1-(5-isoquinolinesulfonyl)-2-methylpiperazine and rottlerin

1-(5-isoquinolinesulfonyl)-2-methylpiperazine has been researched along with rottlerin in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (85.71)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
Alpini, G; Alvaro, D; Benedetti, A; Francis, H; Glaser, SS; Lesage, GD; Marucci, L; Marzioni, M; Patel, T; Phinizy, JL1
Alpini, G; Alvaro, D; Barbaro, B; Francis, H; Glaser, S; LeSage, G; Mancino, MG; Marzioni, M; Mauldin, J; Phinizy, JL; Rashid, S; Roskams, T; Stoica, G; Ueno, Y1
Blanquet, PR; Derer, P; Mariani, J1
Morgan, NG; Scarpello, JH; Smith, SA; Tadayyon, M; Welters, HJ1
Anderson, JM; Macewan, SR; McNally, AK1
Chieng, YC; Hoon, LS; Hsum, YW; Mooi, LY; Soo, KK; Yew, WT1

Other Studies

7 other study(ies) available for 1-(5-isoquinolinesulfonyl)-2-methylpiperazine and rottlerin

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Insulin inhibits secretin-induced ductal secretion by activation of PKC alpha and inhibition of PKA activity.
    Hepatology (Baltimore, Md.), 2002, Volume: 36, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Benzopyrans; Bile; Bile Canaliculi; Bile Ducts; Calcium; Chelating Agents; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Enzyme Inhibitors; Hypoglycemic Agents; Insulin; Isoenzymes; Male; Protein Kinase C; Protein Kinase C-alpha; Rats; Rats, Inbred F344; Receptor, Insulin; Secretin

2002
Dopaminergic inhibition of secretin-stimulated choleresis by increased PKC-gamma expression and decrease of PKA activity.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 284, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Animals; Benzophenanthridines; Benzopyrans; Bicarbonates; Bile; Bile Ducts, Intrahepatic; Chelating Agents; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Down-Regulation; Egtazic Acid; Enzyme Inhibitors; Epithelium; Liver; Male; Phenanthridines; Protein Kinase C; Quinolines; Rats; Rats, Inbred F344; Receptors, Dopamine D2; Secretin

2003
A calcium/calmodulin kinase pathway connects brain-derived neurotrophic factor to the cyclic AMP-responsive transcription factor in the rat hippocampus.
    Neuroscience, 2003, Volume: 118, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Androstadienes; Animals; Antibodies; Benzophenanthridines; Benzopyrans; Blotting, Western; Brain-Derived Neurotrophic Factor; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Carbazoles; Cell Nucleus; Chromones; Cyclic AMP Response Element-Binding Protein; Cytosol; Enzyme Inhibitors; Flavonoids; Hippocampus; Imidazoles; Immunohistochemistry; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Male; Morpholines; Naphthalenes; Phenanthridines; Phosphorylation; Precipitin Tests; Protein Serine-Threonine Kinases; Pyridines; Pyrroles; Rats; Signal Transduction; Time Factors; Tyrphostins; Wortmannin

2003
Evidence that protein kinase Cdelta is not required for palmitate-induced cytotoxicity in BRIN-BD11 beta-cells.
    Journal of molecular endocrinology, 2004, Volume: 32, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Apoptosis; Benzopyrans; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cell Survival; Cells, Cultured; Down-Regulation; Enzyme Inhibitors; Insulin; Insulin Secretion; Islets of Langerhans; Palmitates; Phorbol Esters; Phosphorylation; Protein Kinase C; Protein Kinase C-delta; Signal Transduction

2004
Foreign body-type multinucleated giant cell formation requires protein kinase C beta, delta, and zeta.
    Experimental and molecular pathology, 2008, Volume: 84, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Benzopyrans; Carbazoles; Cell Fusion; Cells, Cultured; Enzyme Inhibitors; Giant Cells, Foreign-Body; Humans; Indoles; Isoenzymes; Isoquinolines; Macrophages; Maleimides; Monocytes; Naphthalenes; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-delta; Signal Transduction

2008
Suppressive effect of maslinic acid on PMA-induced protein kinase C in human B-lymphoblastoid cells.
    Asian Pacific journal of cancer prevention : APJCP, 2012, Volume: 13, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Anticarcinogenic Agents; Benzopyrans; Cells, Cultured; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Isoenzymes; Oleanolic Acid; Precursor Cells, B-Lymphoid; Protein Kinase C; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Triterpenes; Ursolic Acid

2012