1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazole has been researched along with thapsigargin in 106 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 44 (41.51) | 18.2507 |
2000's | 50 (47.17) | 29.6817 |
2010's | 11 (10.38) | 24.3611 |
2020's | 1 (0.94) | 2.80 |
Authors | Studies |
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Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Demaurex, N; Krause, KH; Lew, DP | 1 |
Grinstein, S; Mahaut-Smith, MP; Mason, MJ | 1 |
Musgrave, IF; Schultz, G; Seifert, R | 1 |
Shuttleworth, TJ | 1 |
Berggren, PO; Chow, SC; Gahm, A; Kass, GE; Llopis, J; Orrenius, S; Webb, DL | 1 |
Bressler, J; Forman, S; Goldstein, GW | 1 |
Cabello, OA; Schilling, WP | 1 |
Grinstein, S; Mason, MJ | 1 |
Doan, TN; Elliott, SJ; Gentry, DL; Taylor, AA | 1 |
Törnquist, K | 1 |
Hymel, LJ; Mason, MJ; Mayer, B | 1 |
Hughes, BP; Strazzari, MJ | 1 |
Elton, TS; Guest, LL; Marchase, RB; Rivera, AA; White, CR | 1 |
Rüegg, UT; Skutella, M | 1 |
Chernaya, G; Reeves, JP; Vázquez, M | 1 |
Krautwurst, D; Musgrave, I; Seifert, R; Wenzel-Seifert, K | 1 |
Dohi, T; Kitayama, S; Morita, K; Okamoto, H; Shibata, K | 1 |
Hisayama, T; Inoue, S; Kida, K; Kondoh, W; Moritoki, H; Takeuchi, S | 1 |
Andriantsitohaina, R; Lagaud, GJ; Stoclet, JC | 1 |
Gleispach, H; Huber, E; Leis, HJ; Windischhofer, W; Zach, D; Ziermann, L | 1 |
Dietl, P; Friedrich, F; Haller, T; Wirleitner, B | 1 |
Kankaanranta, H; Kosonen, O; Luomala, M; Moilanen, E | 1 |
David-Dufilho, M; Devynck, MA; Iouzalen, L; Lantoine, F; Millanvoye-Van Brussel, E; Pernollet, MG | 1 |
Grudt, TJ; Henderson, G; Usowicz, MM | 1 |
Gill, DL; Short, AD; Waldron, RT | 1 |
Hobson, S; Kohn, EC; Rodland, KD; Wersto, RP | 1 |
Hinkle, PM; Kerper, LE | 1 |
Helmke, RJ; Martinez, JR; Mörk, AC; Zhang, GH | 1 |
Zimmermann, B | 1 |
Ogino, K; Takagi, K; Takemoto, M; Tomita, T | 1 |
Yang, CM | 1 |
Hawkins, T; Kubista, H; Moss, SE | 1 |
Ho, CM; Jan, CR; Tseng, CJ; Wu, SN | 2 |
Goldfine, H; Wadsworth, SJ | 1 |
Iversen, JG; Nicolaysen, G; Wassdal, I | 1 |
Enoki, T; Furutani, H; Hasegawa, H; Hashimoto, N; Ishikawa, M; Iwamuro, Y; Masaki, T; Minowa, T; Miwa, S; Okamoto, Y; Okazawa, M; Zhang, XF | 1 |
Dugué, B; Titievsky, A; Törnquist, K; Tuominen, R; Vainio, P | 1 |
Chiu, CT; Luo, SF; Pan, SL; Tsai, YJ; Wang, CC; Wu, WB; Yang, CM | 1 |
Fujishima, M; Hirano, K; Hirano, M; Kanaide, H; Kawasaki, J; Nishimura, J | 1 |
Bueb, JL; Tschirhart, EJ; Zardini, DM | 1 |
Hirano, H; Shigenobu, K; Tanaka, H; Tanaka, Y; Taniguchi, H | 1 |
Guan, Z; Saqr, HE; Stokes, BT; Yates, AJ | 1 |
Ayman, S; Gibson, A; McFadzean, I; Wallace, P | 1 |
Hasegawa, A; Ito, S; Nakazato, Y; Ohta, T; Yasuda, W | 1 |
Chin, TY; Chueh, SH | 1 |
Auld, A; Barritt, GJ; Brereton, HM; Chen, J; Gregory, RB; Wang, YJ | 1 |
Aaronson, PI; Hague, D; Robertson, TP; Ward, JP | 1 |
Dora, KA; Garland, CJ; Hill, PB; Hughes, AD | 1 |
Jenner, S; Sage, SO | 1 |
Igarashi, T; Imai, T; Otsuka, K; Shigenobu, K; Takayanagi, K; Tanaka, H; Tanaka, Y; Yamaki, F | 1 |
French, JN; Gilbert, M; Knox, SJ; Rangaswami, AA; Walleczek, J; Williams, SS | 1 |
Bruce, JI; Elliott, AC | 1 |
Freyssinet, JM; Kunzelmann-Marche, C; Martínez, MC | 1 |
Choi, SY; Kim, KT; Kim, YH; Lee, YK | 1 |
Fewtrell, C; Mahmoud, SF | 1 |
Chien, C; Chiu, C; Hsiao, L; Huang, SC; Liang, K; Wang, C; Yang, C | 1 |
Iwamuro, Y; Lee, K; Miwa, S; Morita, H; Okamoto, Y; Zhang, XF | 1 |
Alojado, ME; Knöpfel, T; Strata, P; Tempia, F | 1 |
Chang, HT; Cheng, JS; Chou, KJ; Huang, JK; Jan, CR; Law, YP; Lee, KC; Su, W; Tang, KY; Tseng, LL; Wang, JL | 1 |
Fernandes, F; Gibson, A; McFadzean, I; Wallace, P | 1 |
Enoki, T; Hashimoto, N; Kawanabe, Y; Masaki, T; Okamoto, Y | 1 |
Baird, AW; O'Riordan, AM; Quinn, T | 1 |
Guse, AH; Mayr, GW; Potter, BV; Schöttelndreier, H | 1 |
Groschner, K; Kakishita, E; Marumo, M; Suehiro, A; Wakabayashi, I | 1 |
Cooper, DM; Fagan, KA; Gu, C; Hu, B; Smith, KE | 1 |
Benham, CD; Calver, AR; Davis, JB; Kelsell, RE; Mattei, C; Medhurst, AD; Pangalos, MN; Randall, AD; Riccio, A | 1 |
Fukui, H; Kadowaki, M; Sekiguchi, F; Sugimori, S; Sunano, S; Takaki, M; Yoneda, S | 1 |
Benedetti, A; Gamberucci, A; Giunti, R; Giurisato, E; McIntosh, DP; Pizzo, P; Tassi, M | 1 |
Abu-Basha, EA; Cheng, H; Ding, J; Hsu, WH; Ioudina, M; Yibchok-anun, S | 1 |
Bates, DO; Glass, CA | 1 |
Hirohashi, N; Vacquier, VD | 1 |
Hayashi, H; Honjo, H; Ito, S; Katoh, H; Kodama, I; Kume, H; Shimokata, K | 1 |
Breitner, JC; Cook, DG; Kinney, GA; Spain, WJ; Yang, Y | 1 |
Bristulf, J; Owman, C; Sabirsh, A | 1 |
Ajioka, H; Horie, S; Kunieda, K; Murayama, T; Someya, A | 1 |
Campos-Toimil, M; Elíes, J; Orallo, F | 1 |
Kreutz, R; Liu, D; Scholze, A; Tepel, M; Wehland-von-Trebra, M; Zhu, Z; Zidek, W | 1 |
Bartegi, A; Ben-Amor, N; Pariente, JA; Redondo, PC; Rosado, JA; Salido, GM | 1 |
London, FS; Marcinkiewicz, M; Walsh, PN | 1 |
Alfonso, A; Botana, LM; Escribano, L; Francisca, SJ; Orfao, A; Pernas-Sueiras, O; Vieytes, MR | 1 |
Kuwahara, M | 1 |
Kachoei, BA; Kaczmarek, LK; Knox, RJ; Levy, S; Magoski, NS; Uthuza, D | 1 |
Cabrera, JA; Hong, F; Hong, Z; Nelson, DP; Olschewski, A; Varghese, A; Weir, EK | 1 |
Chrones, T; Kovac, JR; Sims, SM | 1 |
Jumarie, C; Labelle, D; Moreau, R | 1 |
Ding, X; Murray, PA; Yang, M | 1 |
Azuma, T; Hirayama, T; Hisatsune, J; Isomoto, H; Kurazono, H; Moss, J; Mukaida, N; Mukhopadhyay, AK; Nakayama, M; Sap, J; Yahiro, K; Yamaoka, Y; Yamasaki, E | 1 |
Friis, S; Mathes, C; Schrøder, RL; Sunesen, M; Willumsen, NJ | 1 |
Dhondt, A; Glorieux, G; Leybaert, L; Schepers, E; Vanholder, R | 1 |
Baba, Y; Kurosaki, T; Morita, T; Tanimura, A; Tojyo, Y | 1 |
Araki, M; Inui, T; Kubota, T; Miyamoto, M; Mori, Y; Nimura, Y; Takenaka, H; Watanabe, M | 1 |
Feng, SL; Li, BX; Li, TT; Li, YQ; Pan, ZW; Sun, YH; Xu, CQ; Yang, BF | 1 |
Sham, JS; Yip, KP | 1 |
Chai, KL; Chen, WC; Cheng, HH; Cheng, JS; Chien, JM; Chou, CT; Fang, YC; Jan, CR; Kuo, CC; Kuo, LN; Lu, T; Pan, CC; Shu, SS; Tsai, WL; Yeh, JH | 1 |
Huang, X; Lai, X; Lu, X; Ye, Y; Zeng, X; Zeng, Y; Zhang, Y | 1 |
Huang, X; Lai, X; Tang, X; Wu, X; Ye, Y; Zeng, X; Zeng, Y; Zhang, Y | 1 |
Goto, K; Marumo, M; Nakano, T; Takeda, Y; Wakabayashi, I | 1 |
Chang, HT; Chen, IS; Chou, CT; Hsu, SS; Jan, CR; Kuo, CC; Liao, WC; Liu, SI; Mok, KT; Tsai, JY | 1 |
Bannister, JP; Bulley, S; Burris, SK; Jaggar, JH; Jangsangthong, W; Neeb, ZP; Thomas-Gatewood, CM | 1 |
Hadley, SH; Hooper, JS; Mathews, A; Taylor-Clark, TE | 1 |
Alkhani, H; Ase, AR; Grant, R; Groschner, K; O'Donnell, D; Séguéla, P | 1 |
Cai, C; Cai, G; Meng, X; Shen, Q; Tang, S; Wang, X; Yang, X; Yu, C; Zou, F | 1 |
Gruszczynska-Biegala, J; Kuznicki, J; Maciag, F; Majewski, L; Sladowska, M; Strucinska, K | 1 |
106 other study(ies) available for 1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazole and thapsigargin
Article | Year |
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Small molecule regulators of autophagy identified by an image-based high-throughput screen.
Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers | 2007 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Cyclopiazonic acid depletes intracellular Ca2+ stores and activates an influx pathway for divalent cations in HL-60 cells.
Topics: Biological Transport; Calcium; Calcium-Transporting ATPases; Cations, Divalent; Cell Line; Cell Membrane Permeability; Fura-2; Hydroquinones; Imidazoles; Indoles; Mycotoxins; N-Formylmethionine Leucyl-Phenylalanine; Terpenes; Thapsigargin | 1992 |
The role of intracellular Ca2+ in the regulation of the plasma membrane Ca2+ permeability of unstimulated rat lymphocytes.
Topics: Aminoquinolines; Animals; Calcium; Calcium-Transporting ATPases; Cell Membrane; Cell Membrane Permeability; Concanavalin A; Fluorescent Dyes; Imidazoles; Indoles; Kinetics; Male; Rats; Rats, Inbred Strains; Spectrometry, Fluorescence; T-Lymphocytes; Terpenes; Thapsigargin; Thymus Gland | 1991 |
Maitotoxin activates cation channels distinct from the receptor-activated non-selective cation channels of HL-60 cells.
Topics: Bucladesine; Cadmium; Calcium; Cations; Fluorescent Dyes; Fura-2; Gadolinium; Humans; Imidazoles; Ion Channels; Manganese; Marine Toxins; N-Formylmethionine Leucyl-Phenylalanine; Oxocins; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Tumor Cells, Cultured | 1994 |
Temporal relationships between Ca2+ store mobilization and Ca2+ entry in an exocrine cell.
Topics: Animals; Calcium; Calcium-Transporting ATPases; Carbachol; Ducks; Fluorescent Dyes; Imidazoles; Indoles; Inositol 1,4,5-Trisphosphate; Ion Transport; Manganese; Salt Gland; Terpenes; Thapsigargin | 1994 |
Two separate plasma membrane Ca2+ carriers participate in receptor-mediated Ca2+ influx in rat hepatocytes.
Topics: Animals; Calcium; Calcium Channels; Calcium-Binding Proteins; Cell Membrane; Culture Media; Imidazoles; Liver; Male; Rats; Rats, Wistar; Receptors, Cell Surface; Terpenes; Thapsigargin; Type C Phospholipases; Vasopressins | 1994 |
Phospholipid metabolism in neural microvascular endothelial cells after exposure to lead in vitro.
Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Brain; Calcium; Capillaries; Cattle; Cells, Cultured; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Inositol Phosphates; Ionomycin; Lead; Marine Toxins; Molecular Sequence Data; Oxocins; Phospholipids; Phosphorylcholine; Protein Kinase C; Terpenes; Thapsigargin | 1994 |
Vectorial Ca2+ flux from the extracellular space to the endoplasmic reticulum via a restricted cytoplasmic compartment regulates inositol 1,4,5-trisphosphate-stimulated Ca2+ release from internal stores in vascular endothelial cells.
Topics: Animals; Biological Transport; Bradykinin; Calcium; Calcium-Transporting ATPases; Cattle; Cell Compartmentation; Cells, Cultured; Cytoplasm; Egtazic Acid; Endoplasmic Reticulum; Endothelium, Vascular; Extracellular Space; Humans; Hydroquinones; Imidazoles; Inositol 1,4,5-Trisphosphate; Terpenes; Thapsigargin | 1993 |
Ionomycin activates electrogenic Ca2+ influx in rat thymic lymphocytes.
Topics: Animals; Calcium; Calcium-Transporting ATPases; Cells, Cultured; Cytosol; Imidazoles; Ionomycin; Kinetics; Male; Potassium Chloride; Rats; Rats, Wistar; Sodium Chloride; T-Lymphocytes; Terpenes; Thapsigargin; Thymus Gland | 1993 |
Hydrogen peroxide activates agonist-sensitive Ca(2+)-flux pathways in canine venous endothelial cells.
Topics: Adenosine Triphosphate; Animals; Calcium; Dogs; Endothelium, Vascular; Hydrogen Peroxide; Imidazoles; Inosine Triphosphate; Ionomycin; Jugular Veins; Lanthanum; Nickel; Signal Transduction; Terpenes; Thapsigargin | 1994 |
ATP-induced entry of calcium in thyroid FRTL-5 cells. Studies with phorbol myristate acetate and thapsigargin.
Topics: Adenosine Triphosphate; Animals; Biological Transport, Active; Calcium; Cell Line; Enzyme Activation; Imidazoles; Ionomycin; Protein Kinase C; Rats; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Thyroid Gland | 1993 |
Inhibition of Ca2+ transport pathways in thymic lymphocytes by econazole, miconazole, and SKF 96365.
Topics: Animals; Biological Transport; Calcium; Calcium-Transporting ATPases; Cell Membrane Permeability; Cells, Cultured; Cytochrome P-450 Enzyme Inhibitors; Econazole; Fluorescence; Imidazoles; Lymphocytes; Male; Miconazole; Oxidation-Reduction; Proton Pump Inhibitors; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Terpenes; Thapsigargin; Thymus Gland | 1993 |
Evidence that the Ca2+ inflow pathway in hepatocytes stimulated by thapsigargin is similar to that activated by vasopressin.
Topics: Animals; Calcium; Cell Membrane; Cells, Cultured; Dimethyl Sulfoxide; Enzyme Activation; Imidazoles; Kinetics; Liver; Male; Phosphorylases; Platelet Aggregation Inhibitors; Rats; Sensitivity and Specificity; Stimulation, Chemical; Terpenes; Thapsigargin; Vasopressins; Zinc | 1993 |
Hyperglycemia alters cytoplasmic Ca2+ responses to capacitative Ca2+ influx in rat aortic smooth muscle cells.
Topics: Adenosine Triphosphate; Angiotensin II; Animals; Aorta; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cells, Cultured; Cytoplasm; Hyperglycemia; Imidazoles; Male; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; Sarcoplasmic Reticulum; Terpenes; Thapsigargin | 1995 |
Increase of empty pool-activated Ca2+ influx using an intracellular Ca2+ chelating agent.
Topics: Animals; Arginine Vasopressin; Biological Transport; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cell Compartmentation; Cell Membrane; Cells, Cultured; Chelating Agents; Cytoplasm; Egtazic Acid; Enzyme Inhibitors; Imidazoles; Kinetics; Muscle, Smooth, Vascular; Nifedipine; Rats; Terpenes; Thapsigargin | 1996 |
Sodium-calcium exchange and store-dependent calcium influx in transfected chinese hamster ovary cells expressing the bovine cardiac sodium-calcium exchanger. Acceleration of exchange activity in thapsigargin-treated cells.
Topics: Animals; Barium; Biological Transport; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Carrier Proteins; Cattle; CHO Cells; Clone Cells; Cricetinae; Culture Media; Enzyme Inhibitors; Genetic Vectors; Imidazoles; Kinetics; Myocardium; Organelles; Recombinant Proteins; Sodium; Sodium-Calcium Exchanger; Terpenes; Thapsigargin; Transfection | 1996 |
Thapsigargin activates univalent- and bivalent-cation entry in human neutrophils by a SK&F I3 96365- and Gd3+-sensitive pathway and is a partial secretagogue: involvement of pertussis-toxin-sensitive G-proteins and protein phosphatases 1/2A and 2B in the
Topics: Cations; Female; Gadolinium; GTP-Binding Proteins; Humans; Imidazoles; Ion Transport; Male; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Pertussis Toxin; Phosphoprotein Phosphatases; Signal Transduction; Terpenes; Thapsigargin; Virulence Factors, Bordetella | 1996 |
Ca2+ entry induced by calcium influx factor and its regulation by protein kinase C in rabbit neutrophils.
Topics: Adrenal Glands; Alkaloids; Animals; Azepines; Calcium; Calcium Channel Blockers; Cattle; Chromaffin Granules; Enzyme Inhibitors; Imidazoles; Ion Transport; Neutrophils; Platelet Activating Factor; Protein Kinase C; Rabbits; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Triazoles | 1996 |
Inhibition by SK&F96365 of NO-mediated relaxation induced by Ca2(+) -ATPase inhibitors in rat thoracic aorta.
Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cyclic GMP; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Indoles; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nickel; Nitric Oxide; Rats; Rats, Wistar; Terpenes; Thapsigargin | 1996 |
Calcium handling and purinoceptor subtypes involved in ATP-induced contraction in rat small mesenteric arteries.
Topics: Adenosine Triphosphate; Animals; Caffeine; Calcium; Calcium Channel Blockers; Imidazoles; Male; Mesenteric Arteries; Muscle Contraction; Nitrendipine; Pertussis Toxin; Platelet Aggregation Inhibitors; Purinergic Agonists; Purinergic Antagonists; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Purinergic; Terpenes; Thapsigargin; Vascular Resistance; Virulence Factors, Bordetella | 1996 |
Inhibition of prostanoid formation in intact cells by 2,5-di-(tert-butyl)-1,4-benzohydroquinone, a blocker of Ca(2+)-ATPases.
Topics: Arachidonic Acid; Blood Platelets; Bradykinin; Calcimycin; Calcium-Transporting ATPases; Cell Line; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Humans; Imidazoles; In Vitro Techniques; Ionophores; Platelet Aggregation Inhibitors; Prostaglandins; Thapsigargin | 1996 |
Two different store-operated Ca2+ entry pathways in MDCK cells.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Dogs; Electric Conductivity; Imidazoles; Inositol 1,4,5-Trisphosphate; Lanthanum; Potassium Channels; Thapsigargin | 1996 |
Inhibition by fenamates of calcium influx and proliferation of human lymphocytes.
Topics: Analysis of Variance; Anti-Inflammatory Agents, Non-Steroidal; Calcium; Cell Division; Concanavalin A; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flufenamic Acid; Humans; Imidazoles; Lymphocytes; Manganese; ortho-Aminobenzoates; Tetradecanoylphorbol Acetate; Thapsigargin | 1996 |
SK&F 96365 inhibits intracellular Ca2+ pumps and raises cytosolic Ca2+ concentration without production of nitric oxide and von Willebrand factor.
Topics: Adenosine Triphosphate; Biological Transport; Blood Platelets; Calcium; Calcium Channel Blockers; Calcium Radioisotopes; Calcium-Transporting ATPases; Cells, Cultured; Cytoplasm; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epithelial Cells; Epithelium; Humans; Imidazoles; Intracellular Membranes; Nitric Oxide; Thapsigargin; Umbilical Veins; von Willebrand Factor | 1996 |
Ca2+ entry following store depletion in SH-SY5Y neuroblastoma cells.
Topics: Barium; Calcium; Cell Membrane Permeability; Imidazoles; Inositol 1,4,5-Trisphosphate; Lanthanum; Manganese; Muscarinic Agonists; Neuroblastoma; Neurons; Oxotremorine; Strontium; Thapsigargin; Tumor Cells, Cultured | 1996 |
Store-operated Ca2+ entry and coupling to Ca2+ pool depletion in thapsigargin-resistant cells.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cell Compartmentation; Cells, Cultured; Cricetinae; Cricetulus; Cytosol; Drug Resistance; Endoplasmic Reticulum; Enzyme Inhibitors; Imidazoles; Ionomycin; Ionophores; Lysophospholipids; Thapsigargin | 1997 |
Thapsigargin-induced gene expression in nonexcitable cells is dependent on calcium influx.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Chloramphenicol O-Acetyltransferase; Endothelin-1; Enzyme Activation; Gene Expression Regulation; Genes, fos; Genes, Reporter; Imidazoles; Rats; Thapsigargin; Triazoles | 1997 |
Cellular uptake of lead is activated by depletion of intracellular calcium stores.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Enzyme Inhibitors; Fluorescent Dyes; Humans; Hydroquinones; Imidazoles; Indoles; Lanthanum; Lead; Rats; Spectrometry, Fluorescence; Thapsigargin | 1997 |
Regulation of cytosolic free Ca2+ in cultured rat alveolar macrophages (NR8383).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Calcium; Calcium-Transporting ATPases; Cells, Cultured; Cytosol; Enzyme Inhibitors; Imidazoles; Inositol 1,4,5-Trisphosphate; Macrophages, Alveolar; Membrane Potentials; Rats; Receptors, Purinergic P2; Thapsigargin; Zymosan | 1997 |
Calcium store depletion activates two distinct calcium entry pathways in secretory cells of the blowfly salivary gland.
Topics: Animals; Biological Transport; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Chelating Agents; Diptera; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Inhibitors; Gadolinium; Imidazoles; Ion Channel Gating; Lanthanum; Microsomes; Salivary Glands; Serotonin; Thapsigargin; Time Factors | 1998 |
Comparison of contractions produced by carbachol, thapsigargin and cyclopiazonic acid in the guinea-pig tracheal muscle.
Topics: Animals; Cadmium; Calcium Channel Blockers; Carbachol; Female; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Isoproterenol; Male; Muscle Contraction; Nitroprusside; Thapsigargin; Trachea | 1998 |
Dissociation of intracellular Ca2+ release and Ca2+ entry response to 5-hydroxytryptamine in cultured canine tracheal smooth muscle cells.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cells, Cultured; Dogs; Enzyme Inhibitors; Imidazoles; Indoles; Inositol Phosphates; Kinetics; Lanthanum; Membrane Potentials; Muscle, Smooth; Serotonin; Signal Transduction; Thapsigargin; Trachea | 1998 |
Characterisation of calcium signalling in DT40 chicken B-cells.
Topics: Animals; B-Lymphocytes; Calcium; Calcium Signaling; Cell Line; Cell Membrane; Chickens; Dose-Response Relationship, Drug; Hydrogen Peroxide; Imidazoles; Immunoglobulin M; Thapsigargin; Verapamil | 1998 |
Mechanism of rise and decay of thapsigargin-evoked calcium signals in MDCK cells.
Topics: Animals; Bradykinin; Calcium; Calcium Signaling; Calcium-Transporting ATPases; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cell Line; Dogs; Econazole; Egtazic Acid; Endoplasmic Reticulum; Gadolinium; Hydrogen-Ion Concentration; Imidazoles; Indoles; Lanthanum; Manganese; Mitochondria; Sodium; Thapsigargin | 1999 |
Multiple effects of 1-[beta-[3-(4-methoxyphenyl)propoxy]-4-methoxyphenethyl]-1H-imidazole hydrochloride (SKF 96365) on Ca2+ signaling in MDCK cells: depletion of thapsigargin-sensitive Ca2+ store followed by capacitative Ca2+ entry, activation of a direct
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Signaling; Cell Line; Dogs; Electric Conductivity; Endoplasmic Reticulum; Fluorometry; Fura-2; Imidazoles; Kidney; Thapsigargin; Uridine Triphosphate | 1999 |
Listeria monocytogenes phospholipase C-dependent calcium signaling modulates bacterial entry into J774 macrophage-like cells.
Topics: Bacterial Proteins; Calcium Channel Blockers; Calcium Signaling; Cell Line; Cytosol; Imidazoles; Listeria monocytogenes; Macrophages; Mutagenesis; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide Phospholipase C; Thapsigargin; Type C Phospholipases; Vacuoles | 1999 |
Mechanisms of the relaxant and contractile responses to bradykinin in rat duodenum.
Topics: Acetylcholine; Animals; Apamin; Bradykinin; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Charybdotoxin; Duodenum; Enzyme Inhibitors; Estrenes; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Channel Blockers; Pyrrolidinones; Rats; Signal Transduction; Thapsigargin; Type C Phospholipases | 1999 |
Activation of three types of voltage-independent Ca2+ channel in A7r5 cells by endothelin-1 as revealed by a novel Ca2+ channel blocker LOE 908.
Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cations; Cells, Cultured; Drug Interactions; Endothelin-1; Imidazoles; Ionomycin; Isoquinolines; Patch-Clamp Techniques; Rats; Thapsigargin | 1999 |
Redox modulation of intracellular free calcium concentration in thyroid FRTL-5 cells: evidence for an enhanced extrusion of calcium.
Topics: Animals; Barium; Calcium; Calcium-Transporting ATPases; Cell Line; Enzyme Activation; Hydrogen-Ion Concentration; Imidazoles; Membrane Potentials; Mercaptoethanol; Oxidation-Reduction; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Binding; Protein Kinase C; Rats; Staurosporine; tert-Butylhydroperoxide; Tetradecanoylphorbol Acetate; Thapsigargin; Thimerosal; Thyroid Gland; Vanadates | 1999 |
Bradykinin-induced phosphoinositide hydrolysis and Ca2+ mobilization in canine cultured tracheal epithelial cells.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Calcium Channel Blockers; Cells, Cultured; Cholera Toxin; Dogs; Enzyme Inhibitors; Epithelial Cells; Estrenes; Female; Hydrolysis; Imidazoles; Male; Pertussis Toxin; Phosphatidylinositols; Pyrrolidinones; Receptor, Bradykinin B2; Thapsigargin; Trachea; Type C Phospholipases; Virulence Factors, Bordetella | 1999 |
Troglitazone inhibits the capacitative Ca2+ entry in endothelial cells.
Topics: Adenosine Triphosphate; Animals; Aorta; Bradykinin; Calcium; Calcium Channel Blockers; Cells, Cultured; Chromans; Diltiazem; Endothelin-1; Endothelium, Vascular; Enzyme Inhibitors; Imidazoles; Swine; Thapsigargin; Thiazoles; Thiazolidinediones; Time Factors; Troglitazone; Vasodilator Agents | 1999 |
Release of O2- by human umbilical cord blood-derived eosinophils: role of intra- and extracellular calcium.
Topics: Calcium; Calcium Channel Blockers; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Eosinophils; Fetal Blood; Humans; Imidazoles; Ionomycin; Magnesium; N-Formylmethionine Leucyl-Phenylalanine; Nickel; Oxygen; Platelet Activating Factor; Respiratory Burst; Spectrometry, Fluorescence; Thapsigargin | 1999 |
Possible involvement of Ca2+ entry and its pharmacological characteristics responsible for endothelium-dependent, NO-mediated relaxation induced by thapsigargin in guinea-pig aorta.
Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Extracellular Space; Female; Guinea Pigs; Imidazoles; In Vitro Techniques; Male; Nickel; Nitric Oxide; Potassium; Thapsigargin; Vasodilation | 1999 |
Mechanisms through which PDGF alters intracellular calcium levels in U-1242 MG human glioma cells.
Topics: Becaplermin; Brain Neoplasms; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Elapid Venoms; Endoplasmic Reticulum; Enzyme Inhibitors; Flufenamic Acid; Glioma; Humans; Imidazoles; Ion Transport; Masoprocol; Neoplasm Proteins; Nicardipine; Nimodipine; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Peptides; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Ryanodine; Thapsigargin; Tumor Cells, Cultured; Verapamil | 1999 |
Thapsigargin-induced tone and capacitative calcium influx in mouse anococcygeus smooth muscle cells.
Topics: Animals; Cadmium; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Fluorescence; Fura-2; Genistein; Imidazoles; In Vitro Techniques; Male; Manganese; Mice; Muscle Contraction; Muscle, Smooth; Thapsigargin; Time Factors; Verapamil | 1999 |
Effects of inhibitors for tyrosine kinase and non-selective cation channel on capacitative Ca(2+) entry in rat ileal smooth muscle.
Topics: Alkaloids; Animals; Benzylisoquinolines; Caffeine; Calcium; Calcium Channels; Enzyme Inhibitors; Genistein; Ileum; Imidazoles; Male; Muscle Contraction; Muscle, Smooth; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Thapsigargin; Tyrphostins | 2000 |
Distinct Ca(2+) signalling mechanisms induced by ATP and sphingosylphosphorylcholine in porcine aortic smooth muscle cells.
Topics: Adenosine; Adenosine Triphosphate; Animals; Aorta; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Cyclic AMP; Egtazic Acid; Estrenes; Imidazoles; Ionomycin; Manganese; Muscle, Smooth, Vascular; Phosphorylcholine; Pyrrolidinones; Sphingosine; Staurosporine; Swine; Thapsigargin; Thionucleosides; Thionucleotides; Virulence Factors, Bordetella | 2000 |
Store-operated Ca(2+) inflow in Reuber hepatoma cells is inhibited by voltage-operated Ca(2+) channel antagonists and, in contrast to freshly isolated hepatocytes, does not require a pertussis toxin-sensitive trimeric GTP-binding protein.
Topics: Animals; Brefeldin A; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Calmodulin; Chelating Agents; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Inhibitors; Gadolinium; Heterotrimeric GTP-Binding Proteins; Hydroquinones; Imidazoles; Indoles; Liver; Pertussis Toxin; Sulfonamides; Thapsigargin; Tumor Cells, Cultured; Virulence Factors, Bordetella | 2000 |
Voltage-independent calcium entry in hypoxic pulmonary vasoconstriction of intrapulmonary arteries of the rat.
Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Chelating Agents; Diltiazem; Dinucleoside Phosphates; Egtazic Acid; Electric Stimulation; Enzyme Inhibitors; Hypoxia; Imidazoles; In Vitro Techniques; Ion Channel Gating; Lanthanum; Male; Membrane Potentials; Nifedipine; Phosphodiesterase Inhibitors; Pulmonary Artery; Pulmonary Circulation; Rats; Rats, Wistar; Ryanodine; Thapsigargin; Vasoconstriction; Verapamil | 2000 |
The involvement of intracellular Ca(2+) in 5-HT(1B/1D) receptor-mediated contraction of the rabbit isolated renal artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Actin Cytoskeleton; Animals; Caffeine; Calcium; Calcium Channel Blockers; Capillary Permeability; Dose-Response Relationship, Drug; Female; Fluorescence; Fura-2; Imidazoles; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Potassium; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Renal Artery; Serotonin; Thapsigargin; Vasoconstrictor Agents | 2000 |
Two pathways for store-mediated calcium entry in human platelets.
Topics: Androstadienes; Biological Transport; Blood Platelets; Calcium; Calcium Channel Blockers; Calcium Signaling; Chelating Agents; Econazole; Egtazic Acid; Enzyme Inhibitors; Humans; Imidazoles; Ionomycin; Ionophores; Lanthanum; Manganese; Phosphorylation; Protein-Tyrosine Kinases; Thapsigargin; Tyrosine; Wortmannin | 2000 |
Comparison of the Ca2+ entry channels responsible for mechanical responses of guinea-pig aorta to noradrenaline and thapsigargin using SK&F 96365 and LOE 908.
Topics: Acetamides; Animals; Aorta, Thoracic; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Cytoplasm; Enzyme Inhibitors; Extracellular Space; Female; Guinea Pigs; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Thapsigargin; Type C Phospholipases | 2000 |
Bcl-2 overexpression results in enhanced capacitative calcium entry and resistance to SKF-96365-induced apoptosis.
Topics: Apoptosis; Calcium; Calcium Channel Blockers; Calcium Channels; Dose-Response Relationship, Drug; Drug Resistance; Electric Conductivity; Electric Impedance; Endoplasmic Reticulum; Enzyme Inhibitors; HL-60 Cells; Humans; Imidazoles; Ion Channel Gating; Jurkat Cells; Membrane Potentials; Ouabain; Proto-Oncogene Proteins c-bcl-2; Thapsigargin; Transfection | 2000 |
Pharmacological evaluation of the role of cytochrome P450 in intracellular calcium signalling in rat pancreatic acinar cells.
Topics: Animals; Calcium Signaling; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Enzyme Induction; Fatty Acids, Unsaturated; Imidazoles; Indoles; Ketoconazole; Male; Pancreas; Proadifen; Rats; Rats, Sprague-Dawley; Sincalide; Thapsigargin | 2000 |
Regulation of phosphatidylserine transbilayer redistribution by store-operated Ca2+ entry: role of actin cytoskeleton.
Topics: Actins; Annexin A5; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Cytochalasin D; Cytoskeleton; Enzyme Inhibitors; Humans; Imidazoles; Lanthanum; Lipid Bilayers; Miconazole; Phosphatidylserines; Thapsigargin; Tumor Cells, Cultured | 2001 |
Chlorpromazine inhibits store-operated calcium entry and subsequent noradrenaline secretion in PC12 cells.
Topics: Algorithms; Animals; Antipsychotic Agents; Calcium; Calcium Channel Blockers; Calcium Signaling; Calcium-Transporting ATPases; Chlorpromazine; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Imidazoles; Inositol 1,4,5-Trisphosphate; Manganese; Norepinephrine; PC12 Cells; Rats; Thapsigargin | 2001 |
Microdomains of high calcium are not required for exocytosis in RBL-2H3 mucosal mast cells.
Topics: Animals; Antifungal Agents; Antigens; Antimycin A; Calcimycin; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Enzyme Inhibitors; Exocytosis; Imidazoles; Ionophores; Lanthanum; Mast Cells; Mucous Membrane; Oligomycins; Potassium; Rats; Serotonin; Spectrometry, Fluorescence; Thapsigargin; Tumor Cells, Cultured | 2001 |
Mechanisms of bradykinin-mediated Ca(2+) signalling in canine cultured corneal epithelial cells.
Topics: Animals; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Cholera Toxin; Dogs; Enzyme Inhibitors; Epithelium, Corneal; Estrenes; Imidazoles; Pertussis Toxin; Pyrrolidinones; Thapsigargin; Type C Phospholipases; Virulence Factors, Bordetella | 2001 |
Failure of endothelin-1 to activate store-operated Ca2+ channels by lack of mobilization from intracellular Ca2+ stores in cultured bovine adrenal chromaffin cells.
Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cattle; Cells, Cultured; Chromaffin Cells; Endothelin-1; Enzyme Inhibitors; Imidazoles; Ion Channels; Isoquinolines; Thapsigargin | 2001 |
Characterization of the mGluR(1)-mediated electrical and calcium signaling in Purkinje cells of mouse cerebellar slices.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Signaling; Calcium-Transporting ATPases; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Imidazoles; Indoles; Mice; Mice, Inbred ICR; Nimodipine; Organ Culture Techniques; Patch-Clamp Techniques; Purkinje Cells; Receptors, Metabotropic Glutamate; Resorcinols; Sarcoplasmic Reticulum; Sodium; Thapsigargin | 2001 |
Fendiline mobilizes intracellular Ca2+ in Chang liver cells.
Topics: Calcium; Calcium Channel Blockers; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cell Line; Dose-Response Relationship, Drug; Estrenes; Fendiline; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate; Liver; Phosphodiesterase Inhibitors; Pyrrolidinones; Thapsigargin; Time Factors; Type C Phospholipases | 2001 |
Selective inhibition of thapsigargin-induced contraction and capacitative calcium entry in mouse anococcygeus by trifluoromethylphenylimidazole (TRIM).
Topics: Animals; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Synthase; Nitroarginine; Potassium; Thapsigargin | 2001 |
Ca(2+) channels activated by endothelin-1 in CHO cells expressing endothelin-A or endothelin-B receptors.
Topics: Acetamides; Adenosine Triphosphatases; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; CHO Cells; Cricetinae; Electrophysiology; Endothelin-1; Enzyme Inhibitors; Imidazoles; Inositol Phosphates; Isoquinolines; Patch-Clamp Techniques; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Thapsigargin | 2001 |
Role of prostaglandin E(2) and Ca(2+) in bradykinin induced contractions of guinea-pig gallbladder in vitro.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Channels; Cations, Divalent; Culture Media; Dinoprostone; Gallbladder; Guinea Pigs; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Piroxicam; Thapsigargin | 2001 |
Mechanisms involved in alpha6beta1-integrin-mediated Ca(2+) signalling.
Topics: Adenosine Diphosphate Ribose; Calcium Channel Blockers; Calcium Signaling; Cyclic ADP-Ribose; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Humans; Imidazoles; Integrin alpha6beta1; Integrins; Jurkat Cells; Kinetics; Laminin; Pyrimidines; Pyrrolidinones; src-Family Kinases; T-Lymphocytes; Thapsigargin; Type C Phospholipases | 2001 |
Extracellular pH affects platelet aggregation associated with modulation of store-operated Ca(2+) entry.
Topics: Blood Platelets; Calcium; Calcium Channel Blockers; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Ion Transport; Platelet Aggregation; Thapsigargin | 2001 |
Residence of adenylyl cyclase type 8 in caveolae is necessary but not sufficient for regulation by capacitative Ca(2+) entry.
Topics: Adenylyl Cyclases; Calcium; Calcium Channel Blockers; Caveolae; Cell Line; Cholesterol; Colforsin; Cyclic AMP; Humans; Imidazoles; Ionomycin; Kinetics; Mutagenesis; Recombinant Proteins; Sequence Deletion; Thapsigargin; Transfection | 2002 |
Cloning and functional expression of human short TRP7, a candidate protein for store-operated Ca2+ influx.
Topics: Amino Acid Sequence; Brain; Calcium; Calcium Channel Blockers; Cell Line; Central Nervous System; Cloning, Molecular; DNA, Complementary; Enzyme Inhibitors; Epitopes; Exons; Female; Gene Library; Humans; Imidazoles; Ion Channels; Kidney; Male; Manganese; Membrane Proteins; Molecular Sequence Data; Oligonucleotides, Antisense; Phylogeny; Pituitary Gland; Protein Binding; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology, Amino Acid; Thapsigargin; Time Factors; Tissue Distribution; Transfection; TRPM Cation Channels | 2002 |
Rhythmic spontaneous contractions in the rat proximal colon.
Topics: Animals; Anti-Arrhythmia Agents; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Colon; Enzyme Inhibitors; Gastrointestinal Motility; Imidazoles; In Vitro Techniques; Indoles; Male; Myenteric Plexus; Nicardipine; Proto-Oncogene Proteins c-kit; Rats; Rats, Mutant Strains; Rats, Wistar; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Thapsigargin | 2001 |
Diacylglycerol activates the influx of extracellular cations in T-lymphocytes independently of intracellular calcium-store depletion and possibly involving endogenous TRP6 gene products.
Topics: Barium; Blotting, Western; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cations; Cell Line; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Imidazoles; Jurkat Cells; Membrane Potentials; Phytohemagglutinins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Strontium; T-Lymphocytes; Thapsigargin; Time Factors; TRPC Cation Channels | 2002 |
Mechanisms of bradykinin-induced glucagon release in clonal alpha-cells In-R1-G9: involvement of Ca(2+)-dependent and -independent pathways.
Topics: Animals; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Chelating Agents; Clone Cells; Cricetinae; Egtazic Acid; Endoplasmic Reticulum; Enzyme Inhibitors; Estrenes; Glucagon; Glucagonoma; GTP-Binding Proteins; Heparin; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Mesocricetus; Microinjections; Pancreatic Neoplasms; Pertussis Toxin; Phospholipase D; Pyrrolidinones; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thapsigargin; Tumor Cells, Cultured; Type C Phospholipases | 2002 |
Role of endothelial Ca2+ stores in the regulation of hydraulic conductivity of Rana microvessels in vivo.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Capillary Permeability; Endoplasmic Reticulum; Endothelium, Vascular; Enzyme Inhibitors; Imidazoles; Indoles; Ionomycin; Male; Mesentery; Microcirculation; Nickel; Rana temporaria; Sarcoplasmic Reticulum; Thapsigargin | 2003 |
Store-operated calcium channels trigger exocytosis of the sea urchin sperm acrosomal vesicle.
Topics: Acrosome; Acrosome Reaction; Actins; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Exocytosis; Fucose; Hydrogen-Ion Concentration; Imidazoles; Kinetics; Male; Sea Urchins; Secretory Vesicles; Sulfuric Acids; Thapsigargin | 2003 |
ML-9, a myosin light chain kinase inhibitor, reduces intracellular Ca2+ concentration in guinea pig trachealis.
Topics: Androstadienes; Animals; Azepines; Calcium; Calcium Channel Blockers; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Isometric Contraction; Male; Methacholine Chloride; Muscarinic Agonists; Muscle, Smooth; Myosin-Light-Chain Kinase; Potassium; Potassium Channel Blockers; Thapsigargin; Trachea; Wortmannin | 2004 |
Presenilin-1 and intracellular calcium stores regulate neuronal glutamate uptake.
Topics: Amino Acid Transport System X-AG; Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Biological Transport; Caffeine; Calcium; Calcium Channel Blockers; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Endopeptidases; Enzyme Activators; Enzyme Inhibitors; Excitatory Amino Acid Transporter 3; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Imidazoles; Intracellular Fluid; Kainic Acid; Membrane Proteins; Mice; Mice, Knockout; Neurons; Presenilin-1; Protein Kinase C; Symporters; Thapsigargin | 2004 |
Exploring the pharmacology of the leukotriene B4 receptor BLT1, without the confounding effects of BLT2.
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Cytosol; Dantrolene; Dose-Response Relationship, Drug; Estrenes; Fatty Alcohols; Glycols; HeLa Cells; Humans; Imidazoles; Indoles; Intracellular Space; Maleimides; Nickel; Nifedipine; Plasmids; Propranolol; Protein Kinase Inhibitors; Pyrrolidinones; Receptors, Leukotriene B4; Staurosporine; Tetradecanoylphorbol Acetate; Thapsigargin; Transfection | 2004 |
Lafutidine-induced increase in intracellular ca(2+) concentrations in PC12 and endothelial cells.
Topics: Acetamides; Animals; Calcium; Calcium Chloride; Capsaicin; Dose-Response Relationship, Drug; Endothelial Cells; Humans; Imidazoles; Immunoblotting; Intracellular Fluid; PC12 Cells; Piperidines; Pyridines; Rats; Thapsigargin; Time Factors | 2005 |
Trans- and cis-resveratrol increase cytoplasmic calcium levels in A7r5 vascular smooth muscle cells.
Topics: Animals; Aorta; Calcium; Cell Line; Cytoplasm; Drug Synergism; Embryo, Mammalian; Imidazoles; Muscle, Smooth, Vascular; Nickel; Nifedipine; Rats; Resveratrol; Stereoisomerism; Stilbenes; Thapsigargin | 2005 |
Increased transient receptor potential channel TRPC3 expression in spontaneously hypertensive rats.
Topics: Animals; Blotting, Western; Calcium; Calcium Channel Blockers; Imidazoles; Male; Monocytes; Rats; Rats, Inbred SHR; Rats, Inbred WKY; RNA Interference; RNA, Small Interfering; Thapsigargin; Transfection; TRPC Cation Channels | 2005 |
A role for 5,6-epoxyeicosatrienoic acid in calcium entry by de novo conformational coupling in human platelets.
Topics: 8,11,14-Eicosatrienoic Acid; Actins; Antibodies; Blood Platelets; Boron Compounds; Calcium; Calcium Channels; Cell Membrane; Cell Membrane Permeability; Cytochalasin D; Cytochrome P-450 Enzyme System; Cytoskeleton; Enzyme Activation; Humans; Hydrogen Peroxide; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Lanthanum; Manganese; Nickel; Protein-Tyrosine Kinases; Receptors, Cytoplasmic and Nuclear; Thapsigargin; TRPC Cation Channels | 2006 |
PAR-1-stimulated factor IXa binding to a small platelet subpopulation requires a pronounced and sustained increase of cytoplasmic calcium.
Topics: Blood Platelets; Calcium; Cytoplasm; Factor IXa; Humans; Imidazoles; Ion Transport; Lanthanum; Macrocyclic Compounds; Oxazoles; Protein Binding; Receptor, PAR-1; Thapsigargin | 2006 |
Calcium-pH crosstalks in the human mast cell line HMC-1: intracellular alkalinization activates calcium extrusion through the plasma membrane Ca2+-ATPase.
Topics: Ammonium Chloride; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cell Line; Cell Membrane; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Imidazoles; Mast Cells; Nickel; Thapsigargin | 2006 |
Store-mediated calcium entry in pleural mesothelial cells.
Topics: Actins; Animals; Calcium; Cell Shape; Cells, Cultured; Cytochalasin D; Cytoskeleton; Depsipeptides; Epithelial Cells; Imidazoles; Marine Toxins; Microscopy, Confocal; Nifedipine; Oxazoles; Pleura; Rats; Thapsigargin | 2006 |
A store-operated Ca(2+) influx pathway in the bag cell neurons of Aplysia.
Topics: Anilides; Animals; Aplysia; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Electrophysiology; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Indicators and Reagents; Indoles; Inositol 1,4,5-Trisphosphate; Lanthanum; Macrocyclic Compounds; Membrane Potentials; Neurons; Nickel; Oxazoles; Ryanodine Receptor Calcium Release Channel; Thapsigargin; Thiadiazoles | 2006 |
Role of store-operated calcium channels and calcium sensitization in normoxic contraction of the ductus arteriosus.
Topics: Animals; Arachidonic Acids; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Cytosol; Ductus Arteriosus; Endocannabinoids; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoquinolines; Maleimides; Menthol; Mibefradil; Muscle Contraction; Nifedipine; Niflumic Acid; Oxidation-Reduction; Oxygen; Patch-Clamp Techniques; Polyunsaturated Alkamides; Potassium Channels; Protein Serine-Threonine Kinases; Rabbits; rho-Associated Kinases; Ruthenium Red; Sulfonamides; Tetraethylammonium; Thapsigargin; Thiourea | 2006 |
Temporal and spatial dynamics underlying capacitative calcium entry in human colonic smooth muscle.
Topics: Acetylcholine; Aged; Calcium; Calcium Channel Blockers; Calcium Signaling; Calcium-Transporting ATPases; Cholinergic Agents; Colon; Enzyme Inhibitors; Female; Humans; Imidazoles; Indoles; Lanthanum; Male; Membrane Potentials; Microscopy, Fluorescence; Muscle Contraction; Muscle, Smooth; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Thapsigargin; Time Factors | 2008 |
Capacitative calcium entry and proliferation of human osteoblast-like MG-63 cells.
Topics: Animals; Becaplermin; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Cycle; Cell Line; Cell Proliferation; Cell Survival; Electric Capacitance; Gene Expression Regulation; Humans; Imidazoles; Mice; Osteoblasts; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Serum; Thapsigargin; Transient Receptor Potential Channels | 2007 |
Differential effects of intravenous anesthetics on capacitative calcium entry in human pulmonary artery smooth muscle cells.
Topics: Anesthetics, Intravenous; Calcium; Calcium Channel Blockers; Calcium Channels; Carcinogens; Cells, Cultured; Enzyme Inhibitors; Humans; Imidazoles; Muscle, Smooth, Vascular; Protein Kinase C; Protein-Tyrosine Kinases; Pulmonary Artery; Signal Transduction; Tetradecanoylphorbol Acetate; Thapsigargin; Tyrphostins | 2008 |
Molecular characterization of Helicobacter pylori VacA induction of IL-8 in U937 cells reveals a prominent role for p38MAPK in activating transcription factor-2, cAMP response element binding protein, and NF-kappaB activation.
Topics: Activating Transcription Factor 2; Active Transport, Cell Nucleus; Bacterial Proteins; Butylated Hydroxyanisole; Cell Nucleus; Cyclic AMP Response Element-Binding Protein; Dantrolene; Egtazic Acid; Enzyme Activation; Helicobacter pylori; Humans; Imidazoles; Interleukin-8; NF-kappa B; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Promoter Regions, Genetic; Sulfones; Thapsigargin; U937 Cells; Up-Regulation | 2008 |
Automated patch-clamp technique: increased throughput in functional characterization and in pharmacological screening of small-conductance Ca2+ release-activated Ca2+ channels.
Topics: Animals; Automation; Calcium; Cell Line; Dose-Response Relationship, Drug; Egtazic Acid; Electrophysiology; Imidazoles; Inhibitory Concentration 50; Inositol 1,4,5-Trisphosphate; Ionomycin; Patch-Clamp Techniques; Platelet Aggregation Inhibitors; Rats; Thapsigargin | 2008 |
Role of symmetric dimethylarginine in vascular damage by increasing ROS via store-operated calcium influx in monocytes.
Topics: Angiotensin-Converting Enzyme Inhibitors; Anticoagulants; Arginine; Calcium; Calcium Channel Blockers; Calcium Channels; Captopril; Edetic Acid; Enzyme Inhibitors; Humans; Imidazoles; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Reactive Oxygen Species; Respiratory Burst; Thapsigargin; Vascular Diseases | 2009 |
A Stim1-dependent, noncapacitative Ca2+-entry pathway is activated by B-cell-receptor stimulation and depletion of Ca2+.
Topics: Animals; B-Lymphocytes; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Chickens; Enzyme Inhibitors; Genistein; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Jurkat Cells; Lanthanum; Membrane Glycoproteins; Protein-Tyrosine Kinases; Recombinant Fusion Proteins; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Thapsigargin; Time Factors; Transfection | 2009 |
Ca(2+) regulation of endocochlear potential in marginal cells.
Topics: Amiloride; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cochlea; Egtazic Acid; Endolymph; Epithelial Sodium Channels; Evoked Potentials, Auditory; Furosemide; Guinea Pigs; Imidazoles; Nifedipine; Sodium Channel Blockers; Sodium Potassium Chloride Symporter Inhibitors; Thapsigargin; TRPC Cation Channels | 2009 |
Calcium-sensing receptor activation contributed to apoptosis stimulates TRPC6 channel in rat neonatal ventricular myocytes.
Topics: Animals; Apoptosis; Calcium; Calcium Channel Blockers; Gadolinium; Heart Ventricles; Imidazoles; Muscle Cells; Rats; Rats, Wistar; Receptors, Calcium-Sensing; Thapsigargin; TRPC Cation Channels | 2010 |
Mechanisms of vasopressin-induced intracellular Ca2+ oscillations in rat inner medullary collecting duct.
Topics: Animals; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Calcium Signaling; Cyclic ADP-Ribose; Gadolinium; Imidazoles; Inositol 1,4,5-Trisphosphate; Kidney Medulla; Kidney Tubules, Collecting; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Ryanodine Receptor Calcium Release Channel; Thapsigargin | 2011 |
Effect of diindolylmethane on Ca(2+) movement and viability in HA59T human hepatoma cells.
Topics: Apoptosis; Calcium; Calcium Channel Blockers; Carcinoma, Hepatocellular; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Econazole; Endoplasmic Reticulum; Fura-2; Humans; Hydroquinones; Imidazoles; Indoles; Liver Neoplasms; Nifedipine; Phospholipases A2; Protein Kinase C; Tetrazolium Salts; Thapsigargin | 2011 |
The anti-inflammatory effect of the SOCC blocker SK&F 96365 on mouse lymphocytes after stimulation by Con A or PMA/ionomycin.
Topics: Animals; Anti-Inflammatory Agents; Antigens, CD; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Cycle; Cell Proliferation; Cells, Cultured; Concanavalin A; Cytokines; Dose-Response Relationship, Drug; Female; Fluoresceins; Fluorescent Dyes; Imidazoles; Inflammation; Ionomycin; Lymphocyte Activation; Lymphocyte Count; Membrane Potential, Mitochondrial; Mice; Mice, Inbred BALB C; Mitochondria; Signal Transduction; Succinimides; T-Lymphocytes; Tetradecanoylphorbol Acetate; Thapsigargin | 2011 |
Calcium influx blocked by SK&F 96365 modulates the LPS plus IFN-γ-induced inflammatory response in murine peritoneal macrophages.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Chemokine CCL2; Escherichia coli; Female; Imidazoles; Inflammation; Interferon-gamma; Interleukin-10; Interleukin-1beta; Interleukin-6; Ionomycin; Lipopolysaccharides; Macrophages, Peritoneal; Membrane Potential, Mitochondrial; Mice; Mice, Inbred BALB C; NF-kappa B; Nitric Oxide; Phagocytosis; Protein Transport; Reactive Oxygen Species; Thapsigargin; Tumor Necrosis Factor-alpha | 2012 |
Inhibition of thrombin-induced Ca²⁺ influx in platelets by R59949, an inhibitor of diacylglycerol kinase.
Topics: Blood Platelets; Butanols; Calcium; Calcium Channel Blockers; Cell Membrane; Diacylglycerol Kinase; Hemostatics; Humans; Imidazoles; Phosphatidic Acids; Piperidines; Plant Extracts; Platelet Aggregation; Propranolol; Quinazolinones; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thapsia; Thapsigargin; Thrombin | 2012 |
Effect of phenethyl isothiocyanate on Ca2+ movement and viability in MDCK canine renal tubular cells.
Topics: Animals; Apoptosis; Calcium; Calcium Signaling; Cell Survival; Cytosol; Dogs; Econazole; Egtazic Acid; Enzyme Inhibitors; Imidazoles; Isothiocyanates; Kidney Tubules; Madin Darby Canine Kidney Cells; Nifedipine; Thapsigargin | 2012 |
TMEM16A/ANO1 channels contribute to the myogenic response in cerebral arteries.
Topics: Animals; Anoctamin-1; Blood Pressure; Calcium Channel Blockers; Calcium Signaling; Cerebral Arteries; Cerebrovascular Circulation; Chloride Channels; Chlorides; HEK293 Cells; Humans; Imidazoles; Male; Myocytes, Smooth Muscle; Nimodipine; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; RNA, Small Interfering; Thapsigargin; Vasoconstriction | 2012 |
Store-operated calcium entry in vagal sensory nerves is independent of Orai channels.
Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Endoplasmic Reticulum; Enzyme Inhibitors; Gene Expression Regulation; Imidazoles; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Confocal; ORAI1 Protein; Sensory Receptor Cells; Thapsigargin; Time Factors; Transient Receptor Potential Channels; TRPA1 Cation Channel; Vagus Nerve | 2013 |
Contribution of TRPC3 to store-operated calcium entry and inflammatory transductions in primary nociceptors.
Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ganglia, Spinal; Gene Expression Regulation; Imidazoles; Male; Membrane Potentials; Nociceptors; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2Y2; Signal Transduction; Spinal Cord; Thapsigargin; Time Factors; TRPC Cation Channels; Type C Phospholipases | 2014 |
Mitochondrial Ca²⁺ uniporter is critical for store-operated Ca²⁺ entry-dependent breast cancer cell migration.
Topics: Breast Neoplasms; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Line, Tumor; Cell Movement; Female; Gene Expression Regulation, Neoplastic; Humans; Imidazoles; Mitochondria; Ruthenium Red; Thapsigargin | 2015 |
STIM Protein-NMDA2 Receptor Interaction Decreases NMDA-Dependent Calcium Levels in Cortical Neurons.
Topics: Animals; Calcium; Calcium Signaling; Cerebral Cortex; Down-Regulation; HEK293 Cells; HeLa Cells; Humans; Imidazoles; Models, Biological; N-Methylaspartate; Neurons; Protein Binding; Protein Subunits; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; RNA, Small Interfering; Stromal Interaction Molecule 1; Stromal Interaction Molecule 2; Thapsigargin | 2020 |