(3h)2-carbomethoxy-3-(4-fluorophenyl)tropane has been researched along with mazindol in 18 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 9 (50.00) | 18.2507 |
| 2000's | 9 (50.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Reith, ME; Selmeci, G | 1 |
| Kuhar, MJ; Pögün, S; Scheffel, U | 1 |
| London, ED; Mantione, CR; Ritz, MC | 1 |
| Patel, A | 1 |
| Chan, B; Chen, CA; Dannals, RF; Folio, T; Ravert, HT; Ricaurte, GA; Scheffel, U; Shaya, EK; Wong, DF; Yung, B | 1 |
| Boja, JW; Houlihan, WJ; Kopajtic, TA; Kuhar, MJ; Parrino, VA | 1 |
| Reith, ME; Xu, C | 1 |
| Coffey, LL; Reith, ME; Wu, Q | 1 |
| Dannals, RF; Hatzidimitriou, G; Mathews, WB; McCann, UD; Musachio, J; Ravert, HT; Ricaurte, GA; Villemagne, V; Wong, DF; Yuan, J | 1 |
| Bonnet, JJ; Corera, AT; Costentin, J | 1 |
| Dutta, AK; Madras, BK; Reith, ME | 1 |
| Bonnet, JJ; Costentin, J; Do-Régo, JC; Tidjane Corera, A | 1 |
| Chen, N; Reith, ME; Vaughan, RA | 1 |
| Berfield, JL; Ferrer, JV; Javitch, JA; Reith, ME; Wang, LC | 1 |
| Lin, Z; Uhl, GR | 1 |
| Enyedy, IJ; Johnson, KM; Wang, J; Wang, S; Zaman, WA | 1 |
| Houlihan, WJ; Kelly, L | 1 |
| Bondi, CD; Kozikowski, AP; Kulkarni, SS; Newman, AH; Pan, S; Surratt, CK; Ukairo, OT | 1 |
18 other study(ies) available for (3h)2-carbomethoxy-3-(4-fluorophenyl)tropane and mazindol
| Article | Year |
|---|---|
Radiolabeling of dopamine uptake sites in mouse striatum: comparison of binding sites for cocaine, mazindol, and GBR 12935.
Topics: Animals; Binding Sites; Buffers; Cocaine; Corpus Striatum; Dopamine; Drug Interactions; Ethylmaleimide; Kinetics; Male; Mazindol; Membranes; Mice; Mice, Inbred BALB C; Phosphates; Piperazines; Radioligand Assay; Temperature; Tritium; Tromethamine | 1992 |
Cocaine displaces [3H]WIN 35,428 binding to dopamine uptake sites in vivo more rapidly than mazindol or GBR 12909.
Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Injections, Intravenous; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Piperazines; Radioimmunoassay; Receptors, Drug | 1991 |
Spermine interacts with cocaine binding sites on dopamine transporters.
Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Paroxetine; Rats; Rats, Inbred F344; Receptors, Drug; Serotonin; Serotonin Plasma Membrane Transport Proteins; Spermine | 1994 |
Characterization of [125I]RTI-55 binding to dog caudate dopamine transporter.
Topics: Animals; Binding, Competitive; Carrier Proteins; Caudate Nucleus; Cell Membrane; Cholic Acids; Citalopram; Cocaine; Desipramine; Dogs; Dopamine Plasma Membrane Transport Proteins; Filtration; Iodine Radioisotopes; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Protein Binding; Solubility | 1993 |
In vivo imaging of baboon and human dopamine transporters by positron emission tomography using [11C]WIN 35,428.
Topics: Adult; Affect; Aged; Aged, 80 and over; Animals; Blood Pressure; Brain; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Electrocardiography; Female; Humans; Ligands; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Middle Aged; Nerve Endings; Nerve Tissue Proteins; Papio; Pulse; Receptors, Dopamine; Tomography, Emission-Computed | 1993 |
Halogenated mazindol analogs as potential inhibitors of the cocaine binding site at the dopamine transporter.
Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats | 1996 |
WIN 35,428 and mazindol are mutually exclusive in binding to the cloned human dopamine transporter.
Topics: Binding, Competitive; Carrier Proteins; Cloning, Molecular; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Models, Chemical; Nerve Tissue Proteins; Radioligand Assay; Recombinant Proteins; Tritium; Tumor Cells, Cultured | 1997 |
Cations affect [3H]mazindol and [3H]WIN 35,428 binding to the human dopamine transporter in a similar fashion.
Topics: Animals; Carrier Proteins; Cations, Divalent; Cations, Monovalent; Cell Membrane; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Glioma; Humans; Kinetics; Lithium; Magnesium; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mercury; Nerve Tissue Proteins; Potassium; Protein Binding; Rats; Sodium; Tritium; Tumor Cells, Cultured; Zinc | 1997 |
Brain dopamine neurotoxicity in baboons treated with doses of methamphetamine comparable to those recreationally abused by humans: evidence from [11C]WIN-35,428 positron emission tomography studies and direct in vitro determinations.
Topics: Animals; Carbon Radioisotopes; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Humans; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Neostriatum; Nerve Tissue Proteins; Neurotoxins; Papio; Substance-Related Disorders; Tomography, Emission-Computed; Tritium | 1998 |
Binding of uptake blockers to the neuronal dopamine transporter: further investigation about cationic and anionic requirements.
Topics: Animals; Anions; Binding Sites; Cations; Cocaine; Corpus Striatum; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Mazindol; Rats; Rats, Sprague-Dawley | 2000 |
Synthesis and preliminary characterization of a high-affinity novel radioligand for the dopamine transporter.
Topics: Animals; Benzhydryl Compounds; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Female; Ligands; Macaca mulatta; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Piperazines; Piperidines; Radioligand Assay; Tritium | 2001 |
Differential sensitivity to NaCl for inhibitors and substrates that recognize mutually exclusive binding sites on the neuronal transporter of dopamine in rat striatal membranes.
Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dextroamphetamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Sodium Chloride | 2001 |
The role of conserved tryptophan and acidic residues in the human dopamine transporter as characterized by site-directed mutagenesis.
Topics: Amino Acid Sequence; Amino Acid Substitution; Aspartic Acid; Carrier Proteins; Cell Line; Cocaine; Conserved Sequence; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Kinetics; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Protein Structure, Secondary; Radioligand Assay; Recombinant Proteins; Transfection; Tritium; Tryptophan | 2001 |
The uptake inhibitors cocaine and benztropine differentially alter the conformation of the human dopamine transporter.
Topics: Benztropine; Binding Sites; Binding, Competitive; Carrier Proteins; Cell Membrane; Cocaine; Cysteine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Indicators and Reagents; Kinetics; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mesylates; Models, Molecular; Nerve Tissue Proteins; Protein Conformation | 2001 |
Dopamine transporter mutants with cocaine resistance and normal dopamine uptake provide targets for cocaine antagonism.
Topics: Amino Acid Substitution; Animals; Binding, Competitive; Chlorocebus aethiops; Cocaine; COS Cells; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Drug Resistance; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Motor Proteins; Mutation; Nerve Tissue Proteins; Transfection; Tritium | 2002 |
Discovery of substituted 3,4-diphenyl-thiazoles as a novel class of monoamine transporter inhibitors through 3-D pharmacophore search using a new pharmacophore model derived from mazindol.
Topics: Binding Sites; Biphenyl Compounds; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Ligands; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Norepinephrine; Serotonin; Structure-Activity Relationship; Thiazoles | 2002 |
Assessment of mazindane, a pro-drug form of mazindol, in assays used to define cocaine treatment agents.
Topics: Analysis of Variance; Animals; Binding, Competitive; Cell Membrane; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Isoindoles; Macaca mulatta; Male; Mazindol; Mice; Motor Activity; Neurotransmitter Agents; Proadifen; Rats; Rats, Sprague-Dawley; Tritium | 2003 |
Recognition of benztropine by the dopamine transporter (DAT) differs from that of the classical dopamine uptake inhibitors cocaine, methylphenidate, and mazindol as a function of a DAT transmembrane 1 aspartic acid residue.
Topics: Amino Acid Substitution; Animals; Aspartic Acid; Benztropine; Binding, Competitive; CHO Cells; Cocaine; Cricetinae; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Immunohistochemistry; Kinetics; Ligands; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Methylphenidate; Microscopy, Confocal; Models, Molecular; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Transfection | 2005 |