Assay ID | Title | Year | Journal | Article |
AID1347154 | Primary screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1508630 | Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident proteome: Secreted ER Calcium Modulated Protein (SERCaMP) assay | 2021 | Cell reports, 04-27, Volume: 35, Issue:4
| A target-agnostic screen identifies approved drugs to stabilize the endoplasmic reticulum-resident proteome. |
AID414232 | Inhibition of human group 6A iPLA2 by mixed micelle-based assay | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes. |
AID414231 | Inhibition of human group 4A cPLA2 by mixed micelle-based assay | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes. |
AID646965 | Inhibition of human endothelial lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate at 50 uM after 1 hr by vesicle assay | 2012 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 22, Issue:3
| Design and synthesis of boronic acid inhibitors of endothelial lipase. |
AID414230 | Inhibition of human group 5 sPLA2 at 0.091 mol fraction by mixed micelle-based assay | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes. |
AID414228 | Inhibition of human group 4A cPLA2 at 0.091 mol fraction by mixed micelle-based assay | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes. |
AID414229 | Inhibition of human group 6A iPLA2 at 0.091 mol fraction by mixed micelle-based assay | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes. |
AID158962 | Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uM | 2000 | Bioorganic & medicinal chemistry letters, Feb-07, Volume: 10, Issue:3
| Synthesis and enzyme inhibitory activities of a series of lipidic diamine and aminoalcohol derivatives on cytosolic and secretory phospholipases A2. |
AID646966 | Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate at 50 uM after 1 hr by vesicle assay | 2012 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 22, Issue:3
| Design and synthesis of boronic acid inhibitors of endothelial lipase. |
AID158963 | Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uM | 2000 | Bioorganic & medicinal chemistry letters, Feb-07, Volume: 10, Issue:3
| Synthesis and enzyme inhibitory activities of a series of lipidic diamine and aminoalcohol derivatives on cytosolic and secretory phospholipases A2. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |