brussee, J; de Graaf, O; de Vries, H; Göblyös, A; Ijzerman, AP; Link, R; Mantri, M; Mulder-Krieger, T; van Veldhoven, J; von Frijtag Drabbe Künzel, JK1
Cappellacci, L; Franchetti, P; Grifantini, M; Kachler, S; Klotz, KN; Lavecchia, A; Luongo, L; Maione, S; Marabese, I; Petrelli, R; Vita, P1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
El-Tayeb, A; Inamdar, GS; Li, W; Müller, CE; Scheiff, AB; Sudarsanam, V; Vasu, KK; Yerande, SG1
Federico, S; Jacobson, KA; Jayasekara, PS; Kozma, E; Moro, S; Paoletta, S; Spalluto, G; Squarcialupi, L1
Terre'Blanche, G; Van der Walt, MM1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Cox, BF; Lappe, RW; Merkel, LA; Perrone, MH; Rivera, LM1
Brink, A; Fuder, H; Meincke, M; Tauber, U1
Földes, FF; Nagano, O; Nakatsuka, H; Ohta, Y; Reich, D; Sperlagh, B; Vizi, ES1
O'Regan, MH; Perkins, LM; Phillis, JW; Simpson, RE1
Herzer, WA; Jackson, EK; Kuan, CJ1
IJzerman, AP; Jacobson, KA; Van Galen, PJ1
Domenici, MR; Frank, C; Sagratella, S; Scotti de Carolis, A; Zeng, YC1
Czernilofsky, A; Dumont, JE; Ensinger, HA; Lefort, A; Libert, F; Mendla, KD; Van Sande, J; Vassart, G1
Hourani, SM; Kitchen, I; Nicholls, J1
Barraco, RA; Phillis, JW1
Barraco, RA; Normile, HJ1
Lothman, EW; Stringer, JL1
Badger, EW; Bristol, JA; Bruns, RF; Fergus, JH; Hartman, JD; Hays, SJ; Huang, CC; Santay, LA1
Starke, K; Stoffel, D; von Kügelgen, I1
Imaizumi, M; Miyazaki, S; Onodera, K1
Apaya, RP; IJzerman, AP; Price, SL; Soudijn, W; van der Wenden, EM1
Späth, L; Starke, K; von Kügelgen, I1
Martin, PL; Potts, AA1
Carter, M; Jacobson, KA; Ji, XD; Paul, IA; Von Lubitz, DK1
Alexander, SP; Hill, SJ; Iredale, PA1
Broad, RM; Cook, MA1
Carter, M; Jacobson, KA; Paul, IA; Von Lubitz, DK1
Joad, JP; Kott, KS1
Bruns, RF; Montamat, SC; Mudumbi, RV; Vestal, RE1
Halfhide, EJ; Hourani, SM; Kitchen, I; Lee, BS; Nicholls, J1
Hill, SJ; Peakman, MC1
Dickenson, JM; Hill, SJ; Megson, AC; Townsend-Nicholson, A1
Broad, RM; Fredholm, BB1
Brownhill, VR; Hourani, SM; Kitchen, I3
Berger, M; Christoffel, F; Gebicke-Haerter, PJ; Northoff, H; Timmer, J; Van Calker, D1
Gonçalves, J; Queiroz, G1
Jackson, EK; Kusaka, H; Pfeifer, CA; Tofovic, SP1
Andrés, A; Fernández, M; Ros, M; Sanz, JM; Vendite, D1
Hettinger-Smith, BD; Leid, M; Murray, TF1
Brownhill, VR; Hourani, SM; Kitchen, I; Peachey, JA1
Abe, T; Gutterman, DD; Morgan, DA1
Guimarães, S; Moura, D; Vaz-da-Silva, MJ1
Gupta, YK; Malhotra, J2
Cooke, MJ; Fisher, A; Fraser, CM; Stone, TW; Thompson, ID2
Berger, M; Biber, K; Gebicke-Härter, PJ; Klotz, KN; van Calker, D1
Koch, H; Starke, K; von Kügelgen, I1
Coffey, D; Cronstein, BN; Fisher, R; Lahita, RG; Merrill, JT; Salmon, J; Schreibman, D; Shen, C; Zakharenko, O1
Chopde, CT; Ghosh, AK; Mandhane, SN1
Antal, K; Cseppentö, A; Kovács, P; Szabó, JZ; Szentmiklósi, AJ; Ujfalusi, A1
Buxton, IL; Cheek, DJ; Smith, AD; Westfall, DP1
Hourani, SM; Nicholls, J1
Fulga, I; Stone, TW1
Amanatullah, DF; Clair, T; Liotta, LA; Schetz, JA; Stracke, ML; Woodhouse, EC1
Hettinger, BD; Leid, M; Murray, TF1
Bockaert, J; Manzoni, O; Pujalte, D; Williams, J1
Han, DH; Hansen, PA; Holloszy, JO; Nolte, LA1
Beukers, MW; Dalpiaz, A; IJzerman, AP; Schofield, PR; Townsend-Nicholson, A1
Chessell, IP; Dowd, E; Humphrey, PP; McQueen, DS1
Hourani, SM; Kitchen, I; Peachey, JA1
Coupar, IM1
Cattarini, G; Florio, T; Maragliano, A; Schettini, G; Thellung, S1
IJzerman, AP; Kourounakis, AP; van der Klein, PA1
Davis, JM; Gute, DC; Jones, S; Korthuis, RJ; Krsmanovic, A1
Cunha, RA; Lopes, LV; Ribeiro, JA1
Costentin, J; El Yacoubi, M; Ledent, C; Parmentier, M; Vaugeois, JM1
Agostinho, P; Caseiro, P; Cunha, RA; Duarte, EP; Oliveira, CR; Rego, AC1
Fain, JN; Rice, AM; Rivkees, SA1
Jacks, SM; Kapicka, CL; Montamat, SC; Mudumbi, RV; Olson, RD; Vestal, RE1
Materi, LM; Rasmusson, DD; Semba, K1
Dickenson, JM; Germack, R1
Brand, A; Eschke, D; Nieber, K; Vissiennon, Z1
Koos, BJ; Maeda, T1
Barrière, H; Bidet, M; Cuiller, B; Poujeol, C; Poujeol, P; Rubera, I; Tauc, M; Verheecke-Mauze, C1
Cunha, RA; de Mendonça, A; Ribeiro, JA; Sebastião, AM1
Allgaier, C; Brand, A; Eger, K; Eschke, D; Hess, S; Nieber, K; Scheibler, P1
Dickenson, JM; Robinson, AJ1
Hancox, JC; Hinde, AK; Zhang, YH1
Matsumoto, K; Murakami, Y; Tabata, K; Watanabe, H1
Blauth, E; Cassel, JC; Feuerstein, TJ; Jackisch, R; Kelche, C; Sehmisch, S; Thorn, D1
Nakata, H; Saitoh, O; Yoshioka, K1
Jan, C; Koos, BJ; Maeda, T1
Coupar, IM; Tran, BL1
Brooke, RE; Deuchars, J; Deuchars, SA1
Biondi, C; Dalpiaz, A; Forni, F; Pavan, B; Scatturin, A; Vandelli, MA1
Dar, MS1
Hamann, M; Richter, A1
Cheng, JT; Chi, TC; Liu, IM1
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R1
Allen, CN; Honda, K; Ikeda, M; Inoué, S; Sagara, M; Sekino, Y; Shirao, T; Yoshioka, T1
Dai, LJ; Kang, HS; Kerstan, D; Quamme, GA; Ritchie, G1
Furue, H; Kumamoto, E; Lao, LJ; Luo, C; Yoshimura, M1
Battastini, AM; Bonan, CD; Choi, H; Izquierdo, I; Mello e Souza, T; Pereira, GS; Rodrigues, C; Sarkis, JJ; Vinadé, ER1
Allescher, HD; Dunkel, R; Schusdziarra, V; Storr, M; Thammer, J1
Antoniou, K; Ferré, S; Fuxe, K; Goldberg, SR; Justinova, Z; Karcz-Kubicha, M; Müller, CE; Pezzola, A; Popoli, P; Quarta, D; Reggio, R; Solinas, M; Terasmaa, A1
Burki, N; Gu, Q; Hong, JL; Lee, LY; Ruan, T1
Coelho, JE; Costenla, AR; Cunha, RA; de Mendonça, A; Lopes, LV; Oliveira, CR; Parada, A; Rebola, N; Soares-da-Silva, P1
Christie, MJ; Hack, SP; Vaughan, CW1
Battastini, AM; Bonan, CD; Crema, L; da Silva Torres, IL; Dalmaz, C; De Leon Nunes, M; Ferreira, MB; Sarkis, JJ1
Goulart, EC; Kaster, MP; Rodrigues, AL; Rosa, AO; Rosso, MM; Santos, AR1
Nowak, TS; Sorimachi, T1
Avsar, E; Empson, RM1
Fujita, T; Kawasaki, Y; Kumamoto, E; Liu, T1
de Ligt, RA; IJzerman, AP; Klaasse, E; Leurs, R; Lorenzen, A; Milligan, G; Roerink, SF1
Goto, W; Hirao, M; Ikeda, T; Kobayashi, T; Oku, H; Sugiyama, T1
Cao, Y; Jin, L; Meng, F; Sun, WC; Wang, LZ; Zhu, XZ1
Higa, K; Higuchi, H; Iihoshi, M; Nitahara, K; Shono, S; Vizi, ES1
Bonan, CD; Cammarota, M; Izquierdo, I; Pereira, GS; Rossato, JI; Sarkis, JJ1
Kogi, K; Konno, T; Nagai, A; Nakahata, N; Uchibori, T1
Beukers, MW; de Grip, WJ; Ijzerman, AP; Klaasse, EC; Roerink, SF; van den Hout, G1
Cao, C; Han, JH; Kim, SH; Kim, SZ; Yuan, K1
Dalpiaz, A; Heitman, LH; IJzerman, AP; Mulder-Krieger, T; Spanjersberg, RF; von Frijtag Drabbe Künzel, JK1
Cao, Y; Jin, L; Sun, WC; Xie, KQ; Zhu, XZ1
Cao, Y; Xie, KQ; Zhu, XZ1
Kubota, Y; Kunitomo, M; Mizuno, H; Morikawa, T; Nakamura, K; Shinozuka, K; Tanaka, N1
Bonen, A; Dyck, DJ; Graham, TE; Greer, F; Lally, JS; Thong, FS1
Fewell, JE; Gillis, AM; Zhang, C1
Cunha-Reis, D; Ribeiro, JA; Sebastião, AM1
Inoue, K; Miyazaki, N; Nakatsuka, T; Nohda, K; Takeda, D; Yoshida, M1
Kelty, JD; Shields, EJ; Vandam, RJ1
Almeida, RS; Carrettiero, DC; Fior-Chadi, DR1
Kaczynska, K; Szereda-Przestaszewska, M1
Church, JE; Coupar, IM; Pouton, CW; Rose'Meyer, RB; Urmaliya, VB; White, PJ1
Bertram, EH; Hargus, NJ; Patel, MK1
Inscho, EW; Osmond, DA1
Cui, Y; Gong, QJ; Li, YY; Liu, CC; Liu, XG; Liu, Y; Wang, J; Wei, XH; Xin, WJ1
Ledent, C; Pouton, CW; Short, JL; Urmaliya, VB; White, PJ1
Cechova, S; Elsobky, AM; Venton, BJ1
Albensi, BC; Parkinson, FE; Xiong, W; Zhang, D1
Atas, HC; Biber, K; Normann, C; Serchov, T; van Calker, D1
Golab, F; Katebi, M; Mehdizadeh, M; Mohamadzadeh, F; Soleimani, M; Zamani, M1
Cascalheira, JF; Sebastião, AM; Serpa, A1
Nascimento, F; Ribeiro, JA; Sebastião, AM1
Kumei, S; Miyagishi, S; Nozu, T; Ohhira, M; Okumura, T; Takakusaki, K1
Dastjerdi, MN; Mardani, M; Ra, MZ; Valiani, A1

Reviews

2 review(s) available for 1,3-dipropyl-8-cyclopentylxanthine and n(6)-cyclopentyladenosine

ArticleYear
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
    Journal of medicinal chemistry, 1992, Feb-07, Volume: 35, Issue:3

    Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship

1992
Fluorescent ligands for adenosine receptors.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Boron Compounds; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Humans; Ligands; Protein Binding; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1

2013

Other Studies

150 other study(ies) available for 1,3-dipropyl-8-cyclopentylxanthine and n(6)-cyclopentyladenosine

ArticleYear
A steric and electrostatic comparison of three models for the agonist/antagonist binding site on the adenosine A1 receptor.
    Journal of medicinal chemistry, 1992, Feb-21, Volume: 35, Issue:4

    Topics: Adenosine; Binding Sites; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Models, Molecular; Molecular Conformation; Molecular Structure; Purinergic Antagonists; Receptors, Purinergic; Regression Analysis; Structure-Activity Relationship; Xanthine; Xanthines

1992
8-Polycycloalkyl-1,3-dipropylxanthines as potent and selective antagonists for A1-adenosine receptors.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cell Membrane; Corpus Striatum; Guinea Pigs; Humans; Molecular Conformation; Molecular Structure; Prosencephalon; Purinergic Antagonists; Rats; Receptors, Purinergic; Stereoisomerism; Structure-Activity Relationship; Xanthines

1992
Molecular cloning and characterization of the human A3 adenosine receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Nov-01, Volume: 90, Issue:21

    Topics: Adenosine; Amino Acid Sequence; Animals; Binding, Competitive; CHO Cells; Cloning, Molecular; Consensus Sequence; Corpus Striatum; Cricetinae; DNA Primers; Gene Expression; Humans; Iodobenzenes; Kinetics; Liver; Lung; Molecular Sequence Data; Polymerase Chain Reaction; Rats; Receptors, Purinergic P1; Sequence Homology, Amino Acid; Sheep; Transfection

1993
Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Base Composition; Binding, Competitive; CHO Cells; Cricetinae; Guanylate Cyclase; Humans; Phenethylamines; Phenylisopropyladenosine; Receptors, Purinergic P1; Stereoisomerism; Structure-Activity Relationship; Transfection; Xanthines

1998
Identification of the adenine binding site of the human A1 adenosine receptor.
    The Journal of biological chemistry, 1999, Feb-05, Volume: 274, Issue:6

    Topics: Adenine; Amides; Amino Acid Sequence; Amino Acids; Binding Sites; DNA, Complementary; Humans; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Receptors, Purinergic P1

1999
Lignans isolated from valerian: identification and characterization of a new olivil derivative with partial agonistic activity at A(1) adenosine receptors.
    Journal of natural products, 2002, Volume: 65, Issue:10

    Topics: Animals; CHO Cells; Cricetinae; Cyclic AMP; GABA-A Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Lignans; Plant Roots; Purinergic P1 Receptor Agonists; Rats; Serotonin Antagonists; Valerian

2002
A "locked-on," constitutively active mutant of the adenosine A1 receptor.
    European journal of pharmacology, 2005, Mar-07, Volume: 510, Issue:1-2

    Topics: Adenosine; Animals; Binding, Competitive; Cell Line; Cell Membrane; Chlorocebus aethiops; Colforsin; COS Cells; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Humans; Kinetics; Mutation; Plasmids; Radioligand Assay; Receptor, Adenosine A1; Sodium; Sulfur Radioisotopes; Theophylline; Thiophenes; Transfection; Tritium; Xanthines

2005
A series of ligands displaying a remarkable agonistic-antagonistic profile at the adenosine A1 receptor.
    Journal of medicinal chemistry, 2005, Mar-24, Volume: 48, Issue:6

    Topics: Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Aminopyridines; Animals; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dioxoles; Ligands; Models, Molecular; Radioligand Assay; Structure-Activity Relationship

2005
2,6,8-trisubstituted 1-deazapurines as adenosine receptor antagonists.
    Journal of medicinal chemistry, 2007, Feb-22, Volume: 50, Issue:4

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Antagonists; Animals; CHO Cells; Cricetinae; Cricetulus; Humans; Imidazoles; Pyridines; Radioligand Assay; Structure-Activity Relationship

2007
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
A new generation of adenosine receptor antagonists: from di- to trisubstituted aminopyrimidines.
    Bioorganic & medicinal chemistry, 2008, Mar-15, Volume: 16, Issue:6

    Topics: Amines; Cyclic AMP; Humans; Purinergic P1 Receptor Antagonists; Pyrimidines; Receptor, Adenosine A1; Receptor, Adenosine A2A; Structure-Activity Relationship

2008
2-Amino-6-furan-2-yl-4-substituted nicotinonitriles as A2A adenosine receptor antagonists.
    Journal of medicinal chemistry, 2008, Aug-14, Volume: 51, Issue:15

    Topics: Adenosine A2 Receptor Antagonists; Amines; Animals; Cell Line; Cricetinae; Cyclic AMP; Furans; Humans; Models, Molecular; Molecular Structure; Nicotinic Acids; Nitriles; Receptor, Adenosine A2A; Structure-Activity Relationship

2008
N6-Cycloalkyl- and N6-bicycloalkyl-C5'(C2')-modified adenosine derivatives as high-affinity and selective agonists at the human A1 adenosine receptor with antinociceptive effects in mice.
    Journal of medicinal chemistry, 2009, Apr-23, Volume: 52, Issue:8

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenylyl Cyclases; Analgesics; Animals; CHO Cells; Cricetinae; Cricetulus; Cyclopentanes; Humans; Mice; Models, Molecular; Norbornanes; Pain Measurement; Radioligand Assay; Stereoisomerism; Structure-Activity Relationship

2009
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Adenosine A1 Receptor Antagonists; Animals; Drug Design; Humans; Molecular Structure; Rats; Receptor, Adenosine A1; Stereoisomerism; Structure-Activity Relationship; Thiazoles

2010
1,3,7-Triethyl-substituted xanthines--possess nanomolar affinity for the adenosine A1 receptor.
    Bioorganic & medicinal chemistry, 2015, Oct-15, Volume: 23, Issue:20

    Topics: Adenosine A1 Receptor Antagonists; Dose-Response Relationship, Drug; Humans; Molecular Structure; Protein Binding; Receptor, Adenosine A1; Structure-Activity Relationship; Xanthines

2015
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Demonstration of vasorelaxant activity with an A1-selective adenosine agonist in porcine coronary artery: involvement of potassium channels.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Adenosine; Animals; Brain; Coronary Vessels; Cyclic GMP; In Vitro Techniques; Nitric Oxide; Potassium; Potassium Channels; Rats; Receptors, Purinergic; Swine; Vasodilator Agents; Xanthines

1992
Purinoceptor-mediated modulation by endogenous and exogenous agonists of stimulation-evoked [3H]noradrenaline release on rat iris.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: Adenosine; Animals; Electric Stimulation; In Vitro Techniques; Iris; Male; Norepinephrine; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Synaptic Transmission; Theophylline; Xanthines

1992
Presynaptic A1-purinoceptor-mediated inhibitory effects of adenosine and its stable analogues on the mouse hemidiaphragm preparation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:2

    Topics: 2-Chloroadenosine; Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Diaphragm; Dipyridamole; Electric Stimulation; In Vitro Techniques; Magnesium; Male; Mice; Muscle Contraction; Neuromuscular Junction; Phrenic Nerve; Purinergic Antagonists; Receptors, Purinergic; Synapses; Synaptic Transmission; Theophylline; Tritium; Tubocurarine; Xanthines

1992
Excitatory transmitter amino acid release from the ischemic rat cerebral cortex: effects of adenosine receptor agonists and antagonists.
    Journal of neurochemistry, 1992, Volume: 58, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aspartic Acid; Brain Ischemia; Cerebral Cortex; Glutamates; Glutamic Acid; Male; Neurotransmitter Agents; Purinergic Antagonists; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Triazoles; Xanthines

1992
An experimental paradigm for investigating the role of endogenous adenosine/A1 receptor interactions in vivo.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Adenosine; Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Male; Phenethylamines; Purinergic Antagonists; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic; Stereoisomerism; Xanthines

1992
Molecular modeling of adenosine receptors. I. The ligand binding site on the A1 receptor.
    Drug design and discovery, 1992, Volume: 9, Issue:1

    Topics: Adenosine; Amino Acid Sequence; Animals; Bacteriorhodopsins; Dogs; GTP-Binding Proteins; Histidine; Ligands; Models, Chemical; Models, Molecular; Molecular Sequence Data; Protein Binding; Receptors, Purinergic; Xanthines

1992
Effects of adenosinergic drugs on hypoxia-induced electrophysiological changes in rat hippocampal slices.
    Life sciences, 1992, Volume: 51, Issue:13

    Topics: Adenosine; Animals; Caffeine; Dizocilpine Maleate; Electrophysiology; Hippocampus; Hypoxia; In Vitro Techniques; Male; Membrane Potentials; Phenethylamines; Phenylisopropyladenosine; Potassium; Purinergic Antagonists; Rats; Rats, Inbred Strains; Synapses; Xanthines

1992
Cloning and functional characterization of a human A1 adenosine receptor.
    Biochemical and biophysical research communications, 1992, Sep-16, Volume: 187, Issue:2

    Topics: Adenosine; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; DNA; DNA Probes; Dogs; Hippocampus; Humans; Molecular Sequence Data; Nucleic Acid Hybridization; Receptors, Purinergic; Sequence Homology, Nucleic Acid; Transfection; Xanthines

1992
Characterization of P1-purinoceptors on rat duodenum and urinary bladder.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Duodenum; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Urinary Bladder; Vasodilator Agents; Xanthines

1992
Subtypes of adenosine receptors in the brainstem mediate opposite blood pressure responses.
    Neuropharmacology, 1991, Volume: 30, Issue:4

    Topics: Adenosine; Animals; Antihypertensive Agents; Blood Pressure; Brain Stem; Dose-Response Relationship, Drug; Male; Phenethylamines; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Triazoles; Xanthines

1991
N6-cyclopentyladenosine impairs passive avoidance retention by selective action at A1 receptors.
    Brain research bulletin, 1991, Volume: 27, Issue:1

    Topics: Adenosine; Animals; Avoidance Learning; Drug Interactions; Electroshock; Male; Memory; Mice; Receptors, Purinergic; Time Factors; Water Deprivation; Xanthines

1991
A1 adenosinergic modulation alters the duration of maximal dentate activation.
    Neuroscience letters, 1990, Oct-16, Volume: 118, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Animals; Electric Stimulation; Hippocampus; Limbic System; Male; Rats; Rats, Inbred Strains; Receptors, Purinergic; Seizures; Time Factors; Xanthines

1990
Binding of the A1-selective adenosine antagonist 8-cyclopentyl-1,3-dipropylxanthine to rat brain membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:1

    Topics: Adenosine; Animals; Brain; Cell Membrane; Female; Kinetics; Nucleosides; Rats; Xanthines

1987
P2-purinoceptor-mediated inhibition of noradrenaline release in rat atria.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antihypertensive Agents; Atropine; Desipramine; Dose-Response Relationship, Drug; Electric Stimulation; Heart Atria; Indomethacin; Male; Norepinephrine; Phenethylamines; Protein Synthesis Inhibitors; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Receptors, Purinergic P2; Suramin; Triazines; Xanthines; Yohimbine

1995
Effects of xanthine derivatives in a light/dark test in mice and the contribution of adenosine receptors.
    Methods and findings in experimental and clinical pharmacology, 1994, Volume: 16, Issue:9

    Topics: Adenosine; Animals; Antihypertensive Agents; Anxiety; Behavior, Animal; Caffeine; Darkness; Drug Interactions; Light; Male; Mice; Phenethylamines; Purinergic P1 Receptor Antagonists; Structure-Activity Relationship; Theophylline; Xanthines

1994
Relative binding orientations of adenosine A1 receptor ligands--a test case for Distributed Multipole Analysis in medicinal chemistry.
    Journal of computer-aided molecular design, 1995, Volume: 9, Issue:1

    Topics: Adenosine; Computer Graphics; Drug Design; Electrochemistry; Kinetics; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Xanthines

1995
Evidence for P2-purinoceptor-mediated inhibition of noradrenaline release in rat brain cortex.
    British journal of pharmacology, 1994, Volume: 113, Issue:3

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Cerebral Cortex; Male; Norepinephrine; Rats; Rats, Wistar; Receptors, Purinergic P1; Receptors, Purinergic P2; Tetrodotoxin; Xanthines; Yohimbine

1994
The endothelium of the rat renal artery plays an obligatory role in A2 adenosine receptor-mediated relaxation induced by 5'-N-ethylcarboxamidoadenosine and N6-cyclopentyladenosine.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arginine; Endothelium, Vascular; Glyburide; In Vitro Techniques; Indomethacin; Isoproterenol; Male; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Renal Artery; Renal Circulation; Theophylline; Vasodilator Agents; Xanthines

1994
Chronic adenosine A1 receptor agonist and antagonist: effect on receptor density and N-methyl-D-aspartate induced seizures in mice.
    European journal of pharmacology, 1994, Feb-21, Volume: 253, Issue:1-2

    Topics: Adenosine; Animals; Binding Sites; Injections, Subcutaneous; Male; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylaspartate; Receptors, Purinergic P1; Seizures; Xanthines

1994
Coupling of a transfected human brain A1 adenosine receptor in CHO-K1 cells to calcium mobilisation via a pertussis toxin-sensitive mechanism.
    British journal of pharmacology, 1994, Volume: 111, Issue:4

    Topics: Adenosine; Animals; Brain; Calcium; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Pertussis Toxin; Receptors, Purinergic P1; Transfection; Virulence Factors, Bordetella; Xanthines

1994
Inhibition of neurotransmitter release from enteric nerve endings by 2-[p-(carboxyethyl)-phenethylamino]-5'-N-ethylcarboxamido-adenosine (CGS-21680) and related adenosine analogs: lack of simple competition by antagonists.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Adenosine; Animals; Female; Guinea Pigs; In Vitro Techniques; Male; Myenteric Plexus; Neurotransmitter Agents; Phenethylamines; Purinergic Antagonists; Receptors, Purinergic; Xanthines

1993
Effects of N6-cyclopentyl adenosine and 8-cyclopentyl-1,3-dipropylxanthine on N-methyl-D-aspartate induced seizures in mice.
    European journal of pharmacology, 1993, Nov-16, Volume: 249, Issue:3

    Topics: Adenosine; Animals; Drug Interactions; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylaspartate; Seizures; Survival Rate; Temperature; Xanthines

1993
Effect of adenosine receptor ligands on cAMP content in human airways and peripheral lung.
    American journal of respiratory cell and molecular biology, 1993, Volume: 9, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adolescent; Adult; Aged; Child; Cromolyn Sodium; Cyclic AMP; Female; Humans; Ligands; Lung; Male; Middle Aged; Phenethylamines; Receptors, Purinergic; Respiratory System; Theophylline; Xanthines

1993
Cardiac functional responses to adenosine by PD 81,723, an allosteric enhancer of the adenosine A1 receptor.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 2

    Topics: Adenosine; Allosteric Regulation; Animals; Atrial Function; Depression, Chemical; Drug Synergism; Heart; Heart Atria; Heart Rate; Male; Myocardial Contraction; Rats; Rats, Sprague-Dawley; Receptors, Purinergic; Theophylline; Thiophenes; Xanthines

1993
Characterization and ontogeny of P1-purinoceptors on rat vas deferens.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Aging; Animals; Animals, Newborn; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle Development; Muscle, Smooth; Norepinephrine; Rats; Rats, Wistar; Receptors, Purinergic; Tetrodotoxin; Vas Deferens; Vasodilator Agents; Xanthines

1993
Adenosine A1 receptor-mediated changes in basal and histamine-stimulated levels of intracellular calcium in primary rat astrocytes.
    British journal of pharmacology, 1995, Volume: 115, Issue:5

    Topics: Adenosine; Animals; Animals, Newborn; Astrocytes; Calcium; Cells, Cultured; Histamine; Histamine Agonists; Image Processing, Computer-Assisted; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Purinergic P1; Xanthines

1995
Synergy between the inositol phosphate responses to transfected human adenosine A1-receptors and constitutive P2-purinoceptors in CHO-K1 cells.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Cattle; Cells, Cultured; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Humans; Inositol Phosphates; Pertussis Toxin; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Uridine Triphosphate; Virulence Factors, Bordetella; Xanthines

1995
A1, but not A2A, adenosine receptors modulate electrically stimulated [14C]acetylcholine release from rat cortex.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 277, Issue:1

    Topics: 2-Chloroadenosine; Acetylcholine; Adenosine; Animals; Cerebral Cortex; Electric Stimulation; In Vitro Techniques; Male; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Xanthines

1996
Selective enhancement by an adenosine A1 receptor agonist of agents inducing contraction of the rat vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adenosine; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Bradykinin; Carbachol; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Potassium Chloride; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Serotonin; Tyramine; Vas Deferens; Xanthines

1996
Differential distribution of adenosine A2 receptors in the epididymal and prostatic portions of the rat vas deferens.
    European journal of pharmacology, 1996, May-06, Volume: 303, Issue:1-2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dose-Response Relationship, Drug; Drug Interactions; Male; Rats; Rats, Wistar; Receptors, Purinergic P1; Vas Deferens; Xanthines

1996
Both adenosine A1- and A2-receptors are required to stimulate microglial proliferation.
    Neurochemistry international, 1996, Volume: 29, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Animals, Newborn; Cell Division; Cells, Cultured; Microglia; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Receptors, Purinergic P1; Thymidine; Xanthines

1996
Purinoceptor modulation of noradrenaline release in rat tail artery: tonic modulation mediated by inhibitory P2Y- and facilitatory A2A-purinoceptors.
    British journal of pharmacology, 1996, Volume: 117, Issue:1

    Topics: Adenosine; Adenosine Deaminase; Adenosine Triphosphate; Animals; Arteries; Male; Norepinephrine; Phenethylamines; Rats; Rats, Wistar; Receptors, Purinergic; Tail; Thioinosine; Thionucleotides; Xanthines

1996
Central effects of caffeine on renal renin secretion and norepinephrine spillover.
    Journal of cardiovascular pharmacology, 1996, Volume: 28, Issue:2

    Topics: Adenosine; Animals; Caffeine; Central Nervous System Stimulants; Hydralazine; Injections, Intraventricular; Kidney; Male; Norepinephrine; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Renin; Vasodilator Agents; Xanthines

1996
Adenosine A1 receptors in cultured cerebellar granule cells: role of endogenous adenosine.
    Journal of neurochemistry, 1996, Volume: 67, Issue:4

    Topics: Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Animals, Newborn; Cell Membrane; Cells, Cultured; Cerebellum; Colforsin; Cyclic AMP; GTP-Binding Proteins; Kinetics; Neurons; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Time Factors; Xanthines

1996
Chronic exposure to adenosine receptor agonists and antagonists reciprocally regulates the A1 adenosine receptor-adenylyl cyclase system in cerebellar granule cells.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: 2-Chloroadenosine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; Cerebellum; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Kinetics; Neurons; Phenylisopropyladenosine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Theophylline; Time Factors; Xanthines

1996
The ontogenetic profiles of the pre- and postjunctional adenosine receptors in the rat vas deferens.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Age Factors; Animals; Animals, Suckling; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Development; Muscle, Smooth; Neuroeffector Junction; Rats; Rats, Wistar; Receptors, Purinergic P1; Vas Deferens; Xanthines

1996
Differential ontogeny of adenosine receptors in the longitudinal muscle and muscularis mucosae of the rat isolated duodenum.
    European journal of pharmacology, 1996, Dec-19, Volume: 317, Issue:2-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Duodenum; Intestinal Mucosa; Male; Muscle Development; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

1996
Role of adenosine receptor subtypes in neural stunning of sympathetic coronary innervation.
    The American journal of physiology, 1997, Volume: 272, Issue:1 Pt 2

    Topics: Adenosine; Animals; Coronary Vessels; Dogs; Female; Male; Myocardial Stunning; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Sympathetic Nervous System; Theobromine; Theophylline; Vasoconstriction; Xanthines

1997
Adenosine and the endothelium-dependent modulation of 3H-noradrenaline release in the canine pulmonary artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:6

    Topics: Adenosine; Animals; Dogs; Electric Stimulation; Endothelin-1; Endothelium, Vascular; Female; Isotope Labeling; Male; Neuromuscular Junction; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Norepinephrine; Potassium; Potassium Channels; Pulmonary Artery; Purinergic P1 Receptor Antagonists; Suramin; Tetraethylammonium; Tetraethylammonium Compounds; Tritium; Xanthines

1995
Effect of adenosine receptor modulation on pentylenetetrazole-induced seizures in rats.
    British journal of pharmacology, 1997, Volume: 120, Issue:2

    Topics: Adenosine; Animals; Blood Pressure; Body Temperature; Heart Rate; Male; Pentylenetetrazole; Rats; Rats, Wistar; Receptors, Purinergic P1; Seizures; Xanthines

1997
Purine modulation of dizocilpine effects on spontaneous alternation.
    Psychopharmacology, 1997, Volume: 130, Issue:4

    Topics: Adenosine; Animals; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Maze Learning; Memory; Mice; Muscarinic Antagonists; Receptors, Purinergic P1; Scopolamine; Xanthines

1997
Adenosine A1 receptor-mediated activation of phospholipase C in cultured astrocytes depends on the level of receptor expression.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jul-01, Volume: 17, Issue:13

    Topics: Adenosine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Animals; Astrocytes; Brain; Cells, Cultured; Cyclic AMP; Enzyme Activation; Excitatory Amino Acid Antagonists; Extracellular Space; Glutamates; Inositol Phosphates; Intercellular Signaling Peptides and Proteins; Peptides; Rats; Receptors, Adrenergic, alpha; Receptors, Purinergic P1; RNA, Messenger; Type C Phospholipases; Virulence Factors, Bordetella; Wasp Venoms; Xanthines

1997
P2-receptor-mediated inhibition of noradrenaline release in the rat hippocampus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:6

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Electric Stimulation; Hippocampus; In Vitro Techniques; Isotope Labeling; Male; Norepinephrine; Phenethylamines; Rats; Rats, Wistar; Receptors, Purinergic P2; Thionucleotides; Triazines; Tritium; Xanthines; Yohimbine

1997
Adenosine A1 receptor promotion of multinucleated giant cell formation by human monocytes: a mechanism for methotrexate-induced nodulosis in rheumatoid arthritis.
    Arthritis and rheumatism, 1997, Volume: 40, Issue:7

    Topics: Adenosine; Antirheumatic Agents; Arthritis, Rheumatoid; Cells, Cultured; Humans; Methotrexate; Monocytes; Receptors, Purinergic P1; Rheumatoid Nodule; Tetradecanoylphorbol Acetate; Theobromine; Xanthines

1997
Adenosine A2 receptors modulate haloperidol-induced catalepsy in rats.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Catalepsy; Dopamine Antagonists; Haloperidol; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Scopolamine; Theobromine; Theophylline; Xanthines

1997
Regulation of purinoceptors in guinea pig pulmonary artery: functional evidences.
    Acta physiologica Hungarica, 1996, Volume: 84, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Female; Guinea Pigs; Pulmonary Artery; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic; Vasoconstriction; Vasodilation; Xanthines

1996
Competition of adenine nucleotides for a 1,3-[3H]-dipropyl-8-cyclopentylxanthine binding site in rat vas deferens.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:7

    Topics: 2-Chloroadenosine; Adenine Nucleotides; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding Sites; Binding, Competitive; In Vitro Techniques; Kinetics; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Vas Deferens; Xanthines

1997
The involvement of adenosine receptors in the effect of dizocilpine on mice in the elevated plus-maze.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1997, Volume: 7, Issue:4

    Topics: Adenosine; Animals; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic P1; Xanthines

1997
Characterization of adenosine receptors on rat ileum, ileal longitudinal muscle and muscularis mucosae.
    European journal of pharmacology, 1997, Nov-05, Volume: 338, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Electric Stimulation; Ileum; Intestinal Mucosa; Male; Muscle, Smooth; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Vasodilator Agents; Xanthines

1997
Comparison of an adenosine A1 receptor agonist and antagonist on the rat EEG.
    Neuroscience letters, 1998, Mar-06, Volume: 244, Issue:1

    Topics: Adenosine; Animals; Electroencephalography; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Xanthines

1998
Adenosine receptor mediates motility in human melanoma cells.
    Biochemical and biophysical research communications, 1998, May-29, Volume: 246, Issue:3

    Topics: Adenosine; Adenosine Monophosphate; Animals; Chemotaxis; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Humans; Melanoma, Experimental; Pertussis Toxin; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Transfection; Virulence Factors, Bordetella; Xanthines

1998
Cyclopentyladenosine-induced homologous down-regulation of A1 adenosine receptors (A1AR) in intact neurons is accompanied by receptor sequestration but not a reduction in A1AR mRNA expression or G protein alpha-subunit content.
    Journal of neurochemistry, 1998, Volume: 71, Issue:1

    Topics: Adenosine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cells, Cultured; Cerebellum; Down-Regulation; Gene Expression; GTP-Binding Protein alpha Subunits, Gs; Neurons; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; RNA, Messenger; Theophylline; Tritium; Xanthines

1998
Decreased presynaptic sensitivity to adenosine after cocaine withdrawal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Oct-01, Volume: 18, Issue:19

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Affinity Labels; Animals; Cocaine; Dipyridamole; Dopamine Uptake Inhibitors; Excitatory Postsynaptic Potentials; Glutamic Acid; Hippocampus; Male; Nucleus Accumbens; Phosphodiesterase Inhibitors; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Substance Withdrawal Syndrome; Substance-Related Disorders; Theophylline; Thioinosine; Vasodilator Agents; Xanthines

1998
Removal of adenosine decreases the responsiveness of muscle glucose transport to insulin and contractions.
    Diabetes, 1998, Volume: 47, Issue:11

    Topics: Adenosine; Adenosine Deaminase; Adenylyl Cyclase Inhibitors; Animals; Biological Transport; Cyclic AMP; Drug Synergism; Glucose; Glucose Transporter Type 4; Insulin; Male; Monosaccharide Transport Proteins; Muscle Contraction; Muscle Proteins; Muscle, Skeletal; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

1998
Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A1 receptors.
    Biochemical pharmacology, 1998, Dec-01, Volume: 56, Issue:11

    Topics: Adenosine; Alanine; Amino Acid Substitution; Animals; Binding, Competitive; CHO Cells; Cricetinae; Entropy; Humans; Kinetics; Point Mutation; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Receptors, Purinergic P1; Theophylline; Thermodynamics; Threonine; Transfection; Xanthines

1998
Adenosine A1 receptor-mediated excitation of nociceptive afferents innervating the normal and arthritic rat knee joint.
    British journal of pharmacology, 1998, Volume: 125, Issue:6

    Topics: Action Potentials; Adenosine; Adenosine Triphosphate; Analgesics; Animals; Arthritis, Experimental; Hypolipidemic Agents; Knee Joint; Male; Neurons, Afferent; Nociceptors; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

1998
Ontogeny of adenosine receptors in the longitudinal muscle and muscularis mucosae of the rat distal colon.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Aging; Animals; Autoradiography; Binding Sites; Binding, Competitive; Colon; Male; Muscle Contraction; Muscle Development; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Purinergic P1; Subcellular Fractions; Vasodilator Agents; Xanthines

1999
Characterization and tissue location of the neural adenosine receptor in the rat ileum.
    British journal of pharmacology, 1999, Volume: 126, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analysis of Variance; Animals; Female; Ileum; Male; Neurons; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

1999
Effect of adenosinergic modulation on the anticonvulsant effect of phenobarbitone and carbamazepine.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:2

    Topics: Adenosine; Animals; Anticonvulsants; Carbamazepine; Convulsants; Drug Combinations; Male; Pentylenetetrazole; Phenobarbital; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Seizures; Theophylline; Xanthines

1999
Polydeoxyribonucleotides enhance the proliferation of human skin fibroblasts: involvement of A2 purinergic receptor subtypes.
    Life sciences, 1999, Volume: 64, Issue:18

    Topics: Adenosine; Calcium; Cell Division; Cytophotometry; Deoxyribonucleosides; Deoxyribonucleotides; Fibroblasts; Fura-2; Humans; Oligodeoxyribonucleotides; Placenta; Receptors, Purinergic P1; Second Messenger Systems; Theobromine; Xanthines

1999
Allosteric modulation of the adenosine A(1) receptor. Synthesis and biological evaluation of novel 2-amino-3-benzoylthiophenes as allosteric enhancers of agonist binding.
    Journal of medicinal chemistry, 1999, Sep-09, Volume: 42, Issue:18

    Topics: Adenosine; Allosteric Regulation; Animals; Binding, Competitive; Brain; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Thiophenes; Xanthines

1999
Ischemic preconditioning prevents postischemic P-selectin expression in the rat small intestine.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Adenosine; Adenosine Deaminase; Animals; Antibodies, Monoclonal; Ischemia; Ischemic Preconditioning; Jejunum; Male; Organ Specificity; P-Selectin; Protein Kinase C; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Reperfusion; Theobromine; Xanthines

1999
Cross talk between A(1) and A(2A) adenosine receptors in the hippocampus and cortex of young adult and old rats.
    Journal of neurophysiology, 1999, Volume: 82, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Aging; Animals; Binding, Competitive; Cerebral Cortex; Electrophysiology; Hippocampus; In Vitro Techniques; Male; Phenethylamines; Protein Kinase C; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor Cross-Talk; Receptor, Adenosine A2A; Receptors, Purinergic P1; Synaptic Membranes; Triazines; Triazoles; Xanthines

1999
The anxiogenic-like effect of caffeine in two experimental procedures measuring anxiety in the mouse is not shared by selective A(2A) adenosine receptor antagonists.
    Psychopharmacology, 2000, Volume: 148, Issue:2

    Topics: Adenosine; Administration, Oral; Animals; Anxiety; Behavior, Animal; Caffeine; Darkness; Drug Administration Schedule; Injections, Intraperitoneal; Light; Male; Maze Learning; Mice; Mice, Knockout; Neuroprotective Agents; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Reaction Time; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2000
Adenosine modulation of D-[3H]aspartate release in cultured retina cells exposed to oxidative stress.
    Neurochemistry international, 2000, Volume: 36, Issue:3

    Topics: Adenosine; Adenosine Deaminase; Animals; Ascorbic Acid; Aspartic Acid; Calcium; Cells, Cultured; Chick Embryo; Drug Synergism; Kinetics; Oxidative Stress; Phenethylamines; Potassium; Potassium Chloride; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Retina; Theobromine; Tritium; Xanthines

2000
A1 adenosine receptor activation increases adipocyte leptin secretion.
    Endocrinology, 2000, Volume: 141, Issue:4

    Topics: Adenosine; Adipocytes; Animals; Culture Techniques; Dipyridamole; Gene Expression; Leptin; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; RNA, Messenger; Xanthines

2000
Effects of cyclopentyladenosine on isoproterenol response in adult and senescent cardiac tissue from Fischer 344 rats.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:2

    Topics: Adenosine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Agonists; Aging; Animals; Cardiotonic Agents; Electric Stimulation; Heart; Heart Atria; Heart Ventricles; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Xanthines

2000
Inhibition of synaptically evoked cortical acetylcholine release by adenosine: an in vivo microdialysis study in the rat.
    Neuroscience, 2000, Volume: 97, Issue:2

    Topics: Acetylcholine; Adenosine; Analysis of Variance; Animals; Caffeine; Cerebral Cortex; Chromatography, High Pressure Liquid; Dipyridamole; Male; Microdialysis; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Synapses; Xanthines

2000
Activation of protein kinase B by the A(1)-adenosine receptor in DDT(1)MF-2 cells.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adenosine; Androstadienes; Animals; Calcium; Cell Line; Chromones; Cricetinae; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Imidazoles; Indoles; Insulin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Morpholines; Pertussis Toxin; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyridines; Receptors, Purinergic P1; Virulence Factors, Bordetella; Wortmannin; Xanthines

2000
Adenosine A(1) and A(3) receptors mediate inhibition of synaptic transmission in rat cortical neurons.
    Neuropharmacology, 2001, Volume: 40, Issue:1

    Topics: Adenosine; Animals; Cerebral Cortex; Drug Interactions; Electric Stimulation; Female; In Vitro Techniques; Male; Neurons; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Rats; Rats, Wistar; Receptor, Adenosine A3; Receptors, Purinergic P1; Synaptic Transmission; Triazoles; Xanthines

2001
Adenosine A(2A) receptors mediate cardiovascular responses to hypoxia in fetal sheep.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:1

    Topics: Adenosine; Animals; Blood Gas Analysis; Blood Pressure; Female; Fetal Hypoxia; Heart Rate; Hydrogen-Ion Concentration; Phenethylamines; Pregnancy; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sheep; Triazines; Triazoles; Xanthines

2001
Extracellular adenosine modulates a volume-sensitive-like chloride conductance in immortalized rabbit DC1 cells.
    American journal of physiology. Renal physiology, 2001, Volume: 280, Issue:1

    Topics: Adenosine; Animals; Cell Line; Cell Membrane; Cell Size; Chloride Channels; Gadolinium; Guanosine 5'-O-(3-Thiotriphosphate); Hypotonic Solutions; Iodine Radioisotopes; Kidney Tubules; Lanthanum; Manganese; Membrane Potentials; Patch-Clamp Techniques; Rabbits; Receptors, Purinergic P1; Recombinant Proteins; Transfection; Xanthines

2001
Modification of adenosine modulation of synaptic transmission in the hippocampus of aged rats.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Adenosine; Adenosine Deaminase; Aging; Animals; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Hippocampus; Hypoxia; In Vitro Techniques; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Synaptic Transmission; Xanthines

2000
Effect of an adenosine A(1) receptor agonist and a novel pyrimidoindole on membrane properties and neurotransmitter release in rat cortical and hippocampal neurons.
    Neurochemistry international, 2001, Volume: 38, Issue:5

    Topics: Adenosine; Animals; Hippocampus; In Vitro Techniques; Indoles; Male; Membrane Potentials; Neurons; Neurotransmitter Agents; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Rats; Rats, Wistar; Somatosensory Cortex; Xanthines

2001
Regulation of p42/p44 MAPK and p38 MAPK by the adenosine A(1) receptor in DDT(1)MF-2 cells.
    European journal of pharmacology, 2001, Feb-16, Volume: 413, Issue:2-3

    Topics: Adenosine; Animals; Cell Line; Cricetinae; Enzyme Inhibitors; Hypoglycemic Agents; Insulin; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Muscle, Smooth; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Protein Kinase C; Protein-Tyrosine Kinases; Receptors, Purinergic P1; Signal Transduction; Vasodilator Agents; Xanthines

2001
Anti-adrenergic effect of adenosine on Na(+)-Ca(2+) exchange current recorded from guinea-pig ventricular myocytes.
    Cell calcium, 2001, Volume: 29, Issue:5

    Topics: Adenosine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cells, Cultured; Cholinergic Agonists; GTP-Binding Protein alpha Subunits, Gi-Go; Guinea Pigs; Heart Ventricles; Isoproterenol; Myocardium; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Protein Kinase C; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Signal Transduction; Sodium-Calcium Exchanger; Ventricular Function; Xanthines

2001
Ameliorative effects of paeoniflorin, a major constituent of peony root, on adenosine A1 receptor-mediated impairment of passive avoidance performance and long-term potentiation in the hippocampus.
    Biological & pharmaceutical bulletin, 2001, Volume: 24, Issue:5

    Topics: Adenosine; Animals; Avoidance Learning; Benzoates; Bridged-Ring Compounds; Glucosides; Hippocampus; Long-Term Potentiation; Male; Mice; Monoterpenes; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

2001
Electrically evoked release of glutamate in rat hippocampal slices: effects of various drugs and fimbria-fornix lesions.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:5

    Topics: Action Potentials; Adenosine; Animals; Electric Stimulation; Fornix, Brain; Glutamic Acid; Hippocampus; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Xanthines

2001
Heteromeric association creates a P2Y-like adenosine receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 2001, Jun-19, Volume: 98, Issue:13

    Topics: Adenosine; Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Heterotrimeric GTP-Binding Proteins; Humans; Inositol 1,4,5-Trisphosphate; Kinetics; Macromolecular Substances; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Purinergic P1; Receptors, Purinergic P2; Recombinant Proteins; Transfection; Tritium; Xanthines

2001
Adenosine A(1) and A(2A) receptors modulate sleep state and breathing in fetal sheep.
    Journal of applied physiology (Bethesda, Md. : 1985), 2001, Volume: 91, Issue:1

    Topics: Adenosine; Animals; Fetus; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Respiratory Physiological Phenomena; Sheep; Sleep Stages; Triazines; Triazoles; Xanthines

2001
Withdrawal and bidirectional cross-withdrawal responses in rats treated with adenosine agonists and morphine.
    Life sciences, 2001, Jul-06, Volume: 69, Issue:7

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Behavior, Animal; Female; Injections, Subcutaneous; Male; Morphine; Morphine Dependence; Muscle Contraction; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Theobromine; Xanthines

2001
Adenosine A1 receptors reduce release from excitatory but not inhibitory synaptic inputs onto lateral horn neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Aug-15, Volume: 21, Issue:16

    Topics: Adenosine; Animals; Antibody Specificity; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Immunohistochemistry; In Vitro Techniques; Interneurons; Male; Microscopy, Electron; Neural Inhibition; Patch-Clamp Techniques; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Reaction Time; Receptors, Purinergic P1; Spinal Cord; Sympathetic Nervous System; Synapses; Synaptic Transmission; Thorax; Xanthines

2001
Poly(lactic acid) microspheres for the sustained release of a selective A1 receptor agonist.
    Journal of controlled release : official journal of the Controlled Release Society, 2001, Jun-15, Volume: 73, Issue:2-3

    Topics: Adenosine; Cyclic AMP; Delayed-Action Preparations; Drug Stability; Humans; Lactic Acid; Microspheres; Polyesters; Polymers; Purinergic P1 Receptor Agonists; Xanthines

2001
Modulation of ethanol-induced motor incoordination by mouse striatal A(1) adenosinergic receptor.
    Brain research bulletin, 2001, Jul-01, Volume: 55, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Affinity Labels; Animals; Antihypertensive Agents; Ataxia; Azides; Benzodiazepines; Central Nervous System Depressants; Corpus Striatum; Ethanol; Male; Mice; Mice, Inbred ICR; Microinjections; Motor Activity; Pertussis Toxin; Phenethylamines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Vasodilator Agents; Virulence Factors, Bordetella; Xanthines

2001
Effects of adenosine receptor agonists and antagonists in a genetic animal model of primary paroxysmal dystonia.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Adenosine; Animals; Caffeine; Cricetinae; Disease Models, Animal; Dose-Response Relationship, Drug; Dystonia; Female; Male; Mesocricetus; Muscle Contraction; Mutation; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Theobromine; Theophylline; Triazines; Triazoles; Xanthines

2001
Activation of adenosine A1 receptors by drugs to lower plasma glucose in streptozotocin-induced diabetic rats.
    Autonomic neuroscience : basic & clinical, 2000, Oct-02, Volume: 83, Issue:3

    Topics: Adenosine; Animals; Blood Glucose; Cholesterol; Diabetes Mellitus, Experimental; Dipyridamole; Disease Models, Animal; Dose-Response Relationship, Drug; Glucose; Glycogen; Hypoglycemic Agents; Insulin; Male; Muscle, Skeletal; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Streptozocin; Theophylline; Triglycerides; Xanthines

2000
Neuronal mechanisms of the anoxia-induced network oscillations in the rat hippocampus in vitro.
    The Journal of physiology, 2001, Oct-15, Volume: 536, Issue:Pt 2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; Anesthetics, Local; Animals; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periodicity; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Xanthines

2001
The sulphydryl reagent, N-ethylmaleimide, disrupts sleep and blocks A1 adenosine receptor-mediated inhibition of intracellular calcium signaling in the in vitro ventromedial preoptic nucleus.
    Neuroscience, 2001, Volume: 106, Issue:4

    Topics: Adenosine; Animals; Body Temperature; Calcium; Calcium Channels; Calcium Signaling; Circadian Rhythm; Ethylmaleimide; Fura-2; Glutamic Acid; GTP-Binding Proteins; Hypothalamus; Immunohistochemistry; Male; Neurons; Potassium; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Second Messenger Systems; Sleep; Sulfhydryl Reagents; Tetrodotoxin; Xanthines

2001
Adenosine modulates Mg(2+) uptake in distal convoluted tubule cells via A(1) and A(2) purinoceptors.
    American journal of physiology. Renal physiology, 2001, Volume: 281, Issue:6

    Topics: Adenosine; Adenosine Triphosphate; Aldosterone; Animals; Calcium; Cell Line, Transformed; Cyclic AMP; Enzyme Inhibitors; Ion Transport; Kidney Tubules, Distal; Magnesium; Mice; Parathyroid Hormone; Phenethylamines; Protein Kinase Inhibitors; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theobromine; Xanthines

2001
Adenosine inhibits excitatory transmission to substantia gelatinosa neurons of the adult rat spinal cord through the activation of presynaptic A(1) adenosine receptor.
    Pain, 2001, Volume: 94, Issue:3

    Topics: Adenosine; Age Factors; Analgesics; Animals; Antihypertensive Agents; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Substantia Gelatinosa; Triazines; Triazoles; Xanthines

2001
Blockade of adenosine A1 receptors in the posterior cingulate cortex facilitates memory in rats.
    European journal of pharmacology, 2002, Feb-22, Volume: 437, Issue:3

    Topics: Adenosine; Animals; Avoidance Learning; Dose-Response Relationship, Drug; Gyrus Cinguli; Male; Memory; Purinergic P1 Receptor Antagonists; Rats; Receptors, Purinergic P1; Retention, Psychology; Xanthines

2002
Modulatory effect of adenosine receptors on the ascending and descending neural reflex responses of rat ileum.
    BMC neuroscience, 2002, Dec-20, Volume: 3

    Topics: Adenosine; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Flavins; Gastrointestinal Motility; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Neural Inhibition; Neurons; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Reflex; Tetrodotoxin; Xanthines

2002
Involvement of adenosine A1 and A2A receptors in the motor effects of caffeine after its acute and chronic administration.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:7

    Topics: Adenosine; Amphetamine; Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Theophylline; Time Factors; Triazines; Triazoles; Tritium; Xanthines

2003
Hypersensitivity of pulmonary C fibers induced by adenosine in anesthetized rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2003, Volume: 95, Issue:3

    Topics: Adenosine; Anesthesia; Animals; Body Weight; Bradycardia; Bronchial Hyperreactivity; Capsaicin; Dose-Response Relationship, Drug; Infusions, Intravenous; Lung; Male; Nerve Fibers, Unmyelinated; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Purinergic P1; Xanthines

2003
Decrease of adenosine A1 receptor density and of adenosine neuromodulation in the hippocampus of kindled rats.
    The European journal of neuroscience, 2003, Volume: 18, Issue:4

    Topics: Adenosine; Adenosine Triphosphate; Animals; Blotting, Western; Electrophysiology; Excitatory Postsynaptic Potentials; Hippocampus; Immunohistochemistry; Kindling, Neurologic; Long-Term Potentiation; Male; Neuroprotective Agents; Organ Culture Techniques; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Synaptic Transmission; Synaptosomes; Xanthines

2003
Modulation of GABA release during morphine withdrawal in midbrain neurons in vitro.
    Neuropharmacology, 2003, Volume: 45, Issue:5

    Topics: Action Potentials; Adenosine; Affinity Labels; Animals; Colforsin; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Enkephalins; Enzyme Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Male; Mesencephalon; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Probenecid; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Substance Withdrawal Syndrome; Sulfonamides; Synaptic Transmission; Thioinosine; Time Factors; Uricosuric Agents; Vasodilator Agents; Xanthines

2003
Effect of drugs active at adenosine receptors upon chronic stress-induced hyperalgesia in rats.
    European journal of pharmacology, 2003, Nov-28, Volume: 481, Issue:2-3

    Topics: Adenosine; Animals; Chronic Disease; Hyperalgesia; Male; Pain Measurement; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Stress, Physiological; Xanthines

2003
Adenosine administration produces an antidepressant-like effect in mice: evidence for the involvement of A1 and A2A receptors.
    Neuroscience letters, 2004, Jan-23, Volume: 355, Issue:1-2

    Topics: Adenosine; Animals; Antidepressive Agents; Caffeine; Depressive Disorder; Disease Models, Animal; Female; Male; Mice; Motor Activity; Receptor, Adenosine A1; Receptor, Adenosine A2A; Stress, Psychological; Triazines; Triazoles; Xanthines

2004
Pharmacological manipulations of ATP-dependent potassium channels and adenosine A1 receptors do not impact hippocampal ischemic preconditioning in vivo: evidence in a highly quantitative gerbil model.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2004, Volume: 24, Issue:5

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Female; Gerbillinae; Glyburide; Hippocampus; Ischemic Preconditioning; Membrane Potentials; Potassium Channels; Receptor, Adenosine A1; Xanthines

2004
Adenosine acting via A1 receptors, controls the transition to status epilepticus-like behaviour in an in vitro model of epilepsy.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine Triphosphate; Analysis of Variance; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Hippocampus; In Vitro Techniques; Rats; Rats, Wistar; Receptor, Adenosine A1; Status Epilepticus; Xanthines

2004
Regulation by equilibrative nucleoside transporter of adenosine outward currents in adult rat spinal dorsal horn neurons.
    Brain research bulletin, 2004, Jul-30, Volume: 64, Issue:1

    Topics: 4-Aminopyridine; Adenosine; Animals; Barium; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Equilibrative Nucleoside Transport Proteins; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Posterior Horn Cells; Potassium; Potassium Channel Blockers; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Substantia Gelatinosa; Xanthines

2004
Allosteric modulation and constitutive activity of fusion proteins between the adenosine A1 receptor and different 351Cys-mutated Gi alpha-subunits.
    European journal of pharmacology, 2004, Sep-19, Volume: 499, Issue:1-2

    Topics: Adenosine; Allosteric Site; Animals; Binding, Competitive; Cell Membrane; COS Cells; Cysteine; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Mutation; Radioligand Assay; Receptor, Adenosine A1; Recombinant Fusion Proteins; Sodium Chloride; Sulfur Radioisotopes; Thiophenes; Transfection; Tritium; Xanthines

2004
Effects of adenosine on optic nerve head circulation in rabbits.
    Experimental eye research, 2004, Volume: 79, Issue:5

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A1 Receptor Antagonists; Adenylyl Cyclase Inhibitors; Animals; Caffeine; Capillaries; Dose-Response Relationship, Drug; Glyburide; Injections; Injections, Intravenous; Optic Disk; Phenethylamines; Potassium Channels; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rabbits; Regional Blood Flow; Stimulation, Chemical; Vasodilation; Vitreous Body; Xanthines

2004
Modulating effect of adenosine deaminase on function of adenosine A1 receptors.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine Deaminase; Calcium; Cell Line; Cell Membrane; Embryo, Mammalian; Humans; Kidney; Radioligand Assay; Receptor, Adenosine A1; Signal Transduction; Xanthines

2005
Reversal of neuromuscular effects of adenosine by specific adenosine A1-receptor antagonist in live rats.
    The International journal of neuroscience, 2005, Volume: 115, Issue:3

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Drug Interactions; Drug Synergism; Male; Neuromuscular Junction; Neuromuscular Nondepolarizing Agents; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Sciatic Nerve; Synaptic Transmission; Vecuronium Bromide; Xanthines

2005
Activation of adenosine receptors in the posterior cingulate cortex impairs memory retrieval in the rat.
    Neurobiology of learning and memory, 2005, Volume: 83, Issue:3

    Topics: Adenosine; Animals; Avoidance Learning; Cerebral Cortex; Exploratory Behavior; Gyrus Cinguli; Male; Memory; Microinjections; Phenethylamines; Purinergic Agonists; Purinergic Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2005
2-(1-Hexyn-1-yl)adenosine-induced intraocular hypertension is mediated via K+ channel opening through adenosine A2A receptor in rabbits.
    European journal of pharmacology, 2005, Aug-22, Volume: 518, Issue:2-3

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Alkynes; Animals; Antihypertensive Agents; Caffeine; Decanoic Acids; Glyburide; Hydroxy Acids; Hypotonic Solutions; Intraocular Pressure; Male; Ocular Hypertension; Phenethylamines; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rabbits; Receptor, Adenosine A2A; Sodium Chloride; Time Factors; Xanthines

2005
Allosteric modulators affect the internalization of human adenosine A1 receptors.
    European journal of pharmacology, 2005, Oct-17, Volume: 522, Issue:1-3

    Topics: Adenosine; Allosteric Regulation; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Endocytosis; Humans; Luminescent Proteins; Microscopy, Confocal; Radioligand Assay; Receptor, Adenosine A1; Recombinant Fusion Proteins; Thiadiazoles; Thiazoles; Thiophenes; Transfection; Tritium; Xanthines

2005
Adenosine-stimulated atrial natriuretic peptide release through A1 receptor subtype.
    Hypertension (Dallas, Tex. : 1979), 2005, Volume: 46, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atrial Function; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Xanthines

2005
Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist.
    British journal of pharmacology, 2006, Volume: 147, Issue:5

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Allosteric Regulation; Animals; CHO Cells; Cricetinae; Cyclic AMP; Humans; Nitriles; Pyridines; Radioligand Assay; Receptor, Adenosine A1; Thermodynamics; Xanthines

2006
Activation of adenosine A1 receptor modulates dopamine D1 receptor activity in stably cotransfected human embryonic kidney 293 cells.
    European journal of pharmacology, 2006, Oct-24, Volume: 548, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Alkaline Phosphatase; Benzazepines; Cell Line; Cyclic AMP Response Element-Binding Protein; DNA, Complementary; Dopamine Agonists; Dopamine Antagonists; Humans; Receptor, Adenosine A1; Receptors, Dopamine D1; Transfection; Xanthines

2006
The enhancement of dopamine D1 receptor desensitization by adenosine A1 receptor activation.
    European journal of pharmacology, 2007, May-07, Volume: 562, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine; Binding, Competitive; Cell Line; Cyclic AMP; Dopamine Agonists; Drug Synergism; Humans; Receptor, Adenosine A1; Receptors, Dopamine D1; Time Factors; Transfection; Xanthines

2007
ATP modulates the release of noradrenaline through two different prejunctional receptors on the adrenergic nerves of rat prostate.
    Clinical and experimental pharmacology & physiology, 2007, Volume: 34, Issue:7

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Monophosphate; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Norepinephrine; Presynaptic Terminals; Prostate; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptors, Presynaptic; Receptors, Purinergic P2; Suramin; Sympathetic Nervous System; Thionucleotides; Xanthines

2007
Activation of the A1 adenosine receptor increases insulin-stimulated glucose transport in isolated rat soleus muscle.
    Applied physiology, nutrition, and metabolism = Physiologie appliquee, nutrition et metabolisme, 2007, Volume: 32, Issue:4

    Topics: 3-O-Methylglucose; Adenosine; Adenosine A1 Receptor Antagonists; Animals; Biological Transport; Cell Membrane; Dose-Response Relationship, Drug; Glucose; Glucose Transporter Type 4; In Vitro Techniques; Insulin; Male; Muscle, Skeletal; Rats; Rats, Wistar; Receptor, Adenosine A1; RNA, Messenger; Xanthines

