1,3-dipropyl-8-cyclopentylxanthine has been researched along with n(6)-cyclohexyladenosine in 71 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (1.41) | 18.7374 |
1990's | 48 (67.61) | 18.2507 |
2000's | 17 (23.94) | 29.6817 |
2010's | 5 (7.04) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ijzerman, AP; Soudijn, W; van der Wenden, EM | 1 |
Jacobson, KA; van Galen, PJ; Williams, M | 1 |
Arslan, G; Dionisotti, S; Fredholm, BB; Kull, B; Ongini, E; Zocchi, C | 1 |
Arslan, G; Fredholm, BB; Kull, B; Lorenzen, A; Nilsson, C; Owman, C; Schwabe, U | 1 |
Arend, LJ; Klotz, KN; LeVier, DG; Olson, BA; Schwabe, U; Spielman, WS | 1 |
Lasley, RD; Mentzer, RM | 1 |
Fredholm, BB; Parkinson, FE; van der Ploeg, I | 1 |
Hoppe, E; Reddington, M; Schubert, P; Wasserkort, R | 1 |
Blazynski, C; Mathews, GC; Woods, C | 1 |
Fredholm, BB; Parkinson, FE | 1 |
Galbani, P; Limbruno, U; Mariani, M; Ronca, G; Ronca-Testoni, S; Zucchi, R | 1 |
Jaarsma, D; Korf, J; Sebens, JB | 1 |
Buxton, IL; Schiemann, WP; Westfall, DP | 1 |
Briggs, JP; Schnermann, J; Weihprecht, H | 1 |
Dietrich, MS; Endlich, K; Parekh, N; Steinhausen, M | 1 |
Fastbom, J; Fredholm, BB | 2 |
Bruns, RF; Fergus, JH | 1 |
Briggs, JP; Lorenz, JN; Schnermann, J; Skøtt, O; Weihprecht, H | 1 |
Lee, KS; Reddington, M | 1 |
Arcelli, D; Borasio, PG; Fabbri, E; Ginanni-Corradini, F; Pavan, B; Poli, A | 1 |
Asztely, F; Gustafsson, B; Wigström, H; Xiao, MY | 1 |
Kanayama, T; Kobayashi, M; Koshikawa, N; Murai, T; Takada, K; Tomiyama, K | 1 |
Martin, PL; May, JM | 1 |
Griffith, TM; Randall, MD; Ujiie, H | 1 |
Carter, MF; Jacobson, KA; Ji, XD; Lin, RC; Melman, N; Von Lubitz, DK | 1 |
Yagil, Y | 1 |
Edwards, RM; Spielman, WS | 1 |
Hirawa, N; Ishii, M; Iwamoto, T; Kihara, M; Takagi, N; Toya, Y; Umemura, S | 1 |
Lau, YS; Mouradian, MM | 1 |
Brunner, LC; Cotman, CW; Nguyen, L; Ułas, J | 1 |
Daly, JW; Moni, RW; Romero, FS | 1 |
Constantino, MD; Cunha, RA; Fredholm, BB; Johansson, B; Sebastião, AM | 1 |
Birdsall, NJ; Cohen, FR; Lazareno, S | 1 |
Clanachan, AS; Finegan, BA; Gandhi, M; Lopaschuk, GD | 1 |
Andrés, A; Fernández, M; Ros, M; Sanz, JM; Vendite, D | 1 |
Gagalo, IT; Matuszek, MT | 1 |
Andrés, A; Cubero, A; Fernández, M; Gonzalez-Calero, G; Ros, M; Ruiz, A; Sanz, JM | 1 |
Jacobson, KA; Jiang, JL; Liang, BT; Stambaugh, K | 1 |
Fredholm, BB; Georgiev, V; Johansson, B; Lindström, K | 1 |
Anwer, J; Dar, MS; Meng, ZH | 1 |
Schmidt, JT; Zhang, C | 1 |
Jarrott, B; Krstew, E; Lawrence, AJ | 1 |
Beresewicz, A; Maczewski, M | 1 |
Albinus, M; Finkbeiner, E; Osswald, H; Sosath, B | 1 |
Naghipour, B; Roushan-zamir, F; Shafaghi, B; Zarrindast, MR | 1 |
Grover, LM; Yan, C | 1 |
Gandolfi, O; Lucchi, R; Notari, S; Poli, A; Traversa, U; Zampacavallo, G | 1 |
Heinbockel, T; Pape, HC | 1 |
Sperlágh, B; Vizi, ES; Zsilla, G | 1 |
Elliott, KJ; Rea, MA; Todd Weber, E | 1 |
Dar, MS; DeSanty, KP | 1 |
Georgiev, V; Kambourova, T; Tchekalarova, J | 1 |
Cato, M; Colbert, C; Hallworth, R; Rea, MA | 1 |
Hayslett, JP; Macala, LJ | 1 |
Rea, MA; Sigworth, LA | 1 |
Christopoulos, A; May, LT; Sexton, PM | 1 |
Cunha-Reis, D; Fontinha, BM; Ribeiro, JA; Sebastião, AM | 1 |
Saeed Dar, M | 1 |
Gu, R; Li, W; Shan, H; Wang, J; Wang, WH; Xu, Y; Yang, B; Zhang, Y | 1 |
Brust, TB; Cayabyab, FS; MacVicar, BA | 1 |
Fatokun, AA; Smith, RA; Stone, TW | 1 |
Albasanz, JL; Ferrer, I; Martín, M; Rodríguez, A | 1 |
Binfaré, RW; Budni, J; Lobato, KR; Rodrigues, AL; Rosa, AO; Santos, AR | 1 |
Buck, LT; Pamenter, ME; Shin, DS | 1 |
Marek, GJ | 2 |
Ciocan, D; Constantinescu, AO; Ilie, A; Moldovan, M; Zagrean, AM; Zagrean, L | 1 |
Han, TH; Jang, SH; Lee, SY; Ryu, PD | 1 |
Akbarian, R; Moezi, L; Niknahad, H; Shafaroodi, H | 1 |
Araldi, D; Ferrari, LF; Levine, JD | 1 |
1 review(s) available for 1,3-dipropyl-8-cyclopentylxanthine and n(6)-cyclohexyladenosine
Article | Year |
---|---|
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship | 1992 |
70 other study(ies) available for 1,3-dipropyl-8-cyclopentylxanthine and n(6)-cyclohexyladenosine
Article | Year |
---|---|
A steric and electrostatic comparison of three models for the agonist/antagonist binding site on the adenosine A1 receptor.
Topics: Adenosine; Binding Sites; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Models, Molecular; Molecular Conformation; Molecular Structure; Purinergic Antagonists; Receptors, Purinergic; Regression Analysis; Structure-Activity Relationship; Xanthine; Xanthines | 1992 |
Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261.
Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Cyclic AMP; Humans; Purinergic P1 Receptor Antagonists; Pyrimidines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Species Specificity; Transfection; Triazoles | 1997 |
Differences in the order of potency for agonists but not antagonists at human and rat adenosine A2A receptors.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Humans; Kinetics; PC12 Cells; Phenethylamines; Polymerase Chain Reaction; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Recombinant Proteins; RNA, Messenger; Transcription, Genetic; Transfection; Triazoles; Tritium | 1999 |
Characterization of adenosine A1 receptor in a cell line (28A) derived from rabbit collecting tubule.
Topics: Adenosine; Adenylate Cyclase Toxin; Animals; Binding, Competitive; Brain; Calcium; Cell Line; Cell Membrane; Cyclic AMP; Kidney Medulla; Kidney Tubules, Collecting; Pertussis Toxin; Rabbits; Receptors, Purinergic; Virulence Factors, Bordetella; Xanthines | 1992 |
Adenosine improves recovery of postischemic myocardial function via an adenosine A1 receptor mechanism.
Topics: Adenine Nucleotides; Adenosine; Animals; Hemodynamics; In Vitro Techniques; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Rats; Rats, Wistar; Receptors, Purinergic; Xanthines | 1992 |
Effect of pertussis toxin on radioligand binding to rat brain adenosine A1 receptors.
Topics: Adenosine; Adenosine Diphosphate Ribose; Animals; Autoradiography; Brain; Ethylmaleimide; Guanosine Diphosphate; Magnesium Chloride; Male; Pertussis Toxin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Purinergic; Solubility; Virulence Factors, Bordetella; Xanthines | 1992 |
Modulation of A1 adenosine receptor function in rat brain by the polyamine, spermine.
