Page last updated: 2024-09-03

(endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide and piperidines

(endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide has been researched along with piperidines in 9 studies

Compound Research Comparison

Studies
((endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide)
Trials
((endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide)
Recent Studies (post-2010)
((endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
240040,2355,22114,545

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (77.78)18.2507
2000's1 (11.11)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bockaert, J; Dumuis, A; Ladinsky, H; Monferini, E; Nicola, M; Sebben, M; Turconi, M1
Gebauer, A; Haas, J; Kilbinger, H; Ladinsky, H; Rizzi, CA1
Baxter, GS; Ellis, ES; Gaster, LM; Kennett, GA; Sanger, GJ; Wardle, KA1
Cesana, R; Donetti, A; Ladinsky, H; Rizzi, CA; Sagrada, A; Schiantarelli, P; Schiavi, GB; Schiavone, A1
Bonhaus, DW; DeSouza, A; Eglen, RM; Jakeman, LB; Loury, DN; To, Z; Wong, EH1
Pacenti, P; Schiavone, A; Terrani, S1
Bingham, S; Ellis, ES; Gaster, LM; Rushant, B; Sanger, GJ; Smith, MI; Wardle, KA1
Boulouard, M; Dauphin, F; Lelong, V; Lhonneur, L1
Chinkwo, KA; Coupar, IM; Grabbe, C; Irving, HR; Li, JG; Pouton, CW; Shapiro, M; Tochon-Danguy, N1

Other Studies

9 other study(ies) available for (endo-n-8-methyl-8-azabicyclo(3.2.1)oct-3-yl)-2,3-dihydro-3-ethyl-2-oxo-1h-benzimidazol-1-carboxamide and piperidines

ArticleYear
Azabicycloalkyl benzimidazolone derivatives as a novel class of potent agonists at the 5-HT4 receptor positively coupled to adenylate cyclase in brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:3

    Topics: Adenylyl Cyclases; Animals; Benzimidazoles; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Cyclic AMP; Drug Interactions; Indoles; Mice; Neurons; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron

1991
Benzimidazolones and renzapride facilitate acetylcholine release from guinea-pig myenteric plexus via 5-HT4 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 351, Issue:3

    Topics: Acetylcholine; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Choline; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Myenteric Plexus; Phosphodiesterase Inhibitors; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
The effects of SB 204070, a highly potent and selective 5-HT4 receptor antagonist, on guinea-pig distal colon.
    British journal of pharmacology, 1994, Volume: 112, Issue:3

    Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dimethylphenylpiperazinium Iodide; Dioxanes; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Piperidines; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin Antagonists

1994
Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:4

    Topics: Animals; Anti-Ulcer Agents; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dogs; Dose-Response Relationship, Drug; Female; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle Denervation; Neostriatum; Ondansetron; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Swine; Tumor Cells, Cultured

1994
[3H]BIMU-1, a 5-hydroxytryptamine3 receptor ligand in NG-108 cells, selectively labels sigma-2 binding sites in guinea pig hippocampus.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Animals; Autoradiography; Benzimidazoles; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Guinea Pigs; Hippocampus; Male; Membranes; Mice; Neuroblastoma; Piperidines; Rats; Receptors, Serotonin; Receptors, sigma; Sensitivity and Specificity; Tritium; Tumor Cells, Cultured

1993
Gastric emptying of radionuclide-labeled solid meal in beagle dogs using a scintigraphic method.
    Methods and findings in experimental and clinical pharmacology, 1993, Volume: 15, Issue:7

    Topics: Animals; Anti-Ulcer Agents; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dogs; Eating; Gastric Emptying; Iodine Radioisotopes; Piperidines; Receptors, Serotonin; Scintillation Counting; Time Factors

1993
Selective and functional 5-hydroxytryptamine4 receptor antagonism by SB 207266.
    British journal of pharmacology, 1996, Volume: 118, Issue:3

    Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dogs; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Male; Muscle Contraction; Piperidines; Serotonin; Serotonin Antagonists; Time Factors

1996
BIMU 1 and RS 67333, two 5-HT4 receptor agonists, modulate spontaneous alternation deficits induced by scopolamine in the mouse.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:6

    Topics: Aniline Compounds; Animals; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Locomotion; Male; Memory; Memory Disorders; Mice; Piperidines; Receptors, Serotonin, 5-HT4; Scopolamine; Serotonin 5-HT4 Receptor Agonists

2003
Investigations into the binding affinities of different human 5-HT4 receptor splice variants.
    Pharmacology, 2010, Volume: 85, Issue:4

    Topics: Aniline Compounds; Animals; Benzamides; Benzimidazoles; Benzofurans; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Chlorocebus aethiops; COS Cells; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Indoles; Kinetics; Ligands; Piperidines; Protein Isoforms; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists

2010