Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
acetylcholinesterase | 2 | 0 | 0 | 2 |
pregnane X receptor | 2 | 0 | 0 | 2 |
SMAD family member 2 | 2 | 0 | 0 | 2 |
SMAD family member 3 | 2 | 0 | 0 | 2 |
TDP1 protein | 5 | 0 | 0 | 5 |
GLI family zinc finger 3 | 6 | 0 | 0 | 6 |
Microtubule-associated protein tau | 2 | 0 | 0 | 2 |
AR protein | 7 | 0 | 0 | 7 |
progesterone receptor | 7 | 0 | 0 | 7 |
glucocorticoid receptor [Homo sapiens] | 7 | 0 | 0 | 7 |
retinoic acid nuclear receptor alpha variant 1 | 6 | 0 | 0 | 6 |
retinoid X nuclear receptor alpha | 5 | 0 | 0 | 5 |
estrogen-related nuclear receptor alpha | 4 | 0 | 0 | 4 |
farnesoid X nuclear receptor | 2 | 0 | 0 | 2 |
pregnane X nuclear receptor | 4 | 0 | 0 | 4 |
estrogen nuclear receptor alpha | 7 | 0 | 0 | 7 |
G | 2 | 0 | 0 | 2 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | 5 | 0 | 0 | 5 |
arylsulfatase A | 2 | 0 | 0 | 2 |
euchromatic histone-lysine N-methyltransferase 2 | 2 | 0 | 0 | 2 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 4 | 0 | 0 | 4 |
activating transcription factor 6 | 3 | 0 | 0 | 3 |
nuclear receptor subfamily 1, group I, member 2 | 2 | 0 | 0 | 2 |
chromobox protein homolog 1 | 4 | 0 | 0 | 4 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 4 | 0 | 0 | 4 |
geminin | 4 | 0 | 0 | 4 |
survival motor neuron protein isoform d | 3 | 0 | 0 | 3 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
lamin isoform A-delta10 | 2 | 0 | 0 | 2 |
Voltage-dependent calcium channel gamma-2 subunit | 4 | 0 | 0 | 4 |
Interferon beta | 3 | 0 | 0 | 3 |
HLA class I histocompatibility antigen, B alpha chain | 2 | 0 | 0 | 2 |
Glucocorticoid receptor | 0 | 7 | 0 | 8 |
Sex hormone-binding globulin | 0 | 1 | 5 | 6 |
Glycine receptor subunit alpha-1 | 0 | 6 | 0 | 6 |
Corticosteroid-binding globulin | 0 | 5 | 0 | 5 |
Adenosine receptor A3 | 0 | 2 | 0 | 2 |
Replicase polyprotein 1ab | 0 | 1 | 0 | 1 |
Androgen receptor | 0 | 7 | 1 | 8 |
Alpha-1B adrenergic receptor | 0 | 2 | 0 | 2 |
Glutamate receptor 2 | 4 | 0 | 0 | 4 |
Glycine receptor subunit beta | 0 | 6 | 0 | 6 |
Glycine receptor subunit alpha-2 | 0 | 6 | 0 | 6 |
Glycine receptor subunit alpha-3 | 0 | 6 | 0 | 6 |
Mitogen-activated protein kinase 3 | 0 | 1 | 0 | 1 |
Alpha-1A adrenergic receptor | 0 | 2 | 0 | 2 |
Sodium-dependent dopamine transporter | 0 | 2 | 0 | 2 |
TAR DNA-binding protein 43 | 3 | 0 | 0 | 3 |
Inositol hexakisphosphate kinase 1 | 2 | 0 | 0 | 2 |
cytochrome P450 2C9, partial | 2 | 0 | 0 | 2 |
ATP-dependent phosphofructokinase | 1 | 0 | 0 | 1 |
Chain A, Ferritin light chain | 1 | 0 | 0 | 1 |
hypoxia-inducible factor 1 alpha subunit | 1 | 0 | 0 | 1 |
RAR-related orphan receptor gamma | 4 | 0 | 0 | 4 |
USP1 protein, partial | 1 | 0 | 0 | 1 |
caspase 7, apoptosis-related cysteine protease | 1 | 0 | 0 | 1 |
estrogen receptor 2 (ER beta) | 4 | 0 | 0 | 4 |
nuclear receptor subfamily 1, group I, member 3 | 2 | 0 | 0 | 2 |
67.9K protein | 1 | 0 | 0 | 1 |
peroxisome proliferator-activated receptor delta | 3 | 0 | 0 | 3 |
peroxisome proliferator activated receptor gamma | 3 | 0 | 0 | 3 |
caspase-3 | 1 | 0 | 0 | 1 |
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | 1 | 0 | 0 | 1 |
thyrotropin-releasing hormone receptor | 2 | 0 | 0 | 2 |
v-jun sarcoma virus 17 oncogene homolog (avian) | 3 | 0 | 0 | 3 |
vitamin D3 receptor isoform VDRA | 2 | 0 | 0 | 2 |
thyroid hormone receptor beta isoform 2 | 3 | 0 | 0 | 3 |
heat shock protein beta-1 | 2 | 0 | 0 | 2 |
mitogen-activated protein kinase 1 | 1 | 0 | 0 | 1 |
nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
Cellular tumor antigen p53 | 1 | 0 | 0 | 1 |
Caspase-2 | 0 | 0 | 1 | 1 |
Inositol monophosphatase 1 | 2 | 0 | 0 | 2 |
ATPase family AAA domain-containing protein 5 | 1 | 0 | 0 | 1 |
Ataxin-2 | 1 | 0 | 0 | 1 |
Chain A, HADH2 protein | 3 | 0 | 0 | 3 |
Chain B, HADH2 protein | 3 | 0 | 0 | 3 |
endonuclease IV | 2 | 0 | 0 | 2 |
dopamine D1 receptor | 1 | 0 | 0 | 1 |
thioredoxin reductase | 1 | 0 | 0 | 1 |
GLS protein | 1 | 0 | 0 | 1 |
aldehyde dehydrogenase 1 family, member A1 | 1 | 0 | 0 | 1 |
regulator of G-protein signaling 4 | 1 | 0 | 0 | 1 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | 3 | 0 | 0 | 3 |
peripheral myelin protein 22 isoform 1 | 2 | 0 | 0 | 2 |
atrial natriuretic peptide receptor 1 precursor | 1 | 0 | 0 | 1 |
flap endonuclease 1 | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 3 | 0 | 0 | 3 |
M-phase phosphoprotein 8 | 1 | 0 | 0 | 1 |
muscarinic acetylcholine receptor M1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 3 | 0 | 0 | 3 |
Bile salt export pump | 0 | 3 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit beta-1 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit delta | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit beta-3 | 3 | 0 | 0 | 3 |
Gamma-aminobutyric acid receptor subunit beta-2 | 3 | 0 | 0 | 3 |
Potassium voltage-gated channel subfamily A member 1 | 0 | 0 | 1 | 1 |
GABA theta subunit | 3 | 0 | 0 | 3 |
Multidrug and toxin extrusion protein 1 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit epsilon | 3 | 0 | 0 | 3 |
Chain A, Sex Hormone-Binding Globulin | 0 | 0 | 1 | 1 |
interleukin 8 | 1 | 0 | 0 | 1 |
glp-1 receptor, partial | 1 | 0 | 0 | 1 |
Histone H2A.x | 1 | 0 | 0 | 1 |
potassium voltage-gated channel subfamily H member 2 isoform d | 1 | 0 | 0 | 1 |
transcriptional regulator ERG isoform 3 | 1 | 0 | 0 | 1 |
peripheral myelin protein 22 | 1 | 0 | 0 | 1 |
Plasma kallikrein | 0 | 1 | 0 | 1 |
Progesterone receptor | 0 | 1 | 0 | 1 |
Progesterone receptor | 0 | 1 | 1 | 2 |
Glucocorticoid receptor | 0 | 1 | 0 | 1 |
Mineralocorticoid receptor | 0 | 1 | 0 | 1 |
Sex hormone-binding globulin | 0 | 1 | 0 | 1 |
Androgen receptor | 0 | 2 | 2 | 6 |
Aromatase | 0 | 2 | 0 | 3 |
Androgen receptor | 0 | 1 | 1 | 2 |
Mineralocorticoid receptor | 0 | 1 | 0 | 1 |
Testosterone 17-beta-dehydrogenase 3 | 0 | 1 | 0 | 1 |
Angiotensin-converting enzyme | 0 | 0 | 1 | 1 |
Cannabinoid receptor 2 | 0 | 1 | 0 | 1 |
Nuclear receptor ROR-gamma | 1 | 0 | 0 | 1 |
G-protein coupled bile acid receptor 1 | 0 | 0 | 1 | 1 |
Muscarinic acetylcholine receptor | 0 | 1 | 0 | 1 |
Neuropeptide FF receptor 2 | 0 | 0 | 0 | 1 |
ALK tyrosine kinase receptor | 0 | 1 | 0 | 1 |
Estrogen receptor | 0 | 4 | 1 | 6 |
Polyunsaturated fatty acid lipoxygenase ALOX15 | 0 | 2 | 0 | 2 |
UDP-glucuronosyltransferase 2B7 | 0 | 0 | 0 | 1 |
Sodium-dependent serotonin transporter | 0 | 4 | 0 | 4 |
Alpha-synuclein | 0 | 2 | 0 | 2 |
Solute carrier organic anion transporter family member 1A1 | 0 | 3 | 0 | 4 |
Lanosterol 14-alpha demethylase | 0 | 0 | 1 | 1 |
Olfactory receptor 51E2 | 0 | 0 | 1 | 1 |
UDP-glucuronosyltransferase 1A10 | 0 | 0 | 0 | 1 |
ATAD5 protein, partial | 1 | 0 | 0 | 1 |
NFKB1 protein, partial | 1 | 0 | 0 | 1 |
GALC protein | 2 | 0 | 0 | 2 |
nonstructural protein 1 | 1 | 0 | 0 | 1 |
Bloom syndrome protein isoform 1 | 1 | 0 | 0 | 1 |
hexokinase-4 isoform 1 | 1 | 0 | 0 | 1 |
parathyroid hormone/parathyroid hormone-related peptide receptor precursor | 1 | 0 | 0 | 1 |
glucokinase regulatory protein | 1 | 0 | 0 | 1 |
DNA polymerase iota isoform a (long) | 1 | 0 | 0 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
Rap guanine nucleotide exchange factor 3 | 1 | 0 | 0 | 1 |
Steryl-sulfatase | 0 | 3 | 0 | 4 |
17-beta-hydroxysteroid dehydrogenase type 1 | 0 | 2 | 0 | 3 |
Mu-type opioid receptor | 0 | 0 | 1 | 1 |
5-hydroxytryptamine receptor 2B | 0 | 2 | 0 | 2 |
Mu-type opioid receptor | 0 | 0 | 1 | 1 |
Cytochrome P450 1B1 | 0 | 1 | 0 | 1 |
Estrogen receptor beta | 0 | 1 | 1 | 3 |
Ghrelin O-acyltransferase | 0 | 1 | 0 | 1 |
Broad substrate specificity ATP-binding cassette transporter ABCG2 | 0 | 1 | 0 | 2 |
Estrogen receptor beta | 0 | 0 | 0 | 1 |
Multidrug resistance-associated protein 4 | 0 | 1 | 0 | 1 |
Solute carrier organic anion transporter family member 1A4 | 0 | 0 | 0 | 1 |
Solute carrier organic anion transporter family member 1A5 | 0 | 0 | 0 | 1 |
Solute carrier organic anion transporter family member 2B1 | 0 | 0 | 0 | 1 |
Tyrosine-protein phosphatase non-receptor type 1 | 0 | 0 | 0 | 1 |
Estrogen receptor | 0 | 0 | 0 | 1 |
Sodium/bile acid cotransporter | 0 | 0 | 0 | 1 |
Multidrug resistance-associated protein 1 | 0 | 1 | 0 | 2 |
Solute carrier organic anion transporter family member 1A2 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 20 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 6 | 0 | 1 | 0 | 1 |
Solute carrier organic anion transporter family member | 0 | 0 | 0 | 1 |
Solute carrier organic anion transporter family member 1C1 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 11 | 0 | 0 | 0 | 1 |
Solute carrier organic anion transporter family member 1A1 | 0 | 0 | 0 | 1 |
Solute carrier organic anion transporter family member 1B2 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 1 | 0 | 2 |
Solute carrier organic anion transporter family member 1B1 | 0 | 1 | 0 | 2 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |