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(1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid and picrotoxin

(1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid has been researched along with picrotoxin in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (54.55)29.6817
2010's5 (45.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Grillner, S; Hill, RH; Schmitt, DE1
Hull, C; von Gersdorff, H1
Prada, C; Udin, SB1
Calvo, DJ; Escobar, AL; Goutman, JD1
Duarte, ID; Reis, GM1
Carland, JE; Chebib, M; Johnston, GA1
Denter, DG; Heck, N; Kilb, W; Luhmann, HJ; Riedemann, T; White, R1
Estrada-Mondragón, A; Limón, A; Martínez-Torres, A; Miledi, R; Ochoa-de la Paz, LD1
Chen, S; Li, W; Mehta, B; Snellman, J; Zenisek, D1
Awatramani, GB; Briggman, KL; Hoggarth, A; McLaughlin, AJ; Ronellenfitch, K; Schwab, D; Sethuramanujam, S; Trenholm, S; Vasandani, R1
Biel, M; Hüll, K; Laprell, L; Michalakis, S; Schön, C; Stawski, P; Sumser, MP; Trauner, D1

Other Studies

11 other study(ies) available for (1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid and picrotoxin

ArticleYear
The spinal GABAergic system is a strong modulator of burst frequency in the lamprey locomotor network.
    Journal of neurophysiology, 2004, Volume: 92, Issue:4

    Topics: Algorithms; Animals; Calcium Channel Blockers; Chloride Channels; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Lampreys; Locomotion; Models, Neurological; Nerve Net; Phosphinic Acids; Picrotoxin; Potassium Channels, Calcium-Activated; Propanolamines; Pyridazines; Pyridines; Receptors, GABA; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Spinal Cord

2004
Fast endocytosis is inhibited by GABA-mediated chloride influx at a presynaptic terminal.
    Neuron, 2004, Oct-28, Volume: 44, Issue:3

    Topics: Animals; Bicuculline; Calcium; Cells, Cultured; Chelating Agents; Chlorides; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Endocytosis; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Goldfish; In Vitro Techniques; Ionophores; Membrane Potentials; Microscopy, Electron, Transmission; Models, Neurological; Neural Inhibition; Neurons; Nystatin; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Presynaptic Terminals; Pyridines; Quinoxalines; Retina; Time Factors; Valine

2004
Melatonin decreases calcium levels in retinotectal axons of Xenopus laevis by indirect activation of group III metabotropic glutamate receptors.
    Brain research, 2005, Aug-16, Volume: 1053, Issue:1-2

    Topics: Aniline Compounds; Animals; Antioxidants; Axons; Calcium; Diagnostic Imaging; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Melatonin; Models, Neurological; Phosphinic Acids; Picrotoxin; Potassium Chloride; Pyridines; Receptors, Metabotropic Glutamate; Retinal Ganglion Cells; Superior Colliculi; Tetrahydronaphthalenes; Xanthenes; Xenopus laevis

2005
Analysis of macroscopic ionic currents mediated by GABArho1 receptors during lanthanide modulation predicts novel states controlling channel gating.
    British journal of pharmacology, 2005, Volume: 146, Issue:7

    Topics: Chloride Channels; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Lanthanoid Series Elements; Phosphinic Acids; Picrotoxin; Protein Subunits; Pyridines; Receptors, GABA

2005
Involvement of chloride channel coupled GABA(C) receptors in the peripheral antinociceptive effect induced by GABA(C) receptor agonist cis-4-aminocrotonic acid.
    Life sciences, 2007, Mar-13, Volume: 80, Issue:14

    Topics: Analgesics; Animals; Crotonates; Dinoprostone; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; Hindlimb; Male; Pain Measurement; Pain Threshold; Peripheral Nerves; Phosphinic Acids; Picrotoxin; Potassium Channel Blockers; Pyridines; Rats; Rats, Wistar; Reaction Time; Receptors, GABA

2007
Relative impact of residues at the intracellular and extracellular ends of the human GABAC rho1 receptor M2 domain on picrotoxinin activity.
    European journal of pharmacology, 2008, Feb-02, Volume: 580, Issue:1-2

    Topics: Allosteric Regulation; Animals; Binding Sites; Binding, Competitive; GABA Antagonists; Humans; Mutation; Oocytes; Phosphinic Acids; Picrotoxin; Protein Subunits; Pyridines; Receptors, GABA; Receptors, GABA-B; Sesterterpenes; Xenopus laevis

2008
GABAC receptors are functionally expressed in the intermediate zone and regulate radial migration in the embryonic mouse neocortex.
    Neuroscience, 2010, Apr-28, Volume: 167, Issue:1

    Topics: Animals; Bicuculline; Cell Movement; Crotonates; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neocortex; Neurons; Phosphinic Acids; Picrotoxin; Pyridines; Receptors, GABA; Receptors, GABA-A; RNA, Messenger

2010
Dopamine and serotonin modulate human GABAρ1 receptors expressed in Xenopus laevis oocytes.
    ACS chemical neuroscience, 2012, Feb-15, Volume: 3, Issue:2

    Topics: Animals; Binding, Competitive; Data Interpretation, Statistical; Dopamine; GABA Antagonists; Humans; Membrane Potentials; Octopamine; Oocytes; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Pyridines; Receptors, GABA-A; Receptors, GABA-B; Serotonin; Tyramine; Xenopus laevis

2012
Synaptic ribbons influence the size and frequency of miniature-like evoked postsynaptic currents.
    Neuron, 2013, Feb-06, Volume: 77, Issue:3

    Topics: Alcohol Oxidoreductases; Aminobutyrates; Animals; Biophysics; Co-Repressor Proteins; DNA-Binding Proteins; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glycine Agents; Hibernation; In Vitro Techniques; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Phosphinic Acids; Phosphoproteins; Picrotoxin; Pyridines; Receptors, AMPA; Retina; Sciuridae; Strychnine; Synapses; Visual Pathways; Wakefulness

2013
Specific wiring of distinct amacrine cells in the directionally selective retinal circuit permits independent coding of direction and size.
    Neuron, 2015, Apr-08, Volume: 86, Issue:1

    Topics: Amacrine Cells; Anesthetics, Local; Animals; Excitatory Postsynaptic Potentials; GABA Antagonists; Homeodomain Proteins; Light; Mice; Mice, Transgenic; Nerve Net; Neural Inhibition; Phosphinic Acids; Photic Stimulation; Picrotoxin; Presynaptic Terminals; Pyridines; Retina; Retinal Ganglion Cells; Size Perception; Space Perception; Synapses; Tetrodotoxin; Time Factors; Transcription Factors; Visual Fields

2015
Restoring Light Sensitivity in Blind Retinae Using a Photochromic AMPA Receptor Agonist.
    ACS chemical neuroscience, 2016, Jan-20, Volume: 7, Issue:1

    Topics: Action Potentials; Animals; Animals, Newborn; Blindness; Cyclic Nucleotide-Gated Cation Channels; Disease Models, Animal; GABA Agents; GluK2 Kainate Receptor; HEK293 Cells; Hippocampus; Humans; Light; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Phosphinic Acids; Picrotoxin; Pyridines; Receptors, AMPA; Receptors, Kainic Acid; Retinal Ganglion Cells; rho GTP-Binding Proteins; Rod Opsins; Sesterterpenes

2016