| Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
|---|
| Chain B, pheromone binding protein | 0 | 0 | 1 | 1 |
| Chain A, pheromone binding protein | 0 | 0 | 1 | 1 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | 1 | 0 | 0 | 1 |
| Chain A, RNA-directed RNA polymerase NS5 | 0 | 1 | 0 | 1 |
| acid sphingomyelinase | 1 | 0 | 0 | 1 |
| thioredoxin reductase | 2 | 0 | 0 | 2 |
| USP1 protein, partial | 8 | 0 | 0 | 8 |
| TDP1 protein | 5 | 0 | 0 | 5 |
| vitamin D3 receptor isoform VDRA | 5 | 0 | 0 | 5 |
| importin subunit beta-1 isoform 1 | 1 | 0 | 0 | 1 |
| flap endonuclease 1 | 1 | 0 | 0 | 1 |
| serine/threonine-protein kinase PLK1 | 2 | 0 | 0 | 2 |
| snurportin-1 | 1 | 0 | 0 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | 2 | 0 | 0 | 2 |
| GTP-binding nuclear protein Ran isoform 1 | 1 | 0 | 0 | 1 |
| DNA polymerase eta isoform 1 | 2 | 0 | 0 | 2 |
| DNA polymerase iota isoform a (long) | 1 | 0 | 0 | 1 |
| urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
| plasminogen precursor | 1 | 0 | 0 | 1 |
| urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
| geminin | 4 | 0 | 0 | 4 |
| DNA polymerase kappa isoform 1 | 7 | 0 | 0 | 7 |
| fibroblast growth factor 22 isoform 1 precursor | 0 | 0 | 0 | 1 |
| Mitogen-activated protein kinase 13 | 0 | 1 | 0 | 1 |
| Beta-lactamase | 0 | 1 | 0 | 1 |
| Transthyretin | 0 | 1 | 1 | 4 |
| Fatty acid-binding protein, intestinal | 0 | 2 | 1 | 3 |
| Fatty acid-binding protein, adipocyte | 0 | 6 | 3 | 9 |
| Cyclin-A2 | 0 | 1 | 0 | 1 |
| Cannabinoid receptor 1 | 0 | 1 | 2 | 3 |
| Cyclin-dependent kinase 2 | 0 | 1 | 1 | 2 |
| Choline O-acetyltransferase | 0 | 1 | 0 | 1 |
| Mitogen-activated protein kinase 12 | 0 | 1 | 0 | 1 |
| Guanine nucleotide-binding protein G | 1 | 0 | 0 | 1 |
| Fatty acid-binding protein 5 | 0 | 4 | 2 | 6 |
| Fatty acid-binding protein 5 | 0 | 0 | 3 | 3 |
| Mitogen-activated protein kinase 11 | 0 | 1 | 0 | 1 |
| Mitogen-activated protein kinase 14 | 0 | 1 | 0 | 1 |
| Chain A, Ferritin light chain | 1 | 0 | 0 | 1 |
| phosphopantetheinyl transferase | 4 | 0 | 0 | 4 |
| aldehyde dehydrogenase 1 family, member A1 | 5 | 0 | 0 | 5 |
| Bloom syndrome protein isoform 1 | 2 | 0 | 0 | 2 |
| Fatty-acid amide hydrolase 1 | 0 | 3 | 0 | 3 |
| Fatty-acid amide hydrolase 1 | 0 | 0 | 0 | 1 |
| Potassium channel subfamily K member 3 | 0 | 1 | 0 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | 2 | 0 | 0 | 2 |
| Fatty acid-binding protein, liver | 0 | 1 | 0 | 1 |
| Glutamate receptor 1 | 0 | 0 | 1 | 1 |
| Glutamate receptor 2 | 1 | 0 | 1 | 2 |
| Glutamate receptor 3 | 0 | 0 | 1 | 1 |
| Glutamate receptor 4 | 0 | 0 | 1 | 1 |
| Cannabinoid receptor 1 | 0 | 1 | 0 | 2 |
| Cannabinoid receptor 2 | 0 | 1 | 0 | 2 |
| Alpha-1A adrenergic receptor | 0 | 1 | 0 | 1 |
| Cannabinoid receptor 1 | 0 | 1 | 0 | 1 |
| Histamine H2 receptor | 2 | 0 | 0 | 2 |
| Cannabinoid receptor 2 | 0 | 1 | 0 | 1 |
| Fatty-acid amide hydrolase 1 | 0 | 2 | 0 | 3 |
| Corticotropin-releasing factor receptor 2 | 0 | 1 | 0 | 1 |
| Lanosterol 14-alpha demethylase | 0 | 2 | 0 | 2 |
| Potassium channel subfamily K member 2 | 0 | 1 | 0 | 1 |
| Transient receptor potential cation channel subfamily V member 1 | 0 | 0 | 1 | 2 |
| Cannabinoid receptor 2 | 0 | 1 | 0 | 1 |
| Transient receptor potential cation channel subfamily V member 2 | 0 | 3 | 0 | 3 |
| Chain A, ADIPOCYTE LIPID-BINDING PROTEIN | 0 | 0 | 1 | 1 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 1 | 0 | 0 | 1 |
| Chain A, SERUM ALBUMIN | 0 | 0 | 1 | 1 |
| Chain A, SERUM ALBUMIN | 0 | 0 | 1 | 1 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | 3 | 0 | 0 | 3 |
| Chain A, Beta-lactamase | 1 | 0 | 0 | 1 |
| Chain A, HADH2 protein | 3 | 0 | 0 | 3 |
| Chain B, HADH2 protein | 3 | 0 | 0 | 3 |
| Chain A, 2-oxoglutarate Oxygenase | 2 | 0 | 0 | 2 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | 1 | 0 | 0 | 1 |
| Chain A, Cruzipain | 2 | 0 | 0 | 2 |
| 15-lipoxygenase, partial | 2 | 0 | 0 | 2 |
| Microtubule-associated protein tau | 2 | 0 | 0 | 2 |
| thioredoxin glutathione reductase | 1 | 0 | 0 | 1 |
| euchromatic histone-lysine N-methyltransferase 2 | 3 | 0 | 0 | 3 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | 1 | 0 | 0 | 1 |
| cellular tumor antigen p53 isoform a | 1 | 0 | 0 | 1 |
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | 2 | 0 | 0 | 2 |
| ubiquitin carboxyl-terminal hydrolase 2 isoform a | 1 | 0 | 0 | 1 |
| nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | 1 | 0 | 0 | 1 |
| cytochrome P450 3A4 isoform 1 | 2 | 0 | 0 | 2 |
| histone acetyltransferase KAT2A isoform 1 | 2 | 0 | 0 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | 1 | 0 | 0 | 1 |
| caspase-1 isoform alpha precursor | 2 | 0 | 0 | 2 |
| lamin isoform A-delta10 | 5 | 0 | 0 | 5 |
| Gamma-aminobutyric acid receptor subunit pi | 2 | 0 | 1 | 3 |
| Prostaglandin G/H synthase 1 | 0 | 3 | 0 | 4 |
| Trypsin | 0 | 3 | 0 | 3 |
| Coagulation factor VII | 0 | 3 | 0 | 3 |
| 60 kDa chaperonin | 0 | 1 | 0 | 1 |
| 60 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
| Aromatase | 0 | 3 | 0 | 3 |
| Tissue factor | 0 | 3 | 0 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | 2 | 0 | 1 | 3 |
| Prostaglandin G/H synthase 2 | 0 | 0 | 1 | 2 |
| Nuclear receptor subfamily 4 group A member 2 | 0 | 0 | 2 | 2 |
| 10 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
| Calmodulin | 0 | 0 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | 2 | 0 | 1 | 3 |
| Disintegrin and metalloproteinase domain-containing protein 17 | 1 | 0 | 0 | 1 |
| Prostaglandin G/H synthase 2 | 0 | 3 | 0 | 4 |
| Solute carrier organic anion transporter family member 2A1 | 0 | 0 | 0 | 1 |
| Thiosulfate sulfurtransferase | 0 | 1 | 0 | 1 |
| 60 kDa chaperonin | 0 | 1 | 0 | 1 |
| 10 kDa chaperonin | 0 | 1 | 0 | 1 |
| GABA theta subunit | 2 | 0 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | 2 | 0 | 1 | 3 |
| Solute carrier organic anion transporter family member 1B3 | 0 | 4 | 0 | 6 |
| Cytosolic phospholipase A2 gamma | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 1B1 | 0 | 4 | 0 | 7 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | 1 | 0 | 0 | 1 |
| Caspase-7 | 1 | 0 | 0 | 1 |
| Inositol monophosphatase 1 | 1 | 0 | 0 | 1 |
| Solute carrier organic anion transporter family member 1A4 | 0 | 1 | 0 | 4 |
| Multidrug resistance-associated protein 6 | 0 | 0 | 0 | 1 |
| Solute carrier organic anion transporter family member 1A5 | 0 | 0 | 0 | 3 |
| Endothelin receptor type B | 0 | 1 | 0 | 1 |
| Endothelin-1 receptor | 0 | 2 | 0 | 3 |
| Endothelin-1 receptor | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 1A1 | 0 | 0 | 0 | 1 |
| Endothelin-1 receptor | 0 | 1 | 0 | 1 |
| Canalicular multispecific organic anion transporter 1 | 0 | 1 | 0 | 2 |
| Solute carrier organic anion transporter family member 1B2 | 0 | 0 | 0 | 1 |
| Chain A, Protein (peroxisome Proliferator Activated Receptor (ppar-delta)) | 0 | 1 | 0 | 1 |
| GLS protein | 1 | 0 | 0 | 1 |
| AR protein | 4 | 0 | 0 | 4 |
| regulator of G-protein signaling 4 | 1 | 0 | 0 | 1 |
| peroxisome proliferator activated receptor gamma | 5 | 0 | 0 | 5 |
| thyroid hormone receptor beta isoform 2 | 5 | 0 | 0 | 5 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | 1 | 0 | 0 | 1 |
| Cytochrome P450 1A2 | 0 | 1 | 0 | 1 |
| Retinoic acid receptor RXR-alpha | 0 | 1 | 2 | 3 |
| Peroxisome proliferator-activated receptor gamma | 0 | 0 | 5 | 5 |
| Oxoeicosanoid receptor 1 | 0 | 1 | 0 | 1 |
| Sodium/glucose cotransporter 1 | 0 | 0 | 1 | 1 |
| Sodium/glucose cotransporter 2 | 0 | 1 | 1 | 2 |
| Glucagon-like peptide 1 receptor | 0 | 0 | 1 | 1 |
| Glucagon-like peptide 1 receptor | 0 | 1 | 1 | 2 |
| Glucagon receptor | 0 | 0 | 1 | 1 |
| Glucagon receptor | 0 | 0 | 1 | 1 |
| Glycogen phosphorylase, muscle form | 0 | 1 | 0 | 1 |
| Asialoglycoprotein receptor 1 | 0 | 1 | 1 | 2 |
| N(G),N(G)-dimethylarginine dimethylaminohydrolase 1 | 0 | 1 | 0 | 1 |
| Luciferase | 2 | 0 | 0 | 2 |
| acetylcholinesterase | 3 | 0 | 0 | 3 |
| hypoxia-inducible factor 1 alpha subunit | 2 | 0 | 0 | 2 |
| RAR-related orphan receptor gamma | 4 | 0 | 0 | 4 |
| progesterone receptor | 3 | 0 | 0 | 3 |
| retinoic acid nuclear receptor alpha variant 1 | 3 | 0 | 0 | 3 |
| retinoid X nuclear receptor alpha | 2 | 0 | 0 | 2 |
| estrogen-related nuclear receptor alpha | 5 | 0 | 0 | 5 |
| pregnane X nuclear receptor | 4 | 0 | 0 | 4 |
| estrogen nuclear receptor alpha | 5 | 0 | 0 | 5 |
| aryl hydrocarbon receptor | 3 | 0 | 0 | 3 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 4 | 0 | 0 | 4 |
| activating transcription factor 6 | 2 | 0 | 0 | 2 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | 3 | 0 | 0 | 3 |
| histone deacetylase 9 isoform 3 | 1 | 0 | 0 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | 5 | 0 | 0 | 5 |
| Voltage-dependent calcium channel gamma-2 subunit | 1 | 0 | 0 | 1 |
| SMAD family member 2 | 1 | 0 | 0 | 1 |
| SMAD family member 3 | 1 | 0 | 0 | 1 |
| GLI family zinc finger 3 | 2 | 0 | 0 | 2 |
| caspase 7, apoptosis-related cysteine protease | 1 | 0 | 0 | 1 |
| thyroid stimulating hormone receptor | 1 | 0 | 0 | 1 |
| estrogen receptor 2 (ER beta) | 1 | 0 | 0 | 1 |
| glucocorticoid receptor [Homo sapiens] | 3 | 0 | 0 | 3 |
| farnesoid X nuclear receptor | 3 | 0 | 0 | 3 |
| peroxisome proliferator-activated receptor delta | 3 | 0 | 0 | 3 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | 1 | 0 | 0 | 1 |
| caspase-3 | 1 | 0 | 0 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | 2 | 0 | 0 | 2 |
| heat shock protein beta-1 | 1 | 0 | 0 | 1 |
| Free fatty acid receptor 1 | 0 | 0 | 1 | 1 |
| Sterol O-acyltransferase 1 | 0 | 1 | 0 | 1 |
| Cellular tumor antigen p53 | 4 | 0 | 0 | 4 |
| Fatty acid-binding protein, heart | 0 | 2 | 0 | 2 |
| Seed linoleate 13S-lipoxygenase-1 | 0 | 1 | 0 | 1 |
| Prostaglandin G/H synthase 1 | 0 | 1 | 0 | 1 |
| Adenosine receptor A1 | 0 | 1 | 0 | 1 |
| Tyrosine-protein phosphatase non-receptor type 7 | 0 | 1 | 0 | 1 |
| Sterol O-acyltransferase 1 | 0 | 1 | 0 | 1 |
| Aldo-keto reductase family 1 member C3 | 0 | 1 | 0 | 1 |
| Dual specificity protein phosphatase 3 | 0 | 1 | 0 | 1 |
| Peroxisome proliferator-activated receptor alpha | 2 | 0 | 1 | 3 |
| Free fatty acid receptor 4 | 0 | 0 | 1 | 1 |
| Neurotensin receptor type 1 | 0 | 0 | 1 | 1 |
| Neurotensin receptor type 2 | 0 | 1 | 1 | 3 |
| Myelin basic protein | 0 | 0 | 1 | 1 |
| Neurotensin receptor type 1 | 0 | 1 | 1 | 2 |
| Neurotensin receptor type 1 | 0 | 2 | 2 | 5 |
| Neurotensin receptor type 2 | 0 | 2 | 1 | 3 |
| Sortilin | 0 | 1 | 0 | 1 |
| Chain A, Fatty acid-binding protein, adipocyte | 0 | 1 | 0 | 1 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | 3 | 0 | 0 | 3 |
| nuclear receptor subfamily 1, group I, member 2 | 1 | 0 | 0 | 1 |
| peripheral myelin protein 22 | 2 | 0 | 0 | 2 |
| Acetylcholinesterase | 0 | 1 | 0 | 1 |
| Toll-like receptor 2 | 0 | 1 | 0 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | 0 | 1 | 0 | 1 |
| Olfactory receptor 51E2 | 0 | 0 | 1 | 1 |
| Chain X, Thyroid hormone receptor beta-1 | 0 | 0 | 2 | 2 |
| Chain X, Thyroid hormone receptor beta-1 | 0 | 0 | 2 | 2 |
| apical membrane antigen 1, AMA1 | 2 | 0 | 0 | 2 |
| nuclear receptor subfamily 1, group I, member 3 | 1 | 0 | 0 | 1 |
| EWS/FLI fusion protein | 1 | 0 | 0 | 1 |
| G | 1 | 0 | 0 | 1 |
| thyroid hormone receptor beta isoform a | 2 | 0 | 0 | 2 |
| Nuclear receptor subfamily 1 group I member 2 | 0 | 0 | 1 | 1 |
| Rap guanine nucleotide exchange factor 3 | 1 | 0 | 0 | 1 |
| Interferon beta | 1 | 0 | 0 | 1 |
| HLA class I histocompatibility antigen, B alpha chain | 1 | 0 | 0 | 1 |
| Thyroid hormone receptor alpha | 0 | 2 | 3 | 5 |
| Thyroid hormone receptor beta | 0 | 2 | 3 | 5 |
| Proliferating cell nuclear antigen | 0 | 2 | 0 | 2 |
| UDP-glucuronosyltransferase 1A1 | 0 | 1 | 0 | 1 |
| Malate dehydrogenase, mitochondrial | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 1A2 | 0 | 0 | 0 | 2 |
| Solute carrier organic anion transporter family member 1A3 | 0 | 0 | 0 | 2 |
| Solute carrier organic anion transporter family member 4C1 | 0 | 1 | 0 | 2 |
| Monocarboxylate transporter 8 | 0 | 0 | 0 | 1 |
| Inositol hexakisphosphate kinase 1 | 1 | 0 | 0 | 1 |
| Bile acid receptor | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 1C1 | 0 | 0 | 0 | 1 |
| cytochrome P450 2C9, partial | 1 | 0 | 0 | 1 |
| glp-1 receptor, partial | 1 | 0 | 0 | 1 |
| glucocerebrosidase | 1 | 0 | 0 | 1 |
| chromobox protein homolog 1 | 1 | 0 | 0 | 1 |
| muscleblind-like protein 1 isoform 1 | 1 | 0 | 0 | 1 |
| neuropeptide S receptor isoform A | 1 | 0 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit pi | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit delta | 0 | 1 | 0 | 1 |
| Bile salt export pump | 0 | 1 | 0 | 1 |
| Prothrombin | 0 | 0 | 1 | 1 |
| Androgen receptor | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | 0 | 1 | 0 | 1 |
| Thyroid hormone receptor beta | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-1 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-3 | 0 | 1 | 0 | 1 |
| Adenosine receptor A1 | 0 | 2 | 0 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit epsilon | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | 0 | 1 | 0 | 1 |
| Sigma non-opioid intracellular receptor 1 | 0 | 0 | 1 | 1 |
| Solute carrier organic anion transporter family member 4C1 | 0 | 0 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 4A1 | 0 | 0 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | 0 | 1 | 0 | 1 |
| Solute carrier organic anion transporter family member 1C1 | 0 | 1 | 0 | 1 |
| Gamma-aminobutyric acid receptor subunit theta | 0 | 1 | 0 | 1 |
| Chain A, Glycogen phosphorylase, liver form | 0 | 0 | 1 | 1 |
| Chain A, glycogen phosphorylase, liver form | 0 | 0 | 1 | 1 |
| Chain A, Glycogen phosphorylase, liver form | 0 | 0 | 1 | 1 |
| Chain A, Glycogen phosphorylase, liver form | 0 | 0 | 1 | 1 |
| Solute carrier family 22 member 6 | 0 | 0 | 0 | 1 |
| Solute carrier family 22 member 8 | 0 | 1 | 0 | 1 |
| Solute carrier family 2, facilitated glucose transporter member 9 | 0 | 1 | 1 | 2 |
| Guanine deaminase | 0 | 1 | 0 | 1 |
| [prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |