1-(5-isoquinolinesulfonyl)piperazine and h 89

1-(5-isoquinolinesulfonyl)piperazine has been researched along with h 89 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aherne, GW; Bavetsias, V; Berdini, V; Caldwell, J; Collins, I; Davies, TG; Davis, D; Donald, A; Fonseca, T; Garrett, MD; Hunter, LJ; McDonald, E; Rowlands, MG; Seavers, LC; Woodhead, SJ; Workman, P; Wyatt, PG1
Gerena, L; Geyer, JA; Keenan, SM; Waters, NC; Welsh, WJ; Woodard, CL1

Other Studies

2 other study(ies) available for 1-(5-isoquinolinesulfonyl)piperazine and h 89

ArticleYear
Structure-based design of isoquinoline-5-sulfonamide inhibitors of protein kinase B.
    Bioorganic & medicinal chemistry, 2006, Feb-15, Volume: 14, Issue:4

    Topics: Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Drug Design; Humans; Isoquinolines; Ligands; Molecular Structure; Protein Kinase C; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Structure-Activity Relationship; Sulfonamides

2006
Evaluation of broad spectrum protein kinase inhibitors to probe the architecture of the malarial cyclin dependent protein kinase Pfmrk.
    Bioorganic & medicinal chemistry letters, 2007, Sep-01, Volume: 17, Issue:17

    Topics: Animals; Binding Sites; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinases; Drug Evaluation, Preclinical; Enzyme Inhibitors; Inhibitory Concentration 50; Ligands; Malaria; Molecular Conformation; Naphthalenes; Plasmodium falciparum; Sulfonamides

2007