1-(5-isoquinolinesulfonyl)-2-methylpiperazine and calcimycin
1-(5-isoquinolinesulfonyl)-2-methylpiperazine has been researched along with calcimycin in 135 studies
Research
Studies (135)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 36 (26.67) | 18.7374 |
1990's | 85 (62.96) | 18.2507 |
2000's | 13 (9.63) | 29.6817 |
2010's | 1 (0.74) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
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Hemmings, BA; Monard, D; Stone, SR; Suidan, HS | 1 |
Atluru, D; Atluru, S; Erickson, HH; McVey, DS; Olsen, SC | 1 |
Desai, SN; Letts, GL; Myers, CL; Schembri-King, J; Wallace, RW | 1 |
Bergstrand, H; Karabelas, K; Lundquist, B; Michelsen, P | 1 |
Bargon, J; Crystal, RG; Dalemans, W; Lecocq, JP; Pavirani, A; Trapnell, BC; Yoshimura, K | 1 |
Goto, S; Hagiwara, M; Hidaka, H; Hoshino, T; Hotta, T; Kobayashi, M; Murate, T; Saito, H | 1 |
Koide, Y; Miyachi, H; Sekiguchi, S; Shibata, T; Takemura, Y; Tukemura, Y | 1 |
Kennedy, AR; Umans, RS | 1 |
Ganguly, NK; Gorowara, S; Mahajan, RC; Walia, BN | 1 |
Goto, S; Hidaka, H; Kobayashi, M; Saito, H | 1 |
Calderwood, SK; Price, BD | 1 |
Fusamoto, H; Hayashi, N; Kamada, T; Kasahara, A; Katayama, K; Sasaki, Y; Takehara, T; Towata, T | 1 |
Brown, GE; Lanser, ME; Reed, EB | 1 |
Aragón, C; Casado, M; Giménez, C; Zafra, F | 1 |
Blanchard, LM; Larose, L; Morisset, J; Paquette, B | 1 |
Drexler, HG; Gignac, SM; Hoffbrand, AV; Pettit, GR | 1 |
Bonak, V; Casnellie, JE; Huang, CK; Laramee, GR | 1 |
Bahrami, LH; Lenhard, LW; Pandol, SJ; Perkins, PS | 1 |
Belosevic, M; Daniels, CW | 1 |
Hidaka, H; Hoshino, T; Mizutani, A; Shimizu, S; Yamane, T | 1 |
Casillas, T; Delicado, EG; Miras-Portugal, MT; Sen, RP | 1 |
Caron, L; Grose, JH; Landry, J; Lebel, M | 1 |
Caldwell, CW; Patterson, WP; Yesus, YW | 1 |
Celada, A; Maki, RA | 1 |
Coffee, KA; Cook, JA; Geisel, J; Halushka, PV; Wise, WC | 1 |
Asano, T; Hidaka, H; Ikegaki, I; Mochizuki, D; Satoh, S; Shibuya, M; Sugita, K; Suzuki, Y | 1 |
Smith, NC | 1 |
Ganguly, NK; Khullar, M; Khurana, S; Panigrahi, D; Walia, BN | 1 |
Brown, ML; Cohen, RA; Tesfamariam, B | 1 |
Bement, WM; Capco, DG | 1 |
Cottam, GL; Matsunaga, A; Miller, BC | 1 |
Conquer, J; Mahadevappa, VG | 1 |
Iwasaki, T; Miyata, S; Morita, S; Nagai, K; Shibata, R | 1 |
Ganguly, NK; Garg, UC; Goyal, J; Walia, BN | 1 |
Gimbrone, MA; Hrbolich, JK; Schafer, AI; Zavoico, GB | 1 |
Buschie, M; Drexler, HG; Gignac, SM; Hoffbrand, AV; Pettit, GR | 1 |
Gruenhaupt, D; Peterson, MW | 1 |
Iwata, K; Sasaki, Y | 1 |
Bevan, C; Kinne, RK; Theiss, C | 1 |
Crane, DL; Elliott, MS | 1 |
Manganel, M; Turner, RJ | 1 |
Chijiwa, T; Hagiwara, M; Hidaka, H; Mizutani, A; Terasawa, M; Tokumitsu, H | 1 |
el-Fakahany, EE; Lai, WS; Rogers, TB | 1 |
Brandwein, SR | 1 |
Chan, SO; Wong, SS; Yeung, DC | 1 |
Betts, WH; French, JK; Hurst, NP | 1 |
Pandol, SJ; Schoeffield, MS | 1 |
Conroy, MC; Kennedy, JA; Thueson, DO; Wright, CD | 1 |
Johnson, AL; Tilly, JL | 1 |
Grosman, N; Nielsen, KA | 1 |
Hansen, HS; Jensen, B; Linnebjerg, H | 1 |
Friedman, E; Wang, HY | 1 |
Fuse, I; Iwanaga, T; Tai, HH | 1 |
Hartzell, P; Jondal, M; McConkey, DJ; Orrenius, S | 1 |
Ishimura, Y; Kizaki, H; Muramatsu, J; Odaka, C; Tadakuma, T | 1 |
Kaever, V; Pfannkuche, HJ; Resch, K | 1 |
Halldórsson, H; Kjeld, M; Magnússon, MK; Thorgeirsson, G | 1 |
McMorris, FA; Shin, ML; Shirazi, Y | 1 |
Petty, HR | 1 |
Badwey, JA; Heyworth, PG; Karnovsky, ML | 1 |
Beattie, LL; Cragoe, EJ; Gerrard, JM; Israels, SJ; Lint, D; McNicol, A; Park, J | 1 |
Dandona, P; Jeremy, JY | 2 |
Badwey, JA; Horn, W; Karnovsky, MJ; Karnovsky, ML; Robinson, JM; Soberman, RJ | 1 |
Chik, CL; Ho, AK; Klein, DC | 1 |
Dandona, P; Khokher, MA | 1 |
Fujita, I; Minakami, S; Takeshige, K | 1 |
Maxeiner, B; Pfizenmaier, K; Scheurich, P; Thoma, B; Unglaub, R; Zugmaier, G | 1 |
Kuroki, T; Nose, K; Shibanuma, M | 1 |
el-Fakahany, EE; Lai, WS | 1 |
Ina, Y; Koide, Y; Nezu, N; Yoshida, TO | 1 |
Ikebuchi, H; Suzuki, K; Terao, T; Teshima, R | 1 |
Chapekar, MS; Glazer, RI; Hartman, KD; Knode, MC | 1 |
Daniel, LW; Parker, J; Waite, M | 1 |
Leung, PC; Wang, J | 1 |
Nachmias, VT; Yoshida, K | 1 |
Matsumoto, T; Sha'afi, RI; Tao, W | 1 |
Hoek, JB; Rubin, R; Thomas, AP | 1 |
Fuse, I; Tai, HH | 1 |
Christensen, SB; Fujiki, H; Hirasawa, N; Ohuchi, K; Sugawara, T; Sugimura, T; Tsurufuji, S; Watanabe, M | 1 |
Hogans, BB; Spivak, JL | 1 |
Hidaka, H; Kawamoto, S | 1 |
Craven, PA; DeRubertis, FR; Studer, RK | 1 |
Evans, DL; Jaso-Friedmann, L; Leary, JH | 1 |
Endo, T; Kumegawa, M; Takahashi, Y; Taketani, Y; Yamamoto, S | 1 |
Azuma, Y; Ishimura, Y; Kizaki, H; Onishi, Y; Suzuki, K | 1 |
Reich, H; Sei, Y | 1 |
Ganguly, NK; Kanwar, RK; Kumar, L; Panigrahi, D; Rakesh, J; Walia, BN | 1 |
Papadogiannakis, N | 1 |
Cazaux, CA; Cremaschi, GA; Gorelik, G; Sterin-Borda, L | 1 |
Audette, M; Bouillon, M | 1 |
Boyer, JL; Bruck, R; Nathanson, MH; Roelofsen, H | 1 |
Li, GC; Qian, DH; Tian, M; Zhang, JP | 1 |
Dobrovinskaya, OR; Eidus, LKh; Korystov, YN; Shaposhnikova, VV | 1 |
Andersen, CB; Hansen, AB | 1 |
Andersen, CB; Bouchelouche, PN; Giese, BN; Hansen, AB | 1 |
Mate, KE; Rodger, JC | 1 |
Arao, M; Chihara, K; Fukase, M; Sugimoto, T; Yamaguchi, T | 1 |
Baden, JM; Fujinaga, M; Hoffman, BB | 1 |
Arizono, K; Brady, FO; Peterson, KL | 1 |
Kelly, PT; Malenka, RC; Mauk, MD; Waxham, MN | 1 |
Maurer, JA; McKay, DB; Wenger, BW | 1 |
Amino, K; Fujimoto, T; Honda, Y; Takahashi, M | 1 |
Cohen, S; Li, W; Liu, X; Yanoff, M; Ye, X | 1 |
Hamada, M; Kannan, Y; Kimura, K; Moriyama, M; Musashi, M; Sakurada, K; Shiota, M; Sugano, T | 1 |
Bilski, JJ; Grazul-Bilska, AT; Kirsch, JD; Redmer, DA; Reynolds, LP | 1 |
Bäcker, A; Fandrey, J; Jelkmann, W; Kramer, HJ; Meyer-Lehnert, H; Vogel, V | 1 |
Atsumi, T; Hosoi, K; Kurihara, K; Shioda, Y; Sugita, K; Ueha, T | 1 |
Shimizu, T | 1 |
Ganguly, NK; Kaur, T; Singh, S; Verma, M | 1 |
Inagaki, N; Iwahashi, K; Kitai, H; Kuji, N; Nakatogawa, N; Suzuki, S; Yoshimura, Y | 1 |
Dhawan, V; Ganguly, NK; Kaur, T; Singh, S | 1 |
Eguchi, T; Ishida, H; Ishikawa, Y; Skowronski, MT | 1 |
Ganguly, NK; Gorowara, S; Sapru, S | 1 |
Hori, H; Minaguchi, H; Uemura, T | 1 |
Liu, L | 1 |
Su, JY; Toda, H | 1 |
Hayakawa, A; Nakashima, I; Okamoto, T; Tajiri, H; Yokoyama, I | 1 |
Bershadsky, AD; Berthier, C; Elbaum, M; Grosheva, I; Helfman, DM; Lachish-Zalait, A; Levy, ET; Riveline, D; Shtutman, M | 1 |
Ahmed-Choudhury, J; Coleman, R; Roma, MG | 1 |
Alam, T; Hamawy, MM; Knechtle, SJ; Manthei, ER; Tsuchida, M | 1 |
Howard, EW; Parizi, M; Tomasek, JJ | 1 |
Aikawa, R; Hayashi, D; Komuro, I; Kudoh, S; Mizukami, M; Nagai, R; Shibasaki, F; Shiojima, I; Toko, H; Yazaki, Y; Zhu, W; Zou, Y | 1 |
Davis, J; Schiebinger, R; Yingst, DR | 1 |
Boland, R; Buitrago, C; de Boland, AR; Morelli, S | 1 |
Miyata, Y; Nagano, M; Sato, S; Ui-Tei, K | 1 |
Bungard, D; Lytton, J; Wu, KD | 1 |
Abraham-Podgornik, A; Blankenstein, P; Bondzio, A; Risse, S | 1 |
Bilski, JJ; Grazul-Bilska, AT; Redmer, DA; Reynolds, LP | 1 |
Balaraman, S; Kapoor, P; Madhubala, R; Raj, VS; Saxena, S | 1 |
Ichikawa, A; Mikura, S; Satoh, N; Takasu, Y; Tanaka, S | 1 |
Grinkevich, LN; Lisachev, PD; Merkulova, TI | 1 |
Aikawa, T; Hirose, T; Matsumoto, I; Shimada, T | 1 |
Ark, M; Büyükafşar, K; Cnar, MG; Erol, A; Kubat, H; Tiftik, RN; Ulker, S | 1 |
Bolognesi, G; Bozzato, D; Di Virgilio, F; Ferrari, D; Gulinelli, S; Idzko, M; Pizzirani, C; Salaro, E; Vuerich, M | 1 |
Other Studies
135 other study(ies) available for 1-(5-isoquinolinesulfonyl)-2-methylpiperazine and calcimycin
Article | Year |
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Thrombin causes neurite retraction in neuronal cells through activation of cell surface receptors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Calcimycin; Cyclic AMP; Egtazic Acid; Isoquinolines; Mice; Neurites; Neuroblastoma; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Receptors, Cell Surface; Receptors, Thrombin; Staurosporine; Thrombin; Transcription, Genetic; Tumor Cells, Cultured | 1992 |
Inhibition of equine mononuclear cell proliferation and leukotriene B4 synthesis by a specific 5-lipoxygenase inhibitor, A-63162.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetamides; Animals; Calcimycin; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Horses; Indomethacin; Interleukin-2; Isoquinolines; Leukocytes, Mononuclear; Leukotriene B4; Lipoxygenase Inhibitors; Lymphocyte Activation; Phenyl Ethers; Phytohemagglutinins; Piperazines; Protein Kinase Inhibitors | 1992 |
Discriminatory effects of protein kinase inhibitors and calcium ionophore on endothelial ICAM-1 induction.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Calcimycin; Cell Adhesion Molecules; Cell Survival; Cytokines; Drug Synergism; Endothelium, Vascular; Humans; Intercellular Adhesion Molecule-1; Ionomycin; Isoquinolines; Lipopolysaccharides; Piperazines; Protein Biosynthesis; Protein Kinase Inhibitors; Staurosporine; Tetradecanoylphorbol Acetate | 1992 |
Modulation of human basophil histamine release by protein kinase C inhibitors differs with secretagogue and with inhibitor.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Basophils; Calcimycin; Glyceryl Ethers; Histamine Release; Humans; Indoles; Isoquinolines; Maleimides; Mannitol; Palmitoylcarnitine; Piperazines; Polymyxin B; Protein Kinase C; Sphingosine; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 1992 |
Expression of the cystic fibrosis transmembrane conductance regulator gene can be regulated by protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Cell Line; Colonic Neoplasms; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Activation; Gene Expression Regulation, Neoplastic; Humans; Isoquinolines; Kinetics; Membrane Proteins; Piperazines; Protein Kinase C; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1992 |
Thrombin-induced shape change in human megakaryoblastic leukemic cells, MEG-01, is mediated by protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Azepines; Calcimycin; Cell Size; Cytochalasin B; Humans; Isoquinolines; Megakaryocytes; Phorbol Esters; Piperazines; Protein Kinase C; Thrombin; Tumor Cells, Cultured | 1992 |
Effect of verapamil on the class I major histocompatibility complex antigen expression in K562 chronic myelogenous leukemia cells treated with recombinant human interferon-gamma.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antibodies, Monoclonal; Blotting, Northern; Calcimycin; Calmodulin; Cell Line; Egtazic Acid; Genes, MHC Class I; Genes, myc; Histocompatibility Antigens Class I; Humans; Interferon-gamma; Isoquinolines; Kinetics; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Piperazines; Protein Kinase Inhibitors; Recombinant Proteins; RNA, Neoplasm; Signal Transduction; Sulfonamides; Tumor Necrosis Factor-alpha; Verapamil | 1992 |
Effects of activators and inhibitors of protein kinase C on X-ray induced malignant transformation in vitro.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antipain; Calcimycin; Cell Transformation, Neoplastic; Diglycerides; Enzyme Activation; Isoquinolines; Mice; Mice, Inbred C3H; Neoplasms, Radiation-Induced; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine; Trypsin Inhibitor, Bowman-Birk Soybean | 1992 |
Study on the mechanism of Giardia lamblia induced diarrhoea in mice.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Biological Transport; Calcimycin; Calcium; Chlorides; Diarrhea; Giardia lamblia; Intestinal Mucosa; Isoquinolines; Mice; Piperazines; Protein Kinase C; Sodium; Tetradecanoylphorbol Acetate | 1992 |
[Shape change in human megakaryoblastic leukemia cells, MEG-01].
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actin Cytoskeleton; Calcimycin; Humans; Isoquinolines; Leukemia, Megakaryoblastic, Acute; Megakaryocytes; Microscopy, Electron; Piperazines; Protein Kinase C; Thrombin; Tissue Plasminogen Activator; Tumor Cells, Cultured | 1992 |
Gadd45 and Gadd153 messenger RNA levels are increased during hypoxia and after exposure of cells to agents which elevate the levels of the glucose-regulated proteins.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; DNA Damage; Endoplasmic Reticulum Chaperone BiP; HSP70 Heat-Shock Proteins; Hypoxia; Isoquinolines; Membrane Proteins; Mice; Piperazines; RNA, Messenger; Terpenes; Thapsigargin; Tunicamycin | 1992 |
Signal transduction pathways in the induction of HLA class I antigen expression on Huh 6 cells by interferon-gamma.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calmodulin; Carcinoma, Hepatocellular; Cell Line; Cyclic CMP; Histocompatibility Antigens Class I; Humans; Interferon-gamma; Isoquinolines; Liver Neoplasms; Piperazines; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1991 |
Neutrophil CR3 expression and specific granule exocytosis are controlled by different signal transduction pathways.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Azepines; Bucladesine; Calcimycin; Calcium; Calmodulin; Chlorpromazine; Exocytosis; Gelatinases; Gene Expression Regulation; Humans; In Vitro Techniques; Isoquinolines; Myosin-Light-Chain Kinase; N-Formylmethionine Leucyl-Phenylalanine; Nerve Tissue Proteins; Neutrophils; Pepsin A; Piperazines; Protein Kinase Inhibitors; Receptors, Complement; Receptors, Complement 3b; Signal Transduction; Tetanus Toxin; Up-Regulation | 1991 |
Activation of high-affinity uptake of glutamate by phorbol esters in primary glial cell cultures.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Binding, Competitive; Calcimycin; Cells, Cultured; Diglycerides; Dose-Response Relationship, Drug; Drug Synergism; Glutamates; Glutamic Acid; Isoquinolines; Kinetics; Neuroglia; Neurons; Piperazines; Tetradecanoylphorbol Acetate | 1991 |
Carbamylcholine and phorbol esters desensitize muscarinic receptors by different mechanisms in rat pancreatic acini.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amylases; Animals; Calcimycin; Carbachol; Dose-Response Relationship, Drug; Down-Regulation; Gallic Acid; Isoquinolines; Male; Pancreas; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Secretory Rate; Tetradecanoylphorbol Acetate | 1990 |
Synergistic action of calcium ionophore A23187 and protein kinase C activator bryostatin 1 on human B cell activation and proliferation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antibody Formation; B-Lymphocytes; Bryostatins; Calcimycin; Cell Cycle; Cyclosporins; DNA; Enzyme Activation; Humans; In Vitro Techniques; Isoquinolines; Lactones; Lymphocyte Activation; Macrolides; Piperazines; Protein Kinase C; RNA; Tetradecanoylphorbol Acetate | 1990 |
Protein tyrosine phosphorylation in rabbit peritoneal neutrophils.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aminoquinolines; Animals; Calcimycin; Calcium; Immunoblotting; Isoquinolines; Leukotriene B4; Molecular Weight; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Peritoneal Cavity; Phosphoproteins; Phosphorylation; Phosphotyrosine; Piperazines; Protein Kinase Inhibitors; Rabbits; Tetradecanoylphorbol Acetate; Tyrosine | 1990 |
Intracellular mechanisms involved in short-term regulation of net protein synthesis in pancreatic acini.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amylases; Animals; Calcimycin; Carbachol; DNA Probes; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzymes; Isoquinolines; Lipase; Nucleic Acid Hybridization; Pancreas; Pancreatic Elastase; Phosphatidylcholines; Phospholipases A; Phospholipases A2; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Sincalide; Staurosporine; Tetradecanoylphorbol Acetate | 1991 |
Phagocytosis of Giardia lamblia trophozoites by cytokine-activated macrophages.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bone Marrow Cells; Calcimycin; Cells, Cultured; Cytokines; Giardia lamblia; In Vitro Techniques; Interferon-gamma; Isoquinolines; Lipopolysaccharides; Macrophage Activation; Macrophages; Mice; Mice, Inbred C3H; Phagocytosis; Piperazines; Protein Kinase C; Recombinant Proteins; Tetradecanoylphorbol Acetate | 1992 |
Calcium ion regulates the release of lipase of Fusarium oxysporum.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calcium; Calmodulin; Fusarium; Isoquinolines; Kinetics; Lipase; Piperazines; Protein Kinase Inhibitors; Subcellular Fractions; Sulfonamides | 1991 |
Control of nucleoside transport in neural cells. Effect of protein kinase C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Adrenal Medulla; Animals; Biological Transport; Calcimycin; Caprylates; Cells, Cultured; Diglycerides; Dinucleoside Phosphates; Enzyme Activation; Ethers, Cyclic; Isoquinolines; Kinetics; Okadaic Acid; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate; Triglycerides | 1991 |
Prostacyclin secretion and specific intracellular protein phosphorylation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Bradykinin; Calcimycin; Cattle; Cells, Cultured; Endothelium, Vascular; Epoprostenol; Heat-Shock Proteins; Hot Temperature; Isoquinolines; Phosphoproteins; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Protein Processing, Post-Translational; Secretory Rate; Staurosporine; Tamoxifen; Tetradecanoylphorbol Acetate | 1991 |
Translocation of CD45RA in neutrophils.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antigens, Differentiation; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Cell Membrane; Flow Cytometry; Gene Expression Regulation; Histocompatibility Antigens; Humans; Isoantigens; Isoquinolines; Leukocyte Common Antigens; Neutrophils; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Up-Regulation | 1991 |
IFN-gamma induces the expression of the genes for MHC class II I-A beta and tumor necrosis factor through a protein kinase C-independent pathway.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bone Marrow Cells; Calcimycin; Calmodulin; Gene Expression Regulation; Histocompatibility Antigens Class II; Interferon-gamma; Ionomycin; Isoquinolines; Macrophages; Major Histocompatibility Complex; Mice; Mice, Inbred DBA; Piperazines; Protein Kinase C; RNA, Messenger; Sphingosine; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine; Tumor Necrosis Factor-alpha | 1991 |
Endotoxin-induced arachidonic acid metabolism requires de novo protein synthesis and protein kinase C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Arachidonic Acid; Arachidonic Acids; Bacterial Toxins; Calcimycin; Camptothecin; Cell Survival; Cells, Cultured; Cycloheximide; Dactinomycin; Endotoxins; Enterotoxins; Enzyme Activation; Isoquinolines; Macrophages; Male; Piperazines; Protein Biosynthesis; Protein Kinase C; Rats; Staurosporine; Tetradecanoylphorbol Acetate; Thromboxane B2 | 1991 |
Blockade of intracellular actions of calcium may protect against ischaemic damage to the gerbil brain.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Brain Ischemia; Calcimycin; Calcium Channel Blockers; Cell Death; Dogs; Gerbillinae; In Vitro Techniques; Isoquinolines; Male; Nicardipine; Rats; Rats, Inbred Strains; Vasoconstriction | 1991 |
A role for protein kinase C in the production of free oxygen radicals in response to Nippostrongylus brasiliensis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Diglycerides; Enzyme Activation; Female; Free Radicals; Isoquinolines; Leukocytes; Nematode Infections; Nippostrongylus; Oxygen; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Trifluoperazine | 1991 |
Studies on the mechanism of Salmonella typhimurium enterotoxin-induced diarrhoea.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Arachidonic Acid; Calcimycin; Calcium; Chlorides; Diarrhea; Enterotoxins; Indomethacin; Intestinal Mucosa; Intestine, Small; Isoquinolines; Male; Piperazines; Prostaglandins; Protein Kinase C; Rats; Rats, Inbred Strains; Salmonella typhimurium; Sodium; Tetradecanoylphorbol Acetate; Verapamil; Water-Electrolyte Balance | 1991 |
Elevated glucose impairs endothelium-dependent relaxation by activating protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetylcholine; Animals; Aorta; Calcimycin; Endothelium, Vascular; Enzyme Activation; Glucose; In Vitro Techniques; Isoquinolines; Piperazines; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Vasodilation | 1991 |
Protein kinase C acts downstream of calcium at entry into the first mitotic interphase of Xenopus laevis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Egtazic Acid; Exocytosis; Interphase; Isoquinolines; Oocytes; Piperazines; Protein Kinase C; Signal Transduction; Sphingosine; Sulfonamides; Tetradecanoylphorbol Acetate; Xenopus laevis | 1990 |
Pertussis toxin and H-7 distinguish mechanisms involved in eicosanoid release from lipopolysaccharide-primed macrophages. Eicosanoid release from lipopolysaccharide-primed macrophages.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Arachidonic Acids; Calcimycin; Cells, Cultured; Dinoprostone; Eicosanoids; Female; Isoquinolines; Lipopolysaccharides; Macrophage Activation; Macrophages; Mice; Mice, Inbred BALB C; Pertussis Toxin; Piperazines; SRS-A; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1990 |
Inhibition of protein kinase C by H-7 potentiates the release of oleic, linoleic and arachidonic acids in A23187-stimulated human neutrophils.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cells, Cultured; Fatty Acids; Humans; Isoquinolines; Linoleic Acid; Linoleic Acids; Neutrophils; Oleic Acid; Oleic Acids; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1990 |
Effects of H-7 (protein kinase inhibitor) and phorbol ester on aortic strips from spontaneously hypertensive rats.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Angiotensin II; Animals; Aorta, Thoracic; Calcimycin; Calcium; Dinoprost; Hypertension; In Vitro Techniques; Isoquinolines; Lanthanum; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phorbol Esters; Piperazines; Potassium Chloride; Protein Kinase Inhibitors; Rats; Rats, Inbred SHR; Rats, Inbred WKY | 1990 |
Differences between the mechanisms of action of heat-stable and heat-labile enterotoxins of Escherichia coli.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bacterial Toxins; Biological Transport, Active; Calcimycin; Calcium; Calmodulin; Chlorides; Enterotoxins; Escherichia coli; Escherichia coli Proteins; Ileum; Isoquinolines; Mice; Piperazines; Protein Kinase C; Sodium; Tetradecanoylphorbol Acetate | 1990 |
Enhancement of thrombin- and ionomycin-stimulated prostacyclin and platelet-activating factor production in cultured endothelial cells by a tumor-promoting phorbol ester.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Arachidonic Acids; Calcimycin; Cells, Cultured; Dinoprost; Dinoprostone; Endothelium, Vascular; Epoprostenol; Humans; Ionomycin; Isoquinolines; Phorbol Esters; Phospholipases A; Phospholipases A2; Piperazines; Platelet Activating Factor; Prostaglandin D2; Prostaglandins H; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Thrombin | 1990 |
Expression of proto-oncogene c-jun during differentiation of B-chronic lymphocytic leukemia.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Bryostatins; Calcimycin; Cell Differentiation; Enzyme Activation; Gene Expression; Humans; Isoquinolines; Kinetics; Lactones; Leukemia, Lymphocytic, Chronic, B-Cell; Macrolides; Piperazines; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogenes; RNA, Messenger; Second Messenger Systems; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1990 |
A23187 increases permeability of MDCK monolayers independent of phospholipase activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Cell Line; Cell Membrane Permeability; Choline; Dexamethasone; Dogs; Enzyme Activation; Epithelium; Inositol; Isoquinolines; Kidney; Kinetics; Lipolysis; Mannitol; Phorbol 12,13-Dibutyrate; Phospholipases; Phospholipases A; Phospholipases A2; Piperazines; Protein Kinase C; Quinacrine | 1990 |
Concanavalin A- and fetal-calf-serum-induced rounding and myosin light chain phosphorylation in cultured smooth muscle cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta; Blood; Calcimycin; Calcium; Cells, Cultured; Chickens; Concanavalin A; Culture Media; Cytochalasin B; Cytochalasins; Diltiazem; Egtazic Acid; Gizzard, Avian; Ionomycin; Isoquinolines; Kinetics; Muscle, Smooth; Muscle, Smooth, Vascular; Myosin Subfragments; Phosphorylation; Rabbits; Verapamil | 1990 |
Role of Ca2+ in sorbitol release from rat inner medullary collecting duct (IMCD) cells under hypoosmotic stress.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calmodulin; Isoquinolines; Kidney Medulla; Kidney Tubules; Kidney Tubules, Collecting; Male; Osmotic Pressure; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Sorbitol; Trifluoperazine | 1990 |
Protein kinase C modulation of queuine uptake in cultured human fibroblasts.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Calcimycin; Cells, Cultured; Diglycerides; Enzyme Activation; Fibroblasts; Growth Substances; Guanine; Humans; In Vitro Techniques; Isoquinolines; Male; Phorbol Esters; Phosphatidylserines; Piperazines; Protein Kinase C; Sphingosine; Staurosporine | 1990 |
Agonist-induced activation of Na+/H+ exchange in rat parotid acinar cells is dependent on calcium but not on protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Carbachol; Carrier Proteins; Diglycerides; Epinephrine; Isoquinolines; Male; Parotid Gland; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Sodium-Hydrogen Exchangers; Sulfonamides; Trifluoperazine | 1990 |
KN-62, 1-[N,O-bis(5-isoquinolinesulfonyl)-N-methyl-L-tyrosyl]-4-phenylpiperazi ne, a specific inhibitor of Ca2+/calmodulin-dependent protein kinase II.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Binding Sites; Binding, Competitive; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Chickens; Chromatography, Affinity; Cyclic AMP; Gizzard, Avian; Isoquinolines; Kinetics; Myosin-Light-Chain Kinase; Myosins; Pheochromocytoma; Phosphorylation; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Rats; Tumor Cells, Cultured | 1990 |
Protein kinase C is involved in desensitization of muscarinic receptors induced by phorbol esters but not by receptor agonists.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carbachol; Cyclic GMP; Down-Regulation; Isoquinolines; Mice; N-Methylscopolamine; Neuroblastoma; Parasympathomimetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Receptors, Muscarinic; Scopolamine Derivatives; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Differential regulation of soluble interleukin 1 release and membrane expression by pharmacologic agents.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antibodies; Calcimycin; Calmodulin; Cell Membrane; Diglycerides; Dinoprostone; In Vitro Techniques; Interleukin-1; Isoquinolines; L-Lactate Dehydrogenase; Leukotriene B4; Macrophages; Mice; Mice, Inbred C3H; Nucleotides, Cyclic; Piperazines; Protein Kinase C; Solubility; Sulfonamides; Thymus Gland | 1990 |
Regulation of Ki-ras expression in Reuber H35 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bucladesine; Calcimycin; Calcium; Cell Line; Diglycerides; DNA Probes; Egtazic Acid; Gene Expression Regulation, Neoplastic; Genes, ras; Glucagon; Isoquinolines; Kinetics; Liver Neoplasms, Experimental; Piperazines; Protein Kinase Inhibitors; Rats; RNA, Neoplasm; Tetradecanoylphorbol Acetate; Verapamil | 1990 |
Phorbol 12-myristate 13-acetate, A23187 and L-adrenaline inhibit phospholipid methylation in human monocytes and lymphocytes. Inhibition is independent of oxyradical production and phospholipid hydrolysis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Epinephrine; Free Radicals; Humans; Hydrolysis; Isoquinolines; Lymphocytes; Methylation; Monocytes; Phosphatidylcholines; Phosphatidylethanolamines; Phospholipids; Piperazines; Protein Kinase Inhibitors; S-Adenosylmethionine; Sodium Fluoride; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1990 |
1,2-Diacylglycerol, protein kinase C, and pancreatic enzyme secretion.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amylases; Animals; Arachidonic Acid; Arachidonic Acids; Bombesin; Calcimycin; Carbachol; Dibutyryl Cyclic GMP; Diglycerides; Glycerides; Guinea Pigs; In Vitro Techniques; Isoquinolines; Kinetics; Pancreas; Piperazines; Protein Kinase C; Sincalide; Tetradecanoylphorbol Acetate; Tetragastrin | 1986 |
Specific inhibition of phorbol ester and DiC8-induced histamine release from human basophils by the protein kinase C inhibitors, H-7 and H-9.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Basophils; Calcimycin; Calmodulin; Diglycerides; Glycerides; Histamine Release; Humans; Immunoglobulin E; In Vitro Techniques; Isoquinolines; Kinetics; Perphenazine; Piperazines; Protein Kinase C; Sulfonamides; Tetradecanoylphorbol Acetate | 1987 |
Effects of a phorbol ester, a calcium ionophore, and 3',5'-adenosine monophosphate production on hen granulosa cell plasminogen activator activity.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 1-Methyl-3-isobutylxanthine; Animals; Calcimycin; Chickens; Cyclic AMP; Cycloheximide; Dactinomycin; Female; Granulosa Cells; In Vitro Techniques; Isoquinolines; L-Lactate Dehydrogenase; Luteinizing Hormone; Piperazines; Plasminogen Activators; Progesterone; Protein Kinase C; Sheep; Tetradecanoylphorbol Acetate | 1988 |
The influence of tetradecanoyl-phorbol-acetate (TPA) on histamine release from isolated rat mast cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Diglycerides; Histamine Release; Isoquinolines; Male; Mast Cells; Piperazines; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1988 |
Inhibition by amiloride and by Na+-depletion of A23187-stimulated arachidonic acid and histamine release from rat mast cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amiloride; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Carrier Proteins; Histamine Release; In Vitro Techniques; Isoquinolines; Mast Cells; Piperazines; Protein Kinase C; Rats; Sodium; Sodium-Hydrogen Exchangers; Sphingosine | 1988 |
Effect of age on brain cortical protein kinase C and its mediation of 5-hydroxytryptamine release.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aging; Animals; Calcimycin; Calcium; Cerebral Cortex; Isoquinolines; Piperazines; Protein Kinase C; Rats; Rats, Inbred F344; Serotonin; Tetradecanoylphorbol Acetate | 1989 |
Phorbol ester, 1,2-diacylglycerol, and collagen induce inhibition of arachidonic acid incorporation into phospholipids in human platelets.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 1-Acylglycerophosphocholine O-Acyltransferase; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcimycin; Coenzyme A Ligases; Collagen; Diglycerides; Enzyme Activation; Glycerides; Isoquinolines; Phospholipids; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate; Thromboxane B2 | 1989 |
Inhibition of DNA fragmentation in thymocytes and isolated thymocyte nuclei by agents that stimulate protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Cell Nucleus; Cells, Cultured; Cytosol; DNA; Isoquinolines; Kinetics; Male; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thymus Gland | 1989 |
Activation of a suicide process of thymocytes through DNA fragmentation by calcium ionophores and phorbol esters.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Cell Survival; Cycloheximide; Dactinomycin; DNA Damage; Isoquinolines; Lectins; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Peanut Agglutinin; Phenotype; Piperazines; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1989 |
Modulation of calcium-induced eicosanoid synthesis in mouse peritoneal macrophages by protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Dinoprostone; Fatty Acids, Unsaturated; In Vitro Techniques; Isoquinolines; Macrophages; Mice; Mice, Inbred DBA; Piperazines; Protein Kinase C; SRS-A; Tetradecanoylphorbol Acetate | 1989 |
Endothelial inositol phosphate generation and prostacyclin production in response to G-protein activation by AlF4-.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 6-Ketoprostaglandin F1 alpha; Aluminum; Aluminum Compounds; Arachidonic Acids; Calcimycin; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Endothelium, Vascular; Epoprostenol; Female; Fluorides; Fluorine; GTP-Binding Proteins; Humans; Inositol Phosphates; Isoquinolines; Kinetics; Pertussis Toxin; Piperazines; Pregnancy; Protein Kinase C; Signal Transduction; Sodium Fluoride; Tetradecanoylphorbol Acetate; Umbilical Veins; Virulence Factors, Bordetella | 1989 |
Arachidonic acid mobilization and phosphoinositide turnover by the terminal complement complex, C5b-9, in rat oligodendrocyte x C6 glioma cell hybrids.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Clone Cells; Complement Membrane Attack Complex; Complement System Proteins; Glioma; Humans; Hybrid Cells; Isoquinolines; Neuroglia; Oligodendroglia; Phosphatidylinositols; Piperazines; Protein Kinase C; Quinacrine; Rats | 1989 |
Regulation of RAW264 macrophage morphology and spreading: studies with protein kinase C activators, inhibitors and a cyclic AMP analog.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bucladesine; Calcimycin; Cell Line; Cell Movement; Enzyme Activation; Isoquinolines; Kinetics; Macrophages; Mice; Microscopy, Electron, Scanning; Phenylephrine; Piperazines; Protein Kinase C; Sphingosine; Trifluoperazine | 1989 |
Protein phosphorylation associated with synergistic stimulation of neutrophils.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Diterpenes; Drug Synergism; Guinea Pigs; Hydroxyeicosatetraenoic Acids; Isoquinolines; Molecular Weight; Neutrophils; Phosphoproteins; Phosphorus Radioisotopes; Phosphorylation; Piperazines; Sulfonamides; Superoxides; Terpenes | 1989 |
A role for protein kinase C in the membrane fusion necessary for platelet granule secretion.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amiloride; Blood Platelets; Calcimycin; Carrier Proteins; Cytoplasmic Granules; Diglycerides; Humans; In Vitro Techniques; Isoquinolines; Membrane Fusion; Membrane Potentials; Phosphoproteins; Piperazines; Platelet Aggregation; Protein Kinase C; Sodium-Hydrogen Exchangers; Sphingosine; Tetradecanoylphorbol Acetate | 1989 |
Fluoride but not phorbol esters stimulate rat urinary bladder prostanoid synthesis: investigations into the roles of G proteins and protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Atropine; Bucladesine; Calcimycin; Carbachol; Fluorides; GTP-Binding Proteins; Isoquinolines; Nifedipine; Phorbol Esters; Piperazines; Prostaglandins; Protein Kinase C; Protein Kinase Inhibitors; Rats; Rats, Inbred Strains; Urinary Bladder; Verapamil | 1987 |
Synergistic stimulation of neutrophils. Possible involvement of 5-hydroxy-6,8,11,14-eicosatetraenoate in superoxide release.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Cations, Divalent; Drug Synergism; Guinea Pigs; Hydroxyeicosatetraenoic Acids; Isoquinolines; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Sphingosine; Sulfonamides; Superoxides | 1988 |
Effects of protein kinase inhibitor (1-(5-isoquinolinesulfonyl)-2-methylpiperazine (H7) on protein kinase C activity and adrenergic stimulation of cAMP and cGMP in rat pinealocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Cyclic AMP; Cyclic GMP; Female; In Vitro Techniques; Isoproterenol; Isoquinolines; Norepinephrine; Pineal Gland; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Adrenergic | 1988 |
The effect of polyunsaturated fatty acids on rat adipocyte lipogenesis: the role of protein kinase C, calcium and calmodulin.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adipose Tissue; alpha-Linolenic Acid; Animals; Calcimycin; Calcium; Calmodulin; Cells, Cultured; Insulin; Isoquinolines; Linolenic Acids; Lipids; Male; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Verapamil | 1988 |
Inhibition of neutrophil superoxide formation by 1-(5-isoquinolinesulfonyl)-2-methylpiperazine (H-7), and inhibitor of protein kinase-C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Cytoplasm; Humans; Isoquinolines; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphoproteins; Phosphorylation; Piperazines; Protein Kinase C; Superoxides; Tetradecanoylphorbol Acetate | 1986 |
Rapid modulation of tumor necrosis factor membrane receptors by activators of protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Cells, Cultured; Diglycerides; Glycoproteins; Humans; Isoquinolines; Lymphocyte Activation; Piperazines; Protein Kinase C; Receptors, Cell Surface; Receptors, Tumor Necrosis Factor; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1986 |
Inhibition of proto-oncogene c-fos transcription by inhibitors of protein kinase C and ion transport.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Amiloride; Aminopyridines; Biological Transport, Active; Calcimycin; Humans; Isoquinolines; Phorbol Esters; Piperazines; Potassium; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogenes; Quinidine; RNA, Messenger; Sodium; Tetraethylammonium Compounds; Transcription, Genetic | 1987 |
Phorbol ester-induced inhibition of cyclic GMP formation mediated by muscarinic receptors in murine neuroblastoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carbachol; Cell Line; Cyclic GMP; Dose-Response Relationship, Drug; Histamine; Isoquinolines; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Piperazines; Receptors, Muscarinic; Tetradecanoylphorbol Acetate | 1987 |
Regulation of HLA class II antigen expression: intracellular signaling molecules responsible for the regulation by IFN-gamma and cross-linking of Fc receptors in HL-60 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antigens, Neoplasm; Calcimycin; Calcium; Calmodulin; Cell Line; Cyclic AMP; Gene Expression Regulation; Histocompatibility Antigens Class II; Humans; Immunoglobulin G; Interferon-gamma; Isoquinolines; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Protein Kinase C; Receptors, Fc; Recombinant Proteins; Sulfonamides; Tetradecanoylphorbol Acetate | 1987 |
Possible involvement of phosphorylation of a 36,000-dalton protein of rat basophilic leukemia (RBL-2H3) cell membranes in serotonin release.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Basophils; Calcimycin; Cell Membrane; Diglycerides; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Isoquinolines; Leukemia, Experimental; Molecular Weight; Phosphoproteins; Phosphorylation; Piperazines; Rats; Serotonin; Tetradecanoylphorbol Acetate | 1986 |
Synergistic effect of retinoic acid and calcium ionophore A23187 on differentiation, c-myc expression, and membrane tyrosine kinase activity in human promyelocytic leukemia cell line HL-60.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calmodulin; Cell Differentiation; Cell Line; Cell Membrane; Drug Synergism; Gene Expression Regulation; Hematopoiesis; Humans; Isoquinolines; Leukemia, Myeloid, Acute; Piperazines; Protein-Tyrosine Kinases; Proto-Oncogenes; RNA, Messenger; Sulfonamides; Tretinoin; Trifluoperazine | 1987 |
Evidence of protein kinase C involvement in phorbol diester-stimulated arachidonic acid release and prostaglandin synthesis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Indomethacin; Isoquinolines; Kidney; Lysophosphatidylcholines; Molecular Weight; Phospholipid Ethers; Phosphorylation; Piperazines; Prostaglandins; Protein Kinase C; Tetradecanoylphorbol Acetate | 1987 |
The role of the diacylglycerol-protein kinase C system in mediating adrenoceptor-prostacyclin synthesis coupling in the rat aorta.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta, Thoracic; Calcimycin; Calcium; Calcium Channel Blockers; Diglycerides; Epinephrine; Epoprostenol; Glycerides; In Vitro Techniques; Isoquinolines; Male; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Adrenergic | 1987 |
Role of protein kinase C in luteinizing hormone-releasing hormone (LHRH)-stimulated progesterone production in rat granulosa cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Female; Gonadotropin-Releasing Hormone; Granulosa Cells; In Vitro Techniques; Isoquinolines; Kinetics; Phorbol Esters; Piperazines; Progesterone; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1987 |
Phorbol ester stimulates calcium sequestration in saponized human platelets.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Diphosphate; Alprostadil; Benzofurans; Biological Transport, Active; Blood Platelets; Calcimycin; Calcium; Calcium Radioisotopes; Chelating Agents; Fura-2; Humans; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoquinolines; Kinetics; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate; Thrombin | 1987 |
Demonstration of calcium-dependent phospholipase A2 activity in membrane preparation of rabbit neutrophils. Absence of activation by fMet-Leu-Phe, phorbol 12-myristate 13-acetate and A-kinase.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Cell Membrane; Enzyme Activation; In Vitro Techniques; Isoquinolines; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phospholipases; Phospholipases A; Phospholipases A2; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Rabbits; Tetradecanoylphorbol Acetate | 1988 |
Ethanol-induced phospholipase C activation is inhibited by phorbol esters in isolated hepatocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aminoquinolines; Animals; Calcimycin; Diglycerides; Enzyme Activation; Ethanol; Fluorescent Dyes; Isoquinolines; Liver; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1988 |
Does protein kinase C activation mediate thrombin-induced arachidonate release in human platelets?
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcimycin; Calcium; Enzyme Activation; Gallic Acid; Humans; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoquinolines; Piperazines; Protein Kinase C; Sulfonamides; Tetradecanoylphorbol Acetate; Thrombin; Thromboxane B2 | 1988 |
Analysis of the stimulative effect of thapsigargin, a non-TPA-type tumour promoter, on arachidonic acid metabolism in rat peritoneal macrophages.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Carcinogens; Cytoplasm; In Vitro Techniques; Isoquinolines; Lyngbya Toxins; Macrophages; Male; N-Formylmethionine Leucyl-Phenylalanine; Peritoneal Cavity; Piperazines; Plant Extracts; Protein Kinase Inhibitors; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thapsigargin | 1988 |
Tumor-promoting phorbol esters stimulate the proliferation of interleukin-3 dependent cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Cell Division; Cell Survival; Colony-Stimulating Factors; Enzyme Activation; Granulocyte-Macrophage Colony-Stimulating Factor; Growth Substances; Interleukin-3; Isoquinolines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
1-(5-Isoquinolinesulfonyl)-2-methylpiperazine (H-7) is a selective inhibitor of protein kinase C in rabbit platelets.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Blood Platelets; Blood Proteins; Calcimycin; Calcium; Calmodulin; Isoquinolines; Phosphorylation; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Rabbits; Tetradecanoylphorbol Acetate | 1984 |
Impaired nitric oxide-dependent cyclic guanosine monophosphate generation in glomeruli from diabetic rats. Evidence for protein kinase C-mediated suppression of the cholinergic response.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 1-Methyl-3-isobutylxanthine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alkaloids; Amino Acid Oxidoreductases; Animals; Arginine; Calcimycin; Carbachol; Cyclic GMP; Diabetes Mellitus, Experimental; Female; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Isoquinolines; Kidney Glomerulus; Kinetics; Membrane Proteins; Myristoylated Alanine-Rich C Kinase Substrate; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Phosphates; Phosphorylation; Piperazines; Prostaglandin Endoperoxides, Synthetic; Protein Kinase C; Proteins; Rats; Rats, Sprague-Dawley; Staurosporine; Thromboxane A2 | 1994 |
Pathways of signaling in nonspecific cytotoxic cells: effects of protein kinase and phosphatase inhibitors and evidence for membrane tyrosine phosphorylation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Catfishes; Cell Membrane; Cytotoxicity, Immunologic; Female; Immunity, Cellular; Isoquinolines; Male; Phosphoprotein Phosphatases; Phosphotyrosine; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Signal Transduction; Sulfonamides; Tyrosine | 1994 |
Studies on the induction of cyclooxygenase isozymes by various prostaglandins in mouse osteoblastic cell line with reference to signal transduction pathways.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alprostadil; Animals; Base Sequence; Calcimycin; Cell Line; Cycloheximide; Dexamethasone; Enzyme Induction; Iloprost; Isoenzymes; Isoquinolines; Mice; Molecular Sequence Data; Piperazines; Prostaglandin-Endoperoxide Synthases; Tetradecanoylphorbol Acetate | 1994 |
Biphasic effect of staurosporine on thymocyte apoptosis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Apoptosis; Bucladesine; Calcimycin; Carbazoles; Carcinogens; Cells, Cultured; DNA; DNA Damage; Dose-Response Relationship, Drug; Indole Alkaloids; Isoquinolines; Male; Mice; Mice, Inbred BALB C; Piperazines; Protein Kinase Inhibitors; Radiation-Sensitizing Agents; Staurosporine; Tetradecanoylphorbol Acetate; Thymus Gland; Time Factors | 1995 |
Thapsigargin induces IL-2 receptor alpha-chain in human peripheral and Jurkat T cells via a protein kinase C-independent mechanism.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Base Sequence; Calcimycin; Calcium; Calcium-Transporting ATPases; Cholera Toxin; Colforsin; Drug Synergism; Gene Expression Regulation; Gene Expression Regulation, Leukemic; Humans; Hydroquinones; Isoquinolines; Leukemia-Lymphoma, Adult T-Cell; Molecular Sequence Data; Neoplasm Proteins; NF-kappa B; Piperazines; Protein Kinase C; Receptors, Interleukin-2; RNA, Messenger; RNA, Neoplasm; Signal Transduction; Staurosporine; T-Lymphocytes; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin | 1995 |
Calcium and protein kinase C play an important role in Campylobacter jejuni-induced changes in Na+ and Cl- transport in rat ileum in vitro.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calmodulin; Campylobacter Infections; Campylobacter jejuni; Chlorides; Cyclic AMP; Dantrolene; Diarrhea; Enzyme Activation; Ileum; In Vitro Techniques; Ion Transport; Isoquinolines; Male; Piperazines; Protein Kinase C; Rats; Rats, Wistar; Sodium; Tetradecanoylphorbol Acetate; Verapamil | 1995 |
(-)-Indolactam V-induced mitogenesis in human fetal/neonatal and adult T cells: lower response of neonatal cells and possible regulatory role of monocytes in protein kinase C-mediated pathways.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Fetus; Humans; In Vitro Techniques; Indoles; Infant, Newborn; Isoquinolines; Lactams; Lymphocyte Activation; Monocytes; Phytohemagglutinins; Piperazines; Protein Kinase C; Receptors, Antigen, T-Cell; Signal Transduction; T-Lymphocytes | 1995 |
Down-regulation of beta-adrenergic receptors induced by mitogen activation of intracellular signaling events in lymphocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Concanavalin A; Cyclic AMP; Down-Regulation; Genistein; In Vitro Techniques; Interleukin-2; Intracellular Fluid; Isoflavones; Isoquinolines; Lymphocyte Activation; Mice; Mice, Inbred BALB C; Neuroimmunomodulation; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Receptors, Adrenergic, beta; Signal Transduction; Sulfonamides; T-Lymphocytes | 1995 |
Retinoic acid-stimulated intercellular adhesion molecule-1 expression on SK-N-SH cells: calcium/calmodulin-dependent pathway.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Adhesion Molecules; Enzyme Activation; Humans; Imidazoles; Intercellular Adhesion Molecule-1; Interferon-gamma; Isoquinolines; Neuroblastoma; Piperazines; Protein Kinase C; Sulfonamides; Terpenes; Thapsigargin; Tretinoin; Tumor Cells, Cultured; Up-Regulation | 1994 |
Effects of protein kinase C and cytosolic Ca2+ on exocytosis in the isolated perfused rat liver.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bile; Calcimycin; Calcium; Cytosol; Exocytosis; Horseradish Peroxidase; Hydroquinones; In Vitro Techniques; Isoquinolines; Liver; Male; Perfusion; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Vasopressins | 1994 |
[Inhibitory effects of protein kinase C inhibitor and calmodulin antagonist on tumor necrosis factor production by mouse macrophages].
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calmodulin; Female; Isoquinolines; Lipopolysaccharides; Macrophages, Peritoneal; Mice; Mice, Inbred ICR; Piperazines; Protein Kinase C; Sulfonamides; Tumor Necrosis Factor-alpha | 1993 |
Dependence of thymocyte apoptosis on protein kinase C and phospholipase A2.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Calcimycin; Concanavalin A; DNA; Enzyme Activation; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Phospholipases A; Phospholipases A2; Piperazines; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Thymus Gland | 1994 |
Comparison of the effects of tumour necrosis factor alpha stimulation and phorbol ester treatment on the immunocytochemical staining of intercellular adhesion molecule 1 in human renal carcinoma cell cultures.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Calcimycin; Carcinoma, Renal Cell; Cell Adhesion Molecules; Humans; Immunoenzyme Techniques; Intercellular Adhesion Molecule-1; Isoquinolines; Kidney Neoplasms; Piperazines; Protein Kinase C; Signal Transduction; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1993 |
Role of protein kinase C during interferon-gamma- and phorbol ester-stimulated immunocytochemical expression of ICAM-1 in human renal carcinoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Antigens, CD; Calcimycin; Carcinoma, Renal Cell; Cell Adhesion Molecules; Dose-Response Relationship, Drug; Humans; Immunohistochemistry; Intercellular Adhesion Molecule-1; Interferon-gamma; Isoquinolines; Kidney Neoplasms; Piperazines; Protein Kinase C; Recombinant Proteins; Signal Transduction; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1993 |
Role of diacylglycerols and calcium in the marsupial acrosome reaction.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acrosome; Animals; Calcimycin; Calcium; Cells, Cultured; Dexamethasone; Diglycerides; Exocytosis; Isoquinolines; Male; Marsupialia; Osmolar Concentration; Phorbol Esters; Piperazines; Protein Kinase Inhibitors; Semen; Spermatozoa | 1993 |
Protein kinase C is crucial for the stimulation of sodium-dependent phosphate transport by parathyroid hormone-related peptide in osteoblast-like cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenylyl Cyclases; Animals; Biological Transport; Bone Neoplasms; Calcimycin; Calcium; Cell Line; Colforsin; Cytosol; Humans; Isoquinolines; Kinetics; Osteoblasts; Osteosarcoma; Parathyroid Hormone; Parathyroid Hormone-Related Protein; Phosphates; Piperazines; Protein Kinase C; Proteins; Rats; Sodium; Tetradecanoylphorbol Acetate | 1994 |
Receptor subtype and intracellular signal transduction pathway associated with situs inversus induced by alpha 1 adrenergic stimulation in rat embryos.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Embryo, Mammalian; Female; Isoquinolines; Organ Culture Techniques; Phenylephrine; Piperazines; Pregnancy; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Signal Transduction; Situs Inversus | 1994 |
Inhibitors of Ca2+ channels, calmodulin and protein kinases prevent A23187 and other inductions of metallothionein mRNA in EC3 rat hepatoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 2-Chloroadenosine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Gallic Acid; Isoquinolines; Liver Neoplasms, Experimental; Metallothionein; Norepinephrine; Piperazines; Protein Kinase Inhibitors; Rats; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Verapamil | 1993 |
Calcium/calmodulin-dependent protein kinase II regulates hippocampal synaptic transmission.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Sequence; Animals; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Hippocampus; In Vitro Techniques; Iontophoresis; Isoquinolines; Molecular Sequence Data; Peptide Mapping; Phosphorylation; Piperazines; Prostaglandins E; Protein Kinase Inhibitors; Protein Kinases; Rats; Synapses; Synapsins; Synaptic Transmission | 1993 |
Effects of protein kinase inhibitors on morphology and function of cultured bovine adrenal chromaffin cells: KN-62 inhibits secretory function by blocking stimulated Ca2+ entry.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenal Medulla; Alkaloids; Animals; Benzophenanthridines; Biological Transport; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Catecholamines; Cattle; Cells, Cultured; Enzyme Inhibitors; Indole Alkaloids; Isoquinolines; Phenanthridines; Piperazines; Protein Kinase C; Staurosporine; Substrate Specificity | 1996 |
Redistribution of fodrin in an in vitro wound healing model of the corneal epithelium.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carrier Proteins; Cattle; Cell Membrane; Cells, Cultured; Cornea; Cytoplasm; Egtazic Acid; Epithelial Cells; Epithelium; Isoquinolines; Membrane Proteins; Microfilament Proteins; Microscopy, Fluorescence; Naphthalenes; Piperazines; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Wound Healing | 1995 |
Cultured retinal capillary pericytes die by apoptosis after an abrupt fluctuation from high to low glucose levels: a comparative study with retinal capillary endothelial cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Bucladesine; Calcimycin; Capillaries; Cattle; Cell Survival; Cells, Cultured; Coculture Techniques; DNA; Endothelium, Vascular; Enzyme Inhibitors; Glucose; Isoquinolines; Kinetics; Microscopy, Electron; Muscle, Smooth, Vascular; Niacinamide; Piperazines; Retinal Vessels; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors | 1996 |
Phorbol ester, but not endotoxin, desensitizes mannan-induced glycogenolysis in the perfused rat liver.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aprotinin; Calcimycin; Colforsin; Enzyme Inhibitors; Escherichia coli; Leupeptins; Lipopolysaccharides; Liver; Liver Glycogen; Male; Mannans; Norepinephrine; Perfusion; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1996 |
Gap junctional intercellular communication of bovine luteal cells from several stages of the estrous cycle: effects of prostaglandin F2 alpha, protein kinase C and calcium.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Cattle; Corpus Luteum; Dinoprost; Egtazic Acid; Estrus; Female; Gap Junctions; Luteinizing Hormone; Progesterone; Protein Kinase C; Tissue Plasminogen Activator | 1996 |
Effects of erythropoietin on endothelin-1 synthesis and the cellular calcium messenger system in vascular endothelial cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Cells, Cultured; Endothelin-1; Endothelium, Vascular; Enzyme Inhibitors; Erythropoietin; Gallic Acid; Genistein; Ionophores; Isoflavones; Muscle, Smooth, Vascular; Protein Kinase C; Receptor Protein-Tyrosine Kinases; Recombinant Proteins; Second Messenger Systems; Swine; Verapamil | 1997 |
ATP- and EGF-stimulated phosphatidulinositol synthesis by two different pathways, phospholipase D and diacylglycerol kinase, in A-431 epidermoid carcinoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Bradykinin; Calcimycin; Calcium; Carcinoma, Squamous Cell; Chelating Agents; Choline; Diacylglycerol Kinase; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Humans; Ionophores; Neoplasm Proteins; Pertussis Toxin; Phosphatidic Acids; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Phospholipase D; Phosphotransferases (Alcohol Group Acceptor); Pyrimidinones; Receptors, Purinergic P2; Signal Transduction; Staurosporine; Sulfonamides; Thiazoles; Tumor Cells, Cultured; Type C Phospholipases; Virulence Factors, Bordetella | 1996 |
Reorganization of the cortical actin cytoskeleton during maturation division in the Tubifex egg: possible involvement of protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actin Cytoskeleton; Actins; Animals; Calcimycin; Calcium; Cell Size; Chelating Agents; Cytoskeleton; Egtazic Acid; Enzyme Inhibitors; Fluorescent Dyes; Ionophores; Meiosis; Microinjections; Microscopy, Fluorescence; Oligochaeta; Oocytes; Protein Kinase C; Spectrophotometry; Staurosporine; Tetradecanoylphorbol Acetate | 1997 |
Calcium and protein kinase C play a significant role in response to Shigella toxin in rabbit ileum both in vivo and in vitro.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bacterial Toxins; Calcimycin; Calcium; Cyclic AMP; Cyclic GMP; Electrolytes; Ileum; Indomethacin; Inositol Phosphates; Male; Neutralization Tests; Prostaglandins E; Protein Kinase C; Rabbits; Shiga Toxins; Tetradecanoylphorbol Acetate; Verapamil | 1997 |
Effect of KN-62, a selective inhibitor of calmodulin-dependent kinase II, on mouse oocyte activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Enzyme Inhibitors; Female; Fertilization in Vitro; Fluorescent Dyes; Ionophores; Male; Mice; Mice, Inbred ICR; Oocytes; Protein Kinase Inhibitors | 1997 |
Shigella dysenteriae type 1 toxin induced lipid peroxidation in enterocytes isolated from rabbit ileum.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antioxidants; Bacterial Toxins; Calcimycin; Calcium Channel Blockers; Dantrolene; Dysentery, Bacillary; Enterotoxins; Enzyme Inhibitors; Ileum; In Vitro Techniques; Indomethacin; Ionophores; Lipid Peroxides; Male; Muscle Relaxants, Central; Rabbits; Reactive Oxygen Species; Shiga Toxins; Shigella dysenteriae; Tetradecanoylphorbol Acetate; Verapamil | 1998 |
Acetylcholine acts on M3 muscarinic receptors and induces the translocation of aquaporin5 water channel via cytosolic Ca2+ elevation in rat parotid glands.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetylcholine; Animals; Aquaporin 5; Aquaporins; Atropine; Calcimycin; Calcium; Calcium Channel Blockers; Cytosol; Diamines; Enzyme Inhibitors; Gallic Acid; Ion Channels; Ionophores; Male; Membrane Proteins; Parasympatholytics; Parotid Gland; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Staurosporine | 1998 |
Role of intracellular second messengers and reactive oxygen species in the pathophysiology of V. cholera O139 treated rabbit ileum.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antioxidants; Calcimycin; Calcium; Calcium Channel Blockers; Cholera; Cyclic AMP; Dantrolene; Enzyme Activation; Ileum; Inositol Phosphates; Ionophores; Lipid Peroxidation; Protein Kinase C; Rabbits; Reactive Oxygen Species; Second Messenger Systems; Tetradecanoylphorbol Acetate; Verapamil; Water-Electrolyte Balance | 1998 |
Effects of GnRH on protein kinase C activity, Ca2+ mobilization and steroidogenesis of human granulosa cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calcium; Enzyme Inhibitors; Estradiol; Female; Gonadotropin-Releasing Hormone; Granulosa Cells; Humans; Lipoxygenase Inhibitors; Masoprocol; Progesterone; Protein Kinase C; Steroids; Tetradecanoylphorbol Acetate | 1998 |
Inhibition of lung surfactant secretion by KN-62, a specific inhibitor of the calcium- and calmodulin-dependent protein kinase II.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ionophores; Male; Phosphatidylcholines; Pulmonary Alveoli; Rats; Rats, Sprague-Dawley; Terbutaline; Tetradecanoylphorbol Acetate | 1998 |
Mechanisms of isoflurane-increased submaximum Ca2+-activated force in rabbit skinned femoral arterial strips.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Anesthetics, Inhalation; Animals; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Femoral Artery; In Vitro Techniques; Isoflurane; Male; Myosin Light Chains; Phosphorylation; Protein Kinase C; Rabbits; Vasoconstriction | 1998 |
Protein kinase C-dependent anti-apoptotic mechanism that is associated with high sensitivity to anti-Fas antibody in ovarian cancer cell lines.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antibodies; Apoptosis; Calcimycin; Cell Division; Ceramides; Cyclic AMP-Dependent Protein Kinases; DNA Fragmentation; Enzyme Inhibitors; fas Receptor; Female; Flow Cytometry; Humans; Isoquinolines; Ovarian Neoplasms; Protein Kinase C; Signal Transduction; Sphingomyelin Phosphodiesterase; Sulfonamides; Tetradecanoylphorbol Acetate; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured | 1999 |
Caldesmon inhibits nonmuscle cell contractility and interferes with the formation of focal adhesions.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actomyosin; Animals; Botulinum Toxins; Calcimycin; Calcium-Binding Proteins; Calmodulin-Binding Proteins; Cell Line, Transformed; Cytoskeleton; Enzyme Inhibitors; Gene Expression; Green Fluorescent Proteins; Humans; Ionophores; Luminescent Proteins; Microscopy, Fluorescence; Microtubules; Mutation; Nocodazole; Rats; Thapsigargin; Transfection | 1999 |
The protein kinase inhibitor 1-(5-isoquinolinylsulfonyl)-2-methyl-piperzine (H-7) prevents and reverses Ca(2+)-mediated injury in isolated rat hepatocyte couplets.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Adenosine Triphosphate; Animals; Calcimycin; Calcium; Cell Membrane; Chelating Agents; Cholic Acids; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Inhibitors; Fluoresceins; Fluorescence; Fluorescent Dyes; In Vitro Techniques; Ionophores; Liver; Male; Protein Kinase Inhibitors; Rats; Rats, Wistar; Tight Junctions; Vacuoles | 1999 |
T cell activation up-regulates the expression of the focal adhesion kinase Pyk2: opposing roles for the activation of protein kinase C and the increase in intracellular Ca2+.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; CD28 Antigens; Cell Adhesion Molecules; Cyclosporine; Enzyme Activation; Enzyme Inhibitors; Focal Adhesion Kinase 1; Focal Adhesion Kinase 2; Focal Adhesion Protein-Tyrosine Kinases; Humans; Intracellular Fluid; Ionophores; Jurkat Cells; Lymphocyte Activation; MAP Kinase Kinase Kinase 1; MAP Kinase Kinase Kinases; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Antigen, T-Cell; Signal Transduction; T-Lymphocytes; Tacrolimus; Tetradecanoylphorbol Acetate; Transcription, Genetic; Up-Regulation | 1999 |
Regulation of LPA-promoted myofibroblast contraction: role of Rho, myosin light chain kinase, and myosin light chain phosphatase.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; ADP Ribose Transferases; Alkaloids; Azepines; Botulinum Toxins; Calcimycin; Calcium; Carbazoles; Cells, Cultured; Enzyme Inhibitors; Humans; Indoles; Intracellular Signaling Peptides and Proteins; Ionomycin; Kinetics; Lysophospholipids; Models, Chemical; Muscle Contraction; Muscle, Skeletal; Myosin-Light-Chain Kinase; Myosin-Light-Chain Phosphatase; Naphthalenes; Phosphoprotein Phosphatases; Protein Serine-Threonine Kinases; Recombinant Proteins; rho-Associated Kinases | 2000 |
Ca2+/calmodulin-dependent kinase II and calcineurin play critical roles in endothelin-1-induced cardiomyocyte hypertrophy.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Animals, Newborn; Calcimycin; Calcineurin; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cardiomegaly; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Gene Expression Regulation; Heart; Ionomycin; Kinetics; Models, Cardiovascular; Myocardium; Myosin Heavy Chains; Promoter Regions, Genetic; Rats; Rats, Wistar; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 2000 |
Effects of extracellular calcium and potassium on the sodium pump of rat adrenal glomerulosa cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aldosterone; Animals; Calcimycin; Calcium; Calcium Channels; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cells, Cultured; Enzyme Inhibitors; Extracellular Space; Female; Imidazoles; Intracellular Fluid; Ionophores; Isradipine; Potassium; Rats; Rats, Sprague-Dawley; Rubidium Radioisotopes; Sodium-Potassium-Exchanging ATPase; Staurosporine; Zona Glomerulosa | 2001 |
The stimulation of MAP kinase by 1,25(OH)(2)-vitamin D(3) in skeletal muscle cells is mediated by protein kinase C and calcium.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcitriol; Calcium; Calmodulin; Chick Embryo; Egtazic Acid; Enzyme Activation; Fluphenazine; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Skeletal; Naphthalenes; Neomycin; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Thapsigargin; Type C Phospholipases; Verapamil | 2001 |
Calmodulin-dependent and -independent apoptosis in cell of a Drosophila neuronal cell line.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Calcimycin; Calcium; Calmodulin; Caspases; Cell Line; Chelating Agents; Cycloheximide; Dactinomycin; DNA Fragmentation; Drosophila melanogaster; Egtazic Acid; Enzyme Inhibitors; Ionophores; Neurons; Protein Synthesis Inhibitors; Sulfonamides | 2000 |
Regulation of SERCA Ca2+ pump expression by cytoplasmic Ca2+ in vascular smooth muscle cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta; Blotting, Northern; Calcimycin; Calcium; Calcium-Transporting ATPases; Carrier Proteins; Cells, Cultured; Cytoplasm; Endoplasmic Reticulum Chaperone BiP; Enzyme Inhibitors; Gene Expression; Heat-Shock Proteins; Homeostasis; Ionophores; Male; Molecular Chaperones; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Staurosporine; Thapsigargin | 2001 |
Involvement of intracellular Ca2+ in the regulation of bovine leukemia virus expression.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Cell Line; Enzyme Inhibitors; Gene Expression Regulation, Viral; Ionophores; Kidney; Leukemia Virus, Bovine; NF-kappa B; Protein Kinase C; Signal Transduction; Staurosporine; Terminal Repeat Sequences; Transcription, Genetic | 2001 |
Effects of second messengers on gap junctional intercellular communication of ovine luteal cells throughout the estrous cycle.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Blotting, Western; Bucladesine; Calcimycin; Calcium; Cells, Cultured; Chelating Agents; Culture Media, Conditioned; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Estrous Cycle; Female; Fluorescent Antibody Technique; Gap Junctions; Immunohistochemistry; Ionophores; Luteal Cells; Progesterone; Protein Kinase C; Second Messenger Systems; Sheep; Tetradecanoylphorbol Acetate; Thionucleotides | 2001 |
Effect of Leishmania donovani lipophosphoglycan on ornithine decarboxylase activity in macrophages.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Anti-Bacterial Agents; Bucladesine; Calcimycin; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glycosphingolipids; Leishmania donovani; Leishmaniasis, Visceral; Lipopolysaccharides; Macrophages; Mice; Okadaic Acid; Ornithine Decarboxylase; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors | 2001 |
Antigen-independent induction of histamine synthesis by immunoglobulin E in mouse bone marrow-derived mast cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antigens; Calcimycin; Calcium Signaling; Enzyme Inhibitors; Estrenes; Female; Histamine; Histidine Decarboxylase; Immunoglobulin E; In Vitro Techniques; Interleukin-3; Mast Cells; Mice; Mice, Inbred BALB C; Protein Kinase C; Pyrrolidinones; Receptors, IgE; RNA, Messenger; src-Family Kinases; Tetradecanoylphorbol Acetate; Type C Phospholipases | 2002 |
Formation of AP-1 transcription factors during learning in Helix.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Casein Kinase II; CCAAT-Enhancer-Binding Proteins; Central Nervous System; DNA-Binding Proteins; Drug Interactions; Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Exoribonucleases; Flavonoids; Genistein; Helix, Snails; Ionophores; Learning; Phorbol Esters; Protein Serine-Threonine Kinases; Serotonin; Transcription Factor AP-1 | 2003 |
Platelet-activating factor acts on cortisol secretion by perfused guinea-pig adrenals via calcium-/phospholipid-dependent mechanisms.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenal Glands; Adrenocorticotropic Hormone; Animals; Calcimycin; Calcium; Colforsin; Corticosterone; Cyclic AMP-Dependent Protein Kinases; Diglycerides; Drug Synergism; Enzyme Activation; Guinea Pigs; Hydrocortisone; Ionophores; Isoquinolines; Male; Perfusion; Phospholipid Ethers; Phospholipids; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Pyridinium Compounds; Receptors, G-Protein-Coupled; Secretory Rate | 2005 |
Nitric oxide does not downregulate Rho-kinase (ROCK-2) expression in rat coronary endothelial cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Calcimycin; Cells, Cultured; Coronary Vessels; Down-Regulation; Endothelial Cells; Gene Expression Regulation, Enzymologic; In Vitro Techniques; Male; Microcirculation; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroglycerin; Nitroprusside; Pyridines; Rats; Rats, Wistar; rho-Associated Kinases; Sodium Nitrite; Triazenes | 2008 |
IL-18 associates to microvesicles shed from human macrophages by a LPS/TLR-4 independent mechanism in response to P2X receptor stimulation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetamides; Adenosine Triphosphate; Anti-Bacterial Agents; Calcimycin; Calcium Ionophores; Cell-Derived Microparticles; Humans; Interleukin-18; Lipopolysaccharides; Macrophages; Polymyxin B; Protein Precursors; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Pyridines; Quinolines; Receptors, Purinergic P2X4; Receptors, Purinergic P2X7; Sulfonamides; Tetrazoles; Toll-Like Receptor 4 | 2012 |