1-(5-isoquinolinesulfonyl)-2-methylpiperazine and niacinamide

1-(5-isoquinolinesulfonyl)-2-methylpiperazine has been researched along with niacinamide in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's1 (20.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Cohen, S; Li, W; Liu, X; Yanoff, M; Ye, X1
Jett, M; Yan, Z; Yang, DC1
Hirst, DG; Ruddock, MW1
Chou, AH; Hu, SH; Wang, HL; Wang, SS; Weng, YH; Yeh, TH1

Other Studies

5 other study(ies) available for 1-(5-isoquinolinesulfonyl)-2-methylpiperazine and niacinamide

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Cultured retinal capillary pericytes die by apoptosis after an abrupt fluctuation from high to low glucose levels: a comparative study with retinal capillary endothelial cells.
    Diabetologia, 1996, Volume: 39, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Bucladesine; Calcimycin; Capillaries; Cattle; Cell Survival; Cells, Cultured; Coculture Techniques; DNA; Endothelium, Vascular; Enzyme Inhibitors; Glucose; Isoquinolines; Kinetics; Microscopy, Electron; Muscle, Smooth, Vascular; Niacinamide; Piperazines; Retinal Vessels; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors

1996
Cholera toxin induces tumor necrosis factor alpha production in human monocytes.
    Molecular cell biology research communications : MCBRC, 1999, Volume: 2, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Diphosphate; Benzamides; Cells, Cultured; Cholera Toxin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Isoquinolines; Lymphocytes; Monocytes; Niacinamide; Poly(ADP-ribose) Polymerase Inhibitors; Protein Kinase C; Signal Transduction; Sphingosine; Sulfonamides; Transcription, Genetic; Tumor Necrosis Factor-alpha; Type C Phospholipases

1999
Nicotinamide relaxes vascular smooth muscle by inhibiting myosin light chain kinase-dependent signaling pathways: implications for anticancer efficacy.
    Oncology research, 2004, Volume: 14, Issue:10

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calmodulin; Chickens; Dose-Response Relationship, Drug; Male; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Niacinamide; Oxygen; Peptides; Phenylephrine; Phosphorylation; Rats; Rats, Wistar; Signal Transduction; Time Factors

2004
H1152 promotes the degradation of polyglutamine-expanded ataxin-3 or ataxin-7 independently of its ROCK-inhibiting effect and ameliorates mutant ataxin-3-induced neurodegeneration in the SCA3 transgenic mouse.
    Neuropharmacology, 2013, Volume: 70

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Ataxin-3; Ataxin-7; Brain; Dose-Response Relationship, Drug; Gene Expression; Humans; Indazoles; Mice; Mice, Transgenic; Mutation; Nerve Degeneration; Nerve Tissue Proteins; Neuroprotective Agents; Niacinamide; Nuclear Proteins; Peptides; Proteasome Endopeptidase Complex; Pyridines; rho-Associated Kinases; Transcription Factors

2013