Page last updated: 2024-09-27

Microscopic Polyangiitis

A primary systemic vasculitis of small- and some medium-sized vessels. It is characterized by a tropism for kidneys and lungs, positive association with anti-neutrophil cytoplasmic antibodies (ANCA), and a paucity of immunoglobulin deposits in vessel walls.

Synonyms(1)

Synonym
Microscopic Polyangiitis

Research Excerpts

Overview

ExcerptReference
"Microscopic polyangiitis is an autoimmune small-vessel vasculitis that often manifests as focal and necrotizing glomerulonephritis and renal failure."( Borza, DB; Chang, J; Fugger, L; Hickey, MJ; Holdsworth, SR; Kitching, AR; Ooi, JD, 2012)
"Microscopic polyangiitis is characterized by pauci-immune, necrotizing small-vessel vasculitis and an anti-neutrophil cytoplasmic antibody-associated vasculitis."( Fukushima, M; Imai, Y; Inokuma, T; Inoue, S; Ono, Y; Tamaki, Y; Yoshimura, H, 2013)
"Microscopic polyangiitis is an ANCA-associated vasculitis and affects small sized vessels."( Abouzid, Z; Bayahia, R; Benamar, L; Benjaafar, A; Bouattar, T; Chattahi, M; Ouzeddoun, N; Rouass, L; Sebti, K, 2022)
"Microscopic polyangiitis is a necrotising vasculitis characterised by anti-neutrophil cytoplasmic antibodies against myeloperoxidase."( Kataoka, H; Kondo, M; Mukai, M; Nakanowatari, M; Tomita, T, 2023)
"Microscopic polyangiitis is an important and common component of cytoplasmic antibody-associated vasculitides that can lead to serious morbidity and even death."( Akdam, H; Alp, A; Ersoy, M; Kahraman Çetin, N; Meteoğlu, İ; Yeniçerioğlu, Y, 2023)

Research

Studies (252)

TimeframeStudies, This Condition (%)All Conditions %
pre-19900 (0.00)23.3326
1990's0 (0.00)12.5806
2000's8 (3.17)18.1394
2010's168 (66.67)28.8240
2020's76 (30.16)9.53
DrugIndicatedRelationship StrengthStudiesTrials
salicylic acid0low10
gabexate0low10
leflunomide0low10
nafamostat0low10
corticosterone0low10
isoxazoles0low10
citrulline0low20
azetidyl-2-carboxylic acid0low10
betamethasone valerate0low10
hypochlorous acid0low10
ursodeoxycholic acid0low10
piperacillin0low10
azelnidipine0low10
fluorodeoxyglucose f180low40
mizoribine0low40
methotrexate0medium102
trimethoprim, sulfamethoxazole drug combination0low40
dihydropyridines0low10
resveratrol0low10
tacrolimus0low10
mycophenolic acid0medium133
propylthiouracil0low20
mocetinostat0medium1223
tofacitinib0low10
cardiovascular agents0low10
piperidines0low10
interleukin-80low10
acenocoumarol0low10
nephrin0low10
ganciclovir0low10
eye0low10

Protein Targets (1,024)

ProteinPotency MeasurementsInhibition MeasurementsActivation MeasurementsDrugs
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE5005
Luciferase3003
RAR-related orphan receptor gamma100010
retinoid X nuclear receptor alpha120012
G9009
peroxisome proliferator activated receptor gamma100010
euchromatic histone-lysine N-methyltransferase 2100010
thyroid stimulating hormone receptor6006
chromobox protein homolog 16006
parathyroid hormone/parathyroid hormone-related peptide receptor precursor5005
geminin140014
muscleblind-like protein 1 isoform 15005
Interferon beta120012
HLA class I histocompatibility antigen, B alpha chain 9009
Guanine nucleotide-binding protein G2002
Inositol hexakisphosphate kinase 19009
cytochrome P450 2C9, partial9009
Chain A, TYROSYL-DNA PHOSPHODIESTERASE4004
Chain A, Ferritin light chain3003
interleukin 82002
acetylcholinesterase5005
thioredoxin reductase8008
phosphopantetheinyl transferase5005
SMAD family member 24004
ATAD5 protein, partial4004
Fumarate hydratase4004
SMAD family member 34004
TDP1 protein140014
GLI family zinc finger 3110011
Microtubule-associated protein tau4004
AR protein120012
thioredoxin glutathione reductase2002
nuclear receptor subfamily 1, group I, member 38008
EWS/FLI fusion protein9009
glucocorticoid receptor [Homo sapiens]120012
retinoic acid nuclear receptor alpha variant 1100010
estrogen-related nuclear receptor alpha120012
farnesoid X nuclear receptor7007
pregnane X nuclear receptor110011
estrogen nuclear receptor alpha150015
polyprotein4004
P533003
peroxisome proliferator-activated receptor delta7007
arylsulfatase A5005
IDH16006
aryl hydrocarbon receptor7007
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a100010
activating transcription factor 64004
v-jun sarcoma virus 17 oncogene homolog (avian)6006
Histone H2A.x6006
Bloom syndrome protein isoform 17007
peripheral myelin protein 22 isoform 13003
hemoglobin subunit beta1001
cellular tumor antigen p53 isoform a4004
thyroid hormone receptor beta isoform 2110011
heat shock protein beta-14004
nuclear factor erythroid 2-related factor 2 isoform 1100010
DNA polymerase iota isoform a (long)6006
peripheral myelin protein 226006
survival motor neuron protein isoform d9009
cytochrome P450 3A4 isoform 16006
M-phase phosphoprotein 83003
muscarinic acetylcholine receptor M12002
lamin isoform A-delta109009
Gamma-aminobutyric acid receptor subunit pi6006
ATP-binding cassette sub-family C member 3010010
Multidrug resistance-associated protein 4010011
Bile salt export pump0404
Voltage-dependent calcium channel gamma-2 subunit8008
Bile salt export pump015015
Cellular tumor antigen p539009
Gamma-aminobutyric acid receptor subunit beta-16006
Gamma-aminobutyric acid receptor subunit delta6006
Gamma-aminobutyric acid receptor subunit gamma-26006
Glutamate receptor 28109
Gamma-aminobutyric acid receptor subunit alpha-56006
Gamma-aminobutyric acid receptor subunit alpha-36006
Gamma-aminobutyric acid receptor subunit gamma-16006
Gamma-aminobutyric acid receptor subunit alpha-26006
Gamma-aminobutyric acid receptor subunit alpha-46006
Gamma-aminobutyric acid receptor subunit gamma-36006
Gamma-aminobutyric acid receptor subunit alpha-66006
Nuclear receptor ROR-gamma4004
Gamma-aminobutyric acid receptor subunit alpha-16006
Gamma-aminobutyric acid receptor subunit beta-36006
Gamma-aminobutyric acid receptor subunit beta-26006
GABA theta subunit6006
Canalicular multispecific organic anion transporter 1010010
ATPase family AAA domain-containing protein 59009
Ataxin-29009
Gamma-aminobutyric acid receptor subunit epsilon6006
Protein-arginine deiminase type-40303
hypoxia-inducible factor 1 alpha subunit4004
USP1 protein, partial4004
caspase 7, apoptosis-related cysteine protease3003
estrogen receptor 2 (ER beta)5005
progesterone receptor110011
cytochrome P450 family 3 subfamily A polypeptide 47007
cytochrome P450 2D66006
vitamin D (1,25- dihydroxyvitamin D3) receptor8008
caspase-33003
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a4004
Caspase-71001
caspase-31001
nuclear receptor ROR-gamma isoform 15005
Spike glycoprotein4004
Proton-coupled amino acid transporter 10101
N(G),N(G)-dimethylarginine dimethylaminohydrolase 10101
General amino-acid permease GAP10001
Nitric oxide synthase, brain0101
Nitric oxide synthase, brain 0101
Chain A, HADH2 protein6006
Chain B, HADH2 protein6006
pregnane X receptor2002
NFKB1 protein, partial2002
GALC protein1001
Thrombopoietin2002
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)5005
nonstructural protein 13003
thyroid hormone receptor beta isoform a4004
nuclear factor erythroid 2-related factor 2 isoform 27007
mitogen-activated protein kinase 11001
serine/threonine-protein kinase mTOR isoform 12002
Solute carrier family 22 member 20202
Solute carrier family 22 member 1 0203
Solute carrier family 22 member 30101
Solute carrier family 22 member 30101
Sex hormone-binding globulin0011
Corticosteroid-binding globulin0202
Mineralocorticoid receptor 0224
Androgen receptor0404
C-8 sterol isomerase0101
Solute carrier organic anion transporter family member 1A10101
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase0101
Solute carrier family 22 member 10202
Sigma non-opioid intracellular receptor 10101
Solute carrier family 22 member 20202
cytochrome P450 2D6 isoform 11001
lethal factor (plasmid)2002
Membrane primary amine oxidase 0101
Polyunsaturated fatty acid lipoxygenase ALOX15B2002
Coagulation factor X0202
Plasminogen0404
Coagulation factor XII0202
Urokinase-type plasminogen activator0101
Tissue-type plasminogen activator0101
Serine protease hepsin0303
Histamine H2 receptor3003
Multidrug and toxin extrusion protein 20101
Multidrug and toxin extrusion protein 10101
Thymidine kinase 0101
endonuclease IV1001
ClpP3003
GLS protein3003
aldehyde dehydrogenase 1 family, member A19009
POU domain, class 2, transcription factor 20001
Transitional endoplasmic reticulum ATPase0101
Purine nucleoside phosphorylase0011
Solute carrier family 22 member 60103
glp-1 receptor, partial3003
matrix metalloproteinase 1, partial0011
PPM1D protein5005
Parkin2002
pyruvate kinase2002
nuclear receptor subfamily 1, group I, member 23003
NPC intracellular cholesterol transporter 1 precursor2002
cytochrome P450 2C19 precursor2002
cytochrome P450 2C9 precursor1001
histone deacetylase 9 isoform 32002
huntingtin isoform 23003
ras-related protein Rab-9A2002
urokinase-type plasminogen activator precursor3003
plasminogen precursor3003
urokinase plasminogen activator surface receptor precursor3003
histone acetyltransferase KAT2A isoform 14004
neuropeptide S receptor isoform A1001
Dihydroorotate dehydrogenase (quinone), mitochondrial0101
Integrin beta-33104
Cytochrome P450 1A20202
Aldo-keto reductase family 1 member B10404
Integrin alpha-IIb3104
Amine oxidase [flavin-containing] A0202
Endothelin receptor type B2002
Sodium-dependent noradrenaline transporter 0415
Endothelin-1 receptor2002
Sodium-dependent dopamine transporter 0202
Dihydroorotate dehydrogenase (quinone), mitochondrial0101
Dihydroorotate dehydrogenase (quinone), mitochondrial0101
dopamine D1 receptor2002
atrial natriuretic peptide receptor 1 precursor1001
flap endonuclease 12002
Alkaline phosphatase, tissue-nonspecific isozyme0202
Alkaline phosphatase, placental type0101
Alkaline phosphatase, tissue-nonspecific isozyme 0202
Intestinal-type alkaline phosphatase0101
Intestinal-type alkaline phosphatase0101
5'-nucleotidase0101
Phospholipase A-2-activating protein0101
ATP-dependent phosphofructokinase5005
Chain B, DIHYDROFOLATE REDUCTASE0011
Chain B, DIHYDROFOLATE REDUCTASE0011
Chain B, DIHYDROFOLATE REDUCTASE0011
Chain A, 2-oxoglutarate Oxygenase6006
acid sphingomyelinase1001
15-lipoxygenase, partial1001
67.9K protein3003
Thymidylate synthase 0101
alpha-galactosidase1001
Thymidylate synthase 0101
polyunsaturated fatty acid lipoxygenase ALOX121001
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 14004
vitamin D3 receptor isoform VDRA3003
transcriptional regulator ERG isoform 31001
importin subunit beta-1 isoform 11001
DNA polymerase beta2002
nuclear receptor coactivator 1 isoform 1 [Homo sapiens]0101
snurportin-11001
peptidyl-prolyl cis-trans isomerase NIMA-interacting 13003
DNA polymerase eta isoform 11001
transactivating tegument protein VP16 [Human herpesvirus 1]0101
DNA polymerase kappa isoform 13003
caspase-1 isoform alpha precursor1001
nuclear receptor coactivator 3 isoform a0101
Toll-like receptor 40101
Fatty-acid amide hydrolase 10101
ATP-binding cassette sub-family C member 30102
Dihydrofolate reductase0203
Dihydrofolate reductase0203
Dihydrofolate reductase 0101
Dihydrofolate reductase0101
Dihydrofolate reductase0101
Dihydrofolate reductase0203
Thymidylate synthase0101
Tyrosine-protein kinase ABL10124
Carbonic anhydrase 20314
Thymidylate synthase0202
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Thymidylate synthase0202
5-hydroxytryptamine receptor 2C0203
High mobility group protein B10022
Dihydrofolate reductase0101
Thymidylate synthase0101
Dihydrofolate reductase0224
Glucose-6-phosphate 1-dehydrogenase0101
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Folate receptor beta0101
5-hydroxytryptamine receptor 2A0202
Cytochrome P450 11B1, mitochondrial 0101
Folate receptor alpha0101
Dihydrofolate reductase0202
Histidine decarboxylase0101
Trifunctional purine biosynthetic protein adenosine-30101
Cyclin-dependent kinase 20123
Bifunctional purine biosynthesis protein ATIC0202
Multidrug resistance-associated protein 1 0001
Delta-type opioid receptor0101
Mu-type opioid receptor0101
Kappa-type opioid receptor0101
Reduced folate transporter0202
Folylpolyglutamate synthase, mitochondrial0103
6-phosphogluconate dehydrogenase, decarboxylating0101
Caspase-71001
Solute carrier organic anion transporter family member 1A30001
Dihydrofolate reductase0101
Pteridine reductase 10101
Folylpolyglutamate synthase, mitochondrial0103
Bifunctional dihydrofolate reductase-thymidylate synthase0101
TAR DNA-binding protein 433003
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Canalicular multispecific organic anion transporter 10102
Trifunctional purine biosynthetic protein adenosine-30101
Solute carrier family 22 member 200202
Dihydrofolate reductase 0101
Solute carrier family 22 member 80102
Solute carrier family 22 member 60202
Dihydrofolate reductase0101
ATP-binding cassette sub-family C member 110001
Proton-coupled folate transporter0101
Multidrug resistance associated protein0102
Solute carrier organic anion transporter family member 1B30001
Solute carrier family 22 member 110001
Broad substrate specificity ATP-binding cassette transporter ABCG20102
bromodomain adjacent to zinc finger domain 2B1001
Nuclear receptor subfamily 1 group I member 20022
Glucocorticoid receptor06314
Glycine receptor subunit alpha-10606
Glycine receptor subunit beta0606
Glycine receptor subunit alpha-20606
Glycine receptor subunit alpha-30606
Nuclear receptor subfamily 1 group I member 20011
regulator of G-protein signaling 42002
lysosomal alpha-glucosidase preproprotein2002
glycogen synthase kinase-3 beta isoform 10011
Histone deacetylase 30202
Nuclear receptor corepressor 10101
Integrin beta-10101
Cytochrome P450 3A40505
Leukotriene A-4 hydrolase0202
Cytochrome P450 2D60202
Integrin alpha-40101
Cytochrome P450 2C190303
Histone deacetylase 40101
Potassium voltage-gated channel subfamily H member 20101
Histone deacetylase 10202
Histone deacetylase 70101
Histone deacetylase 20202
Histone deacetylase 11 0101
Histone deacetylase 80101
Histone deacetylase 60101
Histone deacetylase 50101
Nuclear receptor corepressor 20101
Chain A, Inosine-5'-Monophosphate Dehydrogenase 20101
UDP-glucuronosyltransferase 1A90001
Inosine-5'-monophosphate dehydrogenase 20202
Glutamate receptor 10101
Glutamate receptor 30101
Glutamate receptor 40101
Inosine-5'-monophosphate dehydrogenase 1 0202
UDP-glucuronosyltransferase 1A1 0001
Sodium-dependent serotonin transporter0101
Peroxisome proliferator-activated receptor gamma0011
Alpha-synuclein2002
Inosine-5'-monophosphate dehydrogenase0102
UDP-glucuronosyltransferase 1A70001
UDP-glucuronosyltransferase 1A100001
UDP-glucuronosyltransferase 1A80001
Ubiquitin-like modifier activating enzyme 20101
SUMO1 activating enzyme subunit 10101
ubiquitin-like modifier-activating enzyme 10101
SUMO-conjugating enzyme UBC90101
ubiquitin-conjugating enzyme E2 N0101
ubiquitin-conjugating enzyme E2 variant 1 isoform a0101
Prothrombin0101
Complement C1r subcomponent0101
Cationic trypsin0101
Interstitial collagenase0101
Cathepsin D0202
Trypsin-10101
72 kDa type IV collagenase0101
Complement C1s subcomponent0101
Matrix metalloproteinase-90101
Neutrophil collagenase0101
5-hydroxytryptamine receptor 2B0101
Collagenase 30101
Hepatocyte growth factor activator0213
Suppressor of tumorigenicity 14 protein0101
Beta-lactamase 0001
Beta-lactamase 0101
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Metallo-beta-lactamase type 20001
Beta-lactamase 0001
Metallo-beta-lactamase VIM-19 0001
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Voltage-dependent L-type calcium channel subunit alpha-1F0101
Beta-lactamase SHV-10001
Beta-lactamase SHV-10001
Beta-lactamase0001
Beta-lactamase OXA-70001
Kappa-type opioid receptor0001
Solute carrier family 15 member 10101
Voltage-dependent L-type calcium channel subunit alpha-1D 0101
Voltage-dependent L-type calcium channel subunit alpha-1S0101
Voltage-dependent L-type calcium channel subunit alpha-1C0101
Metallo-beta-lactamase VIM-130001
Beta-lactamase 0001
Beta-lactamase 0001
Metallo-beta-lactamase VIM-20001
Beta-lactamase 0001
Beta-lactamase 0001
Class D beta-lactamase0001
Beta-lactamase 0001
Beta-lactamase 0001
Beta-lactamase 0001
Metallo-b-lactamase 0001
BlaVIM-1 0001
Beta-lactamase 0001
Carbapenem-hydrolyzing beta-lactamase KPC0001
Histamine H3 receptor0001
Beta-lactamase class B VIM-2 0001
Beta-lactamase VIM-1 0001
luciferase0001
Fatty acid-binding protein, liver0101
Estrogen receptor0303
Progesterone receptor0203
Glucocorticoid receptor0112
Glucocorticoid receptor0011
Androgen receptor0202
Cytochrome P450 2C9 0303
Glutamine synthetase0011
Histamine H1 receptor0011
Prostaglandin G/H synthase 20314
Nociceptin receptor0011
Cytochrome P450 2J20101
Estrogen receptor beta0202
Chain A, Putative fructose-1,6-bisphosphate aldolase2002
thyroid stimulating hormone receptor1001
NADH-cytochrome b5 reductase 3 0101
Myeloperoxidase0101
Thyroid peroxidase0101
Taste receptor type 2 member 380012
Chain A, Beta-lactamase3003
Chain A, Troponin C, slow skeletal and cardiac muscles0011
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
Chain A, Leukotriene A-4 hydrolase0101
BRCA11001
M18 aspartyl aminopeptidase0101
cathepsin L10101
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)1001
hexokinase-4 isoform 11001
glucokinase regulatory protein1001
atrial natriuretic peptide receptor 2 precursor1001
nuclear factor NF-kappa-B p105 subunit isoform 10011
FAD-linked sulfhydryl oxidase ALR0001
Vif0101
DNA dC->dU-editing enzyme APOBEC-3G isoform 10101
transcription factor p65 isoform 10011
serine/threonine-protein kinase 33 isoform a0011
POsterior Segregation0011
Aryl hydrocarbon receptor0101
Estrogen receptor beta0012
Acetylcholinesterase0101
Polyphenol oxidase 20203
Carbonic anhydrase 120202
Lysine-specific histone demethylase 1A0101
Transient receptor potential cation channel subfamily A member 10112
Carbonic anhydrase 10303
Myc proto-oncogene protein0102
Transthyretin0011
Cytochrome P450 1A10101
Amyloid-beta precursor protein0112
Prostaglandin G/H synthase 10112
Tyrosine-protein kinase Lck0213
Cholinesterase0101
Carbonic anhydrase 30202
ATP-dependent translocase ABCB10102
Luciferin 4-monooxygenase0101
Neuronal acetylcholine receptor subunit alpha-40101
DNA polymerase alpha catalytic subunit0101
Polyunsaturated fatty acid 5-lipoxygenase0101
Breakpoint cluster region protein0113
Tyrosinase0202
Aromatase0202
Ornithine decarboxylase0101
Neuronal acetylcholine receptor subunit beta-20101
Tyrosinase0101
Ribosyldihydronicotinamide dehydrogenase [quinone]0224
Protein kinase C alpha type0123
Tyrosine-protein phosphatase non-receptor type 10204
5-hydroxytryptamine receptor 1A0102
Estrogen receptor0012
Nuclear factor NF-kappa-B p105 subunit0101
Acetylcholinesterase0202
Carbonic anhydrase 40202
Prostaglandin G/H synthase 10202
Carbonic anhydrase 60202
Sucrase-isomaltase, intestinal0101
Amine oxidase [flavin-containing] B0101
Dipeptidyl peptidase 40101
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 10101
Nitric oxide synthase, inducible0101
Carbonic anhydrase 5A, mitochondrial0202
Carbonic anhydrase 70202
Cannabinoid receptor 10101
D(1A) dopamine receptor1001
Alpha-glucosidase MAL120101
Prostaglandin G/H synthase 20101
Cholinesterase0101
Inositol monophosphatase 11001
Nuclear factor NF-kappa-B p100 subunit 0101
Squalene synthase0101
Transcription factor p650101
cAMP-specific 3',5'-cyclic phosphodiesterase 4B0001
Bcl-2-like protein 10101
Serine/threonine-protein kinase PAK 10112
Nuclear factor erythroid 2-related factor 20012
Cytochrome P450 1B10202
Carbonic anhydrase 90202
N1L 0101
NAD(P)H dehydrogenase [quinone] 10002
Tubulin beta-2B chain0101
Lysosomal alpha-glucosidase0101
Transient receptor potential cation channel subfamily A member 10101
Similar to alpha-tubulin isoform 1 0101
Similar to alpha-tubulin isoform 1 0101
NAD-dependent protein deacetylase sirtuin-20011
Carbonic anhydrase 130101
Rap guanine nucleotide exchange factor 41001
NAD-dependent protein deacetylase sirtuin-10013
Carbonic anhydrase 150202
Prenyltransferase homolog0001
NAD-dependent protein deacetylase sirtuin-3, mitochondrial0011
Carbonic anhydrase 140202
Zinc finger protein mex-50011
Carbonic anhydrase 5B, mitochondrial0202
large T antigen0101
chaperonin-containing TCP-1 beta subunit homolog1001
Inhibitor of nuclear factor kappa-B kinase subunit beta0012
Solute carrier family 22 member 60101
5'-AMP-activated protein kinase subunit beta-20001
Albumin0112
Polymerase acidic protein0011
Stromelysin-10011
Tyrosine-protein phosphatase YopH0101
Aldo-keto reductase family 1 member B10101
Prolyl 4-hydroxylase subunit alpha-10101
Cystathionine gamma-lyase0101
5'-AMP-activated protein kinase subunit gamma-10012
5'-AMP-activated protein kinase catalytic subunit alpha-20012
Xanthine dehydrogenase/oxidase0101
5'-AMP-activated protein kinase catalytic subunit alpha-10012
Carbonic anhydrase0101
Solute carrier family 22 member 70001
Nicotinate phosphoribosyltransferase0101
Ubiquitin-like domain-containing CTD phosphatase 10101
Carbonic anhydrase 130101
5'-AMP-activated protein kinase subunit gamma-30001
5'-AMP-activated protein kinase subunit gamma-20012
5'-AMP-activated protein kinase subunit beta-10001
UDP-glucuronosyltransferase 2B70001
Cytochrome P450 3A50101
UDP-glucuronosyltransferase 1A40001
Serine/threonine-protein kinase mTOR0112
Peptidyl-prolyl cis-trans isomerase FKBP1A0213
Peptidyl-prolyl cis-trans isomerase FKBP1B0011
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform0101
Peptidyl-prolyl cis-trans isomerase FKBP50101
Splicing factor 3B subunit 30101
Solute carrier organic anion transporter family member 1B10101
Chain A, Tyrosine-protein kinase0101
Chain A, Tyrosine-protein kinase0101
Chain A, Tyrosine-protein kinase JAK20101
Leukotriene C4 synthase0011
tyrosine-protein kinase Yes1001
Serine/threonine-protein kinase Sgk10101
Bone morphogenetic protein receptor type-1B0011
Membrane-associated progesterone receptor component 10011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform0011
Serine/threonine-protein kinase PLK40011
Serine/threonine-protein kinase 250011
ATP-dependent RNA helicase DDX3X0011
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta0011
Pyridoxal kinase0011
Citron Rho-interacting kinase0011
Serine/threonine-protein kinase RIO30011
Dual specificity mitogen-activated protein kinase kinase 70112
Serine/threonine-protein kinase Chk10112
Peripheral plasma membrane protein CASK0011
Aurora kinase A0011
Cyclin-G-associated kinase0011
Serine/threonine-protein kinase DCLK10011
Inhibitor of nuclear factor kappa-B kinase subunit alpha0011
Muscle, skeletal receptor tyrosine-protein kinase0011
Ephrin type-B receptor 60011
Peroxisomal acyl-coenzyme A oxidase 30011
Mitogen-activated protein kinase 130112
3-phosphoinositide-dependent protein kinase 10011
Mitogen-activated protein kinase kinase kinase 130011
Death-associated protein kinase 30011
Mitogen-activated protein kinase kinase kinase 70011
Receptor-interacting serine/threonine-protein kinase 20011
Mitotic checkpoint serine/threonine-protein kinase BUB10011
NUAK family SNF1-like kinase 10011
Dynamin-like 120 kDa protein, mitochondrial0011
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma0011
Tyrosine-protein kinase JAK20327
Rho-associated protein kinase 20112
Serine/threonine-protein kinase ULK10011
Serine/threonine-protein kinase/endoribonuclease IRE10011
Ribosomal protein S6 kinase alpha-50112
U5 small nuclear ribonucleoprotein 200 kDa helicase0011
Ribosomal protein S6 kinase alpha-40011
Serine/threonine-protein kinase 160011
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma0011
Serine/threonine-protein kinase PAK 30011
Cyclin-dependent kinase-like 50011
Serine/threonine-protein kinase 17B0011
Serine/threonine-protein kinase 100011
Serine/threonine-protein kinase D30011
Cyclin-dependent kinase 140011
Mitogen-activated protein kinase kinase kinase 60011
Serine/threonine-protein kinase OSR10011
Mitogen-activated protein kinase kinase kinase kinase 40011
Serine/threonine-protein kinase LATS10011
Serine/threonine-protein kinase PAK 40011
Serine/threonine-protein kinase Chk20011
Epidermal growth factor receptor0112
RAF proto-oncogene serine/threonine-protein kinase0011
Receptor tyrosine-protein kinase erbB-20112
High affinity nerve growth factor receptor0011
ADP/ATP translocase 20011
Protein kinase C beta type0011
Insulin receptor0112
Tyrosine-protein kinase Fyn0011
Cyclin-dependent kinase 10011
Glycogen phosphorylase, liver form0011
Tyrosine-protein kinase Fes/Fps0011
Macrophage colony-stimulating factor 1 receptor0011
Tyrosine-protein kinase Yes0011
Tyrosine-protein kinase Lyn0011
Proto-oncogene tyrosine-protein kinase receptor Ret0011
Insulin-like growth factor 1 receptor0011
Signal recognition particle receptor subunit alpha0011
Cytochrome c1, heme protein, mitochondrial0011
Hepatocyte growth factor receptor0011
Tyrosine-protein kinase HCK0011
Proto-oncogene tyrosine-protein kinase ROS0011
Platelet-derived growth factor receptor beta0011
Tyrosine-protein kinase Fgr0011
Wee1-like protein kinase 20011
Uncharacterized serine/threonine-protein kinase SBK30011
Serine/threonine-protein kinase A-Raf0011
Cytochrome P450 2C80101
Mast/stem cell growth factor receptor Kit0011
Glycogen phosphorylase, brain form0011
Serine/threonine-protein kinase pim-10011
Fibroblast growth factor receptor 10011
DNA topoisomerase 2-alpha0011
Cytochrome P450 2A60101
Myosin light chain kinase, smooth muscle0011
Cyclin-dependent kinase 40011
ADP/ATP translocase 30011
Proto-oncogene tyrosine-protein kinase Src0011
Insulin receptor-related protein0011
Serine/threonine-protein kinase B-raf0011
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform0011
Platelet-derived growth factor receptor alpha0011
Tyrosine-protein kinase Fer0011
cAMP-dependent protein kinase catalytic subunit alpha0011
Vascular endothelial growth factor receptor 1 0011
General transcription and DNA repair factor IIH helicase subunit XPD0011
Interferon-induced, double-stranded RNA-activated protein kinase0011
Casein kinase II subunit alpha'0011
Ras-related protein Rab-6A0011
Serine/threonine-protein kinase MAK0011
Cyclin-dependent kinase 11B0011
Ephrin type-A receptor 10011
Fibroblast growth factor receptor 20011
Receptor tyrosine-protein kinase erbB-30011
Multifunctional protein ADE20011
Fibroblast growth factor receptor 40011
Fibroblast growth factor receptor 30011
cAMP-dependent protein kinase catalytic subunit gamma0011
cAMP-dependent protein kinase catalytic subunit beta0011
Ferrochelatase, mitochondrial0011
Ribosomal protein S6 kinase beta-10112
Tyrosine-protein kinase JAK10327
Protein kinase C eta type0011
Beta-adrenergic receptor kinase 10011
Probable ATP-dependent RNA helicase DDX60011
Activin receptor type-2A0011
Mitogen-activated protein kinase 3 0011
MAP/microtubule affinity-regulating kinase 30011
Deoxycytidine kinase0011
Mitogen-activated protein kinase 10011
Ephrin type-A receptor 20011
Ephrin type-A receptor 30011
Ephrin type-A receptor 80011
Ephrin type-B receptor 20011
Leukocyte tyrosine kinase receptor0011
Non-receptor tyrosine-protein kinase TYK20327
Wee1-like protein kinase0011
Heme oxygenase 20011
Tyrosine-protein kinase receptor UFO0011
Mitogen-activated protein kinase 40011
S-adenosylmethionine synthase isoform type-20011
DnaJ homolog subfamily A member 10011
RAC-alpha serine/threonine-protein kinase0112
RAC-beta serine/threonine-protein kinase0011
G protein-coupled receptor kinase 40011
Dual specificity protein kinase TTK0011
Tyrosine-protein kinase receptor Tie-10011
Vascular endothelial growth factor receptor 30011
Vascular endothelial growth factor receptor 20011
Dual specificity mitogen-activated protein kinase kinase 20011
Receptor-type tyrosine-protein kinase FLT30011
Bone morphogenetic protein receptor type-1A0011
Activin receptor type-1B0011
TGF-beta receptor type-10011
Serine/threonine-protein kinase receptor R30011
TGF-beta receptor type-20011
Tyrosine-protein kinase CSK0112
Glycine--tRNA ligase0011
Protein kinase C iota type0011
Exosome RNA helicase MTR40011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform0112
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform0011
Megakaryocyte-associated tyrosine-protein kinase0011
Tyrosine-protein kinase Tec0112
Tyrosine-protein kinase TXK0112
Tyrosine-protein kinase ABL20011
Tyrosine-protein kinase FRK0011
Tyrosine-protein kinase ZAP-700011
Tyrosine-protein kinase SYK0011
26S proteasome regulatory subunit 6B0011
Mitogen-activated protein kinase 80112
Mitogen-activated protein kinase 90011
Dual specificity mitogen-activated protein kinase kinase 40011
Dual specificity mitogen-activated protein kinase kinase 30011
Casein kinase I isoform alpha0011
Casein kinase I isoform delta0011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 0011
MAP kinase-activated protein kinase 20112
Cyclin-dependent kinase 80011
Elongation factor Tu, mitochondrial0011
Cysteine--tRNA ligase, cytoplasmic0011
Casein kinase I isoform epsilon0011
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial0011
Dual specificity protein kinase CLK10011
Dual specificity protein kinase CLK20011
Dual specificity protein kinase CLK30011
Glycogen synthase kinase-3 alpha0011
Glycogen synthase kinase-3 beta0112
Cyclin-dependent kinase 70011
Cyclin-dependent kinase 90011
Tyrosine-protein kinase Blk0112
Interleukin-1 receptor-associated kinase 10011
Ribosomal protein S6 kinase alpha-30112
Cytoplasmic tyrosine-protein kinase BMX0112
cAMP-dependent protein kinase catalytic subunit PRKX0011
Serine/threonine-protein kinase Nek20011
Serine/threonine-protein kinase Nek30011
Serine/threonine-protein kinase Nek40011
Tyrosine-protein kinase JAK30328
Dual specificity mitogen-activated protein kinase kinase 60011
Serine/threonine-protein kinase PLK10011
Death-associated protein kinase 10011
LIM domain kinase 10011
LIM domain kinase 20011
Mitogen-activated protein kinase 120112
Mitogen-activated protein kinase 100011
Tyrosine--tRNA ligase, cytoplasmic0011
Ephrin type-B receptor 30011
Ephrin type-A receptor 50011
Ephrin type-B receptor 40011
Ephrin type-B receptor 10011
Ephrin type-A receptor 40011
Adenylate kinase 2, mitochondrial0011
Adenosine kinase0011
Hormonally up-regulated neu tumor-associated kinase0011
Serine/threonine-protein kinase SIK10011
Receptor-interacting serine/threonine-protein kinase 40011
Ras-related protein Rab-100011
Cell division control protein 2 homolog0011
Actin-related protein 30011
Calcium-dependent protein kinase 10011
GTP-binding nuclear protein Ran0011
Tubulin alpha-1A chain0011
Casein kinase II subunit alpha0011
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta0011
SRSF protein kinase 20011
Casein kinase I isoform gamma-20011
Mitogen-activated protein kinase kinase kinase 90011
Serine/threonine-protein kinase PknB0011
Cyclin-dependent kinase 30011
Cyclin-dependent kinase-like 10011
Cyclin-dependent kinase 60011
Cyclin-dependent-like kinase 5 0112
Cyclin-dependent kinase 160011
Cyclin-dependent kinase 170011
Glutamate receptor ionotropic, NMDA 2B0101
ATP-dependent 6-phosphofructokinase, platelet type0011
Protein kinase C epsilon type0011
Dual specificity mitogen-activated protein kinase kinase 10011
Angiopoietin-1 receptor0011
Mitogen-activated protein kinase kinase kinase 100011
DNA topoisomerase 2-beta0011
Protein kinase C theta type0011
Activin receptor type-10011
Macrophage-stimulating protein receptor0011
Focal adhesion kinase 10011
Protein kinase C delta type0011
Tyrosine-protein kinase BTK0112
Tyrosine-protein kinase receptor TYRO30011
Cyclin-dependent kinase 180011
Activated CDC42 kinase 10011
Epithelial discoidin domain-containing receptor 10011
Tyrosine-protein kinase ITK/TSK0112
Myotonin-protein kinase0011
Mitogen-activated protein kinase kinase kinase kinase 20011
Mitogen-activated protein kinase kinase kinase 120011
Tyrosine-protein kinase Mer0011
Serine/threonine-protein kinase 40011
Dual specificity mitogen-activated protein kinase kinase 50011
Mitogen-activated protein kinase 70011
Serine/threonine-protein kinase PAK 20011
Serine/threonine-protein kinase 30011
Mitogen-activated protein kinase kinase kinase 10011
cGMP-dependent protein kinase 20011
Integrin-linked protein kinase0011
Rho-associated protein kinase 10011
Non-receptor tyrosine-protein kinase TNK10011
Serine/threonine-protein kinase PRP4 homolog0011
Serine/threonine-protein kinase ATR0011
Receptor-interacting serine/threonine-protein kinase 10011
Calcium/calmodulin-dependent protein kinase type II subunit beta0011
Calcium/calmodulin-dependent protein kinase type II subunit gamma0011
Calcium/calmodulin-dependent protein kinase type II subunit delta0011
Dual specificity tyrosine-phosphorylation-regulated kinase 1A0011
Activin receptor type-2B0011
Bone morphogenetic protein receptor type-20011
Protein-tyrosine kinase 60011
cGMP-dependent protein kinase 1 0011
Cyclin-dependent kinase 130011
Calcium/calmodulin-dependent protein kinase type 10011
Inhibitor of nuclear factor kappa-B kinase subunit epsilon0011
Protein-tyrosine kinase 2-beta0011
Maternal embryonic leucine zipper kinase0011
Chromodomain-helicase-DNA-binding protein 40011
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial0101
Serine/threonine-protein kinase D10011
Serine/threonine-protein kinase 380011
Receptor tyrosine-protein kinase erbB-40112
Ribosomal protein S6 kinase alpha-20011
Ephrin type-A receptor 70011
Ribosomal protein S6 kinase alpha-10011
Dual specificity testis-specific protein kinase 10011
Myosin light chain kinase, smooth muscle0011
Mitogen-activated protein kinase 110112
Serine/threonine-protein kinase STK110011
Rhodopsin kinase GRK10011
NT-3 growth factor receptor0011
Serine/threonine-protein kinase N10011
Serine/threonine-protein kinase N20011
Mitogen-activated protein kinase 140112
Calcium/calmodulin-dependent protein kinase type IV0011
Mitogen-activated protein kinase kinase kinase 110011
BDNF/NT-3 growth factors receptor0011
Mitogen-activated protein kinase 60011
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform0011
Discoidin domain-containing receptor 20011
AP2-associated protein kinase 10011
Myosin light chain kinase 30011
Uncharacterized aarF domain-containing protein kinase 50011
Serine/threonine-protein kinase SBK10011
Mitogen-activated protein kinase kinase kinase 190011
Putative heat shock protein HSP 90-beta 20011
Serine/threonine-protein kinase TNNI3K0011
Rab-like protein 30011
Leucine-rich repeat serine/threonine-protein kinase 20011
Sigma intracellular receptor 20101
Serine/threonine-protein kinase MRCK alpha0011
Tyrosine-protein kinase JAK30101
Tyrosine-protein kinase JAK20101
Tyrosine-protein kinase JAK30101
Serine/threonine-protein kinase MRCK gamma0011
Acyl-CoA dehydrogenase family member 100011
Serine/threonine-protein kinase Nek50011
Serine/threonine-protein kinase ULK30011
Dual serine/threonine and tyrosine protein kinase0011
Mitogen-activated protein kinase kinase kinase 150011
Uncharacterized protein FLJ452520011
Serine/threonine-protein kinase/endoribonuclease IRE20011
Serine/threonine-protein kinase MARK20011
ATP-dependent RNA helicase DHX300011
Serine/threonine-protein kinase TAO10011
STE20-related kinase adapter protein alpha0011
Myosin-140011
AarF domain-containing protein kinase 10011
Serine/threonine-protein kinase tousled-like 20011
Serine/threonine-protein kinase 32C0011
Serine/threonine-protein kinase pim-30011
Serine/threonine-protein kinase VRK20011
Myosin light chain kinase family member 40011
Homeodomain-interacting protein kinase 10011
Calcium/calmodulin-dependent protein kinase type 1D0011
Mitogen-activated protein kinase kinase kinase kinase 30011
Cyclin-dependent kinase-like 30011
MAP kinase-activated protein kinase 50112
Serine/threonine-protein kinase BRSK20011
Serine/threonine-protein kinase NIM10011
Serine/threonine-protein kinase ULK20011
Misshapen-like kinase 10011
Serine/threonine-protein kinase DCLK20011
Calcium/calmodulin-dependent protein kinase kinase 10011
Casein kinase I isoform alpha-like0011
Homeodomain-interacting protein kinase 40011
Myosin-IIIa0011
Ankyrin repeat and protein kinase domain-containing protein 10011
Serine/threonine-protein kinase Nek110011
Atypical kinase COQ8A, mitochondrial0011
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma0011
Mitogen-activated protein kinase 150011
Serine/threonine-protein kinase Nek90011
Serine/threonine-protein kinase BRSK10011
Serine/threonine-protein kinase 350011
Serine/threonine-protein kinase Nek70011
Rhodopsin kinase GRK70011
Serine/threonine-protein kinase 32A0011
Myosin-IIIb0011
ATP-dependent RNA helicase DDX10011
Dual specificity tyrosine-phosphorylation-regulated kinase 20011
Cyclin-dependent kinase-like 20011
Mitogen-activated protein kinase kinase kinase kinase 10011
Serine/threonine-protein kinase Sgk30011
Atypical kinase COQ8B, mitochondrial0011
Aurora kinase B0011
MAP/microtubule affinity-regulating kinase 40011
Calcium/calmodulin-dependent protein kinase type 1G0011
Serine/threonine-protein kinase Nek10011
Cyclin-dependent kinase 150011
PAS domain-containing serine/threonine-protein kinase0011
Calcium/calmodulin-dependent protein kinase kinase 20011
EKC/KEOPS complex subunit TP53RK0011
Dual specificity testis-specific protein kinase 20011
SRSF protein kinase 10011
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase0011
Mitogen-activated protein kinase kinase kinase 50011
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha0011
Mitogen-activated protein kinase kinase kinase 30011
Eukaryotic translation initiation factor 2-alpha kinase 10011
Serine/threonine-protein kinase RIO10011
MAP kinase-interacting serine/threonine-protein kinase 10011
Serine/threonine-protein kinase RIO20011
Cyclin-dependent kinase 190011
Transient receptor potential cation channel subfamily M member 60011
Testis-specific serine/threonine-protein kinase 10011
Serine/threonine-protein kinase 330011
Nucleolar GTP-binding protein 10011
Serine/threonine-protein kinase D20011
Serine/threonine-protein kinase DCLK30011
NUAK family SNF1-like kinase 20011
RNA cytidine acetyltransferase0011
Serine/threonine-protein kinase SIK20011
Myosin light chain kinase 2, skeletal/cardiac muscle0011
STE20-like serine/threonine-protein kinase 0011
Serine/threonine-protein kinase TAO30011
Homeodomain-interacting protein kinase 20011
Tyrosine-protein kinase Srms0011
Homeodomain-interacting protein kinase 30011
Serine/threonine-protein kinase PLK30011
dCTP pyrophosphatase 10011
Dual specificity protein kinase CLK40011
MAP kinase-interacting serine/threonine-protein kinase 20011
Serine/threonine-protein kinase Nek60011
Casein kinase I isoform gamma-10011
Serine/threonine-protein kinase PAK 60011
SNF-related serine/threonine-protein kinase0011
Serine/threonine-protein kinase LATS20011
Serine/threonine-protein kinase 360011
Phenylalanine--tRNA ligase beta subunit0011
BMP-2-inducible protein kinase0011
Midasin0011
Interleukin-1 receptor-associated kinase 40011
Serine/threonine-protein kinase 32B0011
Mitogen-activated protein kinase kinase kinase 200011
Cyclin-dependent kinase 120011
Serine/threonine-protein kinase PLK20011
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 130011
Serine/threonine-protein kinase MARK10011
Serine/threonine-protein kinase pim-20011
Serine/threonine-protein kinase PAK 50011
Serine/threonine-protein kinase 260011
eIF-2-alpha kinase GCN20011
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial0011
Serine/threonine-protein kinase NLK0011
Phosphatidylinositol 4-kinase beta0011
Serine/threonine-protein kinase 17A0011
STE20/SPS1-related proline-alanine-rich protein kinase0011
Ephrin type-A receptor 60011
Serine/threonine-protein kinase TBK10112
Septin-90011
Death-associated protein kinase 20011
Ribosomal protein S6 kinase alpha-60011
TRAF2 and NCK-interacting protein kinase0011
Serine/threonine-protein kinase tousled-like 10011
Serine/threonine-protein kinase TAO20011
Long-chain-fatty-acid--CoA ligase 50011
ALK tyrosine kinase receptor0011
SRSF protein kinase 30011
Serine/threonine-protein kinase ICK0011
Cyclin-dependent kinase 11A0011
Aurora kinase C0011
Calcium/calmodulin-dependent protein kinase type II subunit alpha0011
RAC-gamma serine/threonine-protein kinase0011
Serine/threonine-protein kinase 38-like0011
Microtubule-associated serine/threonine-protein kinase 10011
Serine/threonine-protein kinase SIK30011
Mitogen-activated protein kinase kinase kinase 20011
Thyroid hormone receptor-associated protein 30011
Dual specificity tyrosine-phosphorylation-regulated kinase 1B0011
Mitogen-activated protein kinase kinase kinase kinase 50011
Receptor-interacting serine/threonine-protein kinase 30011
Serine/threonine-protein kinase MRCK beta0011
Interleukin-1 receptor-associated kinase 30011
Serine/threonine-protein kinase 240011
Casein kinase I isoform gamma-30011
Mitogen-activated protein kinase kinase kinase 40011
Ubiquitin carboxyl-terminal hydrolase 20101
Vitamin D3 receptor0112
Ileal sodium/bile acid cotransporter0101
Sodium/bile acid cotransporter0101
G-protein coupled bile acid receptor 10011
Bile acid receptor0011
CDGSH iron-sulfur domain-containing protein 10202
M1-family alanyl aminopeptidase0101
Albumin0011
Proprotein convertase subtilisin/kexin type 70101
Vitamin K epoxide reductase complex subunit 1-like protein 10101
Vitamin K epoxide reductase complex subunit 10101
Protease 0101
Vitamin K epoxide reductase complex subunit 1-like protein 10101
Vitamin K epoxide reductase complex subunit 1 0202
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023]