| Assay ID | Title | Year | Journal | Article |
|---|
| AID213285 | Compound was tested for inhibition of thrombin | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID1558644 | Inhibition of human plasmin | 2020 | Journal of medicinal chemistry, 02-27, Volume: 63, Issue:4
| Fibrinolysis Inhibitors: Potential Drugs for the Treatment and Prevention of Bleeding. |
| AID267981 | Inhibition of uPA | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| AID159999 | Compound was tested for inhibition of plasma kallikrein | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID164134 | Compound was tested for inhibition of protein Ca | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID213514 | Compound was tested for inhibition of tryptase | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID267984 | Inhibition of f10a | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| AID215190 | Compound was tested for inhibition of trypsin | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID1265736 | Inhibition of uPA (unknown origin) | 2015 | Journal of medicinal chemistry, Dec-10, Volume: 58, Issue:23
| Discovery and SAR of Novel and Selective Inhibitors of Urokinase Plasminogen Activator (uPA) with an Imidazo[1,2-a]pyridine Scaffold. |
| AID158487 | Compound was tested for inhibition of plasminogen activator urokinase (microPa) | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID644382 | Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior substrate addition measured for 10 mins by spectrophotometry | 2012 | Bioorganic & medicinal chemistry, Feb-15, Volume: 20, Issue:4
| Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA). |
| AID644389 | Selectivity ratio of Ki for recombinant tPA to Ki for human uPA | 2012 | Bioorganic & medicinal chemistry, Feb-15, Volume: 20, Issue:4
| Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA). |
| AID51334 | Compound was tested for inhibition of Coagulation factor X | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID644385 | Inhibition of human plasma thrombin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior substrate addition measured for 10 mins by spectrophotometry | 2012 | Bioorganic & medicinal chemistry, Feb-15, Volume: 20, Issue:4
| Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA). |
| AID644384 | Inhibition of recombinant tPA using H-D-Ile-Pro-Arg-pNA.2HCl as substrate preincubated for 15 mins prior substrate addition measured for 10 mins by spectrophotometry | 2012 | Bioorganic & medicinal chemistry, Feb-15, Volume: 20, Issue:4
| Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA). |
| AID267980 | Inhibition of matriptase | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| AID267982 | Inhibition of plasmin | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| AID267983 | Inhibition of thrombin | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| AID644383 | Inhibition of human plasma plasmin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior substrate addition measured for 10 mins by spectrophotometry | 2012 | Bioorganic & medicinal chemistry, Feb-15, Volume: 20, Issue:4
| Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA). |
| AID312586 | Inhibition of uPA | 2008 | Journal of medicinal chemistry, Jan-24, Volume: 51, Issue:2
| Fragment-based discovery of mexiletine derivatives as orally bioavailable inhibitors of urokinase-type plasminogen activator. |
| AID158138 | Compound was tested for inhibition of plasmin | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID228984 | Compound was tested for inhibition of sc-tissue plasminogen activator | 1999 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 9, Issue:21
| 3-Amidinophenylalanine-based inhibitors of urokinase. |
| AID1798368 | Determination of Inhibition Constants from Article 10.1021/jm051272l: \\Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase.\\ | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |