Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
interleukin 8 | 3 | 0 | 0 | 3 |
TDP1 protein | 6 | 0 | 0 | 6 |
GLI family zinc finger 3 | 6 | 0 | 0 | 6 |
AR protein | 4 | 0 | 0 | 4 |
aldehyde dehydrogenase 1 family, member A1 | 5 | 0 | 0 | 5 |
EWS/FLI fusion protein | 3 | 0 | 0 | 3 |
retinoic acid nuclear receptor alpha variant 1 | 5 | 0 | 0 | 5 |
estrogen-related nuclear receptor alpha | 5 | 0 | 0 | 5 |
farnesoid X nuclear receptor | 2 | 0 | 0 | 2 |
pregnane X nuclear receptor | 4 | 0 | 0 | 4 |
estrogen nuclear receptor alpha | 6 | 0 | 0 | 6 |
G | 1 | 0 | 0 | 1 |
cytochrome P450 2D6 | 1 | 0 | 0 | 1 |
peroxisome proliferator activated receptor gamma | 3 | 0 | 0 | 3 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | 4 | 0 | 0 | 4 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
activating transcription factor 6 | 1 | 0 | 0 | 1 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | 2 | 0 | 0 | 2 |
thyroid hormone receptor beta isoform 2 | 4 | 0 | 0 | 4 |
heat shock protein beta-1 | 2 | 0 | 0 | 2 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 3 | 0 | 0 | 3 |
DNA polymerase iota isoform a (long) | 1 | 0 | 0 | 1 |
geminin | 5 | 0 | 0 | 5 |
streptokinase A precursor | 0 | 0 | 3 | 3 |
lethal factor (plasmid) | 1 | 0 | 0 | 1 |
Dihydroxyacetone phosphate acyltransferase | 0 | 0 | 0 | 2 |
ATP-binding cassette sub-family C member 3 | 0 | 5 | 0 | 5 |
Multidrug resistance-associated protein 4 | 0 | 5 | 0 | 5 |
Bile salt export pump | 0 | 7 | 0 | 7 |
Interferon beta | 1 | 0 | 0 | 1 |
HLA class I histocompatibility antigen, B alpha chain | 1 | 0 | 0 | 1 |
30S ribosomal protein S6 | 0 | 3 | 1 | 4 |
30S ribosomal protein S7 | 0 | 3 | 1 | 4 |
50S ribosomal protein L15 | 0 | 3 | 1 | 4 |
Cellular tumor antigen p53 | 4 | 0 | 0 | 4 |
Cytochrome P450 3A4 | 0 | 2 | 0 | 2 |
50S ribosomal protein L10 | 0 | 3 | 1 | 4 |
50S ribosomal protein L11 | 0 | 3 | 1 | 4 |
50S ribosomal protein L7/L12 | 0 | 3 | 1 | 4 |
50S ribosomal protein L19 | 0 | 3 | 1 | 4 |
50S ribosomal protein L1 | 0 | 3 | 1 | 4 |
50S ribosomal protein L20 | 0 | 3 | 1 | 4 |
50S ribosomal protein L27 | 0 | 3 | 1 | 4 |
50S ribosomal protein L28 | 0 | 3 | 1 | 4 |
50S ribosomal protein L29 | 0 | 3 | 1 | 4 |
50S ribosomal protein L31 | 0 | 3 | 1 | 4 |
50S ribosomal protein L31 type B | 0 | 3 | 1 | 4 |
50S ribosomal protein L32 | 0 | 3 | 1 | 4 |
50S ribosomal protein L33 | 0 | 3 | 1 | 4 |
50S ribosomal protein L34 | 0 | 3 | 1 | 4 |
50S ribosomal protein L35 | 0 | 3 | 1 | 4 |
50S ribosomal protein L36 | 0 | 3 | 1 | 4 |
30S ribosomal protein S10 | 0 | 3 | 1 | 4 |
30S ribosomal protein S11 | 0 | 3 | 1 | 4 |
30S ribosomal protein S12 | 0 | 3 | 1 | 4 |
30S ribosomal protein S13 | 0 | 3 | 1 | 4 |
30S ribosomal protein S16 | 0 | 3 | 1 | 4 |
30S ribosomal protein S18 | 0 | 3 | 1 | 4 |
30S ribosomal protein S19 | 0 | 3 | 1 | 4 |
30S ribosomal protein S20 | 0 | 3 | 1 | 4 |
30S ribosomal protein S2 | 0 | 3 | 1 | 4 |
30S ribosomal protein S3 | 0 | 3 | 1 | 4 |
30S ribosomal protein S4 | 0 | 3 | 1 | 4 |
30S ribosomal protein S5 | 0 | 3 | 1 | 4 |
30S ribosomal protein S8 | 0 | 3 | 1 | 4 |
30S ribosomal protein S9 | 0 | 3 | 1 | 4 |
50S ribosomal protein L13 | 0 | 3 | 1 | 4 |
50S ribosomal protein L14 | 0 | 3 | 1 | 4 |
50S ribosomal protein L16 | 0 | 3 | 1 | 4 |
50S ribosomal protein L23 | 0 | 3 | 1 | 4 |
30S ribosomal protein S15 | 0 | 3 | 1 | 4 |
50S ribosomal protein L17 | 0 | 3 | 1 | 4 |
50S ribosomal protein L21 | 0 | 3 | 1 | 4 |
50S ribosomal protein L30 | 0 | 3 | 1 | 4 |
50S ribosomal protein L6 | 0 | 3 | 1 | 4 |
30S ribosomal protein S14 | 0 | 3 | 1 | 4 |
30S ribosomal protein S17 | 0 | 3 | 1 | 4 |
30S ribosomal protein S1 | 0 | 3 | 1 | 4 |
50S ribosomal protein L18 | 0 | 3 | 1 | 4 |
50S ribosomal protein L2 | 0 | 3 | 1 | 4 |
50S ribosomal protein L3 | 0 | 3 | 1 | 4 |
50S ribosomal protein L24 | 0 | 3 | 1 | 4 |
50S ribosomal protein L4 | 0 | 3 | 1 | 4 |
50S ribosomal protein L22 | 0 | 3 | 1 | 4 |
50S ribosomal protein L5 | 0 | 3 | 1 | 4 |
30S ribosomal protein S21 | 0 | 3 | 1 | 4 |
50S ribosomal protein L25 | 0 | 3 | 1 | 4 |
50S ribosomal protein L36 2 | 0 | 3 | 1 | 4 |
Inositol hexakisphosphate kinase 1 | 1 | 0 | 0 | 1 |
Methionine--tRNA ligase, mitochondrial | 0 | 0 | 1 | 1 |
cytochrome P450 2C9, partial | 1 | 0 | 0 | 1 |
Luciferase | 1 | 0 | 0 | 1 |
hypoxia-inducible factor 1 alpha subunit | 1 | 0 | 0 | 1 |
RAR-related orphan receptor gamma | 2 | 0 | 0 | 2 |
nuclear receptor subfamily 1, group I, member 3 | 2 | 0 | 0 | 2 |
progesterone receptor | 3 | 0 | 0 | 3 |
retinoid X nuclear receptor alpha | 3 | 0 | 0 | 3 |
peroxisome proliferator-activated receptor delta | 2 | 0 | 0 | 2 |
v-jun sarcoma virus 17 oncogene homolog (avian) | 3 | 0 | 0 | 3 |
Histone H2A.x | 2 | 0 | 0 | 2 |
lamin isoform A-delta10 | 1 | 0 | 0 | 1 |
Voltage-dependent calcium channel gamma-2 subunit | 1 | 0 | 0 | 1 |
Glutamate receptor 2 | 1 | 0 | 0 | 1 |
Nuclear receptor ROR-gamma | 2 | 0 | 0 | 2 |
Chain A, HADH2 protein | 3 | 0 | 0 | 3 |
Chain B, HADH2 protein | 3 | 0 | 0 | 3 |
endonuclease IV | 1 | 0 | 0 | 1 |
dopamine D1 receptor | 1 | 0 | 0 | 1 |
thioredoxin reductase | 2 | 0 | 0 | 2 |
pregnane X receptor | 2 | 0 | 0 | 2 |
GLS protein | 1 | 0 | 0 | 1 |
regulator of G-protein signaling 4 | 1 | 0 | 0 | 1 |
glucocorticoid receptor [Homo sapiens] | 4 | 0 | 0 | 4 |
euchromatic histone-lysine N-methyltransferase 2 | 3 | 0 | 0 | 3 |
peripheral myelin protein 22 isoform 1 | 1 | 0 | 0 | 1 |
atrial natriuretic peptide receptor 1 precursor | 1 | 0 | 0 | 1 |
chromobox protein homolog 1 | 1 | 0 | 0 | 1 |
flap endonuclease 1 | 2 | 0 | 0 | 2 |
survival motor neuron protein isoform d | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 1 | 0 | 0 | 1 |
M-phase phosphoprotein 8 | 1 | 0 | 0 | 1 |
muscarinic acetylcholine receptor M1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 1 | 1 | 0 | 2 |
Glucocorticoid receptor | 0 | 4 | 1 | 5 |
Sex hormone-binding globulin | 0 | 0 | 1 | 1 |
Glycine receptor subunit alpha-1 | 0 | 4 | 0 | 4 |
Corticosteroid-binding globulin | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit delta | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 1 | 1 | 0 | 2 |
Glycine receptor subunit beta | 0 | 4 | 0 | 4 |
Glycine receptor subunit alpha-2 | 0 | 4 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 1 | 1 | 0 | 2 |
Glycine receptor subunit alpha-3 | 0 | 4 | 0 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-3 | 1 | 1 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-2 | 1 | 1 | 0 | 2 |
Potassium voltage-gated channel subfamily A member 1 | 0 | 0 | 1 | 1 |
TAR DNA-binding protein 43 | 1 | 0 | 0 | 1 |
GABA theta subunit | 1 | 1 | 0 | 2 |
Multidrug and toxin extrusion protein 1 | 0 | 2 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit epsilon | 1 | 1 | 0 | 2 |
Chain A, Beta-lactamase | 1 | 0 | 0 | 1 |
Motilin receptor | 0 | 0 | 1 | 1 |
acid sphingomyelinase | 1 | 0 | 0 | 1 |
low molecular weight phosphotyrosine protein phosphatase isoform c | 0 | 1 | 0 | 1 |
serine/threonine-protein kinase PLK1 | 1 | 0 | 0 | 1 |
Motilin receptor | 0 | 1 | 1 | 2 |
Rap guanine nucleotide exchange factor 3 | 1 | 0 | 0 | 1 |
Albumin | 0 | 0 | 2 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
60 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Cytochrome P450 2C9 | 0 | 1 | 0 | 1 |
Chitinase B | 0 | 1 | 0 | 1 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Low molecular weight phosphotyrosine protein phosphatase | 0 | 1 | 0 | 1 |
Cytochrome P450 2J2 | 0 | 1 | 0 | 1 |
10 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Potassium voltage-gated channel subfamily H member 2 | 0 | 2 | 0 | 2 |
Cytochrome P450 1B1 | 0 | 1 | 0 | 1 |
Thiosulfate sulfurtransferase | 0 | 1 | 0 | 1 |
Lanosterol 14-alpha demethylase | 0 | 1 | 0 | 1 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
10 kDa chaperonin | 0 | 1 | 0 | 1 |
Canalicular multispecific organic anion transporter 1 | 0 | 4 | 0 | 4 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 1 | 0 | 0 | 1 |
Chain A, 2-oxoglutarate Oxygenase | 1 | 0 | 0 | 1 |
Chain A, Ferritin light chain | 1 | 0 | 0 | 1 |
arylsulfatase A | 1 | 0 | 0 | 1 |
STE24 | 0 | 0 | 0 | 1 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 2 | 2 | 0 | 0 | 2 |
parathyroid hormone/parathyroid hormone-related peptide receptor precursor | 1 | 0 | 0 | 1 |
CAAX prenyl protease | 0 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
Trypsin | 0 | 0 | 0 | 1 |
DNA gyrase subunit A | 0 | 1 | 0 | 2 |
DNA gyrase subunit B | 0 | 1 | 0 | 2 |
DNA gyrase subunit B | 0 | 1 | 0 | 2 |
DNA gyrase subunit A | 0 | 1 | 0 | 2 |
Chain A, TYROSYL-DNA PHOSPHODIESTERASE | 1 | 0 | 0 | 1 |
thioredoxin glutathione reductase | 1 | 0 | 0 | 1 |
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | 1 | 0 | 0 | 1 |
estrogen receptor 2 (ER beta) | 1 | 0 | 0 | 1 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 1 | 0 | 0 | 1 |
vitamin D3 receptor isoform VDRA | 2 | 0 | 0 | 2 |
nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
Bile salt export pump | 0 | 1 | 0 | 1 |
Enoyl-[acyl-carrier-protein] reductase [NADH] | 0 | 0 | 0 | 1 |
Protein-arginine deiminase type-4 | 0 | 3 | 0 | 3 |
thyroid stimulating hormone receptor | 1 | 0 | 0 | 1 |
67.9K protein | 1 | 0 | 0 | 1 |
cytochrome P450 2C19 precursor | 1 | 0 | 0 | 1 |
cytochrome P450 2C9 precursor | 1 | 0 | 0 | 1 |
thyroid hormone receptor beta isoform a | 1 | 0 | 0 | 1 |
Endothelin-1 receptor | 0 | 2 | 0 | 2 |
Endothelin-1 receptor | 0 | 1 | 0 | 1 |
Histamine H2 receptor | 1 | 0 | 0 | 1 |
90-kda heat shock protein beta HSP90 beta, partial | 0 | 1 | 0 | 1 |
estrogen receptor beta isoform 1 | 0 | 1 | 0 | 1 |
heat shock protein HSP 90-alpha isoform 2 | 0 | 1 | 0 | 1 |
tyrosine-protein phosphatase non-receptor type 7 isoform 2 | 0 | 1 | 0 | 1 |
Tetracycline resistance protein, class B | 0 | 0 | 0 | 1 |
Muscarinic acetylcholine receptor M2 | 0 | 1 | 0 | 1 |
72 kDa type IV collagenase | 0 | 1 | 0 | 1 |
Stromelysin-1 | 0 | 1 | 0 | 1 |
Multidrug transporter MdfA | 0 | 1 | 0 | 1 |
Alpha-1B adrenergic receptor | 0 | 1 | 0 | 1 |
Neutrophil collagenase | 0 | 1 | 0 | 1 |
Alpha-1D adrenergic receptor | 0 | 1 | 0 | 1 |
Alpha-synuclein | 0 | 1 | 0 | 1 |
Alpha-1A adrenergic receptor | 0 | 1 | 0 | 1 |
Collagenase 3 | 0 | 1 | 0 | 1 |
Cannabinoid receptor 1 | 0 | 1 | 0 | 1 |
Integrase | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 0 | 0 | 1 |
P2Y purinoceptor 12 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 11 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 7 | 0 | 0 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |