1-(5-isoquinolinesulfonyl)-2-methylpiperazine and trifluoperazine

1-(5-isoquinolinesulfonyl)-2-methylpiperazine has been researched along with trifluoperazine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19906 (16.67)18.7374
1990's26 (72.22)18.2507
2000's4 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hegemann, L; Kurscheid-Reich, D; Wohlfeil, S1
Dzwonczyk, S; Grover, GJ; Sargent, CA; Sleph, PG; Smith, MA1
Kennedy, AR; Umans, RS1
Imanaka, T; Itoga, H; Okawa, S; Suga, T; Watanabe, T1
Frizzell, RA; Worrell, RT1
Celada, A; Maki, RA1
Broquet, P; Carret, JP; Louisot, P; Peschard, MJ; Richard, M; Vignon, E1
Balda, MS; Cereijido, M; Contreras, RG; García-Sáinz, JA; González-Mariscal, L; Macias-Silva, M; Torres-Marquez, ME1
Smith, NC1
Abe, K; Katoh, N; Matsuno, K; Miyazaki, T; Sakurada, K; Tanaka, M; Uehara, Y1
Bevan, C; Kinne, RK; Theiss, C1
Manganel, M; Turner, RJ1
Brown, EJ; Gresham, HD; Mormol, JS; Zheleznyak, A1
Gabbay, RA; Lebovitz, HE; Siconolfi-Baez, L1
Petty, HR1
Dormer, RL; Goodchild, MC; McPherson, MA; Shori, DK1
Bright, EC; Colombani, PM; Hess, AD; Wells, M1
Devenyi, ZJ; Holian, A; Jordan, MK; Nguyen, HV1
Hoffman, MD; Wright, CD1
Chapekar, MS; Glazer, RI; Hartman, KD; Knode, MC1
Gukovskaya, AS; Pandol, SJ1
Sanderson, MJ; Schweitzer, ES; Wasterlain, CG1
Basu, U; Bennett, GS; Hollander, BA; Quintana, R; Rodriguez, R1
Bouzinba-Segard, H; Castagna, M; Fan, XT; Perderiset, M1
Dunlop, J; Ennis, C; Minchin, MC; Rossiter, J1
Ganapathi, R; Grabowski, D; Hidaka, H; Kawamura, K; Krivacic, K1
Fukushima, T; Hamada, T; Ono, M; Shibata, S; Shimazoe, T; Watanabe, A; Watanabe, S1
Castrucci, AM; da Silva, MA; Josefsson, L; Nery, LE1
Bernal, RM; Muñoz, ML; Santos, JI; Tovar, R1
Chen, J; Hoffman, BB; Hu, ZW; Lin, R1
Chen, YZ; Xing, BR; Zhu, BG1
Gadea, A; López-Colomé, AM1
Basavappa, S; Chang, CB; Huang, CC; Lim, PH; Liu, JY1
Dohovics, R; Hermann, A; Janáky, R; Oja, SS; Saransaari, P; Varga, V1
Fukushi, H; Morishima, Y; Shirasaki, Y; Takano, H1
Fu, XZ; Meng, FJ; Zhang, GY; Zhang, QG1

Other Studies

36 other study(ies) available for 1-(5-isoquinolinesulfonyl)-2-methylpiperazine and trifluoperazine

ArticleYear
Effect of protein kinase inhibitors on ACTH-stimulated aldosterone production in rat zona glomerulosa cells.
    Life sciences, 1992, Volume: 51, Issue:14

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenocorticotropic Hormone; Aldosterone; Alkaloids; Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Isoquinolines; Piperazines; Protein Kinase Inhibitors; Rats; Rats, Inbred Strains; Staurosporine; Trifluoperazine; Zona Glomerulosa

1992
Effect of calmodulin and protein kinase C inhibitors on globally ischemic rat hearts.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Analysis of Variance; Animals; Benzimidazoles; Calmodulin; Coronary Disease; Heart; In Vitro Techniques; Isoquinolines; L-Lactate Dehydrogenase; Male; Myocardial Contraction; Naphthalenes; Piperazines; Polycyclic Compounds; Polymyxin B; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine; Sulfonamides; Trifluoperazine

1992
Effects of activators and inhibitors of protein kinase C on X-ray induced malignant transformation in vitro.
    European journal of cancer (Oxford, England : 1990), 1992, Volume: 28A, Issue:4-5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antipain; Calcimycin; Cell Transformation, Neoplastic; Diglycerides; Enzyme Activation; Isoquinolines; Mice; Mice, Inbred C3H; Neoplasms, Radiation-Induced; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine; Trypsin Inhibitor, Bowman-Birk Soybean

1992
Involvement of calmodulin- and protein kinase C-related mechanism in an induction process of peroxisomal fatty acid oxidation-related enzymes by hypolipidemic peroxisome proliferators.
    Biochimica et biophysica acta, 1992, Apr-30, Volume: 1135, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bezafibrate; Body Weight; Calmodulin; Catalase; Cells, Cultured; Clofibrate; Diethylhexyl Phthalate; Electrophoresis, Polyacrylamide Gel; Isoquinolines; Kinetics; Liver; Male; Membrane Proteins; Microbodies; Molecular Weight; Organ Size; Oxidation-Reduction; Piperazines; Protein Kinase C; Pyrimidines; Rats; Rats, Inbred Strains; Reference Values; Trifluoperazine

1992
CaMKII mediates stimulation of chloride conductance by calcium in T84 cells.
    The American journal of physiology, 1991, Volume: 260, Issue:4 Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Line; Chloride Channels; Colon; Imidazoles; Ion Channels; Ionomycin; Isoquinolines; Kinetics; Membrane Proteins; Peptide Fragments; Phloretin; Piperazines; Protein Kinase C; Protein Kinases; Sphingosine; Trifluoperazine

1991
IFN-gamma induces the expression of the genes for MHC class II I-A beta and tumor necrosis factor through a protein kinase C-independent pathway.
    Journal of immunology (Baltimore, Md. : 1950), 1991, Jan-01, Volume: 146, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bone Marrow Cells; Calcimycin; Calmodulin; Gene Expression Regulation; Histocompatibility Antigens Class II; Interferon-gamma; Ionomycin; Isoquinolines; Macrophages; Major Histocompatibility Complex; Mice; Mice, Inbred DBA; Piperazines; Protein Kinase C; RNA, Messenger; Sphingosine; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine; Tumor Necrosis Factor-alpha

1991
Calmodulin-dependent collagenase and proteoglycanase activities in chondrocytes from human osteoarthritic cartilage.
    Biochemical and biophysical research communications, 1991, Feb-14, Volume: 174, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calmodulin; Cartilage, Articular; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Microbial Collagenase; Middle Aged; Osteoarthritis; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine

1991
Assembly and sealing of tight junctions: possible participation of G-proteins, phospholipase C, protein kinase C and calmodulin.
    The Journal of membrane biology, 1991, Volume: 122, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenylate Cyclase Toxin; Animals; Calcium; Calmodulin; Carbachol; Cells, Cultured; Electric Conductivity; Epithelial Cells; Epithelium; GTP-Binding Proteins; Intercellular Junctions; Isoquinolines; Kidney; Membrane Potentials; Neomycin; Pertussis Toxin; Piperazines; Polymyxin B; Protein Kinase C; Trifluoperazine; Type C Phospholipases; Virulence Factors, Bordetella

1991
A role for protein kinase C in the production of free oxygen radicals in response to Nippostrongylus brasiliensis.
    Parasitology research, 1991, Volume: 77, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Diglycerides; Enzyme Activation; Female; Free Radicals; Isoquinolines; Leukocytes; Nematode Infections; Nippostrongylus; Oxygen; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Trifluoperazine

1991
Phosphorylation of coagulation factor II by phospholipid/Ca(2+)-dependent protein kinase (protein kinase C).
    Biochemical and biophysical research communications, 1991, May-15, Volume: 176, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acids; Animals; Cattle; Gossypol; Humans; Isoquinolines; Kinetics; Palmitoylcarnitine; Phosphorylation; Piperazines; Protein Kinase C; Prothrombin; Spleen; Swine; Thrombin; Trifluoperazine

1991
Role of Ca2+ in sorbitol release from rat inner medullary collecting duct (IMCD) cells under hypoosmotic stress.
    Biochemical and biophysical research communications, 1990, Jul-31, Volume: 170, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calmodulin; Isoquinolines; Kidney Medulla; Kidney Tubules; Kidney Tubules, Collecting; Male; Osmotic Pressure; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Sorbitol; Trifluoperazine

1990
Agonist-induced activation of Na+/H+ exchange in rat parotid acinar cells is dependent on calcium but not on protein kinase C.
    The Journal of biological chemistry, 1990, Mar-15, Volume: 265, Issue:8

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Carbachol; Carrier Proteins; Diglycerides; Epinephrine; Isoquinolines; Male; Parotid Gland; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Sodium-Hydrogen Exchangers; Sulfonamides; Trifluoperazine

1990
Studies on the molecular mechanisms of human neutrophil Fc receptor-mediated phagocytosis. Evidence that a distinct pathway for activation of the respiratory burst results in reactive oxygen metabolite-dependent amplification of ingestion.
    The Journal of biological chemistry, 1990, May-15, Volume: 265, Issue:14

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Biological Factors; Bucladesine; Cholera Toxin; Colony-Stimulating Factors; Cytokines; Enzyme Activation; Granulocyte-Macrophage Colony-Stimulating Factor; Growth Substances; Humans; Immunoglobulin G; Isoquinolines; Neutrophils; Opsonin Proteins; Phagocytosis; Piperazines; Protein Kinase C; Receptors, Fc; Signal Transduction; Superoxides; Trifluoperazine; Tumor Necrosis Factor-alpha; Virulence Factors, Bordetella

1990
Calcium-dependent protein kinase activity is decreased in diabetic rat sciatic nerve.
    Endocrinology, 1990, Volume: 127, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Chromatography, Gel; Diabetes Mellitus, Experimental; Diglycerides; Enzyme Activation; Isoquinolines; Male; Phosphatidylserines; Phospholipids; Piperazines; Polymyxin B; Protein Kinase C; Rats; Rats, Inbred Strains; Sciatic Nerve; Sulfonamides; Trifluoperazine

1990
Regulation of RAW264 macrophage morphology and spreading: studies with protein kinase C activators, inhibitors and a cyclic AMP analog.
    Biochimica et biophysica acta, 1989, Aug-15, Volume: 1012, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bucladesine; Calcimycin; Cell Line; Cell Movement; Enzyme Activation; Isoquinolines; Kinetics; Macrophages; Mice; Microscopy, Electron, Scanning; Phenylephrine; Piperazines; Protein Kinase C; Sphingosine; Trifluoperazine

1989
Defective phosphorylation of a calmodulin-binding protein in cystic-fibrosis submandibular glands.
    The Biochemical journal, 1989, Oct-15, Volume: 263, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Adolescent; Adult; Calcineurin; Calmodulin-Binding Proteins; Cyclic AMP; Cystic Fibrosis; Enzyme Activation; Humans; Isoquinolines; Phosphoprotein Phosphatases; Phosphorylation; Piperazines; Protein Kinase C; Submandibular Gland; Trifluoperazine

1989
Drug-drug interaction between cyclosporine and agents affecting calcium-dependent lymphocyte proliferation.
    Transplantation proceedings, 1989, Volume: 21, Issue:1 Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium Channel Blockers; Cells, Cultured; Cyclosporins; Drug Interactions; Humans; Imidazoles; Isoquinolines; Lymphocyte Activation; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine; Verapamil

1989
Inhibition of macrophage activation by isoquinolinesulfonamides, phenothiazines, and a napthalenesulfonamide.
    Journal of cellular physiology, 1988, Volume: 137, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Fluphenazine; Guinea Pigs; Isoquinolines; Macrophage Activation; Macrophages; Male; Naphthalenes; Phenothiazines; Phosphatidylinositols; Piperazines; Protein Kinase Inhibitors; Pulmonary Alveoli; Sulfonamides; Superoxides; Trifluoperazine

1988
Comparison of the roles of calmodulin and protein kinase C in activation of the human neutrophil respiratory burst.
    Biochemical and biophysical research communications, 1987, Jan-15, Volume: 142, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calmodulin; Humans; Isoquinolines; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oxygen Consumption; Piperazines; Protein Kinase C; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate; Trifluoperazine

1987
Synergistic effect of retinoic acid and calcium ionophore A23187 on differentiation, c-myc expression, and membrane tyrosine kinase activity in human promyelocytic leukemia cell line HL-60.
    Molecular pharmacology, 1987, Volume: 31, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calmodulin; Cell Differentiation; Cell Line; Cell Membrane; Drug Synergism; Gene Expression Regulation; Hematopoiesis; Humans; Isoquinolines; Leukemia, Myeloid, Acute; Piperazines; Protein-Tyrosine Kinases; Proto-Oncogenes; RNA, Messenger; Sulfonamides; Tretinoin; Trifluoperazine

1987
Dual regulation of cGMP formation by calcium in pancreatic acinar cells.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Oxidoreductases; Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Cyclic GMP; Cytosol; Guanylate Cyclase; Guinea Pigs; Homeostasis; Imidazoles; In Vitro Techniques; Isoquinolines; Kinetics; Nitric Oxide Synthase; Pancreas; Piperazines; Protein Kinase C; Staurosporine; Sulfonamides; Trifluoperazine

1995
Inhibition of regulated catecholamine secretion from PC12 cells by the Ca2+/calmodulin kinase II inhibitor KN-62.
    Journal of cell science, 1995, Volume: 108 ( Pt 7)

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Isoquinolines; Kinetics; Membrane Potentials; Norepinephrine; PC12 Cells; Piperazines; Protein Kinase C; Rats; Trifluoperazine

1995
Differential sensitivity to inhibitors discriminates between two types of kinases responsible for in vivo phosphorylation of different sites in the carboxy-terminal tail of chicken neurofilament-M.
    Molecular and cellular neurosciences, 1994, Volume: 5, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Sequence; Animals; Carbazoles; Chick Embryo; Ganglia, Spinal; Indole Alkaloids; Isoquinolines; Lithium Chloride; Molecular Sequence Data; Neurofilament Proteins; Phosphorylation; Piperazines; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Sphingosine; Staurosporine; Trifluoperazine

1994
Synergy between phorbol esters and retinoic acid in inducing protein kinase C activation.
    Biochemical and biophysical research communications, 1994, Oct-14, Volume: 204, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Brain; Chlorpromazine; Cytosol; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Isoquinolines; Kinetics; Phosphorylation; Piperazines; Protein Binding; Protein Kinase C; Rats; Sulfonamides; Tetradecanoylphorbol Acetate; Tretinoin; Trifluoperazine; Tritium

1994
The effect of 3 calmodulin antagonists on K(+)-stimulated neurotransmitter release from rat cortical slices.
    Biochemical Society transactions, 1993, Volume: 21, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calmodulin; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Kinetics; Piperazines; Potassium; Rats; Serotonin; Sulfonamides; Trifluoperazine

1993
Cellular events involved in the sensitization of etoposide-resistant cells by inhibitors of calcium-calmodulin-dependent processes. Role for effects on apoptosis, DNA cleavable complex, and phosphorylation.
    Biochemical pharmacology, 1996, Dec-24, Volume: 52, Issue:12

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antineoplastic Agents; Apoptosis; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; DNA Topoisomerases, Type II; Drug Resistance; Enzyme Inhibitors; Etoposide; HL-60 Cells; Humans; Topoisomerase II Inhibitors; Trifluoperazine

1996
The involvement of calmodulin and Ca2+/calmodulin-dependent protein kinase II in the circadian rhythms controlled by the suprachiasmatic nucleus.
    Neuroscience letters, 1997, May-09, Volume: 227, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Analysis of Variance; Animals; Biomarkers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Circadian Rhythm; Drug Evaluation, Preclinical; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Nerve Tissue Proteins; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Suprachiasmatic Nucleus; Trifluoperazine

1997
Cellular signalling of PCH-induced pigment aggregation in the crustacean Macrobrachium potiuna erythrophores.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1997, Volume: 167, Issue:8

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Chromatophores; Colforsin; Cyclosporine; In Vitro Techniques; Invertebrate Hormones; Neomycin; Okadaic Acid; Oligopeptides; Palaemonidae; Pigments, Biological; Pyrrolidonecarboxylic Acid; Signal Transduction; Trifluoperazine

1997
Possible role of calmodulin in excystation of Giardia lamblia.
    Parasitology research, 1998, Volume: 84, Issue:9

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Calcium; Calmodulin; Child; Enzyme Activation; Feces; Giardia lamblia; Giardiasis; Humans; Protein Kinase C; Sulfonamides; Trifluoperazine

1998
alpha1-adrenergic receptor activation of c-fos expression in transfected rat-1 fibroblasts: role of Ca2+.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenergic alpha-1 Receptor Antagonists; Animals; Calcium; Calmodulin; Doxazosin; Egtazic Acid; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Genes, fos; Imidazoles; Kinetics; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-fos; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Sulfonamides; Transcription, Genetic; Trifluoperazine

1999
Effect of calcium on the uptake of glutamate by synaptosomes: possible involvement of two different mechanisms.
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:3-4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cerebral Cortex; Chelating Agents; Egtazic Acid; Electrophysiology; Enzyme Inhibitors; Glutamic Acid; Male; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Sodium Channels; Synaptosomes; Tetrodotoxin; Trifluoperazine

1999
Regulation of glycine transport in cultured Müller cells by Ca2+/calmodulin-dependent enzymes.
    Annals of the New York Academy of Sciences, 1999, Apr-30, Volume: 868

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Transport Systems, Neutral; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Carrier Proteins; Cell Line; Chick Embryo; Enzyme Inhibitors; Glycine Plasma Membrane Transport Proteins; Imidazoles; Kinetics; Sulfonamides; Trifluoperazine

1999
Effects of calcium, calmodulin, protein kinase C and protein tyrosine kinases on volume-activated taurine efflux in human erythroleukemia cells.
    Journal of cellular physiology, 2001, Volume: 189, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Biological Transport; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Size; Enzyme Inhibitors; Erythroid Precursor Cells; Humans; Hypotonic Solutions; K562 Cells; Kinetics; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Protein Kinase C; Protein-Tyrosine Kinases; Sulfonamides; Taurine; Trifluoperazine

2001
Regulation of glutamatergic neurotransmission in the striatum by presynaptic adenylyl cyclase-dependent processes.
    Neurochemistry international, 2003, Volume: 42, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Bucladesine; Calcium; Calmodulin; Corpus Striatum; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Feedback; Female; Glutamic Acid; Imidazoles; Imines; Isoenzymes; Isoproterenol; Isoquinolines; Kainic Acid; Male; Mice; N-Methylaspartate; Nerve Tissue Proteins; Propranolol; Receptors, Adrenergic, beta; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Presynaptic; Second Messenger Systems; Sulfonamides; Synaptic Transmission; Trifluoperazine

2003
Calmodulin and calmodulin-dependent kinase II mediate neuronal cell death induced by depolarization.
    Brain research, 2003, Feb-07, Volume: 962, Issue:1-2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Benzylamines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Death; Cells, Cultured; Cerebral Cortex; Egtazic Acid; Enzyme Inhibitors; Fetus; Kinetics; Membrane Potentials; Neurons; NG-Nitroarginine Methyl Ester; Nifedipine; Nitriles; Pyrethrins; Rats; Sulfonamides; Tacrolimus; Trifluoperazine; Veratridine

2003
NMDA receptor-mediated immediate Ser831 phosphorylation of GluR1 through CaMKIIalpha in rat hippocampus during early global ischemia.
    Neuroscience research, 2004, Volume: 48, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Analysis of Variance; Animals; Blotting, Western; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cytosol; Densitometry; Dopamine Antagonists; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Hippocampus; Hypoxia-Ischemia, Brain; Male; Nifedipine; Phosphorylation; Precipitin Tests; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Serine; Synaptosomes; Time Factors; Trifluoperazine

2004