| Assay ID | Title | Year | Journal | Article |
|---|
| AID239678 | In vitro inhibition of [3H]nisoxetine binding to norepinephrine transporter expressed in human kidney cells | 2005 | Journal of medicinal chemistry, Jun-30, Volume: 48, Issue:13
| Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. |
| AID344678 | Displacement of [3H]MADAM from SERT in rat brain cortex membrane | 2008 | Bioorganic & medicinal chemistry, Oct-01, Volume: 16, Issue:19
| Docking study, synthesis, and in vitro evaluation of fluoro-MADAM derivatives as SERT ligands for PET imaging. |
| AID456161 | Displacement of [3H]citalopram from human cloned SERT expressed in HEK293 cells | 2010 | Bioorganic & medicinal chemistry, Jan-01, Volume: 18, Issue:1
| Synthesis and in vitro evaluation of fluorinated diphenyloxide derivatives and sulfur analogs as serotonin transporter ligands. |
| AID239682 | In vitro inhibition of [3H]citalopram binding to human serotonin transporter expressed in human HEK293 cells | 2005 | Journal of medicinal chemistry, Jun-30, Volume: 48, Issue:13
| Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. |
| AID344682 | Displacement of [3H]GBR-12935 from human cloned DAT expressed in HEK293 cells | 2008 | Bioorganic & medicinal chemistry, Oct-01, Volume: 16, Issue:19
| Docking study, synthesis, and in vitro evaluation of fluoro-MADAM derivatives as SERT ligands for PET imaging. |
| AID145540 | Inhibition of [3H]nisoxetine binding to norepinephrine transporter (NET) of rat cortical homogenates | 2002 | Journal of medicinal chemistry, Mar-14, Volume: 45, Issue:6
| Substituted diphenyl sulfides as selective serotonin transporter ligands: synthesis and in vitro evaluation. |
| AID361595 | Displacement of [3H]citalopram from human SERT expressed in HEK293 cells | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| 3-(4-(6-Fluoroalkoxy-3,4-dihydroisoquinoline-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitriles for SERT imaging: chemical synthesis, evaluation in vitro and radiofluorination. |
| AID239411 | In vitro displacement of [3H]nisoxetine from human norepinephrine transporter expressed in HEK293 cells | 2005 | Journal of medicinal chemistry, Apr-07, Volume: 48, Issue:7
| Fluorinated diaryl sulfides as serotonin transporter ligands: synthesis, structure-activity relationship study, and in vivo evaluation of fluorine-18-labeled compounds as PET imaging agents. |
| AID65810 | Inhibition of [3H]-GBR-12,935 binding to dopamine transporter (DAT) of rat striatal membranes | 2002 | Journal of medicinal chemistry, Mar-14, Volume: 45, Issue:6
| Substituted diphenyl sulfides as selective serotonin transporter ligands: synthesis and in vitro evaluation. |
| AID200776 | In vitro binding affinity in LLC-PK1 cells by SERT binding assay by using [125I]IDAM as a radioligand | 2002 | Journal of medicinal chemistry, Oct-10, Volume: 45, Issue:21
| New PET imaging agent for the serotonin transporter: [(18)F]ACF (2-[(2-amino-4-chloro-5-fluorophenyl)thio]-N,N-dimethyl-benzenmethanamine). |
| AID309075 | Displacement of [3H]WIN-35428 from DAT in rat brain | 2007 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 17, Issue:17
| New fluoro-diphenylchalcogen derivatives to explore the serotonin transporter by PET. |
| AID309074 | Displacement of [3H]paroxetine from SERT in rat brain | 2007 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 17, Issue:17
| New fluoro-diphenylchalcogen derivatives to explore the serotonin transporter by PET. |
| AID239293 | In vitro displacement of [3H]GBR-12935 from human dopamine transporter expressed in HEK293 cells | 2005 | Journal of medicinal chemistry, Apr-07, Volume: 48, Issue:7
| Fluorinated diaryl sulfides as serotonin transporter ligands: synthesis, structure-activity relationship study, and in vivo evaluation of fluorine-18-labeled compounds as PET imaging agents. |
| AID253263 | Partition coefficient (logP) | 2005 | Journal of medicinal chemistry, Jun-30, Volume: 48, Issue:13
| Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. |
| AID344683 | Displacement of [3H]nisoxetine from human cloned NET expressed in HEK293 cells | 2008 | Bioorganic & medicinal chemistry, Oct-01, Volume: 16, Issue:19
| Docking study, synthesis, and in vitro evaluation of fluoro-MADAM derivatives as SERT ligands for PET imaging. |
| AID261750 | Inhibitory activity against DAT | 2006 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 16, Issue:5
| Synthesis and in vitro evaluation of novel derivatives of diphenylsulfide as serotonin transporter ligands. |
| AID361596 | Displacement of [3H]paroxetine from human SERT expressed in HEK293 cells | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| 3-(4-(6-Fluoroalkoxy-3,4-dihydroisoquinoline-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitriles for SERT imaging: chemical synthesis, evaluation in vitro and radiofluorination. |
| AID309076 | Displacement of [3H]nisoxetine from NET in rat brain | 2007 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 17, Issue:17
| New fluoro-diphenylchalcogen derivatives to explore the serotonin transporter by PET. |
| AID239342 | In vitro displacement of [3H]paroxetine from human serotonin transporter expressed in HEK293 cells | 2005 | Journal of medicinal chemistry, Apr-07, Volume: 48, Issue:7
| Fluorinated diaryl sulfides as serotonin transporter ligands: synthesis, structure-activity relationship study, and in vivo evaluation of fluorine-18-labeled compounds as PET imaging agents. |
| AID261748 | Displacement of [3H]paroxetine from SERT | 2006 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 16, Issue:5
| Synthesis and in vitro evaluation of novel derivatives of diphenylsulfide as serotonin transporter ligands. |
| AID239662 | In vitro inhibition of [3H]WIN-35428 binding to human dopamine transporter expressed in canine kidney cells | 2005 | Journal of medicinal chemistry, Jun-30, Volume: 48, Issue:13
| Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. |
| AID229007 | Inhibition of [3H]paroxetine binding to serotonin transporter (SERT) of rat cortical membrane | 2002 | Journal of medicinal chemistry, Mar-14, Volume: 45, Issue:6
| Substituted diphenyl sulfides as selective serotonin transporter ligands: synthesis and in vitro evaluation. |
| AID261751 | Inhibitory activity against NET | 2006 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 16, Issue:5
| Synthesis and in vitro evaluation of novel derivatives of diphenylsulfide as serotonin transporter ligands. |
| AID344684 | Partition coefficient, log P in n-octanol/0.02 M phosphate buffer at pH 7.4 | 2008 | Bioorganic & medicinal chemistry, Oct-01, Volume: 16, Issue:19
| Docking study, synthesis, and in vitro evaluation of fluoro-MADAM derivatives as SERT ligands for PET imaging. |
| AID344681 | Displacement of [3H]paroxetine from SERT in rat brain cortex membrane | 2008 | Bioorganic & medicinal chemistry, Oct-01, Volume: 16, Issue:19
| Docking study, synthesis, and in vitro evaluation of fluoro-MADAM derivatives as SERT ligands for PET imaging. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |