1-(3-chlorophenyl)piperazine has been researched along with mdl 100907 in 26 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (3.85) | 18.2507 |
2000's | 15 (57.69) | 29.6817 |
2010's | 10 (38.46) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Dekeyne, A; Girardon, S; Millan, MJ | 1 |
Evans, DC; Hemrick-Luecke, SK | 1 |
Gleason, SD; Leander, JD; Lucaites, VL; Nelson, DL; Shannon, HE | 1 |
Cunningham, KA; Frankel, PS | 1 |
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L | 2 |
Eckler, JR; Rabin, RA; Rice, KC; Winter, JC | 1 |
Clifton, PG; Dalton, GL; Dourish, CT; Kennett, GA; Lee, MD | 1 |
Gráf, M | 1 |
Avison, MJ; Deutch, AY; Gore, JC; Gresch, PJ; Hackler, EA; Sanders-Bush, E; Sengupta, S; Turner, GH | 1 |
Asaka, M; Hattori, T; Katsurada, T; Nagai, K; Ohkawara, T; Sadakane, C; Takeda, H | 1 |
Dzhordzhikiya, RK; Kirillova, VV; Nigmatullina, RR | 1 |
Amitani, H; Asakawa, A; Fujimiya, M; Fujitsuka, N; Hayashi, M; Inui, A; Kojima, S; Sameshima, M | 1 |
Ali, U; Liu, J; Liu, X; Wang, S; Wang, T; Wu, ZH; Zhang, QJ | 1 |
Arai, Y; Chancellor, MB; de Groat, WC; Kaiho, Y; Kamo, I; Kitta, T; Miyazato, M; Sugaya, K; Yoshimura, N | 1 |
Foley, JJ; Walker, EA | 1 |
Gan'shina, TS; Gorbunov, AA; Mirzoian, RS | 1 |
Hajos, M; Kocsis, B; Sörman, E; Wang, D | 1 |
Haider, S; Haleem, DJ; Khaliq, S; Memon, Z; Saleem, S | 1 |
Gao, L; Han, X; Yuan, L; Zhang, Q; Zhou, W; Zhu, Y | 1 |
Fedotova, IuO; Frolova, HO; Ordian, NE; Soboliev, VI | 1 |
Bhutada, P; Deshmukh, P; Dixit, P; Kaulaskar, S; Thakur, K | 1 |
Dvorkin-Gheva, A; Johnson, E; Szechtman, H; Tucci, MC; Wong, M | 1 |
Gwarek, M; Lübbert, H; Schmitz, B; Segelcke, D; Ullmer, C; Zhu, XR | 1 |
Cui, R; Fan, J; Ge, T; Hall, FS; Li, B; Liu, W; Lv, J; Song, Y; Wang, X; Zhang, Z | 1 |
26 other study(ies) available for 1-(3-chlorophenyl)piperazine and mdl 100907
Article | Year |
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Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Discriminative stimulus properties of the novel serotonin (5-HT)2C receptor agonist, RO 60-0175: a pharmacological analysis.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Conditioning, Operant; Ethylamines; Fluorobenzenes; Indoles; Male; Mianserin; Piperazines; Piperidines; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes | 1999 |
Comparison of the potency of MDL 100,907 and SB 242084 in blocking the serotonin (5-HT)(2) receptor agonist-induced increases in rat serum corticosterone concentrations: evidence for 5-HT(2A) receptor mediation of the HPA axis.
Topics: Aminopyridines; Amphetamines; Animals; Corticosterone; Dose-Response Relationship, Drug; Ethylamines; Fluorobenzenes; Hypothalamo-Hypophyseal System; Indoles; Male; Piperazines; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
m-CPP hypolocomotion is selectively antagonized by compounds with high affinity for 5-HT(2C) receptors but not 5-HT(2A) or 5-HT(2B) receptors.
Topics: Amphetamines; Animals; Binding, Competitive; Cell Line; Cricetinae; Fluorobenzenes; Humans; Kinetics; Male; Mice; Mice, Inbred Strains; Motor Activity; Piperazines; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists | 2001 |
m-Chlorophenylpiperazine (mCPP) modulates the discriminative stimulus effects of cocaine through actions at the 5-HT2C receptor.
Topics: Animals; Cocaine; Discrimination Learning; Male; Piperazines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2004 |
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction | 2004 |
m-CPP, a 5-HT2C receptor agonist that modifies the perfusion pressure of the hindquarter vascular bed of anesthetized rat.
Topics: Adrenergic beta-2 Receptor Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Epinephrine; Hindlimb; Male; Methiothepin; Perfusion; Piperazines; Pressure; Propanolamines; Rats; Rats, Wistar; Regional Blood Flow; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Vasoconstriction; Vasodilation | 2005 |
Serotonergic/glutamatergic interactions: potentiation of phencyclidine-induced stimulus control by citalopram.
Topics: Aminopyridines; Analysis of Variance; Animals; Citalopram; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Indoles; Male; Phencyclidine; Piperazines; Rats; Rats, Inbred F344; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2005 |
Serotonin 1B and 2C receptor interactions in the modulation of feeding behaviour in the mouse.
Topics: Aminopyridines; Animals; Feeding Behavior; Female; Indoles; Male; Mice; Mice, Knockout; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Satiety Response; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2006 |
5-HT2c receptor activation induces grooming behaviour in rats: possible correlations with obsessive-compulsive disorder.
Topics: Aminopyridines; Animals; Grooming; Indoles; Male; Obsessive-Compulsive Disorder; Piperazines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2006 |
5-Hydroxytryptamine2C receptor contribution to m-chlorophenylpiperazine and N-methyl-beta-carboline-3-carboxamide-induced anxiety-like behavior and limbic brain activation.
Topics: Aminopyridines; Animals; Anxiety; Behavior, Animal; Carbolines; Indoles; Limbic System; Magnetic Resonance Imaging; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2007 |
Rikkunshito, an herbal medicine, suppresses cisplatin-induced anorexia in rats via 5-HT2 receptor antagonism.
Topics: Acylation; Aminopyridines; Animals; Anorexia; Antineoplastic Agents; Body Weight; Chalcones; Cisplatin; Disease Models, Animal; Dopamine Antagonists; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Eating; Flavones; Gastric Mucosa; Gastrointestinal Agents; Ghrelin; Hesperidin; Indoles; Male; Oligopeptides; Piperazines; Protein Binding; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Ghrelin; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Stomach; Thiophenes; Vagotomy | 2008 |
Adrenergic and serotoninergic regulation of myocardial contractility in patients with various morphofunctional changes in the heart resulting from chronic heart failure.
Topics: Adrenergic Agonists; Epinephrine; Heart Failure; Humans; Hypertrophy, Left Ventricular; Middle Aged; Myocardial Contraction; Piperazines; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Agents | 2007 |
Selective serotonin reuptake inhibitors modify physiological gastrointestinal motor activities via 5-HT2c receptor and acyl ghrelin.
Topics: Animals; Drugs, Chinese Herbal; Eating; Fenfluramine; Fluoxetine; Fluvoxamine; Gastrointestinal Motility; Ghrelin; Growth Hormone; Injections, Intraventricular; Male; Oligopeptides; Paroxetine; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Ghrelin; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2009 |
Subthalamic neurons show increased firing to 5-HT2C receptor activation in 6-hydroxydopamine-lesioned rats.
Topics: Action Potentials; Aminopyridines; Analysis of Variance; Animals; Immunohistochemistry; Indoles; Male; Microelectrodes; Neurons; Oxidopamine; Parkinsonian Disorders; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Subthalamic Nucleus | 2009 |
Role of spinal serotonergic pathways in sneeze-induced urethral continence reflex in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Fluoxetine; Piperazines; Pressure; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT2; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Sneezing; Spiro Compounds; Sulfonamides; Urethra; Urinary Incontinence, Stress | 2009 |
Acquisition session length modulates consolidation effects produced by 5-HT2C ligands in a mouse autoshaping-operant procedure.
Topics: Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Inverse Agonism; Drug Partial Agonism; Indoles; Ligands; Lysergic Acid Diethylamide; Male; Memory; Methysergide; Mianserin; Mice; Piperazines; Pyrazines; Pyridines; Reinforcement Schedule; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2010 |
[Effect of tropoxin on cerebrovascular effects of meta-chlorophenylpiperazine and serotonin].
Topics: Animals; Aza Compounds; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Carotid Artery, Internal; Cerebrovascular Circulation; Drug Interactions; Male; Migraine Disorders; Piperazines; Rats; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction | 2010 |
Control of hippocampal theta rhythm by serotonin: role of 5-HT2c receptors.
Topics: Aminopyridines; Anesthesia; Animals; Brain Stem; Deep Brain Stimulation; Dose-Response Relationship, Drug; Electroencephalography; Hippocampus; Indoles; Male; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Sleep, REM; Theta Rhythm; Time Factors | 2011 |
Influence of serotonergic 5-HT2C receptor antagonist mesulergine in the reversal of memory deficits induced by mCPP.
Topics: Analysis of Variance; Animals; Behavior, Animal; Disease Models, Animal; Ergolines; Male; Maze Learning; Memory Disorders; Memory, Long-Term; Memory, Short-Term; Piperazines; Random Allocation; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2012 |
Serotonin receptor 2C and insulin secretion.
Topics: Aminopyridines; Animals; Blotting, Western; Cell Line, Tumor; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Gene Expression; Humans; Indoles; Insulin; Insulin Secretion; Insulin-Secreting Cells; Islets of Langerhans; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Palmitic Acid; Piperazines; Receptor, Serotonin, 5-HT2C; Reverse Transcriptase Polymerase Chain Reaction; RNA Interference; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2013 |
[Involvement of some subtypes of 5-HT2-receptors in affective behavior in female rats].
Topics: Animals; Animals, Outbred Strains; Anti-Anxiety Agents; Anxiety; Depression; Estrogens; Estrus; Female; Injections, Intraperitoneal; Ketanserin; Piperazines; Proestrus; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2012 |
Effects of agomelatine in a murine model of obsessive-compulsive disorder: interaction with meta-chlorophenylpiperazine, bicuculline, and diazepam.
Topics: Acetamides; Animals; Antidepressive Agents; Behavior, Animal; Bicuculline; Diazepam; Disease Models, Animal; Drug Interactions; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred C57BL; Motor Activity; Obsessive-Compulsive Disorder; Piperazines; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2013 |
5-HT2A/C receptors do not mediate the attenuation of compulsive checking by mCPP in the quinpirole sensitization rat model of obsessive-compulsive disorder (OCD).
Topics: Animals; Compulsive Behavior; Disease Models, Animal; Male; Obsessive-Compulsive Disorder; Piperazines; Quinpirole; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2015 |
BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs.
Topics: Animals; Blood Proteins; Brain; Cell Line; Guinea Pigs; Humans; Indoles; Male; Piperazines; Piperidines; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT2 Receptor Antagonists; Substrate Specificity; Thiophenes; Thioxanthenes; Xanthenes | 2015 |
The role of 5-HT
Topics: Animals; Appetite Depressants; Appetite Regulation; Appetite Stimulants; Behavior, Animal; Corticosterone; Dose-Response Relationship, Drug; Energy Intake; Hyperphagia; Hypothalamus; Leptin; Mice, Inbred ICR; Nerve Tissue Proteins; Neurons; Organ Specificity; Piperazines; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Spiro Compounds; Sulfonamides; Up-Regulation | 2017 |