Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 2 | 0 | 0 | 2 |
Chain A, Beta-lactamase | 2 | 0 | 0 | 2 |
Chain A, 2-oxoglutarate Oxygenase | 2 | 0 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
AR protein | 2 | 0 | 0 | 2 |
apical membrane antigen 1, AMA1 | 2 | 0 | 0 | 2 |
estrogen nuclear receptor alpha | 4 | 0 | 0 | 4 |
Beta-lactamase | 0 | 0 | 0 | 2 |
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | 1 | 0 | 0 | 1 |
DNA polymerase eta isoform 1 | 1 | 0 | 0 | 1 |
DNA polymerase iota isoform a (long) | 1 | 0 | 0 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
DNA polymerase kappa isoform 1 | 1 | 0 | 0 | 1 |
ATP-binding cassette sub-family C member 3 | 0 | 4 | 0 | 4 |
Multidrug resistance-associated protein 4 | 0 | 4 | 0 | 4 |
Bile salt export pump | 0 | 1 | 0 | 1 |
Bile salt export pump | 0 | 5 | 0 | 5 |
Beta-lactamase SHV-1 | 0 | 0 | 0 | 2 |
Beta-lactamase SHV-1 | 0 | 0 | 0 | 2 |
Cytochrome P450 2C9 | 0 | 4 | 0 | 4 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Kappa-type opioid receptor | 0 | 0 | 0 | 2 |
Solute carrier family 15 member 1 | 0 | 2 | 0 | 2 |
Solute carrier family 15 member 1 | 0 | 1 | 0 | 1 |
Cytochrome P450 2J2 | 0 | 3 | 0 | 3 |
B2 metallo-beta-lactamase | 0 | 0 | 0 | 2 |
Solute carrier family 15 member 2 | 0 | 2 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Solute carrier family 15 member 2 | 0 | 2 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 2 |
Canalicular multispecific organic anion transporter 1 | 0 | 4 | 0 | 4 |
Chain A, Avidin | 0 | 0 | 1 | 1 |
Chain A, Protein (streptavidin) | 0 | 0 | 1 | 1 |
Chain B, Protein (streptavidin) | 0 | 0 | 1 | 1 |
Chain A, Streptavidin | 0 | 0 | 1 | 1 |
Chain D, Streptavidin | 0 | 0 | 1 | 1 |
Chain A, Streptavidin | 0 | 0 | 1 | 1 |
Chain D, Streptavidin | 0 | 0 | 1 | 1 |
Chain A, Streptavidin | 0 | 0 | 1 | 1 |
Chain D, Streptavidin | 0 | 0 | 1 | 1 |
Chain A, Streptavidin Complex With Biotin | 0 | 0 | 1 | 1 |
Chain D, Circularly Permuted Core-streptavidin E51/a46 | 0 | 0 | 1 | 1 |
Chain A, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain D, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain A, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain D, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain A, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain D, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain A, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain D, Core-streptavidin | 0 | 0 | 1 | 1 |
Chain A, Avidin | 0 | 0 | 1 | 1 |
Chain A, Streptavidin | 0 | 0 | 1 | 1 |
Chain B, Streptavidin | 0 | 0 | 1 | 1 |
Chain A, Streptavidin | 0 | 0 | 1 | 1 |
Chain B, Streptavidin | 0 | 0 | 1 | 1 |
Chain A, JmjC domain-containing histone demethylation protein 3A | 2 | 0 | 0 | 2 |
RAR-related orphan receptor gamma | 2 | 0 | 0 | 2 |
nonstructural protein 1 | 0 | 1 | 0 | 1 |
green fluorescent protein, partial | 0 | 1 | 0 | 1 |
vitamin D3 receptor isoform VDRA | 1 | 0 | 0 | 1 |
insulin-degrading enzyme isoform 1 | 0 | 0 | 1 | 1 |
Streptavidin | 0 | 0 | 1 | 1 |
Receptor-type tyrosine-protein phosphatase beta | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 1 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase type 2 | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase VIM-11 | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase VIM-2 | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase VIM-19 | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 6 | 0 | 2 | 0 | 2 |
Albumin | 0 | 0 | 2 | 2 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase VIM-13 | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-beta-lactamase VIM-2 | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase Toho-1 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 6 | 0 | 3 | 0 | 3 |
Solute carrier family 22 member 7 | 0 | 1 | 0 | 1 |
Metallo-beta-lactamase | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Metallo-b-lactamase | 0 | 0 | 0 | 1 |
BlaVIM-1 | 0 | 0 | 0 | 1 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 2 | 0 | 2 |
Beta-lactamase | 0 | 0 | 0 | 1 |
Carbapenem-hydrolyzing beta-lactamase KPC | 0 | 0 | 0 | 1 |
Histamine H3 receptor | 0 | 0 | 0 | 1 |
Beta-lactamase class B VIM-2 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 11 | 0 | 2 | 0 | 2 |
Solute carrier family 22 member 8 | 0 | 1 | 0 | 1 |
Beta-lactamase VIM-1 | 0 | 0 | 0 | 1 |
Solute carrier family 22 member 7 | 0 | 1 | 0 | 1 |
Motilin receptor | 0 | 0 | 1 | 1 |
acid sphingomyelinase | 1 | 0 | 0 | 1 |
TDP1 protein | 2 | 0 | 0 | 2 |
GLI family zinc finger 3 | 1 | 0 | 0 | 1 |
estrogen-related nuclear receptor alpha | 2 | 0 | 0 | 2 |
thyroid hormone receptor beta isoform 2 | 2 | 0 | 0 | 2 |
low molecular weight phosphotyrosine protein phosphatase isoform c | 0 | 1 | 0 | 1 |
serine/threonine-protein kinase PLK1 | 1 | 0 | 0 | 1 |
geminin | 2 | 0 | 0 | 2 |
streptokinase A precursor | 0 | 0 | 1 | 1 |
Motilin receptor | 0 | 1 | 1 | 2 |
Rap guanine nucleotide exchange factor 3 | 1 | 0 | 0 | 1 |
30S ribosomal protein S6 | 0 | 2 | 1 | 3 |
30S ribosomal protein S7 | 0 | 2 | 1 | 3 |
50S ribosomal protein L15 | 0 | 2 | 1 | 3 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Cytochrome P450 3A4 | 0 | 3 | 0 | 3 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
50S ribosomal protein L10 | 0 | 2 | 1 | 3 |
50S ribosomal protein L11 | 0 | 2 | 1 | 3 |
50S ribosomal protein L7/L12 | 0 | 2 | 1 | 3 |
50S ribosomal protein L19 | 0 | 2 | 1 | 3 |
50S ribosomal protein L1 | 0 | 2 | 1 | 3 |
50S ribosomal protein L20 | 0 | 2 | 1 | 3 |
50S ribosomal protein L27 | 0 | 2 | 1 | 3 |
50S ribosomal protein L28 | 0 | 2 | 1 | 3 |
50S ribosomal protein L29 | 0 | 2 | 1 | 3 |
50S ribosomal protein L31 | 0 | 2 | 1 | 3 |
50S ribosomal protein L31 type B | 0 | 2 | 1 | 3 |
50S ribosomal protein L32 | 0 | 2 | 1 | 3 |
50S ribosomal protein L33 | 0 | 2 | 1 | 3 |
50S ribosomal protein L34 | 0 | 2 | 1 | 3 |
50S ribosomal protein L35 | 0 | 2 | 1 | 3 |
50S ribosomal protein L36 | 0 | 2 | 1 | 3 |
30S ribosomal protein S10 | 0 | 2 | 1 | 3 |
30S ribosomal protein S11 | 0 | 2 | 1 | 3 |
30S ribosomal protein S12 | 0 | 2 | 1 | 3 |
30S ribosomal protein S13 | 0 | 2 | 1 | 3 |
30S ribosomal protein S16 | 0 | 2 | 1 | 3 |
30S ribosomal protein S18 | 0 | 2 | 1 | 3 |
30S ribosomal protein S19 | 0 | 2 | 1 | 3 |
30S ribosomal protein S20 | 0 | 2 | 1 | 3 |
30S ribosomal protein S2 | 0 | 2 | 1 | 3 |
30S ribosomal protein S3 | 0 | 2 | 1 | 3 |
30S ribosomal protein S4 | 0 | 2 | 1 | 3 |
30S ribosomal protein S5 | 0 | 2 | 1 | 3 |
30S ribosomal protein S8 | 0 | 2 | 1 | 3 |
30S ribosomal protein S9 | 0 | 2 | 1 | 3 |
50S ribosomal protein L13 | 0 | 2 | 1 | 3 |
50S ribosomal protein L14 | 0 | 2 | 1 | 3 |
50S ribosomal protein L16 | 0 | 2 | 1 | 3 |
50S ribosomal protein L23 | 0 | 2 | 1 | 3 |
30S ribosomal protein S15 | 0 | 2 | 1 | 3 |
50S ribosomal protein L17 | 0 | 2 | 1 | 3 |
50S ribosomal protein L21 | 0 | 2 | 1 | 3 |
50S ribosomal protein L30 | 0 | 2 | 1 | 3 |
50S ribosomal protein L6 | 0 | 2 | 1 | 3 |
30S ribosomal protein S14 | 0 | 2 | 1 | 3 |
30S ribosomal protein S17 | 0 | 2 | 1 | 3 |
30S ribosomal protein S1 | 0 | 2 | 1 | 3 |
50S ribosomal protein L18 | 0 | 2 | 1 | 3 |
60 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Chitinase B | 0 | 1 | 0 | 1 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Low molecular weight phosphotyrosine protein phosphatase | 0 | 1 | 0 | 1 |
50S ribosomal protein L2 | 0 | 2 | 1 | 3 |
50S ribosomal protein L3 | 0 | 2 | 1 | 3 |
50S ribosomal protein L24 | 0 | 2 | 1 | 3 |
50S ribosomal protein L4 | 0 | 2 | 1 | 3 |
50S ribosomal protein L22 | 0 | 2 | 1 | 3 |
10 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
50S ribosomal protein L5 | 0 | 2 | 1 | 3 |
30S ribosomal protein S21 | 0 | 2 | 1 | 3 |
50S ribosomal protein L25 | 0 | 2 | 1 | 3 |
Potassium voltage-gated channel subfamily H member 2 | 0 | 1 | 0 | 1 |
Cytochrome P450 1B1 | 0 | 1 | 0 | 1 |
Thiosulfate sulfurtransferase | 0 | 1 | 0 | 1 |
Lanosterol 14-alpha demethylase | 0 | 1 | 0 | 1 |
50S ribosomal protein L36 2 | 0 | 2 | 1 | 3 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
10 kDa chaperonin | 0 | 1 | 0 | 1 |
Multidrug and toxin extrusion protein 1 | 0 | 1 | 0 | 1 |
Menin | 0 | 0 | 1 | 1 |
Lecithin retinol acyltransferase | 0 | 1 | 0 | 1 |
Lethal factor | 0 | 1 | 0 | 1 |
Protein Rev | 0 | 0 | 1 | 1 |
Aminoglycoside 3'-phosphotransferase | 0 | 0 | 0 | 1 |
Tyrosyl-DNA phosphodiesterase 1 | 0 | 1 | 0 | 1 |
Sialidase-4 | 0 | 1 | 0 | 1 |
Sialidase-1 | 0 | 1 | 0 | 1 |
Sialidase-3 | 0 | 1 | 0 | 1 |
Sialidase-2 | 0 | 1 | 0 | 1 |
Luciferase | 1 | 0 | 0 | 1 |
thioredoxin reductase | 1 | 0 | 0 | 1 |
15-lipoxygenase, partial | 1 | 0 | 0 | 1 |
phosphopantetheinyl transferase | 1 | 0 | 0 | 1 |
ATAD5 protein, partial | 1 | 0 | 0 | 1 |
NFKB1 protein, partial | 1 | 0 | 0 | 1 |
GLS protein | 1 | 0 | 0 | 1 |
nuclear receptor subfamily 1, group I, member 3 | 2 | 0 | 0 | 2 |
EWS/FLI fusion protein | 2 | 0 | 0 | 2 |
nonstructural protein 1 | 1 | 0 | 0 | 1 |
retinoic acid nuclear receptor alpha variant 1 | 2 | 0 | 0 | 2 |
pregnane X nuclear receptor | 2 | 0 | 0 | 2 |
G | 2 | 0 | 0 | 2 |
Parkin | 1 | 0 | 0 | 1 |
bromodomain adjacent to zinc finger domain 2B | 1 | 0 | 0 | 1 |
arylsulfatase A | 1 | 0 | 0 | 1 |
euchromatic histone-lysine N-methyltransferase 2 | 1 | 0 | 0 | 1 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 1 | 0 | 0 | 1 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | 1 | 0 | 0 | 1 |
Bloom syndrome protein isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 2D6 isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 2C19 precursor | 1 | 0 | 0 | 1 |
cytochrome P450 2C9 precursor | 1 | 0 | 0 | 1 |
chromobox protein homolog 1 | 1 | 0 | 0 | 1 |
potassium voltage-gated channel subfamily H member 2 isoform d | 1 | 0 | 0 | 1 |
ubiquitin carboxyl-terminal hydrolase 2 isoform a | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 1 | 0 | 0 | 1 |
muscleblind-like protein 1 isoform 1 | 1 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
muscarinic acetylcholine receptor M1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 1 | 0 | 0 | 1 |
Prostaglandin G/H synthase 1 | 0 | 1 | 0 | 1 |
Prostaglandin G/H synthase 2 | 0 | 1 | 0 | 1 |
Interferon beta | 2 | 0 | 0 | 2 |
HLA class I histocompatibility antigen, B alpha chain | 2 | 0 | 0 | 2 |
Prostaglandin G/H synthase 1 | 0 | 1 | 0 | 1 |
Polyunsaturated fatty acid 5-lipoxygenase | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit delta | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 1 | 0 | 0 | 1 |
Prostaglandin G/H synthase 1 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 1 | 0 | 0 | 1 |
Prostaglandin G/H synthase 2 | 0 | 1 | 0 | 1 |
Prostaglandin G/H synthase 2 | 0 | 1 | 0 | 1 |
Alpha-synuclein | 1 | 0 | 0 | 1 |
Histamine H2 receptor | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-3 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-2 | 1 | 0 | 0 | 1 |
Disintegrin and metalloproteinase domain-containing protein 17 | 1 | 0 | 0 | 1 |
TAR DNA-binding protein 43 | 1 | 0 | 0 | 1 |
Prostaglandin G/H synthase 1 | 0 | 1 | 0 | 1 |
GABA theta subunit | 1 | 0 | 0 | 1 |
Inositol hexakisphosphate kinase 1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit epsilon | 1 | 0 | 0 | 1 |
cytochrome P450 2C9, partial | 2 | 0 | 0 | 2 |
ATP-dependent phosphofructokinase | 1 | 0 | 0 | 1 |
progesterone receptor | 1 | 0 | 0 | 1 |
cytochrome P450 family 3 subfamily A polypeptide 4 | 1 | 0 | 0 | 1 |
cytochrome P450 2D6 | 1 | 0 | 0 | 1 |
peroxisome proliferator-activated receptor delta | 1 | 0 | 0 | 1 |
thyroid stimulating hormone receptor | 1 | 0 | 0 | 1 |
Nuclear receptor subfamily 1 group I member 2 | 0 | 0 | 1 | 1 |
Cytochrome P450 1A2 | 0 | 1 | 0 | 1 |
Cytochrome P450 2D6 | 0 | 1 | 0 | 1 |
Cytochrome P450 2C19 | 0 | 1 | 0 | 1 |
Genome polyprotein | 0 | 0 | 1 | 2 |
Genome polyprotein | 0 | 0 | 1 | 1 |
Genome polyprotein | 0 | 0 | 1 | 1 |
Fumarate hydratase | 1 | 0 | 0 | 1 |
polyprotein | 1 | 0 | 0 | 1 |
lamin isoform A-delta10 | 1 | 0 | 0 | 1 |
Butyrophilin subfamily 3 member A1 | 0 | 0 | 1 | 2 |
Carbonic anhydrase 12 | 0 | 1 | 0 | 1 |
Geranylgeranyl pyrophosphate synthase | 0 | 2 | 0 | 3 |
Carbonic anhydrase 1 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 2 | 0 | 1 | 0 | 1 |
72 kDa type IV collagenase | 0 | 1 | 0 | 1 |
Farnesyl pyrophosphate synthase | 0 | 2 | 0 | 2 |
Matrix metalloproteinase-9 | 0 | 1 | 0 | 1 |
Neutrophil collagenase | 0 | 1 | 0 | 1 |
Farnesyl diphosphate synthase | 0 | 1 | 0 | 1 |
Matrix metalloproteinase-14 | 0 | 1 | 0 | 1 |
Farnesyl pyrophosphate synthase | 0 | 2 | 0 | 2 |
Geranylgeranyl pyrophosphate synthase | 0 | 2 | 0 | 2 |
Carbonic anhydrase 9 | 0 | 1 | 0 | 1 |
Farnesyl pyrophosphate synthase | 0 | 1 | 0 | 1 |
H | 0 | 1 | 0 | 1 |
Carbonic anhydrase 14 | 0 | 1 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |