1,3-dipropyl-8-cyclopentylxanthine has been researched along with colforsin in 47 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 2 (4.26) | 18.7374 |
| 1990's | 27 (57.45) | 18.2507 |
| 2000's | 13 (27.66) | 29.6817 |
| 2010's | 5 (10.64) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
| Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
| López-Novoa, JM; Olivera, A; Tomás, M | 1 |
| LeVier, DG; McCoy, DE; Spielman, WS | 1 |
| Arai, A; Lynch, G | 1 |
| Czernilofsky, A; Dumont, JE; Ensinger, HA; Lefort, A; Libert, F; Mendla, KD; Van Sande, J; Vassart, G | 1 |
| Hreniuk, SP; Kaartinen, JM; LaNoue, KF; Martin, LF; Ohisalo, JJ; Ranta, S | 1 |
| Chatzipanteli, K; Orford, M; Saggerson, D; Shepherd, J | 1 |
| Ameri, A; Jurna, I | 1 |
| Wells, JN; Zhang, Y | 1 |
| Alexander, SP; Hill, SJ; Kendall, DA | 1 |
| Dobson, JG; MacDonald, SG; Romano, FD | 1 |
| Gean, PW; Huang, CC | 1 |
| Arcelli, D; Borasio, PG; Fabbri, E; Ginanni-Corradini, F; Pavan, B; Poli, A | 1 |
| Alexander, SP; Curtis, AR; Hill, SJ; Kendall, DA | 1 |
| Akatsuka, Y; Egashira, K; Katsuda, Y; Narishige, T; Shimokawa, H; Takeshita, A; Ueno, H | 1 |
| Alexander, SP; Cartmell, J; Kemp, JA; Kendall, DA | 1 |
| Gupta, RC; Neumann, J; Watanabe, AM | 1 |
| Correia-de-Sá, P; Ribeiro, JA | 1 |
| Bottrill, FE; Hiley, CR; Richardson, PJ; Warnock, J | 1 |
| Andrés, A; Fernández, M; Ros, M; Sanz, JM; Vendite, D | 1 |
| Haws, CM; Krouse, ME; Law, T; Nepomuceno, IB; Nguyen, H; Wakelee, H; Wine, JJ; Xia, Y | 1 |
| Belardinelli, L; Harrison, JK; Jacobson, M; Kollias-Baker, CA; Ozeck, M; Ruble, J; Shryock, JC | 1 |
| Andrés, A; Cubero, A; Fernández, M; Gonzalez-Calero, G; Ros, M; Ruiz, A; Sanz, JM | 1 |
| Bauer, J; Fiebich, BL; Heese, K; Otten, U | 1 |
| Guo, Y; He, Z; Raman, S; Reenstra, WW | 1 |
| Bispham, JR; Hill, SJ; Walker, EM | 1 |
| Gean, PW; Lu, KT | 1 |
| Al-Nakkash, L; Hwang, TC | 1 |
| Habuchi, Y; Morikawa, J; Nishio, M; Tanaka, H; Yamamoto, T | 1 |
| Hsu, KS; Huang, CC; Liang, YC | 1 |
| Dubey, RK; Gillespie, DG; Jackson, EK; Keller, PJ; Mi, Z; Rosselli, M | 1 |
| Andrés, A; Escriche, M; Franco, R; Lluis, C; Martín, M; Ros, M; Ruiz, MA | 1 |
| Doering, A; Middlekauff, HR; Weiss, JN | 1 |
| Greenberg, AG; Kraemer, FB; Xue, B; Zemel, MB | 1 |
| Esselstyn, J; Hertel, C; Lee, R; Lerner, A; Moon, E; Wolda, S | 1 |
| Erdmann, A; Gao, ZG; IJzerman, AP; Jacobson, KA; Kim, SG; Melman, N; Müller, CE | 1 |
| Christie, MJ; Hack, SP; Vaughan, CW | 1 |
| Albasanz, JL; Fernández, M; León, D; Martín, M; Ruíz, MA | 1 |
| de Ligt, RA; IJzerman, AP; Leurs, R; Lorenzen, A; Rivkees, SA | 1 |
| Cao, C; Han, JH; Kim, SH; Kim, SZ; Yuan, K | 1 |
| Albasanz, JL; Ferrer, I; Martín, M; Rodríguez, A | 1 |
| Albasanz, JL; Barrachina, M; Ferrer, I; Martín, M; Perez, S | 1 |
| Chen, CC; Hsu, KS; Huang, CC; Yang, CH | 1 |
| Dobson, JG; Fenton, RA; Ikebe, M; Komatsu, S; Shea, LG | 1 |
| Cascalheira, JF; Sebastião, AM; Serpa, A | 1 |
| Muñoz, MD; Solís, JM | 1 |
47 other study(ies) available for 1,3-dipropyl-8-cyclopentylxanthine and colforsin
| Article | Year |
|---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Effect of adenosine A1 and A2 agonists and antagonists on cAMP and Ca2+ in cultured rat mesangial cells.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Glomerular Mesangium; Purines; Rats; Sulfonamides; Xanthines | 1992 |
Functional localization of adenosine receptor-mediated pathways in the LLC-PK1 renal cell line.
Topics: Adenosine; Calcium; Cell Line; Colforsin; Cyclic AMP; Inositol Phosphates; Intracellular Membranes; Kidney; Receptors, Purinergic; Signal Transduction; Time Factors; Tissue Distribution; Xanthines | 1992 |
Factors regulating the magnitude of long-term potentiation induced by theta pattern stimulation.
Topics: Animals; Colforsin; Electric Stimulation; Evoked Potentials; Hippocampus; Membrane Potentials; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Theta Rhythm; Time Factors; Xanthines | 1992 |
Cloning and functional characterization of a human A1 adenosine receptor.
Topics: Adenosine; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; DNA; DNA Probes; Dogs; Hippocampus; Humans; Molecular Sequence Data; Nucleic Acid Hybridization; Receptors, Purinergic; Sequence Homology, Nucleic Acid; Transfection; Xanthines | 1992 |
Attenuated adenosine-sensitivity and decreased adenosine-receptor number in adipocyte plasma membranes in human obesity.
Topics: Adenosine; Adenylyl Cyclases; Adipose Tissue; Body Weight; Cell Membrane; Colforsin; Cyclic AMP; Enzyme Activation; Glucose; Humans; Isoproterenol; Obesity; Phenylisopropyladenosine; Receptors, Purinergic; Xanthines | 1991 |
Diabetes decreases sensitivity of adipocyte lipolysis to inhibition by Gi-linked receptor agonists.
Topics: Adipose Tissue; Animals; Cell Membrane; Colforsin; Diabetes Mellitus, Experimental; Dinoprostone; Electrophoresis, Polyacrylamide Gel; GTP-Binding Proteins; Immunoblotting; Lipolysis; Male; Niacin; Norepinephrine; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Xanthines | 1991 |
Adenosine A1 and non-A1 receptors: intracellular analysis of the actions of adenosine agonists and antagonists in rat hippocampal neurons.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Electric Stimulation; Electrodes; Hippocampus; Male; Membrane Potentials; Neurons; Phenylisopropyladenosine; Purinergic Antagonists; Rats; Rats, Inbred Strains; Receptors, Purinergic; Synapses; Theophylline; Xanthines | 1991 |
The effects of chronic caffeine administration on peripheral adenosine receptors.
Topics: Adenylyl Cyclases; Adipose Tissue; Animals; Binding Sites; Caffeine; Cell Membrane; Colforsin; Lipolysis; Male; Platelet Aggregation; Rats; Rats, Inbred Strains; Receptors, Purinergic; Xanthines | 1990 |
Differences in the adenosine receptors modulating inositol phosphates and cyclic AMP accumulation in mammalian cerebral cortex.
Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cerebral Cortex; Colforsin; Cyclic AMP; Female; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Kinetics; Lithium; Male; Mice; Receptors, Purinergic; Second Messenger Systems; Xanthines | 1989 |
Adenosine receptor coupling to adenylate cyclase of rat ventricular myocyte membranes.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cells, Cultured; Colforsin; Guanylyl Imidodiphosphate; Heart Ventricles; Isoproterenol; Kinetics; Male; Myocardium; Peptidyl-Dipeptidase A; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline; Xanthines | 1989 |
Cyclic adenosine-3',5'-monophosphate potentiates the synaptic potential mediated by NMDA receptors in the amygdala.
Topics: Amygdala; Animals; Bucladesine; Colforsin; Cyclic AMP; Electric Stimulation; Long-Term Potentiation; Male; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Xanthines | 1995 |
Adenosine analogs inhibit acetylcholine release and cyclic AMP synthesis in the guinea-pig superior cervical ganglion.
Topics: Acetylcholine; Adenosine; Animals; Colforsin; Cyclic AMP; Depression, Chemical; Electric Stimulation; Guinea Pigs; Imidazoles; Phosphodiesterase Inhibitors; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Superior Cervical Ganglion; Sympathetic Nervous System; Xanthines | 1995 |
A1 adenosine receptor inhibition of cyclic AMP formation and radioligand binding in the guinea-pig cerebral cortex.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cerebral Cortex; Colforsin; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Phenylisopropyladenosine; Phosphatidylinositols; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Receptors, Purinergic P1; Sulfonamides; Vasodilator Agents; Xanthines | 1994 |
ATP sensitive potassium channels are involved in adenosine A2 receptor mediated coronary vasodilatation in the dog.
Topics: Acetylcholine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Glyburide; Guanidines; Ion Channel Gating; Pinacidil; Potassium Channels; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P2; Theophylline; Vasodilator Agents; Xanthines | 1994 |
Endogenous adenosine regulates the apparent efficacy of 1-aminocyclopentyl-1S,3R-dicarboxylate inhibition of forskolin-stimulated cyclic AMP accumulation in rat cerebral cortical slices.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cerebral Cortex; Colforsin; Cyclic AMP; Cycloleucine; Female; In Vitro Techniques; Kinetics; Male; Neurotoxins; Rats; Rats, Inbred Strains; Xanthines | 1993 |
Comparison of adenosine and muscarinic receptor-mediated effects on protein phosphatase inhibitor-1 activity in the heart.
Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Carrier Proteins; Colforsin; Depression, Chemical; Enzyme Activation; Enzyme Inhibitors; Female; Guinea Pigs; Heart; Heart Ventricles; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Myocardial Contraction; Myocardium; Phenylisopropyladenosine; Phosphoprotein Phosphatases; Protein Kinases; Proteins; Receptors, Muscarinic; Receptors, Purinergic; Stimulation, Chemical; Ventricular Function; Xanthines | 1993 |
Facilitation of [3H]-ACh release by forskolin depends on A2-adenosine receptor activation.
Topics: Acetylcholine; Adenosine; Adenosine Deaminase; Adenylyl Cyclases; Animals; Colforsin; Diaphragm; Female; In Vitro Techniques; Male; Nerve Endings; Phenethylamines; Phenylisopropyladenosine; Phrenic Nerve; Purinergic Antagonists; Purines; Rats; Rats, Wistar; Receptors, Purinergic; Sulfonamides; Xanthines | 1993 |
Effects of pH on responses to adenosine, CGS 21680, carbachol and nitroprusside in the isolated perfused superior mesenteric arterial bed of the rat.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Carbachol; Colforsin; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Nitroprusside; Perfusion; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Vascular Resistance; Vasoconstrictor Agents; Vasodilator Agents; Xanthines | 1995 |
Adenosine A1 receptors in cultured cerebellar granule cells: role of endogenous adenosine.
Topics: Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Animals, Newborn; Cell Membrane; Cells, Cultured; Cerebellum; Colforsin; Cyclic AMP; GTP-Binding Proteins; Kinetics; Neurons; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Time Factors; Xanthines | 1996 |
Delta F508-CFTR channels: kinetics, activation by forskolin, and potentiation by xanthines.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Line; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; Glycosylation; Iodine; Mice; Mutation; Time Factors; Xanthines | 1996 |
Agonist-independent effect of an allosteric enhancer of the A1 adenosine receptor in CHO cells stably expressing the recombinant human A1 receptor.
Topics: Adenosine; Adenosine Deaminase; Allosteric Regulation; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Recombinant Proteins; Thiophenes; Xanthines | 1997 |
Desensitization and internalization of adenosine A1 receptors in rat brain by in vivo treatment with R-PIA: involvement of coated vesicles.
Topics: Adenosine; Adenylyl Cyclase Inhibitors; Animals; Brain; Coated Vesicles; Colforsin; Enzyme Activation; Guanosine Triphosphate; Immunoblotting; Intracellular Membranes; Male; Microsomes; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Rats, Wistar; Receptors, Purinergic P1; Vasodilator Agents; Xanthines | 1996 |
Nerve growth factor (NGF) expression in rat microglia is induced by adenosine A2a-receptors.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Animals, Newborn; Antihypertensive Agents; Bucladesine; Colforsin; Gene Expression; Microglia; Nerve Growth Factors; Phenethylamines; Polymerase Chain Reaction; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Vasodilator Agents; Xanthines | 1997 |
Cystic fibrosis transmembrane conductance regulator activation by cAMP-independent mechanisms.
Topics: 1-Methyl-3-isobutylxanthine; 3T3 Cells; Animals; Benzimidazoles; Chlorophenols; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Inhibitors; Genistein; Humans; Kinetics; Marine Toxins; Mice; Oxazoles; Phosphopeptides; Phosphorylation; Recombinant Proteins; Sequence Deletion; Transfection; Xanthines | 1998 |
Nonselective effects of the putative phospholipase C inhibitor, U73122, on adenosine A1 receptor-mediated signal transduction events in Chinese hamster ovary cells.
Topics: Animals; Cell Survival; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Inositol Phosphates; Kinetics; Phosphatidylinositols; Pyrrolidinones; Receptors, Purinergic P1; Recombinant Proteins; Signal Transduction; Transfection; Type C Phospholipases; Xanthines | 1998 |
Masking of forskolin-induced long-term potentiation by adenosine accumulation in area CA1 of the rat hippocampus.
Topics: 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Hippocampus; Long-Term Potentiation; Male; Nerve Fibers; Neurons; Probenecid; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Synapses; Thionucleotides; Xanthines | 1999 |
Activation of wild-type and deltaF508-CFTR by phosphodiesterase inhibitors through cAMP-dependent and -independent mechanisms.
Topics: 1-Methyl-3-isobutylxanthine; 3T3 Cells; Animals; Cell Line; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Mice; Milrinone; Mutation; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Thionucleotides; Xanthines | 1999 |
P2 purinoceptors contribute to ATP-induced inhibition of L-type Ca2+ current in rabbit atrial myocytes.
Topics: 1-Methyl-3-isobutylxanthine; 5'-Nucleotidase; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Calcium-Transporting ATPases; Colforsin; Cyclic AMP; Enzyme Inhibitors; Isoproterenol; Myocardium; Patch-Clamp Techniques; Pertussis Toxin; Potassium Channels; Potassium Channels, Voltage-Gated; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rabbits; Receptors, Purinergic P2; Shal Potassium Channels; Suramin; Virulence Factors, Bordetella; Xanthines | 1999 |
A role for extracellular adenosine in time-dependent reversal of long-term potentiation by low-frequency stimulation at hippocampal CA1 synapses.
Topics: Adenosine; Animals; Buspirone; Colforsin; Cyclic AMP; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Least-Squares Analysis; Long-Term Potentiation; Male; Neurons; Piperazines; Purinergic P1 Receptor Antagonists; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Theobromine; Thionucleotides; Time Factors; Xanthines | 1999 |
Estradiol inhibits smooth muscle cell growth in part by activating the cAMP-adenosine pathway.
Topics: Adenosine; Adenylyl Cyclases; Animals; Antihypertensive Agents; Aorta; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; DDT; Enzyme Inhibitors; Estradiol; Fetal Proteins; Male; Muscle, Smooth, Vascular; Proline; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Thionucleotides; Thymidine; Tritium; Xanthines | 2000 |
Adenosine A(1) receptor in cultured neurons from rat cerebral cortex: colocalization with adenosine deaminase.
Topics: Adenosine Deaminase; Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; Embryo, Mammalian; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Kinetics; Neurons; Rats; Rats, Wistar; Receptors, Purinergic P1; Transcription, Genetic; Xanthines | 2000 |
Adenosine enhances neuroexcitability by inhibiting a slow postspike afterhyperpolarization in rabbit vagal afferent neurons.
Topics: Action Potentials; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cadmium; Colforsin; Neurons, Afferent; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rabbits; Receptors, Purinergic P1; Time Factors; Vagus Nerve; Xanthines | 2001 |
Mechanism of intracellular calcium ([Ca2+]i) inhibition of lipolysis in human adipocytes.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Adipocytes; Androstadienes; Bucladesine; Calcium; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Humans; Insulin; Isoproterenol; Lipolysis; Phosphodiesterase Inhibitors; Phosphorylation; Potassium Chloride; Quinolones; Sterol Esterase; Wortmannin; Xanthines | 2001 |
PDE7A is expressed in human B-lymphocytes and is up-regulated by elevation of intracellular cAMP.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; B-Lymphocytes; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Humans; Intracellular Fluid; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Lymphocytic, Chronic, B-Cell; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Antagonists; Spleen; Theophylline; Tumor Cells, Cultured; Up-Regulation; Xanthines | 2002 |
Differential allosteric modulation by amiloride analogues of agonist and antagonist binding at A(1) and A(3) adenosine receptors.
Topics: Adenosine; Allosteric Regulation; Amiloride; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diuretics; Dose-Response Relationship, Drug; Drug Interactions; Humans; Imidazoles; Kinetics; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Transfection; Tritium; Xanthines | 2003 |
Modulation of GABA release during morphine withdrawal in midbrain neurons in vitro.
Topics: Action Potentials; Adenosine; Affinity Labels; Animals; Colforsin; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Enkephalins; Enzyme Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Male; Mesencephalon; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Probenecid; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Substance Withdrawal Syndrome; Sulfonamides; Synaptic Transmission; Thioinosine; Time Factors; Uricosuric Agents; Vasodilator Agents; Xanthines | 2003 |
Down-regulation of rat brain adenosine A1 receptors at the end of pregnancy.
Topics: Adenosine; Adenylyl Cyclases; Aldehyde-Lyases; Animals; Antihypertensive Agents; Binding Sites; Blotting, Northern; Brain; Cell Membrane; Colforsin; Densitometry; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Female; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Immunoblotting; Phenethylamines; Pregnancy; Rats; Rats, Wistar; Receptor, Adenosine A1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tritium; Xanthines | 2004 |
A "locked-on," constitutively active mutant of the adenosine A1 receptor.
Topics: Adenosine; Animals; Binding, Competitive; Cell Line; Cell Membrane; Chlorocebus aethiops; Colforsin; COS Cells; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Humans; Kinetics; Mutation; Plasmids; Radioligand Assay; Receptor, Adenosine A1; Sodium; Sulfur Radioisotopes; Theophylline; Thiophenes; Transfection; Tritium; Xanthines | 2005 |
Adenosine-stimulated atrial natriuretic peptide release through A1 receptor subtype.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atrial Function; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Xanthines | 2005 |
Up-regulation of adenosine A1 receptors in frontal cortex from Pick's disease cases.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Aged; Brain; Cadaver; Cell Membrane; Colforsin; Female; Frontal Lobe; Humans; Male; Occipital Lobe; Pick Disease of the Brain; Receptor, Adenosine A1; RNA, Messenger; Up-Regulation; Xanthines | 2007 |
Up-regulation of adenosine receptors in the frontal cortex in Alzheimer's disease.
Topics: Adenylyl Cyclases; Aged; Aged, 80 and over; Alzheimer Disease; Analysis of Variance; Cell Membrane; Colforsin; Cyclic AMP; Female; Frontal Lobe; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Protein Binding; Receptors, Purinergic P1; Triazines; Triazoles; Tritium; Up-Regulation; Xanthines | 2008 |
Acute stress impairs hippocampal mossy fiber-CA3 long-term potentiation by enhancing cAMP-specific phosphodiesterase 4 activity.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adrenalectomy; Animals; Anti-Inflammatory Agents; Biophysical Phenomena; Colforsin; Corticosterone; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Mice; Mice, Inbred C57BL; Mineralocorticoid Receptor Antagonists; Mossy Fibers, Hippocampal; Phosphodiesterase Inhibitors; Spironolactone; Stress, Psychological; Synaptosomes; Xanthines | 2010 |
Crosstalk between adenosine A1 and β1-adrenergic receptors regulates translocation of PKCε in isolated rat cardiomyocytes.
Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adrenergic beta-1 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Intracellular Signaling Peptides and Proteins; Isoproterenol; Isoquinolines; Membrane Proteins; Myocardium; Myocytes, Cardiac; Organ Culture Techniques; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Protein Transport; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adrenergic, beta-1; Signal Transduction; Sulfonamides; Xanthines | 2012 |
Modulation of cGMP accumulation by adenosine A1 receptors at the hippocampus: influence of cGMP levels and gender.
Topics: Adenosine; Adenosine Deaminase; Animals; Colforsin; Cyclic AMP; Cyclic GMP; Female; Hippocampus; Imidazoles; Male; Nitroprusside; Rats; Rats, Wistar; Receptor, Adenosine A1; Rolipram; Triazines; Xanthines | 2014 |
Characterisation of the mechanisms underlying the special sensitivity of the CA2 hippocampal area to adenosine receptor antagonists.
Topics: Adenylyl Cyclases; Animals; CA1 Region, Hippocampal; CA2 Region, Hippocampal; Caffeine; Colforsin; Excitatory Postsynaptic Potentials; Male; Phosphodiesterase Inhibitors; Purinergic Agonists; Purinergic P1 Receptor Antagonists; Rats, Sprague-Dawley; Receptor, Adenosine A1; Rolipram; Synapses; Tissue Culture Techniques; Xanthines | 2019 |