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(3h)2-carbomethoxy-3-(4-fluorophenyl)tropane and gbr 12935

(3h)2-carbomethoxy-3-(4-fluorophenyl)tropane has been researched along with gbr 12935 in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (80.00)18.2507
2000's3 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hoffman, BJ; Kish, SJ; Niznik, HB; Pristupa, ZB; Wilson, JM1
Reith, ME; Wiener, HL1
Reith, ME; Selmeci, G1
Eshleman, AJ; Janowsky, A; Neve, KA; Neve, RL1
Coen, KM; Corrigall, WA; Kish, SJ; Nobrega, JN; Shannak, K; Wilson, JM1
Abraham, P; Boja, JW; Cadet, JL; Carroll, FI; Kopajtic, TA; Lever, J; Lewin, AH; Seltzman, HH; Wyrick, CD1
Carroll, ME; Dixon, LM; Kish, SJ; Lac, ST; Niznik, HB; Nobrega, JN; Pristupa, ZB; Shannak, K; Wilson, JM1
Becketts, KM; Carroll, FI; de Costa, BR; Dersch, CM; Radesca, LR; Rice, KC; Rothman, RB1
Richfield, EK1
Darmani, NA; Reeves, SL1
Descarries, L; Doucet, G; Lafaille, F; Mrini, A; Soucy, JP1
Bonnet, JJ; Corera, AT; Do RĂ©go, JC1
Carroll, FI; Kimmel, HL; Kuhar, MJ1
Chen, N; Dutta, AK; Maiti, S; Reith, ME; Zhen, J1
Booze, RM; Mactutus, CF; Wallace, DR; Zhu, J1

Other Studies

15 other study(ies) available for (3h)2-carbomethoxy-3-(4-fluorophenyl)tropane and gbr 12935

ArticleYear
Pharmacological heterogeneity of the cloned and native human dopamine transporter: disassociation of [3H]WIN 35,428 and [3H]GBR 12,935 binding.
    Molecular pharmacology, 1994, Volume: 45, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cells, Cultured; Cloning, Molecular; Cocaine; DNA; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Sequence Data; Nerve Tissue Proteins; Piperazines

1994
Determination of radioligand specific activity using competition binding assays.
    Analytical biochemistry, 1992, Nov-15, Volume: 207, Issue:1

    Topics: Animals; Binding, Competitive; Cocaine; Corpus Striatum; Female; Kinetics; Ligands; Male; Mice; Mice, Inbred C57BL; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Tritium

1992
Radiolabeling of dopamine uptake sites in mouse striatum: comparison of binding sites for cocaine, mazindol, and GBR 12935.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:3

    Topics: Animals; Binding Sites; Buffers; Cocaine; Corpus Striatum; Dopamine; Drug Interactions; Ethylmaleimide; Kinetics; Male; Mazindol; Membranes; Mice; Mice, Inbred BALB C; Phosphates; Piperazines; Radioligand Assay; Temperature; Tritium; Tromethamine

1992
Characterization of a recombinant human dopamine transporter in multiple cell lines.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:1

    Topics: Amino Acid Sequence; Animals; Carrier Proteins; Cell Line; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Sequence Data; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Recombinant Proteins; Tritium; Tumor Cells, Cultured

1995
Amygdala dopamine levels are markedly elevated after self- but not passive-administration of cocaine.
    Brain research, 1994, Dec-30, Volume: 668, Issue:1-2

    Topics: Amygdala; Animals; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Administration Schedule; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Piperazines; Rats; Rats, Inbred Strains; Self Stimulation; Serotonin

1994
Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester.
    Molecular pharmacology, 1995, Volume: 47, Issue:4

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley

1995
Heterogeneous subregional binding patterns of 3H-WIN 35,428 and 3H-GBR 12,935 are differentially regulated by chronic cocaine self-administration.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:5 Pt 2

    Topics: Animals; Biogenic Monoamines; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Wistar; Reference Values; Self Administration; Substance Withdrawal Syndrome; Time Factors; Tissue Distribution; Tritium

1994
Studies of the biogenic amine transporters. II. A brief study on the use of [3H]DA-uptake-inhibition to transporter-binding-inhibition ratios for the in vitro evaluation of putative cocaine antagonists.
    Life sciences, 1993, Volume: 53, Issue:17

    Topics: Animals; Biogenic Amines; Biological Transport; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Tritium

1993
Zinc modulation of drug binding, cocaine affinity states, and dopamine uptake on the dopamine uptake complex.
    Molecular pharmacology, 1993, Volume: 43, Issue:1

    Topics: Animals; Binding, Competitive; Buffers; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Ethylmaleimide; In Vitro Techniques; Male; Membrane Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley; Zinc

1993
The stimulatory and inhibitory components of cocaine's actions on the 5-HTP-induced 5-HT2A receptor response.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 55, Issue:3

    Topics: 1-Naphthylamine; 5-Hydroxytryptophan; Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Fluoxetine; Head Movements; Male; Mice; Mice, Inbred ICR; Norepinephrine; Piperazines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Sertraline

1996
Comparative evaluation of [3H]WIN 35428 and [3H]GBR 12935 as markers of dopamine innervation density in brain.
    Synapse (New York, N.Y.), 1997, Volume: 25, Issue:2

    Topics: Animals; Autoradiography; Brain; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Male; Piperazines; Rats; Rats, Sprague-Dawley

1997
Specificity and ion dependence of binding of GBR analogs.
    Methods in enzymology, 1998, Volume: 296

    Topics: Animals; Carrier Proteins; Cell Fractionation; Cell Membrane; Centrifugation, Density Gradient; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Substrate Specificity; Tritium

1998
Dopamine transporter synthesis and degradation rate in rat striatum and nucleus accumbens using RTI-76.
    Neuropharmacology, 2000, Feb-14, Volume: 39, Issue:4

    Topics: Animals; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Fluoxetine; Injections, Intraventricular; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Nucleus Accumbens; Piperazines; Protein Binding; Rats; Rats, Sprague-Dawley; Symporters; Tropanes

2000
Interaction between a hydroxypiperidine analogue of 4-(2-benzhydryloxy-ethyl)-1-(4-fluorobenzyl)piperidine and Aspartate 68 in the human dopamine transporter.
    European journal of pharmacology, 2004, Dec-03, Volume: 506, Issue:1

    Topics: Animals; Aspartic Acid; Benzhydryl Compounds; Binding Sites; Binding, Competitive; Biological Transport; Cell Line; Cell Membrane; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Humans; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Mutation; Nerve Tissue Proteins; Norepinephrine; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Serotonin; Stereoisomerism; Synaptosomes; Tritium

2004
HIV-1 Tat protein-induced rapid and reversible decrease in [3H]dopamine uptake: dissociation of [3H]dopamine uptake and [3H]2beta-carbomethoxy-3-beta-(4-fluorophenyl)tropane (WIN 35,428) binding in rat striatal synaptosomes.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 329, Issue:3

    Topics: Animals; Binding Sites; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Leucine; Male; Piperazines; Protein Binding; Rats; Rats, Sprague-Dawley; Surface Plasmon Resonance; Synaptosomes; tat Gene Products, Human Immunodeficiency Virus

2009