1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine has been researched along with gbr 12935 in 3 studies
Studies (1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine) | Trials (1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine) | Recent Studies (post-2010) (1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine) | Studies (gbr 12935) | Trials (gbr 12935) | Recent Studies (post-2010) (gbr 12935) |
---|---|---|---|---|---|
62 | 0 | 14 | 203 | 1 | 15 |
Protein | Taxonomy | 1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine (IC50) | gbr 12935 (IC50) |
---|---|---|---|
Sodium-dependent noradrenaline transporter | Homo sapiens (human) | 0.713 | |
Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | 0.0038 | |
Sodium-dependent serotonin transporter | Homo sapiens (human) | 1.9995 | |
Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | 0.4033 | |
Small conductance calcium-activated potassium channel protein 2 | Rattus norvegicus (Norway rat) | 0.298 | |
Small conductance calcium-activated potassium channel protein 3 | Rattus norvegicus (Norway rat) | 0.298 | |
Small conductance calcium-activated potassium channel protein 1 | Rattus norvegicus (Norway rat) | 0.298 | |
Sodium-dependent dopamine transporter | Homo sapiens (human) | 0.018 | |
Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 0.017 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (66.67) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Hoffman, BT; Katz, JL; Kopajtic, T; Newman, AH | 1 |
de Costa, B; Jacobson, AE; Reith, ME; Rice, KC | 1 |
Akunne, HC; Baumann, MH; Cadet, JL; Carroll, FI; Char, GU; de Costa, BR; Dersch, CM; Partilla, JS; Rice, KC; Rothman, RB | 1 |
3 other study(ies) available for 1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine and gbr 12935
Article | Year |
---|---|
2D QSAR modeling and preliminary database searching for dopamine transporter inhibitors using genetic algorithm variable selection of Molconn Z descriptors.
Topics: Algorithms; Binding, Competitive; Carrier Proteins; Databases, Factual; Dopamine; Dopamine Plasma Membrane Transport Proteins; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Quantitative Structure-Activity Relationship; Radioligand Assay; Reproducibility of Results; Software | 2000 |
Evidence for mutually exclusive binding of cocaine, BTCP, GBR 12935, and dopamine to the dopamine transporter.
Topics: Animals; Binding Sites; Binding, Competitive; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Female; Phencyclidine; Piperazines; Rats; Rats, Sprague-Dawley | 1992 |
Studies of the biogenic amine transporters. III. Demonstration of two binding sites for [3H]GBR12935 and [3H]BTCP in rat caudate membranes.
Topics: Animals; Binding Sites; Biogenic Amines; Carrier Proteins; Caudate Nucleus; Dopamine Agents; Ligands; Male; Membranes; Oxidopamine; Phencyclidine; Piperazines; Rats; Rats, Sprague-Dawley; Tritium | 1994 |