Page last updated: 2024-09-03

(3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine and kelatorphan

(3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine has been researched along with kelatorphan in 4 studies

Compound Research Comparison

Studies
((3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine)
Trials
((3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine)
Recent Studies (post-2010)
((3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine)
Studies
(kelatorphan)
Trials
(kelatorphan)
Recent Studies (post-2010) (kelatorphan)
5005801

Protein Interaction Comparison

ProteinTaxonomy(3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine (IC50)kelatorphan (IC50)
ThermolysinBacillus thermoproteolyticus0.003
NeprilysinOryctolagus cuniculus (rabbit)0.0036
Leukotriene A-4 hydrolaseHomo sapiens (human)0.005

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19904 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fournié-Zaluski, MC; Peyroux, J; Roques, BP; Schmidt, C; Soleilhac, JM; Xie, J1
Fournié-Zaluski, MC; Hernandez, JF; Roques, BP; Soleilhac, JM1
Bouboutou, R; Chaillet, P; Costentin, J; Coulaud, A; Devin, J; Fournié-Zaluski, MC; Roques, BP; Waksman, G1
Besselievre, R; Bouboutou, R; Chaillet, P; Costentin, J; Coulaud, A; Devin, J; Fournie-Zaluski, MC; Hamel, E; Roques, BP; Waksman, G1

Other Studies

4 other study(ies) available for (3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycine and kelatorphan

ArticleYear
New kelatorphan-related inhibitors of enkephalin metabolism: improved antinociceptive properties.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:7

    Topics: Analgesics; Animals; Dipeptides; Enkephalins; Male; Mice

1989
Retro-inverso concept applied to the complete inhibitors of enkephalin-degrading enzymes.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:9

    Topics: Aminopeptidases; Animals; Brain; CD13 Antigens; Chemical Phenomena; Chemistry; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Hydroxamic Acids; Kidney; Metalloendopeptidases; Molecular Conformation; Neprilysin; Rabbits; Rats; Stereoisomerism; Structure-Activity Relationship; Swine

1988
New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Aminopeptidases; Analgesia; Animals; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Hydroxylamines; Leucine; Male; Mice; Neprilysin; Protease Inhibitors; Rabbits; Rats; Stereoisomerism; Thiorphan; Tiopronin

1985
Kelatorphan: a full inhibitor of enkephalin degrading enzymes. Biochemical and pharmacological properties, regional distribution of enkephalinase in rat brain by use of a tritiated derivative.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Aminopeptidases; Analgesics; Animals; Autoradiography; Brain; Dipeptides; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Enkephalin, Methionine; Glycine; In Vitro Techniques; Mice; Propionates; Rats

1985