Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
RAR-related orphan receptor gamma | 3 | 0 | 0 | 3 |
TDP1 protein | 4 | 0 | 0 | 4 |
estrogen nuclear receptor alpha | 3 | 0 | 0 | 3 |
Liver carboxylesterase 1 | 0 | 0 | 0 | 1 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 3 | 0 | 0 | 3 |
Chain A, TYROSYL-DNA PHOSPHODIESTERASE | 1 | 0 | 0 | 1 |
Chain A, Putative fructose-1,6-bisphosphate aldolase | 1 | 0 | 0 | 1 |
acetylcholinesterase | 2 | 0 | 0 | 2 |
phosphopantetheinyl transferase | 2 | 0 | 0 | 2 |
estrogen receptor 2 (ER beta) | 2 | 0 | 0 | 2 |
G | 3 | 0 | 0 | 3 |
cytochrome P450 2D6 | 2 | 0 | 0 | 2 |
euchromatic histone-lysine N-methyltransferase 2 | 2 | 0 | 0 | 2 |
vitamin D3 receptor isoform VDRA | 2 | 0 | 0 | 2 |
histone-lysine N-methyltransferase 2A isoform 2 precursor | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 2 | 0 | 0 | 2 |
DNA polymerase kappa isoform 1 | 1 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 2 | 0 | 0 | 2 |
Interferon beta | 3 | 0 | 0 | 3 |
HLA class I histocompatibility antigen, B alpha chain | 3 | 0 | 0 | 3 |
Inositol hexakisphosphate kinase 1 | 3 | 0 | 0 | 3 |
cytochrome P450 2C9, partial | 3 | 0 | 0 | 3 |
ATP-dependent phosphofructokinase | 2 | 0 | 0 | 2 |
Thymidine kinase 2 | 0 | 1 | 0 | 1 |
Deoxycytidine kinase | 0 | 0 | 0 | 1 |
Probable deoxycytidylate deaminase | 0 | 0 | 0 | 1 |
Cytidine deaminase | 0 | 0 | 0 | 1 |
AAA family ATPase | 0 | 0 | 0 | 1 |
Reverse transcriptase/RNaseH | 0 | 0 | 1 | 1 |
Chain A, Uracil Phosphoribosyltransferase | 0 | 1 | 0 | 1 |
Luciferase | 2 | 0 | 0 | 2 |
interleukin 8 | 1 | 0 | 0 | 1 |
endonuclease IV | 1 | 0 | 0 | 1 |
glp-1 receptor, partial | 2 | 0 | 0 | 2 |
Skn7p | 0 | 0 | 0 | 1 |
thioredoxin reductase | 2 | 0 | 0 | 2 |
pregnane X receptor | 2 | 0 | 0 | 2 |
hypoxia-inducible factor 1 alpha subunit | 1 | 0 | 0 | 1 |
ATAD5 protein, partial | 1 | 0 | 0 | 1 |
GLI family zinc finger 3 | 2 | 0 | 0 | 2 |
Microtubule-associated protein tau | 2 | 0 | 0 | 2 |
Thrombopoietin | 1 | 0 | 0 | 1 |
AR protein | 3 | 0 | 0 | 3 |
aldehyde dehydrogenase 1 family, member A1 | 2 | 0 | 0 | 2 |
thyroid stimulating hormone receptor | 2 | 0 | 0 | 2 |
nuclear receptor subfamily 1, group I, member 3 | 2 | 0 | 0 | 2 |
progesterone receptor | 1 | 0 | 0 | 1 |
EWS/FLI fusion protein | 2 | 0 | 0 | 2 |
nonstructural protein 1 | 1 | 0 | 0 | 1 |
glucocorticoid receptor [Homo sapiens] | 2 | 0 | 0 | 2 |
retinoic acid nuclear receptor alpha variant 1 | 1 | 0 | 0 | 1 |
retinoid X nuclear receptor alpha | 2 | 0 | 0 | 2 |
estrogen-related nuclear receptor alpha | 1 | 0 | 0 | 1 |
farnesoid X nuclear receptor | 1 | 0 | 0 | 1 |
pregnane X nuclear receptor | 2 | 0 | 0 | 2 |
67.9K protein | 2 | 0 | 0 | 2 |
peroxisome proliferator-activated receptor delta | 2 | 0 | 0 | 2 |
peroxisome proliferator activated receptor gamma | 2 | 0 | 0 | 2 |
arylsulfatase A | 1 | 0 | 0 | 1 |
IDH1 | 2 | 0 | 0 | 2 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 2 | 0 | 0 | 2 |
v-jun sarcoma virus 17 oncogene homolog (avian) | 1 | 0 | 0 | 1 |
Histone H2A.x | 1 | 0 | 0 | 1 |
peripheral myelin protein 22 isoform 1 | 1 | 0 | 0 | 1 |
hemoglobin subunit beta | 1 | 0 | 0 | 1 |
chromobox protein homolog 1 | 2 | 0 | 0 | 2 |
nuclear factor erythroid 2-related factor 2 isoform 2 | 1 | 0 | 0 | 1 |
thyroid hormone receptor beta isoform 2 | 2 | 0 | 0 | 2 |
huntingtin isoform 2 | 1 | 0 | 0 | 1 |
flap endonuclease 1 | 1 | 0 | 0 | 1 |
serine/threonine-protein kinase mTOR isoform 1 | 1 | 0 | 0 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
geminin | 2 | 0 | 0 | 2 |
Vpr | 1 | 0 | 0 | 1 |
peripheral myelin protein 22 | 3 | 0 | 0 | 3 |
survival motor neuron protein isoform d | 2 | 0 | 0 | 2 |
muscleblind-like protein 1 isoform 1 | 1 | 0 | 0 | 1 |
lamin isoform A-delta10 | 3 | 0 | 0 | 3 |
ATP-binding cassette sub-family C member 3 | 0 | 2 | 0 | 2 |
Multidrug resistance-associated protein 4 | 0 | 2 | 0 | 2 |
Voltage-dependent calcium channel gamma-2 subunit | 1 | 0 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 0 | 0 | 1 |
Bile salt export pump | 0 | 3 | 0 | 3 |
Epidermal growth factor receptor | 0 | 2 | 0 | 2 |
Cellular tumor antigen p53 | 3 | 0 | 0 | 3 |
Amyloid-beta precursor protein | 1 | 0 | 0 | 1 |
Thymidylate synthase | 0 | 1 | 0 | 1 |
Aromatase | 0 | 3 | 0 | 3 |
Glutamate receptor 2 | 1 | 0 | 0 | 1 |
Canalicular multispecific organic anion transporter 1 | 0 | 2 | 0 | 2 |
ATPase family AAA domain-containing protein 5 | 1 | 0 | 0 | 1 |
Ataxin-2 | 1 | 0 | 0 | 1 |
HSP40, subfamily A [Plasmodium falciparum 3D7] | 0 | 0 | 0 | 1 |
USP1 protein, partial | 2 | 0 | 0 | 2 |
GALC protein | 1 | 0 | 0 | 1 |
cytochrome P450 family 3 subfamily A polypeptide 4 | 3 | 0 | 0 | 3 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
cytochrome P450 2D6 isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 2C19 precursor | 2 | 0 | 0 | 2 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | 1 | 0 | 0 | 1 |
importin subunit beta-1 isoform 1 | 1 | 0 | 0 | 1 |
mitogen-activated protein kinase 1 | 1 | 0 | 0 | 1 |
snurportin-1 | 1 | 0 | 0 | 1 |
GTP-binding nuclear protein Ran isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit pi | 2 | 0 | 0 | 2 |
Cytochrome P450 1A1 | 0 | 2 | 0 | 2 |
Cytochrome P450 1A2 | 0 | 2 | 0 | 2 |
Cytochrome P450 3A4 | 0 | 1 | 0 | 1 |
Cytochrome P450 2D6 | 0 | 1 | 0 | 1 |
Cytochrome P450 2C9 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit delta | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 2 | 0 | 0 | 2 |
Cytochrome P450 2C19 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-3 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-2 | 2 | 0 | 0 | 2 |
Cytochrome P450 1B1 | 0 | 1 | 0 | 1 |
GABA theta subunit | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit epsilon | 2 | 0 | 0 | 2 |
runt-related transcription factor 1 isoform AML1b | 1 | 0 | 0 | 1 |
core-binding factor subunit beta isoform 2 | 1 | 0 | 0 | 1 |
Carbonic anhydrase 2 | 0 | 1 | 0 | 1 |
Estrogen receptor | 0 | 1 | 0 | 1 |
Steryl-sulfatase | 0 | 1 | 0 | 1 |
Cytochrome P450 11B1, mitochondrial | 0 | 1 | 0 | 1 |
Cytochrome P450 11B2, mitochondrial | 0 | 1 | 0 | 1 |
Amine oxidase [flavin-containing] A | 0 | 1 | 0 | 1 |
Chain A, Beta-lactamase | 2 | 0 | 0 | 2 |
Genome polyprotein | 0 | 1 | 0 | 1 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | 1 | 0 | 0 | 1 |
nuclear receptor subfamily 1, group I, member 2 | 1 | 0 | 0 | 1 |
NPC intracellular cholesterol transporter 1 precursor | 1 | 0 | 0 | 1 |
Tyrosine-protein kinase ABL1 | 0 | 1 | 0 | 1 |
Tubulin alpha-1A chain | 0 | 0 | 1 | 2 |
Tubulin beta chain | 0 | 0 | 1 | 1 |
Tubulin beta-4A chain | 0 | 1 | 1 | 3 |
Receptor tyrosine-protein kinase erbB-2 | 0 | 1 | 0 | 1 |
Integrin beta-3 | 0 | 1 | 0 | 1 |
Tyrosine-protein kinase Fyn | 0 | 1 | 0 | 1 |
Integrin alpha-V | 0 | 1 | 0 | 1 |
Tubulin beta chain | 0 | 1 | 1 | 3 |
ATP-dependent translocase ABCB1 | 0 | 1 | 0 | 3 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
Tubulin alpha-3C chain | 0 | 1 | 1 | 3 |
Botulinum neurotoxin type A | 0 | 1 | 0 | 1 |
Apoptosis regulator Bcl-2 | 0 | 1 | 0 | 1 |
60 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Fibroblast growth factor receptor 1 | 0 | 1 | 0 | 1 |
Proto-oncogene tyrosine-protein kinase Src | 0 | 1 | 0 | 1 |
UDP-glucuronosyltransferase 2B7 | 0 | 1 | 0 | 1 |
UDP-glucuronosyltransferase 1-6 | 0 | 1 | 0 | 1 |
ATP-dependent translocase ABCB1 | 0 | 1 | 0 | 1 |
Substance-K receptor | 0 | 2 | 0 | 2 |
UDP-glucuronosyltransferase 1A1 | 0 | 1 | 0 | 1 |
UDP-glucuronosyltransferase 1A4 | 0 | 1 | 0 | 1 |
Serum paraoxonase/arylesterase 1 | 0 | 1 | 0 | 1 |
Cholecystokinin receptor type A | 0 | 2 | 0 | 2 |
Melanocortin receptor 5 | 0 | 2 | 0 | 2 |
UDP-glucuronosyltransferase 2B10 | 0 | 1 | 0 | 1 |
Delta-type opioid receptor | 0 | 2 | 0 | 2 |
10 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Tubulin alpha-1B chain | 0 | 1 | 1 | 3 |
Tubulin alpha-4A chain | 0 | 1 | 1 | 3 |
Tubulin beta-4B chain | 0 | 1 | 1 | 3 |
Bcl-2-like protein 1 | 0 | 1 | 0 | 1 |
Tyrosine-protein kinase Mer | 0 | 1 | 0 | 1 |
Tubulin beta-3 chain | 0 | 2 | 1 | 4 |
Tubulin beta-2A chain | 0 | 1 | 1 | 3 |
Thiosulfate sulfurtransferase | 0 | 1 | 0 | 1 |
Beta-tubulin | 0 | 1 | 0 | 1 |
Tubulin beta-8 chain | 0 | 1 | 1 | 3 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
Tubulin beta-2B chain | 0 | 0 | 1 | 3 |
Tubulin alpha-3E chain | 0 | 1 | 1 | 3 |
Tubulin alpha-1A chain | 0 | 1 | 1 | 3 |
10 kDa chaperonin | 0 | 1 | 0 | 1 |
Similar to alpha-tubulin isoform 1 | 0 | 0 | 1 | 3 |
Similar to alpha-tubulin isoform 1 | 0 | 0 | 0 | 2 |
Tubulin alpha-1C chain | 0 | 1 | 1 | 3 |
Tubulin beta-6 chain | 0 | 1 | 1 | 3 |
Tubulin beta-2B chain | 0 | 1 | 1 | 3 |
Tubulin beta-1 chain | 0 | 1 | 1 | 3 |
Nucleotide-binding oligomerization domain-containing protein 2 | 0 | 1 | 0 | 1 |
Solute carrier organic anion transporter family member 1B3 | 0 | 2 | 0 | 2 |
Solute carrier organic anion transporter family member 1B1 | 0 | 2 | 0 | 2 |
potassium voltage-gated channel subfamily H member 2 isoform d | 1 | 0 | 0 | 1 |
nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |