(1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid has been researched along with gaboxadol in 6 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (83.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (16.67) | 2.80 |
Authors | Studies |
---|---|
Bang-Andersen, B; Ebert, B; Frølund, B; Hansen, CP; Jensen, AA; Kristiansen, U; Krogsgaard-Larsen, P; Larsen, M; Liljefors, T; Madsen, C; Nielsen, B | 1 |
Chebib, M; Hanrahan, JR; Hibbs, DE; Johnston, GA; Kim, HL; Kumar, RJ; Salam, NK | 1 |
Jonas, P; Jones, MV; Sahara, Y; Westbrook, GL | 1 |
Johnston, GA | 1 |
Platt, B; White, AM | 1 |
Herberholz, J; Pena-Flores, NL; Venuti, LS | 1 |
1 review(s) available for (1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid and gaboxadol
Article | Year |
---|---|
Medicinal chemistry and molecular pharmacology of GABA(C) receptors.
Topics: Amino Acids, Cyclic; Animals; Barbiturates; Crotonates; GABA Agonists; GABA Antagonists; Imidazoles; Isoxazoles; Muscimol; Organophosphorus Compounds; Phosphinic Acids; Pyridines; Receptors, GABA; Receptors, GABA-A | 2002 |
5 other study(ies) available for (1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid and gaboxadol
Article | Year |
---|---|
5-Substituted imidazole-4-acetic acid analogues: synthesis, modeling, and pharmacological characterization of a series of novel gamma-aminobutyric acid(C) receptor agonists.
Topics: Animals; Brain; Cell Line; GABA Agonists; GABA-A Receptor Agonists; Humans; Imidazoles; In Vitro Techniques; Ligands; Membrane Potentials; Models, Molecular; Mutation; Oocytes; Patch-Clamp Techniques; Protein Structure, Tertiary; Protein Subunits; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 2007 |
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.
Topics: Animals; Female; GABA Antagonists; Ligands; Models, Molecular; Molecular Structure; Oocytes; Structure-Activity Relationship; Xenopus laevis | 2008 |
Microscopic kinetics and energetics distinguish GABA(A) receptor agonists from antagonists.
Topics: Animals; Brain; Diffusion; Electrophysiology; Energy Metabolism; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Inhibitory Concentration 50; Isoxazoles; Kinetics; Muscimol; Phosphinic Acids; Protein Binding; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2001 |
Gamma-aminobutyric acid-induced calcium signalling in rat superior collicular neurones.
Topics: Animals; Bicuculline; Calcium; Cells, Cultured; Cytarabine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; Isoxazoles; Neurons; Phosphinic Acids; Pyridines; Rats; Receptors, GABA; Superior Colliculi | 2002 |
Cellular interactions between social experience, alcohol sensitivity, and GABAergic inhibition in a crayfish neural circuit.
Topics: Animals; Astacoidea; Ethanol; GABA Agonists; GABA-A Receptor Antagonists; GABAergic Neurons; Interneurons; Isoxazoles; Phosphinic Acids; Pyridines; Social Behavior; Synaptic Potentials | 2021 |