Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
Chain 1, MANNOSE-BINDING PROTEIN-A | 0 | 0 | 1 | 1 |
Chain A, Galacto-N-biose/lacto-N-biose I transporter substrate-binding protein | 0 | 0 | 1 | 1 |
Putative glycosyltransferase WbgO | 0 | 0 | 0 | 1 |
Chain A, Ferritin light chain | 3 | 0 | 0 | 3 |
thioredoxin reductase | 2 | 0 | 0 | 2 |
TDP1 protein | 4 | 0 | 0 | 4 |
Microtubule-associated protein tau | 2 | 0 | 0 | 2 |
Smad3 | 1 | 0 | 0 | 1 |
aldehyde dehydrogenase 1 family, member A1 | 6 | 0 | 0 | 6 |
alpha-galactosidase | 3 | 0 | 0 | 3 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | 2 | 0 | 0 | 2 |
flap endonuclease 1 | 1 | 0 | 0 | 1 |
DNA polymerase iota isoform a (long) | 3 | 0 | 0 | 3 |
DNA topoisomerase 2-alpha | 0 | 0 | 0 | 1 |
Acetylcholinesterase | 0 | 1 | 0 | 1 |
Carbonic anhydrase 1 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 2 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 4 | 0 | 1 | 0 | 1 |
Carbonic anhydrase | 0 | 1 | 0 | 1 |
Carbonic anhydrase 15 | 0 | 1 | 0 | 1 |
Luciferase | 2 | 0 | 0 | 2 |
interleukin 8 | 4 | 0 | 0 | 4 |
hypoxia-inducible factor 1 alpha subunit | 2 | 0 | 0 | 2 |
RAR-related orphan receptor gamma | 5 | 0 | 0 | 5 |
GLI family zinc finger 3 | 5 | 0 | 0 | 5 |
nuclear receptor subfamily 1, group I, member 3 | 4 | 0 | 0 | 4 |
progesterone receptor | 3 | 0 | 0 | 3 |
retinoic acid nuclear receptor alpha variant 1 | 7 | 0 | 0 | 7 |
retinoid X nuclear receptor alpha | 6 | 0 | 0 | 6 |
estrogen-related nuclear receptor alpha | 5 | 0 | 0 | 5 |
estrogen nuclear receptor alpha | 6 | 0 | 0 | 6 |
peroxisome proliferator-activated receptor delta | 4 | 0 | 0 | 4 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | 4 | 0 | 0 | 4 |
v-jun sarcoma virus 17 oncogene homolog (avian) | 2 | 0 | 0 | 2 |
Histone H2A.x | 3 | 0 | 0 | 3 |
geminin | 5 | 0 | 0 | 5 |
lamin isoform A-delta10 | 5 | 0 | 0 | 5 |
Voltage-dependent calcium channel gamma-2 subunit | 4 | 0 | 0 | 4 |
Cellular tumor antigen p53 | 7 | 0 | 0 | 7 |
Glutamate receptor 2 | 4 | 0 | 0 | 4 |
Nuclear receptor ROR-gamma | 4 | 0 | 0 | 4 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 3 | 0 | 0 | 3 |
Chain A, Putative fructose-1,6-bisphosphate aldolase | 2 | 0 | 0 | 2 |
Chain A, HADH2 protein | 2 | 0 | 0 | 2 |
Chain B, HADH2 protein | 2 | 0 | 0 | 2 |
Chain A, ATP-DEPENDENT DNA HELICASE Q1 | 2 | 0 | 0 | 2 |
Chain A, Cruzipain | 1 | 0 | 0 | 1 |
15-lipoxygenase, partial | 2 | 0 | 0 | 2 |
USP1 protein, partial | 1 | 0 | 0 | 1 |
AR protein | 5 | 0 | 0 | 5 |
caspase 7, apoptosis-related cysteine protease | 2 | 0 | 0 | 2 |
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | 1 | 0 | 0 | 1 |
estrogen receptor 2 (ER beta) | 2 | 0 | 0 | 2 |
cytochrome P450 family 3 subfamily A polypeptide 4 | 2 | 0 | 0 | 2 |
glucocorticoid receptor [Homo sapiens] | 3 | 0 | 0 | 3 |
farnesoid X nuclear receptor | 3 | 0 | 0 | 3 |
pregnane X nuclear receptor | 4 | 0 | 0 | 4 |
peroxisome proliferator activated receptor gamma | 3 | 0 | 0 | 3 |
caspase-3 | 2 | 0 | 0 | 2 |
RAD51 | 0 | 1 | 0 | 1 |
euchromatic histone-lysine N-methyltransferase 2 | 2 | 0 | 0 | 2 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 3 | 0 | 0 | 3 |
activating transcription factor 6 | 3 | 0 | 0 | 3 |
Caspase-7 | 1 | 0 | 0 | 1 |
Bloom syndrome protein isoform 1 | 2 | 0 | 0 | 2 |
vitamin D3 receptor isoform VDRA | 2 | 0 | 0 | 2 |
thyroid hormone receptor beta isoform a | 3 | 0 | 0 | 3 |
caspase-3 | 1 | 0 | 0 | 1 |
thyroid hormone receptor beta isoform 2 | 4 | 0 | 0 | 4 |
huntingtin isoform 2 | 1 | 0 | 0 | 1 |
histone-lysine N-methyltransferase 2A isoform 2 precursor | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 5 | 0 | 0 | 5 |
nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
peripheral myelin protein 22 | 2 | 0 | 0 | 2 |
survival motor neuron protein isoform d | 3 | 0 | 0 | 3 |
cytochrome P450 3A4 isoform 1 | 4 | 0 | 0 | 4 |
caspase-1 isoform alpha precursor | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 4 | 0 | 0 | 4 |
Interferon beta | 1 | 0 | 0 | 1 |
ATP-dependent translocase ABCB1 | 0 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit delta | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 4 | 0 | 0 | 4 |
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 | 0 | 1 | 0 | 1 |
Caspase-7 | 1 | 0 | 0 | 1 |
Spike glycoprotein | 1 | 0 | 1 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 4 | 0 | 0 | 4 |
Growth factor receptor-bound protein 2 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-3 | 4 | 0 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit beta-2 | 4 | 0 | 0 | 4 |
Pantothenate synthetase | 0 | 1 | 0 | 1 |
Discoidin domain-containing receptor 2 | 0 | 1 | 0 | 1 |
Growth factor receptor-bound protein 2 | 0 | 1 | 0 | 1 |
Reverse transcriptase/RNaseH | 0 | 1 | 0 | 1 |
GABA theta subunit | 4 | 0 | 0 | 4 |
Peptide-N(4)-(N-acetyl-beta-glucosaminyl)asparagine amidase | 0 | 0 | 1 | 1 |
ATPase family AAA domain-containing protein 5 | 1 | 0 | 0 | 1 |
Ataxin-2 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit epsilon | 4 | 0 | 0 | 4 |
Cereblon isoform 4 | 0 | 2 | 0 | 2 |
Insulin-like growth factor-binding protein 5 | 0 | 0 | 1 | 1 |
Choline O-acetyltransferase | 0 | 1 | 0 | 1 |
Protein cereblon | 0 | 4 | 0 | 4 |
Chain B, EUKARYOTIC TRANSLATION INITIATION FACTOR 4E | 0 | 0 | 1 | 1 |
Chain B, Pulmonary surfactant-associated protein D | 0 | 1 | 0 | 1 |
Chain A, Pulmonary surfactant-associated protein D | 0 | 1 | 0 | 1 |
parathyroid hormone/parathyroid hormone-related peptide receptor precursor | 1 | 0 | 0 | 1 |
Amyloid-beta precursor protein | 0 | 1 | 0 | 1 |
TAR DNA-binding protein 43 | 1 | 0 | 0 | 1 |
Sodium/myo-inositol cotransporter 2 | 0 | 1 | 0 | 1 |
Chain A, TYROSYL-DNA PHOSPHODIESTERASE | 1 | 0 | 0 | 1 |
Chain A, 2-oxoglutarate Oxygenase | 1 | 0 | 0 | 1 |
GLS protein | 1 | 0 | 0 | 1 |
Thrombopoietin | 2 | 0 | 0 | 2 |
hypothetical protein, conserved | 1 | 0 | 0 | 1 |
regulator of G-protein signaling 4 | 1 | 0 | 0 | 1 |
arylsulfatase A | 2 | 0 | 0 | 2 |
peripheral myelin protein 22 isoform 1 | 2 | 0 | 0 | 2 |
cellular tumor antigen p53 isoform a | 2 | 0 | 0 | 2 |
cytochrome P450 2C19 precursor | 1 | 0 | 0 | 1 |
cytochrome P450 2C9 precursor | 1 | 0 | 0 | 1 |
chromobox protein homolog 1 | 2 | 0 | 0 | 2 |
histone deacetylase 9 isoform 3 | 1 | 0 | 0 | 1 |
DNA polymerase beta | 1 | 0 | 0 | 1 |
ubiquitin carboxyl-terminal hydrolase 2 isoform a | 1 | 0 | 0 | 1 |
M-phase phosphoprotein 8 | 1 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
muscarinic acetylcholine receptor M1 | 2 | 0 | 0 | 2 |
Polyunsaturated fatty acid lipoxygenase ALOX15B | 1 | 0 | 0 | 1 |
Transient receptor potential cation channel subfamily A member 1 | 0 | 0 | 1 | 1 |
Alcohol dehydrogenase E chain | 0 | 1 | 0 | 1 |
Alcohol dehydrogenase S chain | 0 | 1 | 0 | 1 |
Integrin beta-3 | 1 | 0 | 0 | 1 |
Integrin alpha-IIb | 1 | 0 | 0 | 1 |
Histamine H2 receptor | 1 | 0 | 0 | 1 |
Disintegrin and metalloproteinase domain-containing protein 17 | 1 | 0 | 0 | 1 |
ATP-dependent phosphofructokinase | 1 | 0 | 0 | 1 |
acetylcholinesterase | 1 | 0 | 0 | 1 |
pregnane X receptor | 1 | 0 | 0 | 1 |
SMAD family member 2 | 1 | 0 | 0 | 1 |
SMAD family member 3 | 1 | 0 | 0 | 1 |
thyroid stimulating hormone receptor | 2 | 0 | 0 | 2 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | 1 | 0 | 0 | 1 |
potassium voltage-gated channel subfamily H member 2 isoform d | 1 | 0 | 0 | 1 |
heat shock protein beta-1 | 1 | 0 | 0 | 1 |
mitogen-activated protein kinase 1 | 1 | 0 | 0 | 1 |
nuclear factor NF-kappa-B p105 subunit isoform 1 | 1 | 0 | 0 | 1 |
lethal factor (plasmid) | 1 | 0 | 0 | 1 |
Nuclear receptor subfamily 1 group I member 2 | 0 | 1 | 1 | 2 |
Estrogen receptor | 0 | 2 | 1 | 3 |
Glucocorticoid receptor | 0 | 2 | 1 | 3 |
Progesterone receptor | 0 | 2 | 1 | 3 |
Mineralocorticoid receptor | 0 | 2 | 1 | 3 |
Androgen receptor | 0 | 2 | 0 | 2 |
Retinoic acid receptor alpha | 0 | 1 | 1 | 2 |
Retinoic acid receptor beta | 0 | 1 | 1 | 2 |
Thyroid hormone receptor alpha | 0 | 1 | 1 | 2 |
Thyroid hormone receptor beta | 0 | 1 | 1 | 2 |
Vitamin D3 receptor | 0 | 1 | 1 | 2 |
Retinoic acid receptor gamma | 0 | 1 | 1 | 2 |
Retinoic acid receptor RXR-alpha | 0 | 1 | 1 | 2 |
Peroxisome proliferator-activated receptor gamma | 0 | 1 | 1 | 2 |
Oxysterols receptor LXR-beta | 0 | 1 | 1 | 2 |
Peroxisome proliferator-activated receptor delta | 0 | 1 | 1 | 2 |
Peroxisome proliferator-activated receptor alpha | 0 | 1 | 1 | 2 |
Oxysterols receptor LXR-alpha | 0 | 1 | 1 | 2 |
Bile acid receptor | 0 | 1 | 1 | 2 |
Estrogen receptor beta | 0 | 2 | 0 | 2 |
Bile acid receptor | 0 | 2 | 1 | 3 |
NS5 | 0 | 0 | 1 | 1 |
Spike glycoprotein | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 2 | 1 | 0 | 0 | 1 |
glycogen synthase kinase-3 beta isoform 1 | 0 | 0 | 1 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
Transmembrane protease serine 2 | 0 | 0 | 1 | 1 |
ATP-binding cassette sub-family C member 3 | 0 | 1 | 0 | 1 |
Multidrug resistance-associated protein 4 | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1F | 0 | 1 | 0 | 1 |
Bile salt export pump | 0 | 1 | 0 | 1 |
Rap guanine nucleotide exchange factor 3 | 2 | 0 | 0 | 2 |
Polymerase basic protein 2 | 0 | 0 | 1 | 1 |
RNA-directed RNA polymerase catalytic subunit | 0 | 0 | 1 | 1 |
Polymerase acidic protein | 0 | 0 | 1 | 1 |
Procathepsin L | 0 | 0 | 1 | 1 |
Replicase polyprotein 1a | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Adenosine receptor A3 | 0 | 1 | 0 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Adenosylhomocysteinase | 0 | 0 | 0 | 2 |
Adenosine receptor A2a | 0 | 1 | 0 | 1 |
Adenosine receptor A1 | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1D | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1S | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Adenosine receptor A1 | 0 | 1 | 0 | 1 |
Genome polyprotein | 0 | 0 | 1 | 1 |
Canalicular multispecific organic anion transporter 1 | 0 | 1 | 0 | 1 |
Angiotensin-converting enzyme 2 | 0 | 0 | 1 | 1 |
Thymidine kinase | 0 | 1 | 0 | 2 |
Thymidine kinase, cytosolic | 0 | 2 | 0 | 4 |
Thymidine kinase | 0 | 1 | 0 | 2 |
Thymidylate synthase | 0 | 0 | 0 | 1 |
Thymidine phosphorylase | 0 | 0 | 0 | 1 |
Polyunsaturated fatty acid 5-lipoxygenase | 0 | 1 | 0 | 1 |
Glucose-6-phosphate 1-dehydrogenase | 0 | 1 | 0 | 1 |
Thymidine phosphorylase | 0 | 0 | 0 | 1 |
Thymidylate kinase | 0 | 1 | 0 | 1 |
Thymidine kinase, cytosolic | 0 | 0 | 0 | 2 |
Thymidine kinase | 0 | 0 | 0 | 1 |
Thymidylate kinase | 0 | 1 | 0 | 1 |
Thymidine kinase | 0 | 1 | 0 | 2 |
Sterol O-acyltransferase 1 | 0 | 1 | 0 | 1 |
Thymidine kinase | 0 | 0 | 0 | 1 |
Thymidine kinase | 0 | 0 | 0 | 1 |
Chain A, Cytidine Deaminase | 0 | 1 | 0 | 1 |
phosphopantetheinyl transferase | 1 | 0 | 0 | 1 |
nonstructural protein 1 | 1 | 0 | 0 | 1 |
Sodium/nucleoside cotransporter 1 | 0 | 2 | 0 | 2 |
Sodium/nucleoside cotransporter 2 | 0 | 2 | 0 | 2 |
Cytidine deaminase | 0 | 1 | 0 | 1 |
Equilibrative nucleoside transporter 2 | 0 | 2 | 0 | 2 |
Equilibrative nucleoside transporter 1 | 0 | 2 | 0 | 2 |
Uridine-cytidine kinase 1 | 0 | 0 | 0 | 1 |
Solute carrier family 28 member 3 | 0 | 2 | 0 | 2 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |