Page last updated: 2024-09-04

1,1'-biphenyl-4-yl-boronic acid and benzo(b)thiophene-2-boronic acid

1,1'-biphenyl-4-yl-boronic acid has been researched along with benzo(b)thiophene-2-boronic acid in 3 studies

Compound Research Comparison

Studies
(1,1'-biphenyl-4-yl-boronic acid)
Trials
(1,1'-biphenyl-4-yl-boronic acid)
Recent Studies (post-2010)
(1,1'-biphenyl-4-yl-boronic acid)
Studies
(benzo(b)thiophene-2-boronic acid)
Trials
(benzo(b)thiophene-2-boronic acid)
Recent Studies (post-2010) (benzo(b)thiophene-2-boronic acid)
10051703

Protein Interaction Comparison

ProteinTaxonomy1,1'-biphenyl-4-yl-boronic acid (IC50)benzo(b)thiophene-2-boronic acid (IC50)
B2 bradykinin receptorCavia porcellus (domestic guinea pig)0.2
Acyl-protein thioesterase 1Homo sapiens (human)1.4145
Acyl-protein thioesterase 2Homo sapiens (human)1.4145
Chymotrypsinogen ABos taurus (cattle)5
Beta-lactamaseEscherichia coli K-120.2083
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)2.6
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)5
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)5
Fatty-acid amide hydrolase 1Rattus norvegicus (Norway rat)0.15
Monoglyceride lipaseHomo sapiens (human)0.15

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Käsnänen, H; Leppänen, J; Minkkilä, A; Nevalainen, T; Poso, A; Saario, SM1
Fischer, DS; Gerards, T; Inglis, SR; Luxen, A; Schofield, CJ; Teller, N; Woon, EC; Zervosen, A1
Bürger, M; Görmer, K; Hall, D; Hedberg, C; Kondoh, Y; Martinez, NE; Mikoshiba, K; Osada, H; Ozaki, S; Rosin-Steiner, S; Shimizu, T; Tashiro, E; Vetter, IR; Waldmann, H; Watanabe, N; Zimmermann, TJ1

Other Studies

3 other study(ies) available for 1,1'-biphenyl-4-yl-boronic acid and benzo(b)thiophene-2-boronic acid

ArticleYear
Discovery of boronic acids as novel and potent inhibitors of fatty acid amide hydrolase.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Amidohydrolases; Boronic Acids; Dose-Response Relationship, Drug; Drug Discovery; Enzyme Inhibitors; Molecular Structure; Stereoisomerism; Structure-Activity Relationship

2008
Synthesis and evaluation of 3-(dihydroxyboryl)benzoic acids as D,D-carboxypeptidase R39 inhibitors.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Actinomycetales; Anti-Bacterial Agents; Bacterial Proteins; Benzoic Acid; Boronic Acids; Carboxypeptidases; Enzyme Inhibitors; Inhibitory Concentration 50; Structure-Activity Relationship

2009
Boron-based inhibitors of acyl protein thioesterases 1 and 2.
    Chembiochem : a European journal of chemical biology, 2013, Jan-02, Volume: 14, Issue:1

    Topics: Animals; Boron; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Humans; Lipoylation; Madin Darby Canine Kidney Cells; ras Proteins; Thiolester Hydrolases

2013