Topics: Adenosine; Animals; Brain Chemistry; Edetic Acid; Electrophysiology; Hippocampus; In Vitro Techniques; Kinetics; Magnesium; Male; Rats; Rats, Inbred Strains; Receptors, Purinergic; Spermine; Synaptic Transmission; Xanthines | 1991 |
Evidence for the action of endogenous adenosine in the rabbit retina: modulation of the light-evoked release of acetylcholine.
Topics: Acetylcholine; Adenosine; Animals; Binding, Competitive; Light; Phenylisopropyladenosine; Rabbits; Retina; Xanthines | 1992 |
Magnesium-dependent enhancement of endogenous agonist binding to A1 adenosine receptors: a complicating factor in quantitative autoradiography.
Topics: Adenine Nucleotides; Adenosine; Animals; Autoradiography; Corpus Striatum; Magnesium; Male; Rats; Rats, Inbred Strains; Receptors, Purinergic; Xanthines | 1992 |
Effect of ischaemia on cardiac adenosine binding sites.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding Sites; Coronary Disease; In Vitro Techniques; Kinetics; Myocardium; Rats; Rats, Inbred Strains; Receptors, Purinergic; Reference Values; Xanthines | 1991 |
Reduction of adenosine A1-receptors in the perforant pathway terminal zone in Alzheimer hippocampus.
Topics: Adenosine; Aged; Aged, 80 and over; Alzheimer Disease; Autoradiography; Female; Hippocampus; Humans; Male; Middle Aged; Neural Pathways; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Purinergic; Xanthines | 1991 |
Smooth muscle adenosine A1 receptors couple to disparate effectors by distinct G proteins in pregnant myometrium.
Topics: Adenosine; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Inositol Phosphates; Muscle, Smooth; Myometrium; Pertussis Toxin; Pregnancy; Receptors, Purinergic; Type C Phospholipases; Virulence Factors, Bordetella; Xanthines | 1991 |
Inhibition of tubuloglomerular feedback during adenosine1 receptor blockade.
Topics: Adenosine; Adrenergic alpha-Antagonists; Animals; Capillaries; Feedback; Injections; Kidney Glomerulus; Kidney Tubules; Male; Pressure; Rats; Rats, Inbred Strains; Xanthines | 1990 |
Interaction between adenosine and angiotensin II in renal microcirculation.
Topics: Adenosine; Angiotensin II; Animals; Drug Interactions; Female; Kidney Glomerulus; Microcirculation; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Saralasin; Vasoconstriction; Xanthines | 1991 |
Effects of long-term theophylline treatment on adenosine A1-receptors in rat brain: autoradiographic evidence for increased receptor number and altered coupling to G-proteins.
Topics: Adenosine; Animals; Autoradiography; Brain; GTP-Binding Proteins; Male; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline; Xanthines | 1990 |
Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Allosteric Regulation; Animals; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Humans; Models, Biological; Rats; Receptors, Purinergic; Species Specificity; Structure-Activity Relationship; Xanthines | 1990 |
Effect of adenosine1-receptor blockade on renin release from rabbit isolated perfused juxtaglomerular apparatus.
Topics: Adenosine; Animals; In Vitro Techniques; Juxtaglomerular Apparatus; Kinetics; Loop of Henle; Perfusion; Rabbits; Receptors, Purinergic; Renin; Sodium Chloride; Xanthines | 1990 |
Regional differences in the effect of guanine nucleotides on agonist and antagonist binding to adenosine A1-receptors in rat brain, as revealed by autoradiography.
Topics: Adenosine; Animals; Autoradiography; Brain; Guanine Nucleotides; Guanosine Triphosphate; Male; Purinergic Antagonists; Rats; Rats, Inbred Strains; Receptors, Purinergic; Xanthines | 1990 |
1,3-Dipropyl-8-cyclopentylxanthine (DPCPX) inhibition of [3H]N-ethylcarboxamidoadenosine (NECA) binding allows the visualization of putative non-A1 adenosine receptors.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Membranes; Rats; Receptors, Cell Surface; Receptors, Purinergic; Subcellular Fractions; Xanthines | 1986 |
Adenosine analogs inhibit acetylcholine release and cyclic AMP synthesis in the guinea-pig superior cervical ganglion.
Topics: Acetylcholine; Adenosine; Animals; Colforsin; Cyclic AMP; Depression, Chemical; Electric Stimulation; Guinea Pigs; Imidazoles; Phosphodiesterase Inhibitors; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Superior Cervical Ganglion; Sympathetic Nervous System; Xanthines | 1995 |
Effect of adenosine-induced changes in presynaptic release probability on long-term potentiation in the hippocampal CA1 region.
Topics: Adenosine; Animals; Calcium; Electric Stimulation; Electrophysiology; Guinea Pigs; Hippocampus; Long-Term Potentiation; Magnesium; N-Methylaspartate; Neurotransmitter Agents; Presynaptic Terminals; Probability; Reaction Time; Xanthines | 1994 |
Opposite effects of midazolam and beta-carboline-3-carboxylate ethyl ester on the release of dopamine from rat nucleus accumbens measured by in vivo microdialysis.
Topics: Adenosine; Animals; Carbolines; Dopamine; Dose-Response Relationship, Drug; Flumazenil; Ligands; Male; Microdialysis; Midazolam; Nucleus Accumbens; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tetrodotoxin; Theobromine; Xanthines | 1994 |
Identification and functional characterization of A1 and A2 adenosine receptors in the rat vas deferens: a comparison with A1 receptors in guinea pig left atrium and A2 receptors in guinea pig aorta.
Topics: Adenine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta; Guinea Pigs; Heart; In Vitro Techniques; Male; Norbornanes; Phenethylamines; Rats; Receptors, Purinergic P1; Theophylline; Vas Deferens; Xanthines | 1994 |
Modulation of vasodilatation to levcromakalim by adenosine analogues in the rabbit ear: an explanation for hypoxic augmentation.
Topics: Adenosine; Animals; Arginine; Benzopyrans; Blood Pressure; Cromakalim; Drug Synergism; Ear, External; Guanidines; Hypoxia; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Pinacidil; Pyrroles; Rabbits; Regional Blood Flow; Vasodilation; Vasodilator Agents; Xanthines | 1994 |
Chronic administration of selective adenosine A1 receptor agonist or antagonist in cerebral ischemia.
Topics: Adenosine; Animals; Body Temperature; Brain Ischemia; Down-Regulation; Female; Gerbillinae; Hippocampus; Prosencephalon; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Up-Regulation; Xanthines | 1994 |
The effects of adenosine on water and sodium excretion.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Body Water; Diuresis; Infusions, Intra-Arterial; Infusions, Intravenous; Kidney; Male; Natriuresis; Rats; Rats, Wistar; Sodium; Xanthines | 1994 |
Adenosine A1 receptor-mediated inhibition of vasopressin action in inner medullary collecting duct.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arginine Vasopressin; Cyclic AMP; In Vitro Techniques; Kidney Medulla; Kidney Tubules, Collecting; Kinetics; Male; Pertussis Toxin; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Virulence Factors, Bordetella; Xanthines | 1994 |
Identification and characterization of adenosine A1 receptor-cAMP system in human glomeruli.
Topics: Adenosine; Binding, Competitive; Cyclic AMP; Humans; In Vitro Techniques; Kidney Glomerulus; Kinetics; Radioligand Assay; Receptors, Purinergic; Xanthines | 1993 |
Protection against acute MPTP-induced dopamine depletion in mice by adenosine A1 agonist.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 1-Methyl-4-phenylpyridinium; Adenosine; Animals; Corpus Striatum; Dopamine; Kinetics; Male; Mice; Mice, Inbred C57BL; Receptors, Purinergic; Time Factors; Xanthines | 1993 |
Reduced density of adenosine A1 receptors and preserved coupling of adenosine A1 receptors to G proteins in Alzheimer hippocampus: a quantitative autoradiographic study.
Topics: Adenosine; Aged; Aged, 80 and over; Alzheimer Disease; Autoradiography; Dizocilpine Maleate; Female; GTP-Binding Proteins; Hippocampus; Humans; Kinetics; Male; Organ Specificity; Pyramidal Tracts; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic; Tritium; Xanthines | 1993 |
The amphiphilic peptide adenoregulin enhances agonist binding to A1-adenosine receptors and [35S]GTP gamma S to brain membranes.
Topics: Adenosine; Adrenergic alpha-Agonists; Amphibian Proteins; Animals; Antimicrobial Cationic Peptides; Brain; Cell Line; Cell Membrane; Cyclic AMP; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Magnesium Chloride; Peptides; Purinergic P1 Receptor Agonists; Ranidae; Rats; Receptors, Purinergic P1; Sodium Chloride; Sulfur Radioisotopes; Thiophenes; Tritium; Xanthines | 1995 |
Evidence for high-affinity binding sites for the adenosine A2A receptor agonist [3H] CGS 21680 in the rat hippocampus and cerebral cortex that are different from striatal A2A receptors.
Topics: 2-Chloroadenosine; Adenosine; Animals; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; Hippocampus; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Xanthines | 1996 |
The effects of saponin on the binding and functional properties of the human adenosine A1 receptor.
Topics: Adenosine; Animals; Cell Membrane; Cell Membrane Permeability; CHO Cells; Cricetinae; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Protein Binding; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptors, Purinergic P1; Saponins; Xanthines | 1996 |
Inhibition of glycolysis and enhanced mechanical function of working rat hearts as a result of adenosine A1 receptor stimulation during reperfusion following ischaemia.
Topics: Adenosine; Animals; Energy Metabolism; Glycolysis; Heart; Male; Myocardial Ischemia; Myocardial Reperfusion; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Xanthines | 1996 |
Adenosine A1 receptors in cultured cerebellar granule cells: role of endogenous adenosine.
Topics: Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Animals, Newborn; Cell Membrane; Cells, Cultured; Cerebellum; Colforsin; Cyclic AMP; GTP-Binding Proteins; Kinetics; Neurons; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Time Factors; Xanthines | 1996 |
The effect of N6-cyclohexyladenosine and 5'-(N-cyclopropyl)- carboxamidoadenosine on pyrogen fever in rabbits.
Topics: Adenosine; Animals; Blood Pressure; Body Temperature; Female; Fever; Male; Oxygen Consumption; Purinergic P1 Receptor Antagonists; Pyrogens; Rabbits; Xanthines | 1997 |
Desensitization and internalization of adenosine A1 receptors in rat brain by in vivo treatment with R-PIA: involvement of coated vesicles.
Topics: Adenosine; Adenylyl Cyclase Inhibitors; Animals; Brain; Coated Vesicles; Colforsin; Enzyme Activation; Guanosine Triphosphate; Immunoblotting; Intracellular Membranes; Male; Microsomes; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Rats, Wistar; Receptors, Purinergic P1; Vasodilator Agents; Xanthines | 1996 |
A novel cardioprotective function of adenosine A1 and A3 receptors during prolonged simulated ischemia.
Topics: Adenosine; Animals; Cardiotonic Agents; Cell Hypoxia; Cells, Cultured; Chick Embryo; Dihydropyridines; Heart; Heart Ventricles; Myocardial Ischemia; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A3; Receptors, Purinergic P1; Xanthines | 1997 |
A1 and A2A adenosine receptors and A1 mRNA in mouse brain: effect of long-term caffeine treatment.
Topics: Adenosine; Animals; Antihypertensive Agents; Autoradiography; Brain Chemistry; Caffeine; Central Nervous System Stimulants; Cerebellum; Cerebral Cortex; Corpus Striatum; Hippocampus; In Situ Hybridization; Male; Mice; Mice, Inbred Strains; Phenethylamines; Radioligand Assay; Receptors, Purinergic P1; RNA, Messenger; Time Factors; Tritium; Xanthines | 1997 |
The striatal adenosinergic modulation of ethanol-induced motor incoordination in rats: possible role of chloride flux.
Topics: Adenosine; Affinity Labels; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Cerebrospinal Fluid; Chlorides; Corpus Striatum; Ethanol; GABA Modulators; Male; Microdialysis; Motor Activity; Pentobarbital; Radioisotopes; Rats; Rats, Sprague-Dawley; Xanthines | 1997 |
Adenosine A1 receptors mediate retinotectal presynaptic inhibition: uncoupling by C-kinase and role in LTP during regeneration.
Topics: Adenosine; Animals; Calcium; Enzyme Activation; Evoked Potentials, Visual; Goldfish; Long-Term Potentiation; Nerve Crush; Nerve Regeneration; Nifedipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Optic Nerve; Optic Nerve Injuries; Peptides; Pertussis Toxin; Protein Kinase C; Receptors, Purinergic P1; Retina; Spider Venoms; Superior Colliculi; Synaptic Transmission; Virulence Factors, Bordetella; Visual Pathways; Xanthines | 1998 |
Autoradiographic visualisation of axonal transport of adenosine A1 receptors along the rat vagus nerve and characterisation of adenosine A1 receptor binding in the dorsal vagal complex of hypertensive and normotensive rats.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Autoradiography; Axonal Transport; Binding, Competitive; Hypertension; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Purinergic P1; Reference Values; Solitary Nucleus; Vagus Nerve; Xanthines | 1998 |
The role of adenosine and ATP-sensitive potassium channels in the protection afforded by ischemic preconditioning against the post-ischemic endothelial dysfunction in guinea-pig hearts.
Topics: Acetylcholine; Adenosine; Adenosine Triphosphate; Animals; Endothelium, Vascular; Enzyme Inhibitors; Female; Guinea Pigs; Heart; Hemodynamics; In Vitro Techniques; Ischemic Preconditioning, Myocardial; Male; NG-Nitroarginine Methyl Ester; Nitroprusside; Pinacidil; Potassium Channel Blockers; Potassium Channels; Vasodilator Agents; Xanthines | 1998 |
Isolated superfused juxtaglomerular cells from rat kidney: a model for study of renin secretion.
Topics: Adenosine; Adenosine Deaminase; Animals; Cell Separation; Isoenzymes; Juxtaglomerular Apparatus; Male; Perfusion; Rats; Rats, Sprague-Dawley; Renin; Serum Albumin; Time Factors; Xanthines | 1998 |
Effects of adenosine receptor agents on the expression of morphine withdrawal in mice.
Topics: Adenosine; Analysis of Variance; Animals; Behavior, Animal; Diarrhea; Male; Mice; Mice, Inbred Strains; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Substance Withdrawal Syndrome; Theobromine; Xanthines | 1999 |
The modulation of excitatory synaptic transmission by adenosine in area CA1 of the rat hippocampus is temperature dependent.
Topics: Adenosine; Animals; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Temperature; Xanthines | 1999 |
Pharmacological characterization of adenosine A1 receptors and its functional role in brown trout (Salmo trutta) brain.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Brain; Cell Membrane; Glutamic Acid; Guanosine Diphosphate; Kinetics; Neuroprotective Agents; Radioligand Assay; Receptors, Purinergic P1; Synaptosomes; Theophylline; Tritium; Trout; Xanthines | 1999 |
Modulatory effects of adenosine on inhibitory postsynaptic potentials in the lateral amygdala of the rat.
Topics: Adenosine; Amygdala; Animals; Bicuculline; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Long-Evans; Receptors, Purinergic P1; Synaptic Transmission; Xanthines | 1999 |
K(ATP) channel blockers selectively interact with A(1)-adenosine receptor mediated modulation of acetylcholine release in the rat hippocampus.
Topics: 4-Aminopyridine; Acetylcholine; Adenosine; Animals; ATP-Binding Cassette Transporters; Binding, Competitive; Brain Ischemia; Electric Stimulation; Hippocampus; In Vitro Techniques; KATP Channels; Male; Muscarinic Antagonists; Oxotremorine; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Presynaptic; Receptors, Purinergic P1; Xanthines | 2001 |
Adenosine A1 receptors regulate the response of the hamster circadian clock to light.
Topics: Adenosine; Animals; Circadian Rhythm; Cricetinae; Dose-Response Relationship, Drug; Light; Male; Motor Activity; Receptors, Purinergic P1; Suprachiasmatic Nucleus; Xanthines | 2001 |
Involvement of the cerebellar adenosine A(1) receptor in cannabinoid-induced motor incoordination in the acute and tolerant state in mice.
Topics: Adenosine; Analgesics; Animals; Cannabinoids; Cerebellar Ataxia; Cerebellum; Cyclohexanols; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Male; Marijuana Abuse; Mice; Neurons; Phosphodiesterase Inhibitors; Psychomotor Performance; Receptors, Cannabinoid; Receptors, Drug; Receptors, Purinergic P1; Signal Transduction; Tritium; Xanthines | 2001 |
Effects of angiotensin III and angiotensin IV on pentylenetetrazol seizure susceptibility (threshold and kindling): interaction with adenosine A(1) receptors.
Topics: Adenosine; Angiotensin II; Angiotensin III; Angiotensins; Animals; Brain; Convulsants; Disease Susceptibility; Dose-Response Relationship, Drug; Drug Interactions; Epilepsy; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Pentylenetetrazole; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Seizures; Xanthines | 2001 |
Presynaptic adenosine A1 receptors regulate retinohypothalamic neurotransmission in the hamster suprachiasmatic nucleus.
Topics: Adenosine; Animals; Antihypertensive Agents; Circadian Rhythm; Cricetinae; Excitatory Postsynaptic Potentials; Male; Mesocricetus; Neural Inhibition; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Presynaptic; Receptors, Purinergic P1; Retina; Suprachiasmatic Nucleus; Synaptic Transmission; Visual Pathways; Xanthines | 2002 |
Basolateral and apical A1 adenosine receptors mediate sodium transport in cultured renal epithelial (A6) cells.
Topics: Adenosine; Animals; Biological Transport; Cell Line; Cell Membrane; Dimethyl Sulfoxide; Epithelial Cells; Intracellular Membranes; Kidney; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Sodium; Solvents; Xanthines; Xenopus laevis | 2002 |
Adenosine A1 receptors regulate the response of the mouse circadian clock to light.
Topics: Adenosine; Animals; Circadian Rhythm; Dose-Response Relationship, Drug; Immunohistochemistry; Light; Male; Mice; Mice, Inbred C57BL; Mitogen-Activated Protein Kinase 1; Motor Activity; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Suprachiasmatic Nucleus; Xanthines | 2003 |
Effects of urea pretreatment on the binding properties of adenosine A1 receptors.
Topics: Adenosine; Adenosine Deaminase; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Guanylyl Imidodiphosphate; Humans; Kinetics; Ligands; Protein Denaturation; Receptor, Adenosine A1; Temperature; Transfection; Urea; Xanthines | 2005 |
Tonic adenosine A1 and A2A receptor activation is required for the excitatory action of VIP on synaptic transmission in the CA1 area of the hippocampus.
Topics: Adenosine; Adenosine Deaminase; Analysis of Variance; Animals; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neuroprotective Agents; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Synaptic Transmission; Triazines; Triazoles; Vasoactive Intestinal Peptide; Xanthines | 2007 |
Co-modulation of acute ethanol-induced motor impairment by mouse cerebellar adenosinergic A1 and GABA(A) receptor systems.
Topics: Acute Disease; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Alcohol-Induced Disorders, Nervous System; Animals; Central Nervous System Depressants; Cerebellar Ataxia; Cerebellum; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Presynaptic Terminals; Receptor, Adenosine A1; Receptors, GABA-A; Synaptic Transmission; Xanthines | 2006 |
Adenosine stimulates the basolateral 50 pS K channels in the thick ascending limb of the rat kidney.
Topics: Adenosine; Adenosine A2 Receptor Antagonists; Adenylyl Cyclases; Algorithms; Animals; Bucladesine; Caffeine; Dose-Response Relationship, Drug; Enzyme Activation; Female; Kidney; Male; Patch-Clamp Techniques; Phenethylamines; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Adenosine A2; Stimulation, Chemical; Xanthines | 2007 |
C-Jun N-terminal kinase regulates adenosine A1 receptor-mediated synaptic depression in the rat hippocampus.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Animals, Newborn; Baclofen; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; GABA Agonists; Gene Expression; Hippocampus; Hypoxia; In Vitro Techniques; JNK Mitogen-Activated Protein Kinases; Long-Term Synaptic Depression; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Time Factors; Xanthines | 2007 |
Adenosine receptor ligands protect against a combination of apoptotic and necrotic cell death in cerebellar granule neurons.
Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Cell Death; Cell Survival; Cells, Cultured; Cerebellum; Cytarabine; Glutamic Acid; Kynurenic Acid; Necrosis; Neurons; Rats; Rats, Sprague-Dawley; Xanthines | 2008 |
Up-regulation of adenosine A1 receptors in frontal cortex from Pick's disease cases.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Aged; Brain; Cadaver; Cell Membrane; Colforsin; Female; Frontal Lobe; Humans; Male; Occipital Lobe; Pick Disease of the Brain; Receptor, Adenosine A1; RNA, Messenger; Up-Regulation; Xanthines | 2007 |
Involvement of the adenosine A1 and A2A receptors in the antidepressant-like effect of zinc in the forced swimming test.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Aniline Compounds; Animals; Antidepressive Agents; Caffeine; Central Nervous System Stimulants; Dipyridamole; Female; Male; Mice; Motor Activity; Nucleoside Transport Proteins; Receptor, Adenosine A1; Receptor, Adenosine A2A; Swimming; Triazines; Triazoles; Xanthines; Zinc | 2008 |
Adenosine A1 receptor activation mediates NMDA receptor activity in a pertussis toxin-sensitive manner during normoxia but not anoxia in turtle cortical neurons.
Topics: Adenosine; Analysis of Variance; Animals; Anorexia; Anti-Arrhythmia Agents; Cerebral Cortex; Chelating Agents; Decanoic Acids; Drug Interactions; Egtazic Acid; Hydroxy Acids; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pertussis Toxin; Receptor, Adenosine A1; Receptors, N-Methyl-D-Aspartate; Time Factors; Turtles; Xanthines | 2008 |
Activation of adenosine(1) (A(1)) receptors suppresses head shakes induced by a serotonergic hallucinogen in rats.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Amphetamines; Animals; Dose-Response Relationship, Drug; Glutamic Acid; Hallucinogens; Head Movements; Injections, Intraperitoneal; Locomotion; Male; Motor Activity; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Serotonin Receptor Agonists; Xanthines | 2009 |
Endogenous adenosine A1 receptor activation underlies the transient post-ischemic rhythmic delta EEG activity.
Topics: Adenosine; Adenosine A1 Receptor Antagonists; Animals; Delta Rhythm; Disease Models, Animal; Electrocardiography; Electroencephalography; Heart Rate; Ischemic Attack, Transient; Male; Rats; Rats, Wistar; Receptor, Adenosine A1; Statistics, Nonparametric; Theophylline; Xanthines | 2011 |
Adenosine reduces GABAergic IPSC frequency via presynaptic A₁ receptors in hypothalamic paraventricular neurons projecting to rostral ventrolateral medulla.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Afferent Pathways; Animals; Biophysics; Electric Stimulation; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Male; Medulla Oblongata; Neural Inhibition; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Theobromine; Xanthines | 2011 |
Activation of adenosine₁ receptors induces antidepressant-like, anti-impulsive effects on differential reinforcement of low-rate 72-s behavior in rats.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Antidepressive Agents; Autoreceptors; Behavior, Animal; Glutamic Acid; Male; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Reinforcement, Psychology; Synapses; Synaptic Transmission; Xanthines | 2012 |
The interaction of adenosine and morphine on pentylenetetrazole-induced seizure threshold in mice.
Topics: Adenosine; Animals; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Morphine; Naltrexone; Narcotic Antagonists; Pentylenetetrazole; Seizures; Xanthines | 2013 |
Regulation of Expression of Hyperalgesic Priming by Estrogen Receptor α in the Rat.
Topics: 5'-Nucleotidase; Adenosine; Adenosine A1 Receptor Antagonists; Adenosine Monophosphate; Animals; Chronic Pain; Dinoprostone; Disease Models, Animal; DNA, Antisense; Estrogen Receptor alpha; Female; Gene Expression Regulation; Hyperalgesia; Male; Pain Threshold; Rats; Rats, Sprague-Dawley; Ryanodine; Sex Factors; Time Factors; Xanthines | 2017 |