2007
Influence of adenosine A(1)-receptor blockade and vagotomy on the gasping and heart rate response to hypoxia in rats during early postnatal maturation.
    Journal of applied physiology (Bethesda, Md. : 1985), 2007, Volume: 103, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Animals, Newborn; Dose-Response Relationship, Drug; Forelimb; Heart Rate; Hypoxia; Parasympathetic Nervous System; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Reflex; Remission, Spontaneous; Vagotomy; Xanthines

2007
A1 and A2A receptor activation by endogenous adenosine is required for VIP enhancement of K+ -evoked [3H]-GABA release from rat hippocampal nerve terminals.
    Neuroscience letters, 2008, Jan-17, Volume: 430, Issue:3

    Topics: Adenosine; Adenosine Deaminase; Animals; gamma-Aminobutyric Acid; Hippocampus; Male; Phenethylamines; Potassium; Presynaptic Terminals; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptors, Purinergic P1; Synaptic Transmission; Synaptosomes; Tritium; Vasoactive Intestinal Peptide; Xanthines

2008
Adenosine modulates excitatory synaptic transmission and suppresses neuronal death induced by ischaemia in rat spinal motoneurones.
    Pflugers Archiv : European journal of physiology, 2008, Volume: 457, Issue:2

    Topics: Adenosine; Animals; Cell Death; Excitatory Postsynaptic Potentials; In Vitro Techniques; Lumbar Vertebrae; Miniature Postsynaptic Potentials; Motor Neurons; Patch-Clamp Techniques; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptors, Presynaptic; Receptors, Purinergic P1; Sacrum; Spinal Cord; Spinal Cord Ischemia; Synaptic Transmission; Xanthines

2008
Rhythm generation by the pre-Bötzinger complex in medullary slice and island preparations: effects of adenosine A(1) receptor activation.
    BMC neuroscience, 2008, Oct-01, Volume: 9

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Animals, Newborn; Bicuculline; Electrophysiology; Evoked Potentials; Female; In Vitro Techniques; Male; Medulla Oblongata; Mice; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pyridazines; Receptor, Adenosine A1; Respiratory Center; Respiratory Mechanics; Strychnine; Synaptic Transmission; Xanthines

2008
Adenosine modulates alpha2-adrenergic receptors within specific subnuclei of the nucleus tractus solitarius in normotensive and spontaneously hypertensive rats.
    Hypertension research : official journal of the Japanese Society of Hypertension, 2008, Volume: 31, Issue:12

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Intranuclear Space; Male; Protein Binding; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Adenosine A1; Receptors, Adrenergic, alpha-2; Solitary Nucleus; Xanthines

2008
The potential role of the nodose ganglion adenosine A1 receptor in regulation of breathing in anaesthetized rats.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2008, Volume: 59, Issue:4

    Topics: Adenosine; Animals; Blood Pressure; Heart Rate; Male; Nodose Ganglion; Rats; Rats, Wistar; Receptor, Adenosine A1; Respiratory Mechanics; Tidal Volume; Vagotomy; Xanthines

2008
Cardioprotection induced by adenosine A1 receptor agonists in a cardiac cell ischemia model involves cooperative activation of adenosine A2A and A2B receptors by endogenous adenosine.
    Journal of cardiovascular pharmacology, 2009, Volume: 53, Issue:5

    Topics: Acetamides; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Aminopyridines; Animals; Apoptosis; Cardiotonic Agents; Cell Line; Cell Survival; Dihydropyridines; Imidazoles; Myocardial Ischemia; Phenethylamines; Purines; Rats; Triazines; Triazoles; Xanthines

2009
Adenosine A1 receptors presynaptically modulate excitatory synaptic input onto subiculum neurons.
    Brain research, 2009, Jul-14, Volume: 1280

    Topics: Action Potentials; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Central Nervous System Agents; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Presynaptic Terminals; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adenosine A2; Synapses; Synaptic Transmission; Triazines; Triazoles; Xanthines

2009
P2X(1) receptor blockade inhibits whole kidney autoregulation of renal blood flow in vivo.
    American journal of physiology. Renal physiology, 2010, Volume: 298, Issue:6

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine Triphosphate; Animals; Arterioles; Blood Pressure; Dinucleoside Phosphates; Dose-Response Relationship, Drug; Homeostasis; Kidney; Male; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Purinergic P2; Receptors, Purinergic P2X; Renal Circulation; Xanthines

2010
Differential effects of adenosine A1 receptor on pain-related behavior in normal and nerve-injured rats.
    Brain research, 2010, Nov-18, Volume: 1361

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Drug Administration Schedule; Electric Stimulation; Electrophysiology; Escape Reaction; Injections, Intraperitoneal; Long-Term Potentiation; Male; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neuralgia; Pain Threshold; Rats; Rats, Sprague-Dawley; Spinal Nerves; Xanthines

2010
Cooperative cardioprotection through adenosine A1 and A2A receptor agonism in ischemia-reperfused isolated mouse heart.
    Journal of cardiovascular pharmacology, 2010, Volume: 56, Issue:4

    Topics: Acetamides; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Blood Pressure; Cardiotonic Agents; Drug Synergism; In Vitro Techniques; Male; Mice; Mice, Knockout; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocardial Contraction; Myocardial Reperfusion Injury; Phosphorylation; Purines; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2010
A1 receptors self-regulate adenosine release in the striatum: evidence of autoreceptor characteristics.
    Neuroscience, 2010, Dec-29, Volume: 171, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Analysis of Variance; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Electric Stimulation; Electrochemistry; Electrodes, Implanted; Male; Models, Biological; Neural Pathways; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Substantia Nigra; Time Factors; Ventral Tegmental Area; Xanthines

2010
Expression of human equilibrative nucleoside transporter 1 in mouse neurons regulates adenosine levels in physiological and hypoxic-ischemic conditions.
    Journal of neurochemistry, 2011, Volume: 118, Issue:1

    Topics: Action Potentials; Adenosine; Adenosine A1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Equilibrative Nucleoside Transporter 1; Female; Glucose; Glutathione; Hippocampus; Humans; Hypoxia; In Vitro Techniques; Mice; Mice, Transgenic; Neurons; Patch-Clamp Techniques; Protein Binding; Purinergic P1 Receptor Agonists; Statistics, Nonparametric; Synaptic Transmission; Thioinosine; Tritium; Xanthines

2011
Genetically controlled upregulation of adenosine A(1) receptor expression enhances the survival of primary cortical neurons.
    Molecular neurobiology, 2012, Volume: 46, Issue:2

    Topics: Adenosine; Adenosine Deaminase; Animals; Calcium Channels; Cell Survival; Cerebral Cortex; HEK293 Cells; Humans; Mice; N-Methylaspartate; Neurons; Neuroprotective Agents; Neurotoxins; Receptor, Adenosine A1; Tetracycline; Transfection; Up-Regulation; Xanthines

2012
NeuroProtective effects of adenosine receptor agonist coadministration with ascorbic acid on CA1 hippocampus in a mouse model of ischemia reperfusion injury.
    Metabolic brain disease, 2013, Volume: 28, Issue:3

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Antioxidants; Ascorbic Acid; Avoidance Learning; bcl-2-Associated X Protein; Behavior, Animal; Blotting, Western; CA1 Region, Hippocampal; In Situ Nick-End Labeling; Male; Maze Learning; Memory, Short-Term; Mice; Neuroprotective Agents; Proto-Oncogene Proteins c-bcl-2; Receptors, Purinergic P1; Reperfusion Injury; Xanthines

2013
Modulation of cGMP accumulation by adenosine A1 receptors at the hippocampus: influence of cGMP levels and gender.
    European journal of pharmacology, 2014, Dec-05, Volume: 744

    Topics: Adenosine; Adenosine Deaminase; Animals; Colforsin; Cyclic AMP; Cyclic GMP; Female; Hippocampus; Imidazoles; Male; Nitroprusside; Rats; Rats, Wistar; Receptor, Adenosine A1; Rolipram; Triazines; Xanthines

2014
Presymptomatic and symptomatic ALS SOD1(G93A) mice differ in adenosine A1 and A2A receptor-mediated tonic modulation of neuromuscular transmission.
    Purinergic signalling, 2015, Volume: 11, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Amyotrophic Lateral Sclerosis; Animals; Evoked Potentials; Mice; Motor Endplate; Neuromuscular Junction; Phenethylamines; Receptor Cross-Talk; Receptor, Adenosine A1; Receptor, Adenosine A2A; Superoxide Dismutase; Superoxide Dismutase-1; Synaptic Transmission; Xanthines

2015
Adenosine A1 receptors mediate the intracisternal injection of orexin-induced antinociceptive action against colonic distension in conscious rats.
    Journal of the neurological sciences, 2016, Mar-15, Volume: 362

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Analgesics; Animals; Colon; Consciousness; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Male; Orexins; Physical Stimulation; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Reflex; Visceral Pain; Xanthines

2016
Adenosine A1 receptor modifies P53 expression and apoptosis in breast cancer cell line Mcf-7.
    Bratislavske lekarske listy, 2016, Volume: 117, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Apoptosis; Breast Neoplasms; Cell Proliferation; Cell Survival; Gene Expression Profiling; Genes, p53; Humans; MCF-7 Cells; Receptor, Adenosine A1; Xanthines

2016