1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazole has been researched along with 2-aminoethoxydiphenyl borate in 62 studies
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 28 (45.16) | 29.6817 |
2010's | 32 (51.61) | 24.3611 |
2020's | 2 (3.23) | 2.80 |
Authors | Studies |
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Benedetti, A; Gamberucci, A; Giunti, R; Giurisato, E; McIntosh, DP; Pizzo, P; Tassi, M | 1 |
Bonnal, JL; Dewailly, E; Lemonnier, L; Mauroy, B; Prevarskaya, N; Roudbaraki, M; Shuba, Y; Skryma, R; Slomianny, C; Sydorenko, V; Thebault, S | 1 |
Baba, A; Fujisawa, S; Ikegaya, Y; Matsuki, N; Nishiyama, N; Yamada, MK; Yamada, RX; Yasui, T | 1 |
Barajas-López, C; Bazán-Perkins, B; Flores-Soto, E; Montaño, LM | 1 |
Boston, ME; Buescher, ES; Chacon-Cruz, E; Frech, GC; Oelberg, DG | 1 |
Abe, M; Koyama, Y; Santella, L; Yazaki, I | 1 |
Bristulf, J; Owman, C; Sabirsh, A | 1 |
Behra, T; Lhote, P; McManus, B; Poburko, D; Rahimian, R; Ruegg, UT; Szado, T; van Breemen, C | 1 |
Boddy, G; Cho, WJ; Daniel, EE; Willis, A | 1 |
Dumont, L; Fleckenstein-Grün, G; Weirich, J | 1 |
Bartegi, A; Ben-Amor, N; Pariente, JA; Redondo, PC; Rosado, JA; Salido, GM | 1 |
Kiyonaka, S; Mori, Y | 1 |
Folz, RJ; Liu, JQ; Yang, D | 1 |
Jiang, N; Liu, L; Zhang, C; Zhang, YL; Zhang, ZC; Zhang, ZM | 1 |
Cabrera, JA; Hong, F; Hong, Z; Nelson, DP; Olschewski, A; Varghese, A; Weir, EK | 1 |
Farley, JM; Liu, H | 1 |
Asai, K; Imaizumi, Y; Ohya, S; Yamazaki, D | 1 |
Jumarie, C; Labelle, D; Moreau, R | 1 |
Emala, CW; Gallos, G; Goubaeva, F; Mizuta, F; Mizuta, K; Panettieri, RA; Xu, D; Yang, J; Zhu, D | 1 |
Bomben, VC; Sontheimer, HW | 1 |
Delamere, NA; Mandal, A; Shahidullah, M | 1 |
Gu, Y; Meng, F; To, WK | 1 |
Bates, DO; Foster, RR; Mathieson, PW; Saleem, MA; Satchell, SC; Welsh, GI; Ye, Y; Zadeh, MA | 1 |
Chung, L; Moore, SD | 1 |
Hutchins, BI; Kalil, K; Li, L | 1 |
Diana, L; Palleschi, S; Rossi, B; Silvestroni, L | 1 |
Cao, T; Chen, X; Feng, X; He, H; Liu, D; Luo, Z; Ma, L; Ma, S; Tepel, M; Yan, Z; Yang, D; Zhu, Z | 1 |
De Paoli Lacerda, SH; Gelderman, MP; Holada, K; Semberova, J; Simak, J; Simakova, O | 1 |
Hatae, N; Ichikawa, A; Inazumi, T; Kuroiwa, K; Morimoto, K; Segi-Nishida, E; Sugimoto, Y; Tabata, H; Tanaka, S; Yamaoka, K; Yano, A | 1 |
Chen, W; Ke, JB; Wang, Z; Yang, XL | 1 |
Bishara, NB; Ding, H | 1 |
Fang, Y; Kelly, MJ; Qiu, J; Rønnekleiv, OK | 1 |
Fernando Olivera, J; Olivera, JF; Pizarro, G | 1 |
Falck, JR; Jacobs, ER; Li, J; Li, W; Liu, Y; Manthati, VL; Medhora, M; Rao, J; Wang, R; Zhu, D | 1 |
Chai, CY; Chang, WC; Chen, WC; Chiu, YC; Hou, MF; Huang, WC; Juo, SH; Lu, SR; Wang, JY; Wang, YS | 1 |
Li, W; Sun, S; Wu, X; Xue, Y; Zha, L; Zhang, H; Zou, F | 1 |
Grenett, HE; Halloran, BA; Huang, J; Sharifov, OF; Tabengwa, E; Umeda, PK; Urthaler, F; Wolkowicz, PE | 1 |
Donato, J; Elias, CF; Elmquist, JK; Lee, CE; Sohn, JW; Williams, KW; Zhao, JJ | 1 |
Chen, B; Hughes, JD; Liu, H; Perkins, E; Rollins, S | 1 |
Hilton, J; Rae, MG; Sharkey, J | 1 |
Chien, EJ; Lai, JN; Liao, CF; Lin, VH; Tarng, DC; Wang, OY | 1 |
Baran, CN; Girard, BM; May, V; Merriam, LA; Parsons, RL; Roman, CW | 1 |
Cai, C; Chu, X; Meng, X; Tang, S; Wang, X; Zou, F; Zou, M; Zou, W | 1 |
Chang, HC; Chen, YF; Chen, YT; Chiu, WT; Shen, MR; Wang, YK | 1 |
Cao, X; Gao, TM; Li, JH; Li, SJ; Liu, XA; Peng, MR; Wu, CY; Zhao, ST | 1 |
Bonales-Alatorre, E; Delgado-Enciso, I; Dobrovinskaya, O; Moreno-Galindo, EG; Nieto-Pescador, MG; Pottosin, I | 1 |
Endo, T; Komatsu, Y; Yanagawa, Y | 1 |
Chang, WC; Cheng, H; He, H; Kim, M; Lu, F; Mathew, R; Messina, J; Sarnaik, AA; Shen, J; Sun, J; Wang, D; Yang, S | 1 |
Randall, MD; Roberts, RE; Wong, PS | 1 |
Ishii, K; Kimura, H; Koike, S; Ogasawara, Y; Shibuya, N | 1 |
Behuliak, M; Bencze, M; Vavřínová, A; Zicha, J | 1 |
Chan, CM; Chen, Y; Hung, TS; Miller, AL; Shipley, AM; Webb, SE | 1 |
Goto, T; Iwata, Y; Kawada, T; Sun, W; Takahashi, N; Tominaga, M; Uchida, K; Wakabayashi, S | 1 |
Chang, CH; Chiu, SJ; Hsu, WL; Huang, YB; Li, HW; Liang, JL; Lin, MW; Tsai, MH; Wang, CH; Wu, CY; Yen, CJ; Yoshioka, T | 1 |
Edin, F; Hayashi, H; Li, H; Liu, W; Rask-Andersen, H | 1 |
Hishinuma, E; Ishida, H; Ishikawa, T; Saito, SY | 1 |
Cao, Y; Dong, P; Hao, J; Hu, Y; Jiang, L; Liu, Y; Lu, W; Lv, W; Shu, Y; Wang, L; Yang, Z; Zhang, Y | 1 |
Constantino-Jonapa, LA; Del Angel, RM; Dionicio, CL; Ludert, JE; Peña, F; Rosales, R; Ruiz, MC; Vazquez, C; Yocupicio-Monroy, M; Zambrano, JL | 1 |
Chai, CY; Chen, CH; Hsu, WL; Lu, JH; Tsai, MH; Wu, CY; Yen, CJ; Yoshioka, T; Yu, HS | 1 |
Gao, C; Gao, Z; Liu, X; Wei, T; Yan, J; Zhao, W; Zhao, X | 1 |
Diamandakis, D; Krolik, A; Salinska, E; Stafiej, A; Zych, A | 1 |
Albayrak, E; Kocabaş, F; Uslu, M | 1 |
1 review(s) available for 1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazole and 2-aminoethoxydiphenyl borate
Article | Year |
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[TRP channels as targets for novel calcium antagonists].
Topics: Anilides; Boron Compounds; Calcium; Calcium Channel Blockers; Drug Design; Humans; Imidazoles; Second Messenger Systems; Thiadiazoles; TRPC Cation Channels | 2005 |
61 other study(ies) available for 1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazole and 2-aminoethoxydiphenyl borate
Article | Year |
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Diacylglycerol activates the influx of extracellular cations in T-lymphocytes independently of intracellular calcium-store depletion and possibly involving endogenous TRP6 gene products.
Topics: Barium; Blotting, Western; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cations; Cell Line; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Imidazoles; Jurkat Cells; Membrane Potentials; Phytohemagglutinins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Strontium; T-Lymphocytes; Thapsigargin; Time Factors; TRPC Cation Channels | 2002 |
Alpha1-adrenergic receptors activate Ca(2+)-permeable cationic channels in prostate cancer epithelial cells.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Blotting, Western; Boron Compounds; Calcium; Calcium Channel Blockers; Cations; Cell Division; Diglycerides; Dioxanes; Electrophysiology; Epithelial Cells; Humans; Imidazoles; Male; Microscopy, Fluorescence; Prazosin; Prostatic Neoplasms; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; Time Factors; Tumor Cells, Cultured | 2003 |
Activity-evoked capacitative Ca2+ entry: implications in synaptic plasticity.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Dentate Gyrus; Excitatory Postsynaptic Potentials; Imidazoles; Ion Transport; Lanthanum; Long-Term Potentiation; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate | 2003 |
Role of sarcoplasmic reticulum Ca2+ content in Ca2+ entry of bovine airway smooth muscle cells.
Topics: Animals; Boron Compounds; Caffeine; Calcium; Calcium Channel Blockers; Carbachol; Cattle; Dose-Response Relationship, Drug; Gallopamil; Imidazoles; In Vitro Techniques; Lanthanum; Magnesium; Muscarinic Agonists; Muscle, Smooth; Nickel; Phosphodiesterase Inhibitors; Sarcoplasmic Reticulum; Trachea | 2003 |
Surfactant releases internal calcium stores in neutrophils by G protein-activated pathway.
Topics: Boron Compounds; Calcium; Cell Membrane; Cytosol; Gramicidin; GTP-Binding Proteins; Humans; Imidazoles; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Pertussis Toxin; Phospholipids; Potentiometry; Pulmonary Surfactant-Associated Proteins; Pulmonary Surfactants | 2004 |
Mechanisms of calcium elevation in the micromeres of sea urchin embryos.
Topics: Animals; Boron Compounds; Calcium; Calcium Signaling; Embryo, Nonmammalian; Endoplasmic Reticulum; Gadolinium; Imidazoles; Inositol 1,4,5-Trisphosphate; Macrocyclic Compounds; Microtubules; Oxazoles; Sea Urchins | 2004 |
Exploring the pharmacology of the leukotriene B4 receptor BLT1, without the confounding effects of BLT2.
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Cytosol; Dantrolene; Dose-Response Relationship, Drug; Estrenes; Fatty Alcohols; Glycols; HeLa Cells; Humans; Imidazoles; Indoles; Intracellular Space; Maleimides; Nickel; Nifedipine; Plasmids; Propranolol; Protein Kinase Inhibitors; Pyrrolidinones; Receptors, Leukotriene B4; Staurosporine; Tetradecanoylphorbol Acetate; Thapsigargin; Transfection | 2004 |
Basal calcium entry in vascular smooth muscle.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Radioisotopes; Dose-Response Relationship, Drug; Egtazic Acid; Gadolinium; Green Fluorescent Proteins; Imidazoles; Lanthanum; Male; Membrane Proteins; Microscopy, Confocal; Muscle, Smooth, Vascular; Nerve Tissue Proteins; Nifedipine; Rats; Rats, Inbred WKY; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Synaptosomal-Associated Protein 25; TRPC Cation Channels | 2004 |
Comparisons of neural and pacing activities in intestinal segments from W/W++ and W/W(V) mice.
Topics: Anesthetics, Local; Animals; Boron Compounds; Calcium Channel Blockers; Electric Stimulation; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Intestines; Mice; Mice, Inbred BALB C; Mice, Inbred Strains; Mice, Knockout; Muscle, Smooth; Myenteric Plexus; Nerve Block; Nitroarginine; Proto-Oncogene Proteins c-kit; Species Specificity; Tetrodotoxin | 2005 |
Contribution of capacitative and non-capacitative Ca2+-entry to M3-receptor-mediated contraction of porcine coronary smooth muscle.
Topics: Acetamides; Acetylcholine; Animals; Boron Compounds; Calcium; Calcium Channels; Coronary Vessels; Imidazoles; Isoquinolines; Muscle Contraction; Muscle, Smooth, Vascular; Receptor, Muscarinic M3; Swine | 2005 |
A role for 5,6-epoxyeicosatrienoic acid in calcium entry by de novo conformational coupling in human platelets.
Topics: 8,11,14-Eicosatrienoic Acid; Actins; Antibodies; Blood Platelets; Boron Compounds; Calcium; Calcium Channels; Cell Membrane; Cell Membrane Permeability; Cytochalasin D; Cytochrome P-450 Enzyme System; Cytoskeleton; Enzyme Activation; Humans; Hydrogen Peroxide; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Lanthanum; Manganese; Nickel; Protein-Tyrosine Kinases; Receptors, Cytoplasmic and Nuclear; Thapsigargin; TRPC Cation Channels | 2006 |
A novel bronchial ring bioassay for the evaluation of small airway smooth muscle function in mice.
Topics: Animals; Biological Assay; Boron Compounds; Bronchi; Bronchoconstrictor Agents; Calcium Channel Blockers; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Methacholine Chloride; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Papaverine; Potassium Chloride; Respiratory Mucosa; Ryanodine; Stress, Mechanical; Substance P; Vasodilator Agents | 2006 |
Effects of Ca2+ channel blockers on store-operated Ca2+ channel currents of Kupffer cells after hepatic ischemia/reperfusion injury in rats.
Topics: Animals; Boron Compounds; Calcium Channel Blockers; Calcium Channels; Cell Survival; Dose-Response Relationship, Drug; Econazole; Imidazoles; Kupffer Cells; Liver; Male; Miconazole; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Reperfusion Injury | 2006 |
Role of store-operated calcium channels and calcium sensitization in normoxic contraction of the ductus arteriosus.
Topics: Animals; Arachidonic Acids; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Cytosol; Ductus Arteriosus; Endocannabinoids; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoquinolines; Maleimides; Menthol; Mibefradil; Muscle Contraction; Nifedipine; Niflumic Acid; Oxidation-Reduction; Oxygen; Patch-Clamp Techniques; Polyunsaturated Alkamides; Potassium Channels; Protein Serine-Threonine Kinases; Rabbits; rho-Associated Kinases; Ruthenium Red; Sulfonamides; Tetraethylammonium; Thapsigargin; Thiourea | 2006 |
Prostaglandin E2 enhances acetylcholine-induced, Ca2+-dependent ionic currents in swine tracheal mucous gland cells.
Topics: Acetylcholine; Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Carrier Proteins; Cells, Cultured; Charybdotoxin; Colforsin; Dinoprostone; Epithelial Cells; Imidazoles; Ion Channels; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Mucous Membrane; Patch-Clamp Techniques; Peptide Fragments; Peptides; Potassium Channel Blockers; Prostaglandin Antagonists; Swine; Trachea; Xanthones | 2007 |
Characteristics of the ATP-induced Ca2+-entry pathway in the t-BBEC 117 cell line derived from bovine brain endothelial cells.
Topics: Adenosine Triphosphate; Animals; Biological Transport; Blood-Brain Barrier; Boron Compounds; Calcium; Cattle; Cell Line, Transformed; Diglycerides; Dose-Response Relationship, Drug; Endothelial Cells; Imidazoles; Nickel; TRPC Cation Channels | 2007 |
Capacitative calcium entry and proliferation of human osteoblast-like MG-63 cells.
Topics: Animals; Becaplermin; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Cycle; Cell Line; Cell Proliferation; Cell Survival; Electric Capacitance; Gene Expression Regulation; Humans; Imidazoles; Mice; Osteoblasts; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Serum; Thapsigargin; Transient Receptor Potential Channels | 2007 |
Expression and coupling of neurokinin receptor subtypes to inositol phosphate and calcium signaling pathways in human airway smooth muscle cells.
Topics: Boron Compounds; Calcium Signaling; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate; Muscle, Smooth; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Trachea | 2008 |
Inhibition of transient receptor potential canonical channels impairs cytokinesis in human malignant gliomas.
Topics: Biopsy; Blotting, Western; Boron Compounds; Brain Neoplasms; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Glioma; Humans; Imidazoles; Immunohistochemistry; Transient Receptor Potential Channels | 2008 |
Ouabain-induced stimulation of sodium-hydrogen exchange in rat optic nerve astrocytes.
Topics: Amiloride; Ammonium Chloride; Animals; Astrocytes; Boron Compounds; Calcium; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Fluoresceins; Fluorescent Dyes; Hydrogen-Ion Concentration; Imidazoles; Ion Channel Gating; Isoquinolines; Optic Nerve; Ouabain; Rats; Sodium; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sulfonamides | 2008 |
Role of TRP channels and NCX in mediating hypoxia-induced [Ca(2+)](i) elevation in PC12 cells.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gene Expression Regulation; Hypoxia; Imidazoles; Models, Biological; PC12 Cells; Potassium Chloride; Rats; Sodium-Calcium Exchanger; Suramin; Thiourea; TRPC Cation Channels; Verapamil | 2008 |
Flufenamic acid is a tool for investigating TRPC6-mediated calcium signalling in human conditionally immortalised podocytes and HEK293 cells.
Topics: Boron Compounds; Calcium; Calcium Signaling; Cell Line, Transformed; Flufenamic Acid; Humans; Imidazoles; Indomethacin; Intracellular Space; Ion Channel Gating; Niflumic Acid; Podocytes; Transfection; TRPC Cation Channels; TRPC6 Cation Channel | 2009 |
Cholecystokinin excites interneurons in rat basolateral amygdala.
Topics: Amygdala; Analysis of Variance; Animals; Animals, Newborn; Benzodiazepines; Biophysics; Boron Compounds; Cadmium; Calcium; Calcium Channel Blockers; Cholagogues and Choleretics; Cholecystokinin; Electric Stimulation; Imidazoles; In Vitro Techniques; Interneurons; Male; Patch-Clamp Techniques; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Sodium Channel Blockers; Tetraethylammonium; Tetrodotoxin | 2009 |
Wnt5a induces simultaneous cortical axon outgrowth and repulsive axon guidance through distinct signaling mechanisms.
Topics: Analysis of Variance; Animals; Animals, Newborn; Axons; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Signaling; Cell Movement; Cells, Cultured; Cerebral Cortex; Cricetinae; Dose-Response Relationship, Drug; Electroporation; Estrenes; Frizzled Receptors; Green Fluorescent Proteins; Imidazoles; Mesocricetus; Neurons; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptor Protein-Tyrosine Kinases; RNA, Small Interfering; Signal Transduction; Sulfonamides; Time Factors; Wnt Proteins | 2009 |
Di(2-ethylhexyl)phthalate stimulates Ca(2+) entry, chemotaxis and ROS production in human granulocytes.
Topics: Adult; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Signaling; Chemotaxis; Diethylhexyl Phthalate; Drug Antagonism; Econazole; Granulocytes; Humans; Imidazoles; Male; Middle Aged; Plasticizers; Reactive Oxygen Species; Tetradecanoylphorbol Acetate | 2009 |
Increased rhythmicity in hypertensive arterial smooth muscle is linked to transient receptor potential canonical channels.
Topics: Amlodipine; Angiotensin II Type 1 Receptor Blockers; Animals; Arterioles; Benzimidazoles; Benzoates; Biphenyl Compounds; Blood Pressure; Boron Compounds; Calcium; Calcium Channels; Hypertension; Imidazoles; In Vitro Techniques; Muscle, Smooth, Vascular; Norepinephrine; Periodicity; Random Allocation; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Telmisartan; Tetrazoles; TRPC Cation Channels; Verapamil | 2010 |
Carbon nanotubes activate blood platelets by inducing extracellular Ca2+ influx sensitive to calcium entry inhibitors.
Topics: Antigens, CD; Biomarkers; Blood Platelets; Boron Compounds; Calcium; Calcium Channel Blockers; Humans; Imidazoles; Nanotubes, Carbon; P-Selectin; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Tetraspanin 30; Time Factors | 2009 |
Prostaglandin EP3 receptor superactivates adenylyl cyclase via the Gq/PLC/Ca2+ pathway in a lipid raft-dependent manner.
Topics: Adenylyl Cyclases; Animals; Boron Compounds; Calcium; Caveolin 1; Chlorocebus aethiops; COS Cells; Enzyme Activation; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; Humans; Imidazoles; Ionophores; Membrane Microdomains; Pyrrolidinones; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Staurosporine; Type C Phospholipases | 2009 |
Characterization of spontaneous inhibitory postsynaptic currents in cultured rat retinal amacrine cells.
Topics: Amacrine Cells; Animals; Bicuculline; Boron Compounds; Cadmium Chloride; Calcium; Calcium Channel Blockers; Cells, Cultured; Dantrolene; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Imidazoles; Inhibitory Postsynaptic Potentials; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Membrane Potentials; Oxazoles; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2010 |
Glucose enhances expression of TRPC1 and calcium entry in endothelial cells.
Topics: Adenosine Triphosphate; Animals; Antisense Elements (Genetics); Arachidonic Acid; Blotting, Western; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cattle; Cells, Cultured; Endothelial Cells; Gadolinium; Glucose; Imidazoles; Indicators and Reagents; TRPC Cation Channels | 2010 |
Leptin excites proopiomelanocortin neurons via activation of TRPC channels.
Topics: Animals; Appetite; Boron Compounds; Calcium Channel Blockers; Calcium Signaling; Female; Flufenamic Acid; Green Fluorescent Proteins; Hypothalamus; Imidazoles; Ion Channel Gating; Janus Kinase 2; Lanthanum; Leptin; Male; Membrane Potentials; Mice; Mice, Transgenic; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phospholipase C gamma; Pro-Opiomelanocortin; Signal Transduction; Staining and Labeling; TRPC Cation Channels | 2010 |
Two inhibitors of store operated Ca2+ entry suppress excitation contraction coupling in frog skeletal muscle.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Excitation Contraction Coupling; Imidazoles; Muscle, Skeletal; Ranidae | 2010 |
Stable EET urea agonist and soluble epoxide hydrolase inhibitor regulate rat pulmonary arteries through TRPCs.
Topics: Animals; Boron Compounds; Caffeine; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Enzyme Inhibitors; Epoxide Hydrolases; Fatty Acids, Monounsaturated; Female; Imidazoles; Indoles; Lanthanum; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Pulmonary Artery; Rats; Rats, Wistar; Transient Receptor Potential Channels | 2011 |
Histamine regulates cyclooxygenase 2 gene activation through Orai1-mediated NFκB activation in lung cancer cells.
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Line, Tumor; Cyclooxygenase 2; Histamine; Humans; Imidazoles; Lung Neoplasms; NF-kappa B; ORAI1 Protein; RNA Interference; RNA, Small Interfering; Signal Transduction; Transcriptional Activation | 2011 |
Requirement for store-operated calcium entry in sodium butyrate-induced apoptosis in human colon cancer cells.
Topics: Apoptosis; Boron Compounds; Butyrates; Calcium; Calcium Signaling; Cell Line, Tumor; Chelating Agents; Colonic Neoplasms; Egtazic Acid; Endoplasmic Reticulum; Humans; Imidazoles; Membrane Proteins; Neoplasm Proteins; RNA Interference; Stromal Interaction Molecule 1 | 2012 |
Pharmacological evidence for Orai channel activation as a source of cardiac abnormal automaticity.
Topics: Animals; Atrial Function, Left; Azepines; Boron Compounds; Calcium Channel Blockers; Calcium Channels; Calmodulin; Gene Expression Regulation; Heart; Heart Ventricles; Imidazoles; In Vitro Techniques; Myocardium; Naphthalenes; ORAI1 Protein; Rats | 2011 |
The acute effects of leptin require PI3K signaling in the hypothalamic ventral premammillary nucleus.
Topics: Androstadienes; Animals; Boron Compounds; Chromones; Female; Genes, Reporter; Hypothalamus; Imidazoles; KATP Channels; Leptin; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Morpholines; Neurons; Patch-Clamp Techniques; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Subunits; Signal Transduction; TRPC Cation Channels; Wortmannin | 2011 |
Calcium entry via ORAI1 regulates glioblastoma cell proliferation and apoptosis.
Topics: Animals; Apoptosis; Boron Compounds; Calcium; Calcium Channels; Calcium Signaling; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Diethylstilbestrol; Endoplasmic Reticulum; Fura-2; Gene Expression Regulation, Neoplastic; Glioblastoma; Humans; Imidazoles; Membrane Glycoproteins; Membrane Proteins; Neoplasm Proteins; ORAI1 Protein; Rats; RNA, Small Interfering; Stromal Interaction Molecule 1 | 2011 |
Putative TRP channel antagonists, SKF 96365, flufenamic acid and 2-APB, are non-competitive antagonists at recombinant human α1β2γ2 GABA(A) receptors.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Binding, Competitive; Boron Compounds; Flufenamic Acid; GABA-A Receptor Antagonists; HEK293 Cells; Humans; Imidazoles; Receptors, GABA-A; Recombinant Proteins; TRPC Cation Channels | 2012 |
The non-genomic rapid acidification in peripheral T cells by progesterone depends on intracellular calcium increase and not on Na+/H+-exchange inhibition.
Topics: Adult; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Signaling; Cation Transport Proteins; Chelating Agents; Egtazic Acid; Estrenes; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Hydrogen-Ion Concentration; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Male; Nickel; Pertussis Toxin; Progesterone; Protein Kinase C; Pyrrolidinones; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Staurosporine; T-Lymphocytes; Type C Phospholipases; Young Adult | 2012 |
Pretreatment with nonselective cationic channel inhibitors blunts the PACAP-induced increase in guinea pig cardiac neuron excitability.
Topics: Action Potentials; Animals; Boron Compounds; Calcium Channel Blockers; Calcium Signaling; Female; Flufenamic Acid; Guinea Pigs; Heart Conduction System; Imidazoles; Ion Channels; Ion Transport; Laser Capture Microdissection; Male; Membrane Transport Modulators; Neurons; Pituitary Adenylate Cyclase-Activating Polypeptide; Polymerase Chain Reaction; Single-Cell Analysis; TRPC Cation Channels | 2012 |
Store-operated Ca2+ entry (SOCE) plays a role in the polarization of neutrophil-like HL-60 cells by regulating the activation of Akt, Src, and Rho family GTPases.
Topics: Boron Compounds; Calcium Channel Blockers; Calcium Signaling; Cell Polarity; Enzyme Activation; Gene Knockdown Techniques; HL-60 Cells; Humans; Imidazoles; Manganese; Membrane Proteins; N-Formylmethionine Leucyl-Phenylalanine; Neoplasm Proteins; Neutrophils; Proto-Oncogene Proteins c-akt; rho GTP-Binding Proteins; RNA Interference; src-Family Kinases; Stromal Interaction Molecule 1 | 2012 |
The ER Ca²⁺ sensor STIM1 regulates actomyosin contractility of migratory cells.
Topics: Actomyosin; Anilides; Boron Compounds; Calcium; Cell Line, Tumor; Cell Movement; Endoplasmic Reticulum; Humans; Imidazoles; Immunoblotting; Membrane Proteins; Microscopy, Confocal; Neoplasm Proteins; RNA Interference; Stromal Interaction Molecule 1; Thiadiazoles | 2013 |
Store-operated Ca2+ channels blockers inhibit lipopolysaccharide induced astrocyte activation.
Topics: Animals; Astrocytes; Boron Compounds; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cell Proliferation; Cells, Cultured; Female; Glial Fibrillary Acidic Protein; Imidazoles; Interleukin-1beta; Interleukin-6; Lipopolysaccharides; Male; Rats; Rats, Wistar | 2013 |
Mechanosensitive Ca²⁺-permeable channels in human leukemic cells: pharmacological and molecular evidence for TRPV2.
Topics: Amiloride; Boron Compounds; Calcium; Gene Expression; Humans; Imidazoles; Ion Channel Gating; Ion Transport; Jurkat Cells; Leukemia, T-Cell; Magnesium; Mechanotransduction, Cellular; Membrane Potentials; Patch-Clamp Techniques; Potassium; Reverse Transcriptase Polymerase Chain Reaction; RNA Interference; Ruthenium Red; Sodium; TRPV Cation Channels | 2015 |
Substance P Activates Ca2+-Permeable Nonselective Cation Channels through a Phosphatidylcholine-Specific Phospholipase C Signaling Pathway in nNOS-Expressing GABAergic Neurons in Visual Cortex.
Topics: Animals; Anthracenes; Boron Compounds; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agents; GABAergic Neurons; Glutamate Decarboxylase; Imidazoles; In Vitro Techniques; Isoindoles; Mice; Mice, Transgenic; Neurokinin-1 Receptor Antagonists; Nitric Oxide Synthase Type III; Patch-Clamp Techniques; Piperidines; Quinolines; Quinuclidines; Signal Transduction; Substance P; Type C Phospholipases; Visual Cortex | 2016 |
STIM1- and Orai1-mediated Ca(2+) oscillation orchestrates invadopodium formation and melanoma invasion.
Topics: Animals; Boron Compounds; Calcium; Calcium Channels; Calcium Signaling; Cell Line, Tumor; Enzyme Activation; Extracellular Matrix; Humans; Imidazoles; Lung Neoplasms; Matrix Metalloproteinase 14; Matrix Metalloproteinase Inhibitors; MCF-7 Cells; Melanoma; Membrane Proteins; Mice; Mice, Nude; Neoplasm Invasiveness; Neoplasm Proteins; Neoplasm Transplantation; ORAI1 Protein; src-Family Kinases; Stromal Interaction Molecule 1 | 2014 |
Sex differences in the role of transient receptor potential (TRP) channels in endothelium-dependent vasorelaxation in porcine isolated coronary arteries.
Topics: Animals; Boron Compounds; Bradykinin; Calcimycin; Coronary Vessels; Endothelium, Vascular; Female; Gene Expression Regulation; Hydrogen Peroxide; Imidazoles; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Pyrazoles; Sex Characteristics; Sulfonamides; Swine; Transient Receptor Potential Channels; Vasodilation | 2015 |
Polysulfide promotes neuroblastoma cell differentiation by accelerating calcium influx.
Topics: Animals; Boron Compounds; Calcium; Cell Differentiation; Cell Line, Tumor; Imidazoles; Ion Transport; Mice; Neurites; Neuroblastoma; Sulfides; Transient Receptor Potential Channels | 2015 |
Broad-range TRP channel inhibitors (2-APB, flufenamic acid, SKF-96365) affect differently contraction of resistance and conduit femoral arteries of rat.
Topics: Animals; Boron Compounds; Dose-Response Relationship, Drug; Femoral Artery; Flufenamic Acid; Imidazoles; Male; Muscle, Smooth, Vascular; Organ Culture Techniques; Rats; Rats, Wistar; Transient Receptor Potential Channels; Vasoconstriction | 2015 |
Inhibition of SOCE disrupts cytokinesis in zebrafish embryos via inhibition of cleavage furrow deepening.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Signaling; Cleavage Stage, Ovum; Cytokinesis; Embryo, Nonmammalian; Endoplasmic Reticulum; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Zebrafish | 2015 |
Activation of TRPV2 negatively regulates the differentiation of mouse brown adipocytes.
Topics: Adipocytes, Brown; Animals; Boron Compounds; Calcineurin Inhibitors; Calcium Channels; Cell Differentiation; Cells, Cultured; Cyclosporine; HEK293 Cells; Humans; Imidazoles; Lysophosphatidylcholines; Male; Mice; Mice, Inbred C57BL; Tacrolimus; TRPV Cation Channels | 2016 |
A Novel Strategy for TNF-Alpha Production by 2-APB Induced Downregulated SOCE and Upregulated HSP70 in O. tsutsugamushi-Infected Human Macrophages.
Topics: Animals; Boron Compounds; Down-Regulation; HSP70 Heat-Shock Proteins; Humans; Imidazoles; Intracellular Calcium-Sensing Proteins; Macrophages; Membrane Proteins; Mice; Orientia tsutsugamushi; Tumor Necrosis Factor-alpha | 2016 |
The effect of pulsed electric fields on the electrotactic migration of human neural progenitor cells through the involvement of intracellular calcium signaling.
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Signaling; Cell Line; Cell Movement; Cell Survival; Electricity; Humans; Imidazoles; Immunohistochemistry; Intracellular Space; Neural Stem Cells; Neurons; Time-Lapse Imaging | 2016 |
Differential Contribution of Nerve-Derived Noradrenaline to High K
Topics: Acetamides; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Boron Compounds; Calcium; Calcium Channel Blockers; Imidazoles; Ion Channels; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Potassium; Prazosin; Rats, Wistar | 2017 |
Orai1 mediates tumor-promoting store-operated Ca
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Cell Line, Tumor; Gastrointestinal Neoplasms; Gastrointestinal Stromal Tumors; Humans; Imidazoles; MAP Kinase Signaling System; ORAI1 Protein; Proto-Oncogene Proteins c-kit; Risk Factors; Transfection | 2017 |
Dengue virus induced changes in Ca
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Calcium Chelating Agents; Cell Line, Tumor; Cell Membrane; Cell Membrane Permeability; Chlorocebus aethiops; Dengue Virus; Egtazic Acid; Endoplasmic Reticulum; Gene Expression; Hep G2 Cells; Homeostasis; Host-Pathogen Interactions; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Ion Transport; Neoplasm Proteins; ORAI1 Protein; Stromal Interaction Molecule 1; Vero Cells; Vesicular stomatitis Indiana virus; Virus Replication | 2018 |
A potential new approach for treating systemic sclerosis: Dedifferentiation of SSc fibroblasts and change in the microenvironment by blocking store-operated Ca2+ entry.
Topics: Boron Compounds; Calcium Channel Blockers; Calcium Signaling; Cell Dedifferentiation; Cells, Cultured; Cellular Microenvironment; Collagen; Cytoskeleton; Fibroblasts; Humans; Imidazoles; Indomethacin; Scleroderma, Systemic; Skin; Transforming Growth Factor beta1 | 2019 |
Leucine-rich repeat kinase 2 regulates mouse dendritic cell migration by ORAI2.
Topics: Animals; Boron Compounds; Calcium; Calcium Channel Blockers; Cell Movement; Dendritic Cells; Down-Regulation; Gene Expression Regulation; Gene Silencing; Imidazoles; Leucine-Rich Repeat Serine-Threonine Protein Kinase-2; Mice; ORAI2 Protein; Stromal Interaction Molecule 2 | 2019 |
The involvement of TRP channels in memory formation and task retrieval in a passive avoidance task in one-day old chicks.
Topics: Animals; Avoidance Learning; Boron Compounds; Calcium; Chickens; Cognition; Imidazoles; Male; Memory; Neurons; Transient Receptor Potential Channels | 2020 |
Temporal modulation of calcium sensing in hematopoietic stem cells is crucial for proper stem cell expansion and engraftment.
Topics: Animals; Boron Compounds; Calcium; Calcium Signaling; Cell Adhesion Molecules; Cell Cycle; Cell Differentiation; Cell Proliferation; Coculture Techniques; Fetal Blood; Gene Expression Regulation, Developmental; Hematopoietic Stem Cell Transplantation; Hematopoietic Stem Cells; Humans; Imidazoles; Intracellular Calcium-Sensing Proteins; Membrane Proteins; Mice; Receptors, Calcium-Sensing; Receptors, CXCR4 | 2020 |